Page last updated: 2024-08-07 19:46:35
Adenosine receptor A1
[no definition available]
Synonyms
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (100.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| 2-chloro-n(6)cyclopentyladenosine | Sus scrofa (pig) | Ki | 0.0003 | 2 | 2 |
| tecadenoson | Sus scrofa (pig) | Ki | 0.0054 | 2 | 2 |
| trichostatin a | Sus scrofa (pig) | IC50 | 0.2000 | 1 | 1 |
| n(6)-cyclopentyladenosine | Sus scrofa (pig) | Ki | 0.0005 | 2 | 2 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| tecadenoson | Sus scrofa (pig) | EC50 | 0.0316 | 1 | 1 |
| n(6)-cyclopentyladenosine | Sus scrofa (pig) | EC50 | 0.0079 | 1 | 1 |