An alpha-type platelet-derived growth factor receptor that is encoded in the genome of mouse. [OMA:P26618, PRO:DNx]
PDGF-R-alpha;
PDGFR-alpha;
EC 2.7.10.1;
Alpha platelet-derived growth factor receptor;
Alpha-type platelet-derived growth factor receptor;
CD140 antigen-like family member A;
Platelet-derived growth factor alpha receptor
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 6 (54.55) | 18.2507 |
| 2000's | 4 (36.36) | 29.6817 |
| 2010's | 1 (9.09) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| cgp 52411 | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| ag 1295 | Mus musculus (house mouse) | IC50 | 2.9000 | 2 | 2 |
| ag-1296 | Mus musculus (house mouse) | IC50 | 0.8000 | 1 | 1 |
| imatinib | Mus musculus (house mouse) | IC50 | 0.3000 | 1 | 1 |
| 2,3-dimethylquinoxaline | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| staurosporine | Mus musculus (house mouse) | IC50 | 0.0020 | 1 | 1 |
| 2,3-bis(2-pyridinyl)quinoxaline | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| pd 166285 | Mus musculus (house mouse) | IC50 | 0.0589 | 3 | 3 |
| pd 166866 | Mus musculus (house mouse) | IC50 | 50.0000 | 1 | 1 |
| pd 161570 | Mus musculus (house mouse) | IC50 | 0.3600 | 1 | 1 |
| semaxinib | Mus musculus (house mouse) | IC50 | 14.8700 | 3 | 3 |
| orantinib | Mus musculus (house mouse) | IC50 | 18.2571 | 7 | 7 |
| su 11248 | Mus musculus (house mouse) | IC50 | 0.0186 | 7 | 7 |
| su 11652 | Mus musculus (house mouse) | IC50 | 0.0850 | 2 | 2 |
| palladia | Mus musculus (house mouse) | IC50 | 0.0850 | 2 | 2 |
| d-64406 | Mus musculus (house mouse) | IC50 | 0.2000 | 1 | 1 |
| isoalloxazine | Mus musculus (house mouse) | IC50 | 50.0000 | 1 | 1 |
| cgp 53353 | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| cgp 53716 | Mus musculus (house mouse) | IC50 | 0.1000 | 1 | 1 |
| nintedanib | Mus musculus (house mouse) | IC50 | 0.0850 | 1 | 1 |