A urokinase-type plasminogen activator that is encoded in the genome of mouse. [OMA:P06869, PRO:DNx]
U-plasminogen activator;
uPA;
EC 3.4.21.73
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 3 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
gallic acid | Mus musculus (house mouse) | IC50 | 6.6000 | 1 | 1 |
5-(n,n-hexamethylene)amiloride | Mus musculus (house mouse) | Ki | 9.3080 | 1 | 1 |
hexachlorophene | Mus musculus (house mouse) | IC50 | 3.8000 | 1 | 1 |
1,2,5,8-tetrahydroxy anthraquinone | Mus musculus (house mouse) | IC50 | 4.4000 | 1 | 1 |
amiloride | Mus musculus (house mouse) | IC50 | 2.3000 | 1 | 1 |
amiloride | Mus musculus (house mouse) | Ki | 2.3130 | 1 | 1 |
epigallocatechin gallate | Mus musculus (house mouse) | IC50 | 0.0910 | 1 | 1 |
sennoside A | Mus musculus (house mouse) | IC50 | 51.0000 | 1 | 1 |
Epigallocatechin 3,5-Digallate | Mus musculus (house mouse) | IC50 | 0.3300 | 1 | 1 |