Proteins > DNA dC->dU-editing enzyme APOBEC-3F isoform a
Page last updated: 2024-08-07 21:03:04

DNA dC->dU-editing enzyme APOBEC-3F isoform a

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (464)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tyrphostin ag957Homo sapiens (human)Potency17.782810
aristolochic acid iHomo sapiens (human)Potency7.943310
bendiocarbHomo sapiens (human)Potency3.162310
benzo(a)pyreneHomo sapiens (human)Potency4.466810
clioquinolHomo sapiens (human)Potency22.387210
coumaphosHomo sapiens (human)Potency2.818410
dipyridamoleHomo sapiens (human)Potency22.387210
ebselenHomo sapiens (human)Potency35.481310
ellipticineHomo sapiens (human)Potency19.149830
beta-thujaplicinHomo sapiens (human)Potency31.622810
nsc 664704Homo sapiens (human)Potency35.481310
ppm 18Homo sapiens (human)Potency10.000010
vorinostatHomo sapiens (human)Potency7.079510
vincaHomo sapiens (human)Potency11.220210
reserpineHomo sapiens (human)Potency31.622810
chlorquinaldolHomo sapiens (human)Potency6.309610
benzanthroneHomo sapiens (human)Potency15.848910
syrosingopineHomo sapiens (human)Potency22.387210
1-naphthylphenylamineHomo sapiens (human)Potency19.952610
michler's ketoneHomo sapiens (human)Potency2.260920
pyronineHomo sapiens (human)Potency16.320520
n,n,n',n'-tetramethyl-4,4'-methylenedianilineHomo sapiens (human)Potency3.162310
2-aminoanthraquinoneHomo sapiens (human)Potency14.125410
2,4-dihydroxybenzophenoneHomo sapiens (human)Potency3.162310
4'-(chloroacetyl)acetanilideHomo sapiens (human)Potency5.623410
hematoxylinHomo sapiens (human)Potency31.622810
nitrophenideHomo sapiens (human)Potency6.309610
2-anthramineHomo sapiens (human)Potency3.548110
n,n'-diacetylbenzidineHomo sapiens (human)Potency6.309610
2-amino-7-nitrofluoreneHomo sapiens (human)Potency11.220210
ethyl violetHomo sapiens (human)Potency5.623410
6-chrysenamineHomo sapiens (human)Potency6.309610
3-aminofluorantheneHomo sapiens (human)Potency3.960930
nsc 3852Homo sapiens (human)Potency4.441110
nitroxolineHomo sapiens (human)Potency22.387210
hyaluronoglucosaminidaseHomo sapiens (human)Potency35.481310
Bis(2-furanylmethyl) disulfideHomo sapiens (human)Potency35.481310
fenestrelHomo sapiens (human)Potency7.079510
n-acetylamphetamineHomo sapiens (human)Potency2.818410
1-(4-carboxyethylphenyl)-3,3-dimethyltriazeneHomo sapiens (human)Potency0.562310
thymolphthaleinHomo sapiens (human)Potency3.548110
2-n-octyl-4-isothiazolin-3-oneHomo sapiens (human)Potency3.162310
s-2678Homo sapiens (human)Potency25.118910
dinalineHomo sapiens (human)Potency22.387210
butoconazole nitrateHomo sapiens (human)Potency35.481310
nsc 330770Homo sapiens (human)Potency7.509630
topotecan hydrochlorideHomo sapiens (human)Potency35.481310
saquinavir monomethanesulfonateHomo sapiens (human)Potency35.481310
5-AminoacenaphtheneHomo sapiens (human)Potency22.387210
betulinic acidHomo sapiens (human)Potency6.309610
nile redHomo sapiens (human)Potency1.778310
dibenzthioneHomo sapiens (human)Potency5.623410
dabiHomo sapiens (human)Potency35.481310
prazosin hydrochlorideHomo sapiens (human)Potency28.183810
2,2',2''-terpyridineHomo sapiens (human)Potency18.745620
thioxoloneHomo sapiens (human)Potency35.481310
9-methoxyellipticineHomo sapiens (human)Potency5.623410
coumarin 153Homo sapiens (human)Potency4.466810
methyl fluorone blackHomo sapiens (human)Potency3.162310
9-hydroxyphenylfluoronHomo sapiens (human)Potency35.481310
3-aminophenoxazoneHomo sapiens (human)Potency31.622810
5-nitro-1,10-phenanthrolineHomo sapiens (human)Potency35.481310
ergocornineHomo sapiens (human)Potency15.848910
fangchinolineHomo sapiens (human)Potency31.622810
agroclavineHomo sapiens (human)Potency15.848910
5-hydroxybenzofuran-2-oneHomo sapiens (human)Potency35.481310
1-(10h-phenothiazin-2-yl)ethanoneHomo sapiens (human)Potency11.220210
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)Potency6.309610
1-(2-thiazolylazo)-2-naphtholHomo sapiens (human)Potency22.387210
wr 158122Homo sapiens (human)Potency25.118910
difenpiramideHomo sapiens (human)Potency35.481310
3-chloro-6-hydrazino-pyridazineHomo sapiens (human)Potency35.481310
paxillineHomo sapiens (human)Potency31.622810
desethylterbuthylazineHomo sapiens (human)Potency10.000010
n-(phenylthio)-epsilon-caprolactamHomo sapiens (human)Potency35.481310
phacidinHomo sapiens (human)Potency35.481310
c 1303Homo sapiens (human)Potency35.481310
3'-deamino-3'-hydroxydaunorubicinHomo sapiens (human)Potency22.387210
purpactin aHomo sapiens (human)Potency35.481310
alpha-ergocryptineHomo sapiens (human)Potency17.782810
epiberberineHomo sapiens (human)Potency35.481310
2-phenyl-4-oxohydroquinolineHomo sapiens (human)Potency1.900820
2,3,4,4'-tetramethoxy-1,1'-biphenylHomo sapiens (human)Potency2.863120
sb 216763Homo sapiens (human)Potency11.166030
raubasineHomo sapiens (human)Potency14.125410
n-acetyl-1-aminopyreneHomo sapiens (human)Potency22.387210
methyl reserpateHomo sapiens (human)Potency28.183810
nsc 95397Homo sapiens (human)Potency3.548110
1,5-bis(2-methoxyphenyl)penta-1,4-dien-3-oneHomo sapiens (human)Potency4.379730
sirodesmin aHomo sapiens (human)Potency4.900520
pinafideHomo sapiens (human)Potency25.118910
nsc 680410Homo sapiens (human)Potency14.096020
nsc689857Homo sapiens (human)Potency19.373620
nsc697923Homo sapiens (human)Potency3.981110
4-(4-chlorophenyl)-1-methyl-2-(methylthio)-6-oxo-5-pyrimidinecarbonitrileHomo sapiens (human)Potency2.818410
discretamineHomo sapiens (human)Potency11.836220
mometasone furoateHomo sapiens (human)Potency25.118910
grosheiminHomo sapiens (human)Potency6.309610
menadione sodium bisulfite, trihydrateHomo sapiens (human)Potency6.309610
1-[4-amino-3-[2-(1-pyrrolidinyl)ethylthio]-5-thieno[2,3-c]isothiazolyl]ethanoneHomo sapiens (human)Potency10.000010
3-bromo-N-[2-(4-nitroanilino)ethyl]benzamideHomo sapiens (human)Potency15.848910
2-diphenylphosphinopyridineHomo sapiens (human)Potency35.481310
chalconeHomo sapiens (human)Potency6.309610
averufinHomo sapiens (human)Potency14.696630
dibenzylidene acetoneHomo sapiens (human)Potency3.548110
2-[5-(4-butoxyphenyl)-2-tetrazolyl]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency6.273310
3-amino-N-cyclopentyl-6-thiophen-2-yl-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency25.118910
4-[3-(1,3-dioxo-2-isoindolyl)propylamino]-2-methylisoindole-1,3-dioneHomo sapiens (human)Potency24.189430
6-(3,4-dimethoxyphenyl)-4-methoxy-1,3-dimethyl-8-cyclohepta[c]furanoneHomo sapiens (human)Potency3.548110
2-amino-3-cyano-7-(dimethylamino)-4-(3-methoxy-4,5-methylenedioxyphenyl)-4h-chromeneHomo sapiens (human)Potency22.387210
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
2-(3-methylphenyl)sulfonyl-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetonitrileHomo sapiens (human)Potency8.912510
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency22.387210
LSM-28489Homo sapiens (human)Potency35.481310
6-amino-1-(4-fluorophenyl)-3-methyl-4-thiophen-2-yl-5-pyrazolo[3,4-b]pyridinecarbonitrileHomo sapiens (human)Potency35.481310
N2-(1H-benzimidazol-2-yl)benzene-1,2-diamineHomo sapiens (human)Potency2.238710
7-ethoxy-9-nitro-5H-benzo[b][1,4]benzoxazepin-6-oneHomo sapiens (human)Potency25.740020
2-amino-4-(5-methyl-2-furanyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrileHomo sapiens (human)Potency35.481310
7-(diethylamino)-2-oxo-1-benzopyran-3-carbonitrileHomo sapiens (human)Potency3.981110
2-(8-quinolinylthio)acetic acidHomo sapiens (human)Potency17.782810
N-[3-(4-oxo-3,1-benzoxazin-2-yl)phenyl]benzamideHomo sapiens (human)Potency2.818410
n-phenyl-n'-2-pyridylthioureaHomo sapiens (human)Potency22.387210
5-(4-chlorophenyl)-3H-thieno[2,3-d]pyrimidine-4-thioneHomo sapiens (human)Potency3.548110
5-[[5-(diethylamino)-2-furanyl]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dioneHomo sapiens (human)Potency2.136320
4-(4-fluorophenyl)-3H-thiazole-2-thioneHomo sapiens (human)Potency25.118910
N-(2-chlorophenyl)hydrazine-1-carbothioamideHomo sapiens (human)Potency5.623410
1-(3-fluorophenyl)-3-(2-pyridinylmethyl)thioureaHomo sapiens (human)Potency25.118910
3,4,5-trimethoxybenzoic acid [(3,5-dimethyl-4-oxo-1-cyclohexa-2,5-dienylidene)amino] esterHomo sapiens (human)Potency22.387210
1-spiro[2,4-dihydroisoquinoline-3,1'-cyclohexane]thioneHomo sapiens (human)Potency22.387210
6-(4-morpholinyl)naphthalene-2,3-dicarbonitrileHomo sapiens (human)Potency35.481310
6-ethyl-5-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-oneHomo sapiens (human)Potency7.079510
5,6-dimethyl-N-(3-pyridinylmethyl)-4-thieno[2,3-d]pyrimidinamineHomo sapiens (human)Potency2.511910
2-[2-[[benzamido(sulfanylidene)methyl]amino]-4-thiazolyl]acetic acid ethyl esterHomo sapiens (human)Potency28.183810
N-(4-hydroxyphenyl)-3-methoxy-2-naphthalenecarboxamideHomo sapiens (human)Potency35.481310
3-methyl-7-(phenylmethyl)-8-(propan-2-ylthio)purine-2,6-dioneHomo sapiens (human)Potency14.125410
N-(4-methylphenyl)carbamic acid (cyclopentylideneamino) esterHomo sapiens (human)Potency17.782810
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency35.481310
2-(ethylthio)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency3.548110
4-(3-methylphenyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency2.818410
4,5-dimethyl-2-[4-(3-nitrophenyl)-2-thiazolyl]-1H-pyrazol-3-oneHomo sapiens (human)Potency35.481310
4,5-dimethylcyclopenta[c]quinolizine-1,2-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency19.952610
1,4,8-trimethyl-12-quinolino[2,3-b]quinolinamineHomo sapiens (human)Potency7.079510
N-[[(6-methoxy-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency10.000010
1-[(2,4-dichlorophenyl)methyl]-3-phenylthioureaHomo sapiens (human)Potency22.387210
N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency35.481310
N-(2,3-dihydro-1H-inden-5-yl)-2-methyl-3-nitrobenzamideHomo sapiens (human)Potency0.562310
3-amino-2-(4-methoxyphenyl)-7-nitro-1-oxo-4-isoquinolinecarbonitrileHomo sapiens (human)Potency12.589310
1-ethyl-3-(4-methylphenyl)sulfonylthioureaHomo sapiens (human)Potency14.125410
2-(2-furanyl)-3-(4-methylphenyl)imidazo[4,5-b]quinoxalineHomo sapiens (human)Potency19.952610
N2-(4-fluorophenyl)-6-(3-methyl-2-benzofuranyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency25.118910
curcuminHomo sapiens (human)Potency22.387210
N-(3-chloro-4-methylphenyl)-2-(2-formylphenoxy)acetamideHomo sapiens (human)Potency11.220210
1-(4-bromophenyl)-3-(2-fluorophenyl)thioureaHomo sapiens (human)Potency35.481310
2-[[2-[4-(4-chlorophenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-ethyl-4-quinazolinoneHomo sapiens (human)Potency5.623410
2-(4-ethoxyphenyl)-3,4-dimethyl-7-[2-(1-pyrrolidinyl)ethylthio]pyrazolo[3,4-d]pyridazineHomo sapiens (human)Potency22.387210
3-amino-2-[(4-methoxyanilino)-oxomethyl]-4-(4-methoxyphenyl)-6-methyl-5-thieno[2,3-b]pyridinecarboxylic acid ethyl esterHomo sapiens (human)Potency2.802220
1-[[(5-bromo-2-furanyl)-oxomethyl]amino]-3-(2,5-dimethylphenyl)thioureaHomo sapiens (human)Potency6.309610
1-[[[2-(2,4-dichlorophenyl)-4-quinolinyl]-oxomethyl]amino]-3-phenylureaHomo sapiens (human)Potency15.848910
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency22.387210
5-(4-bromophenyl)-N-[[(2-propyl-5-tetrazolyl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
[3-amino-6-thiophen-2-yl-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinyl]-cyclopropylmethanoneHomo sapiens (human)Potency1.141730
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency10.000010
N-[4-(1-pyrrolidinylsulfonyl)phenyl]-2-thiophen-2-ylacetamideHomo sapiens (human)Potency6.309610
3-(4-chlorophenyl)-5-propyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneHomo sapiens (human)Potency14.125410
N2,N7-bis(2,5-dimethylphenyl)-9H-fluorene-2,7-disulfonamideHomo sapiens (human)Potency35.481310
5-nitro-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.548110
2-[(3-cyano-6-methoxy-2-quinolinyl)thio]-N-(2-methyl-1,3-benzothiazol-5-yl)acetamideHomo sapiens (human)Potency21.284330
1-[(7,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-furanylmethyl)-3-(2-methoxyphenyl)thioureaHomo sapiens (human)Potency6.309610
3-pyridinecarboxylic acid [2-(2-furanyl)-4-oxo-1-benzopyran-3-yl] esterHomo sapiens (human)Potency0.631010
2-methyl-N-(4-oxo-2-sulfanylidene-3-thiazolidinyl)benzamideHomo sapiens (human)Potency35.481310
1-[1-ethyl-4-[4-(4-methoxyphenyl)-1-piperazinyl]-6-methyl-2-sulfanylidene-5-pyrimidinyl]ethanoneHomo sapiens (human)Potency10.000010
3-[[[2-(3-methylphenyl)-4-quinolinyl]-oxomethyl]amino]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency19.952610
N-(2-furanylmethyl)-5-methyl-4-phenyl-3-thiophenecarboxamideHomo sapiens (human)Potency17.782810
propanoic acid [4-[[2-furanyl(oxo)methyl]amino]phenyl] esterHomo sapiens (human)Potency6.309610
N-[[3-chloro-2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-methoxy-3-nitrobenzamideHomo sapiens (human)Potency5.623410
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideHomo sapiens (human)Potency5.623410
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineHomo sapiens (human)Potency11.220210
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamineHomo sapiens (human)Potency11.220210
2-(4-chlorophenyl)-N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]acetamideHomo sapiens (human)Potency35.481310
3-methoxy-N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency35.481310
N-(2-methyl-5-nitrophenyl)-4,6-bis(1-pyrrolidinyl)-1,3,5-triazin-2-amineHomo sapiens (human)Potency11.220210
1-[2,3-bis(2-furanyl)-6-quinoxalinyl]-3-[4-(4-morpholinyl)phenyl]thioureaHomo sapiens (human)Potency35.481310
3-(3-oxo-2-benzo[f][1]benzopyranyl)-1-phenyl-4-pyrazolecarboxaldehydeHomo sapiens (human)Potency35.481310
N-(2,3-dimethylphenyl)-2-[[6-(1,3-dioxo-2-isoindolyl)-1,3-benzothiazol-2-yl]thio]acetamideHomo sapiens (human)Potency15.848910
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency35.481310
3-amino-8-methyl-N-[4-(4-morpholinyl)phenyl]-2-thieno[2,3-b]quinolinecarboxamideHomo sapiens (human)Potency16.263830
6-[[2-(4-morpholinyl)-2-oxoethyl]thio]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrileHomo sapiens (human)Potency17.782810
7-methyl-2-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]-3-quinolinecarbonitrileHomo sapiens (human)Potency35.481310
4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineHomo sapiens (human)Potency1.995310
4-(3-chloro-2-thiophenyl)-2-(3-pyridinyl)thiazoleHomo sapiens (human)Potency15.757810
6-methyl-5-[2-(2-methylphenoxy)ethyl]-2-sulfanylidene-1H-pyrimidin-4-oneHomo sapiens (human)Potency1.900820
4-[1-[(3-methoxyphenyl)methyl]-2-benzimidazolyl]-1,2,5-oxadiazol-3-amineHomo sapiens (human)Potency1.413820
3,4-dichloro-N-(2-thiophen-2-ylethyl)benzamideHomo sapiens (human)Potency2.511910
3-(benzenesulfonyl)-2-imino-1-propyl-5-dipyrido[1,2-d-3',4'-f]pyrimidinoneHomo sapiens (human)Potency28.183810
cyqualonHomo sapiens (human)Potency3.548110
syntelinHomo sapiens (human)Potency35.481310
N-[(2-adamantylamino)-sulfanylidenemethyl]hexanamideHomo sapiens (human)Potency10.000010
4-amino-5-[(4-methylphenyl)-oxomethyl]-2-(prop-2-enylamino)-3-thiophenecarbonitrileHomo sapiens (human)Potency35.481310
9-methoxy-6-[(4-methoxyphenyl)methyl]indolo[3,2-b]quinoxalineHomo sapiens (human)Potency10.000010
amn082Homo sapiens (human)Potency35.481310
3-(3-fluoro-4-methoxyphenyl)-5-phenyl-7-furo[3,2-g][1]benzopyranoneHomo sapiens (human)Potency1.983820
1-[2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl]-3-phenylureaHomo sapiens (human)Potency25.118910
1-(6-methyl-2-pyridinyl)-3-(2-phenylethyl)thioureaHomo sapiens (human)Potency6.309610
3-amino-N-(2-fluorophenyl)-6-(2-furanyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency23.808530
1-butyl-3-(4-phenoxyphenyl)thioureaHomo sapiens (human)Potency11.220210
1-(2-methoxyphenyl)-3-[2-[(4-methylphenyl)thio]ethyl]thioureaHomo sapiens (human)Potency22.387210
2-(1,4-dioxo-3H-phthalazin-2-yl)-N-(5-methyl-4-phenyl-2-thiazolyl)acetamideHomo sapiens (human)Potency35.481310
2-(2-furanyl)-4-quinolinecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterHomo sapiens (human)Potency22.387210
2-chloro-1-[2,5-dimethyl-1-(5-methyl-3-isoxazolyl)-3-pyrrolyl]ethanoneHomo sapiens (human)Potency19.837810
4-(4-hydroxyphenyl)-N-(phenylmethyl)-1-piperazinecarbothioamideHomo sapiens (human)Potency3.162310
4-[(3,5-dimethylphenyl)-oxomethyl]-1,3-dihydroquinoxalin-2-oneHomo sapiens (human)Potency0.776720
2,6-dichloro-N-[2-(methylthio)-1,3-benzothiazol-6-yl]benzenesulfonamideHomo sapiens (human)Potency28.183810
N-(3-acetyl-2-methyl-5-benzofuranyl)-N-(8-quinolinylsulfonyl)acetamideHomo sapiens (human)Potency35.481310
2-[3-[(4-chlorophenyl)-oxomethyl]-6-methoxy-4-oxo-1-quinolinyl]-N-(4-fluorophenyl)acetamideHomo sapiens (human)Potency11.220210
5-bromo-N-(6-sulfamoyl-1,3-benzothiazol-2-yl)-2-furancarboxamideHomo sapiens (human)Potency28.183810
2-[[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-oxomethyl]imino-1-(2-methylpropyl)-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency35.481310
2-[(3-methyl-4-oxo-5H-pyrimido[5,4-b]indol-2-yl)thio]-N-(4-methylphenyl)acetamideHomo sapiens (human)Potency15.848910
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[methyl(phenyl)sulfamoyl]benzamideHomo sapiens (human)Potency14.125410
1-[2,3-bis(2-pyridinyl)-6-quinoxalinyl]-3-propylthioureaHomo sapiens (human)Potency35.481310
1-[2-[(2-methylphenyl)methylthio]ethyl]-3-phenylthioureaHomo sapiens (human)Potency35.481310
thiocyanic acid [2-(1-naphthalenyl)-2-oxoethyl] esterHomo sapiens (human)Potency8.912510
mcb-613Homo sapiens (human)Potency6.309610
N-[[5-(1,3-benzothiazol-2-yl)-2-methylanilino]-sulfanylidenemethyl]-1-naphthalenecarboxamideHomo sapiens (human)Potency28.183810
N-[(3-bromoanilino)-sulfanylidenemethyl]-3-phenylpropanamideHomo sapiens (human)Potency35.481310
1-[4-(5-fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]-2-[(4-methyl-2-quinolinyl)thio]ethanoneHomo sapiens (human)Potency35.481310
N-[3-[[diethylamino(sulfanylidene)methyl]thio]-1-oxopropyl]carbamic acid (4-methylphenyl) esterHomo sapiens (human)Potency5.011910
4E2RCatHomo sapiens (human)Potency10.029430
1-[(7-chloro-4-quinolinyl)amino]-3-(2,4-dichlorophenyl)thioureaHomo sapiens (human)Potency35.481310
N1-phenethylhydrazine-1-carbothioamideHomo sapiens (human)Potency10.000010
2-nitrobenzoic acid [1,1,1,3,3,3-hexafluoro-2-[4-[(4-methylphenyl)sulfonylamino]phenyl]propan-2-yl] esterHomo sapiens (human)Potency12.589310
N-[[2-(diethylamino)ethylamino]-sulfanylidenemethyl]-3-(4-methoxyphenyl)-1-phenyl-4-pyrazolecarboxamideHomo sapiens (human)Potency25.118910
[[2-[[4-(4-bromophenyl)-2-thiazolyl]amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterHomo sapiens (human)Potency2.511910
2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-oneHomo sapiens (human)Potency35.481310
N2-(4-methylphenyl)benzene-1,2-diamineHomo sapiens (human)Potency19.952610
N-[[2-(1-cyclohexenyl)ethylamino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency22.387210
1-(2-tert-butylphenyl)-3-cyclohexylthioureaHomo sapiens (human)Potency25.118910
2-[[5-(2-fluoroanilino)-1,3,4-thiadiazol-2-yl]thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency35.481310
2-ethoxy-3-pyridinecarboxylic acid (4-methoxycarbonylphenyl)methyl esterHomo sapiens (human)Potency12.516810
4-hexyl-3-thiophen-2-yl-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency3.548110
N-(3-chloro-2-quinoxalinyl)-2-naphthalenesulfonamideHomo sapiens (human)Potency25.118910
N-[4-(difluoromethylthio)phenyl]-5-[(2-hydroxy-5-methoxyphenyl)-oxomethyl]-2-imino-3-pyrancarboxamideHomo sapiens (human)Potency21.597230
1-(2-chlorophenyl)-3-(3-phenylpropyl)thioureaHomo sapiens (human)Potency35.481310
2-[[(6-chloro-4-oxo-3-prop-2-enyl-2-quinazolinyl)thio]methyl]isoindole-1,3-dioneHomo sapiens (human)Potency35.481310
1-(2-benzofuranyl)-2-[(4-methyl-2-quinolinyl)thio]ethanoneHomo sapiens (human)Potency35.481310
2-(2,4-dichlorophenoxy)-N-[2-(methylthio)phenyl]acetamideHomo sapiens (human)Potency22.387210
N-[4-(2-pyridinyl)-2-thiazolyl]cyclopentanecarboxamideHomo sapiens (human)Potency7.079510
N,N-diethyl-3-[5-(ethylthio)-4-(phenylmethyl)-1,2,4-triazol-3-yl]benzenesulfonamideHomo sapiens (human)Potency35.481310
4-chloro-N-[3-[(3,5-dimethyl-4-isoxazolyl)methylthio]-2-quinoxalinyl]benzenesulfonamideHomo sapiens (human)Potency25.118910
5-(4-(dimethylamino)benzylidene)rhodanineHomo sapiens (human)Potency11.573130
4-amino-5-hydrazino-1,2,4-triazole-3-thiolHomo sapiens (human)Potency3.162310
5-anilino-3-oxo-4-isothiazolecarbonitrileHomo sapiens (human)Potency22.387210
1-(3-methylphenyl)-3-(2-pyridinyl)thioureaHomo sapiens (human)Potency22.387210
1-anilino-3-ethylthioureaHomo sapiens (human)Potency22.387210
xanthane hydrideHomo sapiens (human)Potency2.818410
N-[2-(trifluoromethyl)phenyl]pyrrolidine-1-carbothioamideHomo sapiens (human)Potency19.952610
N'-benzoyl-5-(3,5-dichlorophenoxy)-2-furancarbohydrazideHomo sapiens (human)Potency12.589310
N-(3-chlorophenyl)-2-[[2-(2-pyridinyl)-2,3-dihydro-1,3,4-thiadiazol-5-yl]thio]acetamideHomo sapiens (human)Potency2.818410
5-oxo-3-(4-phenylphenyl)-2H-furan-4-carbonitrileHomo sapiens (human)Potency22.387210
[5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-yl]hydrazineHomo sapiens (human)Potency17.782810
4-[5-chloro-6-methyl-2-(2-pyridinyl)-4-pyrimidinyl]morpholineHomo sapiens (human)Potency35.481310
n-(3-chloro-4-methylphenyl)-4-methyl-1,2,3-thiadiazole-5-carboxamideHomo sapiens (human)Potency0.354810
4-(2-hydroxyphenyl)-8,9-dimethyl-2,3-dihydro-1H-1,5-benzodiazepin-2-oneHomo sapiens (human)Potency11.220210
6-methyl-2-[[(4-methylanilino)-oxomethyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency35.481310
3-[5-[[4-(2-pyridinyl)-1-piperazinyl]sulfonyl]-2-thiophenyl]isoxazoleHomo sapiens (human)Potency25.118910
N-[5-ethyl-3-[(4-methoxyphenyl)-oxomethyl]-2-thiophenyl]-2-(4-methyl-1-piperazinyl)acetamideHomo sapiens (human)Potency5.623410
3-oxo-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)thio]butanoic acid ethyl esterHomo sapiens (human)Potency35.481310
3-(2,4-dimethoxyphenyl)-6-phenyl-2-sulfanylidene-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency5.623410
5-nitro-8-(1-pyrrolidinyl)quinolineHomo sapiens (human)Potency35.481310
2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-phenylacetamideHomo sapiens (human)Potency12.589310
2-[[2-methyl-5-nitro-3-(phenylmethyl)-4-imidazolyl]thio]-6-nitro-1H-benzimidazoleHomo sapiens (human)Potency8.912510
1-[1-(2,3-dihydro-1,4-benzodioxin-3-yl)ethyl]-3-phenylthioureaHomo sapiens (human)Potency3.548110
1-[8-chloro-4-(1-naphthalenyl)-3,3a,4,9b-tetrahydrocyclopenta[c]quinolin-5-yl]ethanoneHomo sapiens (human)Potency35.481310
4-[2,2-bis(1-phenyl-5-tetrazolyl)ethenyl]-N,N-dimethylanilineHomo sapiens (human)Potency22.387210
2-chloro-N-[(2-hydroxy-5-methylanilino)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency15.848910
2-[(4-chlorophenyl)thio]-N-[4-[(2,4-dimethylphenyl)sulfamoyl]phenyl]propanamideHomo sapiens (human)Potency35.481310
1,3,8-trimethyl-5,10-diphenylpyrimido[1,2]pyrrolo[4,5-b]pyridazine-2,4-dioneHomo sapiens (human)Potency20.739520
N-ethyl-N-[2-[(5-nitro-8-quinolinyl)amino]ethyl]benzenesulfonamideHomo sapiens (human)Potency14.125410
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideHomo sapiens (human)Potency35.481310
[4-(benzenesulfonyl)-1-piperazinyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency35.481310
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Potency3.917730
2-methyl-3-phenyl-3H-1,5-benzodiazepin-4-amineHomo sapiens (human)Potency35.481310
4-fluoro-N-[3-[2-nitro-4-(trifluoromethyl)anilino]propyl]benzamideHomo sapiens (human)Potency28.183810
2-[(4-chlorophenyl)sulfonyl-methylamino]-N-(4-methoxy-2-nitrophenyl)acetamideHomo sapiens (human)Potency25.118910
1-(3-chloro-4-methylphenyl)-5-oxo-N-(2-thiazolyl)-3-pyrrolidinecarboxamideHomo sapiens (human)Potency11.220210
[4-(benzenesulfonyl)-1-piperazinyl]-[6-bromo-2-(2-pyridinyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency1.778310
LSM-16248Homo sapiens (human)Potency15.757820
2-[[(4-chlorophenyl)thio]methyl]-5-methylimidazo[1,2-a]pyridineHomo sapiens (human)Potency35.481310
6-(2-chlorophenyl)-3-methyl-2-[4-morpholinyl(oxo)methyl]-1,5,6,7-tetrahydroindol-4-oneHomo sapiens (human)Potency3.165020
4-[[3-[(4-chlorophenyl)sulfonylamino]-2-quinoxalinyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency27.366020
2-cyano-N-(phenylmethyl)-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetamideHomo sapiens (human)Potency6.831320
N-(1,3-benzothiazol-2-yl)-2-oxolanecarboxamideHomo sapiens (human)Potency22.387210
1,3-dimethyl-8-[2-(1-pyrrolidinyl)ethylthio]-6-sulfanylidene-7H-purin-2-oneHomo sapiens (human)Potency3.981110
4-methyl-2-[3-methyl-4-(3-methylphenyl)azo-5-oxo-4H-pyrazol-1-yl]-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
2-[(prop-2-enylthio)-(4,5,6,7-tetrahydro-1H-indol-2-yl)methylidene]propanedinitrileHomo sapiens (human)Potency31.622810
3-methyl-1-(3-propan-2-yloxypropylamino)-4-pyrido[1,2-a]benzimidazolecarbonitrileHomo sapiens (human)Potency35.481310
N-[2-(3-oxo-4H-quinoxalin-2-yl)phenyl]-2-thiophenecarboxamideHomo sapiens (human)Potency17.782810
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(4-methyl-2-thiazolyl)acetamideHomo sapiens (human)Potency12.589310
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolHomo sapiens (human)Potency5.623410
4-[[[(1-ethyl-2-oxo-6-benzo[cd]indolyl)amino]-oxomethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency35.481310
3-[[2-furanyl(oxo)methyl]amino]-N-(4-methoxyphenyl)-2-benzofurancarboxamideHomo sapiens (human)Potency6.309610
N-ethyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(phenylmethyl)propanamideHomo sapiens (human)Potency6.309610
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolHomo sapiens (human)Potency15.848910
3-(4-methoxyphenyl)-3-(1-pyrrolyl)-N-(2-thiazolyl)propanamideHomo sapiens (human)Potency35.481310
2-furanyl-[4-(4-tetrazolo[1,5-a]quinoxalinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency12.589310
8-(2-propoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-oneHomo sapiens (human)Potency3.958210
N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamineHomo sapiens (human)Potency35.481310
[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency22.387210
N-[[3-[(3-chlorophenyl)sulfamoyl]-4-methylanilino]-sulfanylidenemethyl]-4-fluorobenzamideHomo sapiens (human)Potency7.305420
3-[3-(N-ethylanilino)propyl]-6-(4-morpholinyl)-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency35.481310
8-[(1-ethyl-3-piperidinyl)thio]-1,3-dimethyl-6-sulfanylidene-7H-purin-2-oneHomo sapiens (human)Potency22.387210
3-(phenylthio)-1-(1-pyrrolidinyl)-1-propanoneHomo sapiens (human)Potency35.481310
N-(5-acetyl-2-phenyl-4-sulfanylidene-1H-pyrimidin-6-yl)benzamideHomo sapiens (human)Potency11.220210
1-(6-methyl-2-pyridinyl)-3-[3-(trifluoromethyl)phenyl]thioureaHomo sapiens (human)Potency2.818410
1-(3-ethoxypropyl)-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.778310
1,3-diphenyl-4-pyrazolecarboxylic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency25.118910
3-amino-4-(1,3-benzothiazol-2-yl)-N-(3-chloro-2-methylphenyl)-5-phenylimino-2H-thiophene-2-carboxamideHomo sapiens (human)Potency7.079510
2-amino-7-methyl-4-(5-nitro-2-furanyl)-5-oxo-4H-pyrano[3,2-c]pyran-3-carbonitrileHomo sapiens (human)Potency10.000010
3-(1-methyl-2-benzimidazolyl)-1-phenyl-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency35.481310
4-[(4-acetyl-2-methoxyphenyl)methoxy]-3-methoxybenzoic acid [1-(carbamoylamino)-1-oxopropan-2-yl] esterHomo sapiens (human)Potency11.220210
N-[4-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency22.387210
uc-112Homo sapiens (human)Potency19.952610
2-(2-methoxyphenyl)-1-methyl-3,5-dinitro-2H-pyridineHomo sapiens (human)Potency17.782810
N-(1,3-benzodioxol-5-ylmethyl)-4-nitroanilineHomo sapiens (human)Potency35.481310
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolHomo sapiens (human)Potency35.481310
1-[(2,6-dichlorophenyl)methyl]-5-(4-methylphenyl)-2-oxo-3-pyridinecarbonitrileHomo sapiens (human)Potency28.183810
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency10.000010
4-chloro-N-(2-methoxy-1-phenazinyl)benzamideHomo sapiens (human)Potency16.896530
3-(3-bromoanilino)-2-oxo-1H-indole-3-carbonitrileHomo sapiens (human)Potency35.481310
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamideHomo sapiens (human)Potency18.759120
1-ethyl-3-[[2-[(1-methyl-2-benzimidazolyl)thio]-1-oxoethyl]amino]thioureaHomo sapiens (human)Potency4.466810
2-amino-5-(1-benzotriazolyl)-6-methyl-4-phenyl-4H-pyran-3-carbonitrileHomo sapiens (human)Potency25.118910
2-chloro-N-ethyl-N-phenylpropanamideHomo sapiens (human)Potency5.623410
4-methyl-2-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentanoic acid [3-(4-nitrophenyl)-4-oxo-1-benzopyran-7-yl] esterHomo sapiens (human)Potency31.622810
4-(2-fluorophenyl)-5-methyl-2-(2-phenoxyethyl)-1,2,4-triazol-3-oneHomo sapiens (human)Potency6.309610
2-(1H-benzimidazol-2-yl)-5-methyl-4-(phenylmethyl)-4H-pyrazol-3-oneHomo sapiens (human)Potency35.481310
arabino-4-thiouridineHomo sapiens (human)Potency35.481310
N-(1,3-benzothiazol-2-yl)-2-ethylsulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamideHomo sapiens (human)Potency22.387210
N-[6-amino-2,4-dioxo-1-(phenylmethyl)-5-pyrimidinyl]-N-ethyl-2-(2-methyl-2,3-dihydroindol-1-yl)acetamideHomo sapiens (human)Potency35.481310
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyrazinecarboxamideHomo sapiens (human)Potency6.309610
4-(6-methyl-4-phenyl-2-quinazolinyl)-1,3-dihydroquinoxalin-2-oneHomo sapiens (human)Potency8.912510
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideHomo sapiens (human)Potency19.149830
2-pyridinecarboxylic acid [2-[2-(difluoromethoxy)anilino]-2-oxoethyl] esterHomo sapiens (human)Potency35.481310
1-(3,3-dimethylbutan-2-yl)-3-[3-(trifluoromethyl)phenyl]thioureaHomo sapiens (human)Potency31.622810
N,6-dimethyl-2-[[[4-[(2-methyl-1-piperidinyl)sulfonyl]phenyl]-oxomethyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideHomo sapiens (human)Potency35.481310
1-(1-adamantyl)-2-[(1-oxido-2-pyridin-1-iumyl)thio]ethanoneHomo sapiens (human)Potency3.162310
2-(5-bromo-2-thiophenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency35.481310
3-(acetyloxymethyl)-7-[[3-(4-chloro-3,5-dimethyl-1-pyrazolyl)-2-methyl-1-oxopropyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidHomo sapiens (human)Potency12.589310
3-chloro-N-[5-(3-pyridinyl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)Potency31.622810
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-oneHomo sapiens (human)Potency35.481310
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methyl-1-piperidinyl)sulfonyl]benzamideHomo sapiens (human)Potency35.481310
N4-(2,5-dimethoxyphenyl)-N2-(3-methylbutyl)-5-nitropyrimidine-2,4,6-triamineHomo sapiens (human)Potency35.481310
N-[2-(2,4,6-trinitrophenyl)ethyl]anilineHomo sapiens (human)Potency6.309610
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]-4-methylbenzamideHomo sapiens (human)Potency15.862320
2,4-dichloro-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency7.079510
1-benzoyl-5-hydroxy-5-(4-methylphenyl)-4H-pyrazole-3-carboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
2-(3-oxo-2,4-dihydroquinoxalin-1-yl)-2-phenyl-N-(4-propan-2-ylphenyl)acetamideHomo sapiens (human)Potency17.782810
3-(2-methylphenyl)-2-(2-thiazolyl)-5,6,7,7a-tetrahydro-3H-pyrrolo[1,2-c]imidazol-1-oneHomo sapiens (human)Potency10.000010
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideHomo sapiens (human)Potency35.481310
2,6-difluoro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)Potency25.118910
2-(4-chlorophenoxy)-N-(2-thiophen-2-yl-3-imidazo[1,2-a]pyridinyl)acetamideHomo sapiens (human)Potency35.481310
3-chloro-N-[3-(2-methoxyethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency35.481310
4-(1-azepanylsulfonyl)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-hydroxyphenyl]benzamideHomo sapiens (human)Potency14.125410
4-(5-methyl-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)benzoic acid 8-quinolinyl esterHomo sapiens (human)Potency3.548110
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaHomo sapiens (human)Potency5.623410
2-[4-(4-methoxyphenyl)-4-methyl-2,5-dioxo-1-imidazolidinyl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]acetamideHomo sapiens (human)Potency15.848910
6-methoxy-2-methyl-N-[[3-(trifluoromethyl)phenyl]methyl]-4-quinolinamineHomo sapiens (human)Potency14.125410
3,7-dichloro-N-[3-(1-imidazolyl)propyl]-6-methoxy-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency2.818410
5'-bromo-2'-spiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-1H-indole]oneHomo sapiens (human)Potency15.290330
N-(1-benzylpiperidin-4-yl)-2-(pyridin-3-yl)quinazolin-4-amineHomo sapiens (human)Potency35.481310
4-[(2-cyano-1-oxoethyl)amino]benzoic acid [2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl] esterHomo sapiens (human)Potency35.481310
N-(4-bromo-2-fluorophenyl)-2-(2,4-dimethoxyanilino)acetamideHomo sapiens (human)Potency0.562310
3-(1-methyl-2-benzimidazolyl)-1-(3-methylphenyl)-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency10.000010
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-(4,4,6-trimethyl-2-sulfanylidene-1,3-diazinan-1-yl)-1-propanoneHomo sapiens (human)Potency22.387210
N-methyl-2-[[[4-[methyl(phenyl)sulfamoyl]phenyl]-oxomethyl]amino]-6-propyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideHomo sapiens (human)Potency15.004630
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)Potency35.481310
1-[2-[(4-pentoxyphenyl)methylthio]ethyl]-3-phenylthioureaHomo sapiens (human)Potency25.118910
ncgc00099374Homo sapiens (human)Potency1.702530
5-benzoyl-6-methyl-4-[4-(4-morpholinyl)phenyl]-3,4-dihydro-1H-pyrimidin-2-oneHomo sapiens (human)Potency25.118910
quercetin 3-o-methyl etherHomo sapiens (human)Potency13.280420
alpha-linolenic acidHomo sapiens (human)Potency22.387210
rescinnamineHomo sapiens (human)Potency3.162310
sulfuretinHomo sapiens (human)Potency14.125410
caffeic acid phenethyl esterHomo sapiens (human)Potency6.309610
4-hydroxyestradiolHomo sapiens (human)Potency28.183810
2-[[4-methyl-5-[(2-oxo-1,3-benzothiazol-3-yl)methyl]-1,2,4-triazol-3-yl]thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency35.481310
3-(4-chlorophenyl)-1-methyl-N-[3-(1-pyrrolidinyl)propyl]-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency22.387210
4-(4-tetrazolo[1,5-a]quinoxalinyl)morpholineHomo sapiens (human)Potency11.879220
su 6656Homo sapiens (human)Potency2.230130
semaxinibHomo sapiens (human)Potency15.768630
1-(4-methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-oneHomo sapiens (human)Potency6.309610
rd6 5071Homo sapiens (human)Potency0.891310
2-(4-(dimethylamino)styryl)benzothiazoleHomo sapiens (human)Potency35.481310
morusinolHomo sapiens (human)Potency19.952610
3-(dimethylamino)benzoic acid (7-hydroxy-2-oxo-1-benzopyran-4-yl)methyl esterHomo sapiens (human)Potency14.125410
fendiline hydrochlorideHomo sapiens (human)Potency25.118910
2',3,4-trihydroxychalconeHomo sapiens (human)Potency28.183810
2-(dimethylaminostyryl)-1-ethylpyridiniumHomo sapiens (human)Potency22.030930
HTS 01037Homo sapiens (human)Potency14.044110
chloride of pseudoisocyanineHomo sapiens (human)Potency12.589310
5233705 compoundHomo sapiens (human)Potency28.183810
N-[(2-methoxyphenyl)methyl]-6H-indolo[2,3-b]quinoxaline-2-carboxamideHomo sapiens (human)Potency16.213620
6-chloro-4-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-hydroxy-1-benzopyran-2-oneHomo sapiens (human)Potency6.309610
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazineHomo sapiens (human)Potency28.183810
3-amino-5-(4-bromophenyl)-4-pyridazinecarbonitrileHomo sapiens (human)Potency35.481310
2-(1,3-benzoxazol-2-ylamino)-7,7-dimethyl-4-(2-pyridinyl)-1,4,6,8-tetrahydroquinazolin-5-oneHomo sapiens (human)Potency6.309610
(3S)-2-(2-chloro-1-oxoethyl)-1,1-dimethyl-4,9-dihydro-3H-pyrido[3,4-b]indole-3-carboxylic acid methyl esterHomo sapiens (human)Potency15.757810
methiazoleHomo sapiens (human)Potency35.481310
6-ethyl-8-methyl-N-(3-pyridinylmethyl)-3-benzo[b][1,4]benzothiazepinecarboxamideHomo sapiens (human)Potency4.196620
2-[4-ethoxy-2-[2-furanyl(oxo)methyl]imino-1,3-benzothiazol-3-yl]acetic acid methyl esterHomo sapiens (human)Potency8.912510
1-(3-ethylphenyl)-3-(1-naphthalenyl)thioureaHomo sapiens (human)Potency35.481310
org 41841Homo sapiens (human)Potency35.481310
u 74389gHomo sapiens (human)Potency11.220210
enisamium iodideHomo sapiens (human)Potency35.481310
garcinone eHomo sapiens (human)Potency35.481310
N-[1-(5,6-dicyano-3-methyl-2-pyrazinyl)ethyl]-N-phenylacetamideHomo sapiens (human)Potency35.481310
protoapigenoneHomo sapiens (human)Potency5.016120
3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-6-(1-piperidinylsulfonyl)-1,3-benzoxazol-2-oneHomo sapiens (human)Potency17.782810
N-(2-furanylmethyl)-6-propyl-3-benzo[b][1,4]benzothiazepinecarboxamideHomo sapiens (human)Potency1.779820
2-(3-chlorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency3.162310
malyngamide AHomo sapiens (human)Potency17.782810
win 62577Homo sapiens (human)Potency35.481310
4-chloro-N-[3-(3-methyl-1-piperidinyl)propyl]-2-thieno[3,2-c]quinolinecarboxamideHomo sapiens (human)Potency35.481310
5-[[3-bromo-4-[(2-fluorophenyl)methoxy]-5-methoxyphenyl]methylamino]-1,3-dihydrobenzimidazol-2-oneHomo sapiens (human)Potency3.548110
(3aS,5S,9aS)-5-[1-(2-methoxyphenyl)-4-pyrazolyl]-2-phenyl-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-oneHomo sapiens (human)Potency35.481310
N-(2-furanylmethyl)-2-[[4-oxo-3-[3-(1-pyrrolidinyl)propyl]-[1]benzothiolo[3,2-d]pyrimidin-2-yl]thio]acetamideHomo sapiens (human)Potency0.562310
1,2-dihydroacenaphthylen-5-yl-[1-[(6-methyl-2-pyridinyl)methyl]-3-piperidinyl]methanoneHomo sapiens (human)Potency22.387210
1,2-dihydroacenaphthylen-5-yl-[1-(2-pyridinylmethyl)-3-piperidinyl]methanoneHomo sapiens (human)Potency22.387210
N-(4-methylphenyl)-4-tetrazolo[1,5-a]quinoxalinamineHomo sapiens (human)Potency19.952610
1-[4-(3-chlorophenyl)-1-piperazinyl]-3-(diphenylmethyl)oxy-2-propanolHomo sapiens (human)Potency35.481310
2-imino-8-methyl-5-oxo-1-(2-oxolanylmethyl)-N-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideHomo sapiens (human)Potency31.622810
cyclopenolHomo sapiens (human)Potency35.481310
(5S)-1-(4-cyclohexylbutyl)-5-phenyl-4,5-dihydroimidazol-2-amineHomo sapiens (human)Potency35.481310
3-[4-[2-(2-fluorophenyl)ethylamino]-3-nitrophenyl]-3-[[2-(1-naphthalenyl)-1-oxoethyl]amino]propanamideHomo sapiens (human)Potency17.782810
3-[[2-(4-bromophenyl)-1-oxoethyl]amino]-3-[4-[(4-fluorophenyl)methylamino]-3-nitrophenyl]propanamideHomo sapiens (human)Potency23.135330
N-[3-amino-1-[4-[2-(4-methoxyphenyl)ethylamino]-3-nitrophenyl]-3-oxopropyl]-4-bromobenzamideHomo sapiens (human)Potency35.481310
(3R)-7-phenyl-2-(phenylmethyl)-3-[4-(trifluoromethyl)phenyl]-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency35.481310
(3R,3aS,7R,7aS)-7-methyl-3-(2-naphthalenyl)-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency35.481310
(3R)-3-(2-fluoro-5-methylphenyl)-7-phenyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency35.481310
1-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-5-methoxy-isatinHomo sapiens (human)Potency17.782810
2-(2-fluorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency6.309610
N-[5-[methyl-(3-methylphenyl)sulfamoyl]-1,3,4-thiadiazol-2-yl]-2-furancarboxamideHomo sapiens (human)Potency35.481310
4'-epichaetoviridin AHomo sapiens (human)Potency19.952610
(5R)-5-tert-butyl-1-[(3S)-3-[(4-methylphenyl)thio]-3-phenylpropyl]-2-azepanoneHomo sapiens (human)Potency35.481310
3-(4-Amino-3,5-dichlorobenzoyl)-2-(3-amino-3-oxopropyl)-2H-indazole 1-oxideHomo sapiens (human)Potency12.589310
2-[5-(2-fluorophenyl)-2-furanyl]-3-hydroxy-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency35.481310
N-[(5-chloro-8-hydroxy-7-quinolinyl)-cyclopropylmethyl]acetamideHomo sapiens (human)Potency35.481310
N-[(5-fluoro-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideHomo sapiens (human)Potency10.000010
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineHomo sapiens (human)Potency0.562310
2-(3-fluoroanilino)-7-hydroxy-5-oxo-4H-thieno[3,2-b]pyridine-3-carbonitrileHomo sapiens (human)Potency22.387210
4-hydroxy-1-methyl-N'-[(3-methylphenyl)-oxomethyl]-2-oxo-3-quinolinecarbohydrazideHomo sapiens (human)Potency17.782810
3-cinnamoyl-4-hydroxy-6-methyl-2h-pyran-2-oneHomo sapiens (human)Potency1.412510
kf38789Homo sapiens (human)Potency2.818410
azaguanineHomo sapiens (human)Potency5.799720
N-[3-[(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)amino]-1-isoindolylidene]-2-thiophenecarboxamideHomo sapiens (human)Potency13.674030
8-azahypoxanthineHomo sapiens (human)Potency6.316720
1-hydroxyphenazineHomo sapiens (human)Potency35.481310
5-methyl-2-methylsulfanyl-6-propyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency1.122010
glycosminineHomo sapiens (human)Potency3.162310
tn 16Homo sapiens (human)Potency6.137230
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-[2-(methylthio)phenyl]acetamideHomo sapiens (human)Potency0.562310
5-(4-chlorophenyl)-3-(4-nitrophenyl)-1H-pyrazoleHomo sapiens (human)Potency19.952610
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-(3-fluorophenyl)acetamideHomo sapiens (human)Potency35.481310
5-[1-(4-chlorophenyl)-2,5-dimethyl-3-pyrrolyl]-N-methyl-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency35.481310
7-[[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)Potency35.481310