Page last updated: 2024-08-07 18:37:34
Solute carrier family 15 member 1
A solute carrier family 15 member 1 that is encoded in the genome of rat. [OMA:P51574, PRO:DNx]
Synonyms
Intestinal H(+)/peptide cotransporter;
Oligopeptide transporter, small intestine isoform;
Peptide transporter 1;
Proton-coupled dipeptide cotransporter
Research
Bioassay Publications (9)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (66.67) | 18.2507 |
2000's | 2 (22.22) | 29.6817 |
2010's | 1 (11.11) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (38)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
aminolevulinic acid | Rattus norvegicus (Norway rat) | Ki | 2,200.0000 | 1 | 1 |
glyburide | Rattus norvegicus (Norway rat) | Ki | 25.0000 | 1 | 1 |
ampicillin | Rattus norvegicus (Norway rat) | Ki | 47,800.0000 | 1 | 1 |
glycyl-glycyl-glycine | Rattus norvegicus (Norway rat) | Ki | 1,300.0000 | 1 | 1 |
glycylglycine | Rattus norvegicus (Norway rat) | Ki | 860.0000 | 1 | 1 |
cyclacillin | Rattus norvegicus (Norway rat) | Ki | 168.0000 | 1 | 1 |
cephalexin | Rattus norvegicus (Norway rat) | Ki | 4,500.0000 | 1 | 1 |
amoxicillin | Rattus norvegicus (Norway rat) | Ki | 13,000.0000 | 1 | 1 |
cephradine | Rattus norvegicus (Norway rat) | Ki | 8,540.0000 | 1 | 1 |
captopril | Rattus norvegicus (Norway rat) | Ki | 8,700.0000 | 1 | 1 |
cefadroxil anhydrous | Rattus norvegicus (Norway rat) | Ki | 2,170.0000 | 1 | 1 |
omega-aminocaprylic acid | Rattus norvegicus (Norway rat) | Ki | 4,400.0000 | 1 | 1 |
ubenimex | Rattus norvegicus (Norway rat) | Ki | 1,500.0000 | 1 | 1 |
tamiflu | Rattus norvegicus (Norway rat) | IC50 | 18,300.0000 | 1 | 1 |
glycyltryptophan | Rattus norvegicus (Norway rat) | Ki | 1,400.0000 | 1 | 1 |
glycyltyrosine | Rattus norvegicus (Norway rat) | Ki | 210.0000 | 1 | 1 |
glycylleucine | Rattus norvegicus (Norway rat) | Ki | 110.0000 | 1 | 1 |
glycyl-l-phenylalanine | Rattus norvegicus (Norway rat) | Ki | 170.0000 | 1 | 1 |
glycyl-leucyl-tyrosine | Rattus norvegicus (Norway rat) | Ki | 190.0000 | 1 | 1 |
glycylaspartic acid | Rattus norvegicus (Norway rat) | Ki | 300.0000 | 1 | 1 |
beta-aspartylglycine | Rattus norvegicus (Norway rat) | Ki | 50,000.0000 | 1 | 1 |
lysyllysine | Rattus norvegicus (Norway rat) | Ki | 8,000.0000 | 1 | 1 |
alanine-4-nitroanilide | Rattus norvegicus (Norway rat) | Ki | 61.0000 | 1 | 1 |
aspartylglycine | Rattus norvegicus (Norway rat) | Ki | 830.0000 | 1 | 1 |
carnosine | Rattus norvegicus (Norway rat) | Ki | 8,000.0000 | 1 | 1 |
aspartyl-aspartic acid | Rattus norvegicus (Norway rat) | Ki | 990.0000 | 1 | 1 |
glycyllysine | Rattus norvegicus (Norway rat) | Ki | 2,200.0000 | 1 | 1 |
7432 s | Rattus norvegicus (Norway rat) | Ki | 597.0000 | 1 | 1 |
nateglinide | Rattus norvegicus (Norway rat) | IC50 | 160.0000 | 1 | 1 |
cefixime | Rattus norvegicus (Norway rat) | Ki | 6,920.0000 | 1 | 1 |
enalapril | Rattus norvegicus (Norway rat) | Ki | 4,300.0000 | 1 | 1 |
prolylglycine | Rattus norvegicus (Norway rat) | Ki | 13,000.0000 | 1 | 1 |
cefdinir | Rattus norvegicus (Norway rat) | Ki | 11,900.0000 | 1 | 1 |
phenylalanylglycine | Rattus norvegicus (Norway rat) | Ki | 220.0000 | 1 | 1 |
lysylglycine | Rattus norvegicus (Norway rat) | Ki | 910.0000 | 1 | 1 |
glycylhistidine | Rattus norvegicus (Norway rat) | Ki | 1,400.0000 | 1 | 1 |
valacyclovir | Rattus norvegicus (Norway rat) | Ki | 2,600.0000 | 1 | 2 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
cephradine | Rattus norvegicus (Norway rat) | Km | 10,300.0000 | 2 | 2 |
glycylsarcosine | Rattus norvegicus (Norway rat) | Km | 1,080.0000 | 3 | 3 |
7432 s | Rattus norvegicus (Norway rat) | Km | 1,200.0000 | 2 | 2 |