Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
4-methylumbelliferyl acetate | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
phenol | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
1,3-dipropyl-8-(4-sulfophenyl)xanthine | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
pd 173074 | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
hoe 33342 | Homo sapiens (human) | Potency | 30.2586 | 1 | 0 |
cgp 52411 | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
p-chloromercuribenzoic acid | Homo sapiens (human) | Potency | 4.4668 | 1 | 0 |
hydroxyindoleacetic acid | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
8-(4-sulfophenyl)theophylline | Homo sapiens (human) | Potency | 34.8936 | 1 | 0 |
acridone | Homo sapiens (human) | Potency | 29.9033 | 2 | 0 |
ag-1296 | Homo sapiens (human) | Potency | 42.2395 | 1 | 0 |
rtki cpd | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
alfuzosin | Homo sapiens (human) | Potency | 33.7746 | 2 | 0 |
altretamine | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
amlexanox | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
amsacrine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
9-anthroic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
benzylhydrochlorothiazide | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
butacaine | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
calmidazolium | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
cimetidine | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
5,7-dimethoxycoumarin | Homo sapiens (human) | Potency | 22.8741 | 2 | 0 |
4-chloro-N-(2,6-dimethyl-1-piperidinyl)-3-sulfamoylbenzamide | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
clotrimazole | Homo sapiens (human) | Potency | 7.9433 | 1 | 0 |
damnacanthal | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
domperidone | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
ebselen | Homo sapiens (human) | Potency | 32.4648 | 2 | 0 |
flutamide | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
n-(2-(methylamino)ethyl)-5-isoquinolinesulfonamide | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
harmaline | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
hydroxy-2-naphthalenyl-methyl phosphonic acid trisacetoxymethylester | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
amrinone | Homo sapiens (human) | Potency | 1.2589 | 1 | 0 |
iodoacetamide | Homo sapiens (human) | Potency | 22.3872 | 2 | 0 |
kynurenic acid | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
lansoprazole | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
beta-lapachone | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
loratadine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ly 171883 | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
n(1),n(11)-diethylnorspermine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
etoposide phosphate | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
nimesulide | Homo sapiens (human) | Potency | 3.9811 | 1 | 0 |
pinacidil | Homo sapiens (human) | Potency | 3.1623 | 1 | 0 |
pindolol | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
prazosin | Homo sapiens (human) | Potency | 38.0490 | 2 | 0 |
probenecid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ritanserin | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
fenofibrate | Homo sapiens (human) | Potency | 41.6060 | 2 | 0 |
terazosin | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
tolazamide | Homo sapiens (human) | Potency | 5.6234 | 1 | 0 |
triamterene | Homo sapiens (human) | Potency | 30.1763 | 5 | 0 |
tyrphostin a9 | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
papaverine hydrochloride | Homo sapiens (human) | Potency | 3.9811 | 1 | 0 |
cytarabine hydrochloride | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
arginine | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
n,n'-diethylcarbanilide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
aminacrine | Homo sapiens (human) | Potency | 40.0748 | 2 | 0 |
xanthone | Homo sapiens (human) | Potency | 31.8326 | 2 | 0 |
pseudoephedrine | Homo sapiens (human) | Potency | 32.4648 | 2 | 0 |
uvitex swn | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
dehydrothio-4-toluidine | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
pyridostigmine bromide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
2-Phenylethyl 2-aminobenzoate | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
acridines | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
methysergide | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
podophyllotoxin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
physcione | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
aminacrine | Homo sapiens (human) | Potency | 28.1838 | 2 | 0 |
alpha-naphthoflavone | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
ethidium bromide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
amiloride hydrochloride, anhydrous | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
amiloride | Homo sapiens (human) | Potency | 37.3522 | 2 | 0 |
amo-1618 | Homo sapiens (human) | Potency | 2.8184 | 1 | 0 |
diloxanide furoate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
helenalin | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
camptothecin | Homo sapiens (human) | Potency | 15.3211 | 3 | 0 |
1-deoxynojirimycin | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
ribavirin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
10-carboxymethyl-9-acridanone | Homo sapiens (human) | Potency | 23.0856 | 1 | 0 |
terazosin hydrochloride anhydrous | Homo sapiens (human) | Potency | 39.2584 | 2 | 0 |
triclabendazole | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
doxazosin mesylate | Homo sapiens (human) | Potency | 41.8036 | 2 | 0 |
nelfinavir | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
siquil | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
sotalol hydrochloride | Homo sapiens (human) | Potency | 0.1778 | 1 | 0 |
alprenolol hydrochloride | Homo sapiens (human) | Potency | 0.7943 | 1 | 0 |
fluphenazine hydrochloride | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
pyrrolo(1,2-a)quinoxaline | Homo sapiens (human) | Potency | 31.8326 | 2 | 0 |
harmol | Homo sapiens (human) | Potency | 42.2395 | 1 | 0 |
11h-pyrido(2,1-b)quinazolin-11-one | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
amiloride hydrochloride | Homo sapiens (human) | Potency | 16.1936 | 2 | 0 |
prazosin hydrochloride | Homo sapiens (human) | Potency | 41.3363 | 2 | 0 |
5,6-benzocoumarin-3-carboxylic acid ethyl ester | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
masoprocol | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
betamipron | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
tetrandrine | Homo sapiens (human) | Potency | 0.8913 | 1 | 0 |
nodakenin | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
ergocornine | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
irinotecan hydrochloride | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
4'-methoxyflavone | Homo sapiens (human) | Potency | 28.6288 | 2 | 0 |
8-methyl-4-oxo-3-pyrido[1,2-a]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
2-amino-5-bromobenzoic acid | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
2-(1H-benzimidazol-2-yl)aniline | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-methylumbelliferyl butyrate | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
7-(diethylamino)-1-benzopyran-2-one | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-methylumbelliferyl glucuronide | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
7-amino-4-methylcoumarin | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
harmol hydrochloride | Homo sapiens (human) | Potency | 29.9033 | 2 | 0 |
hexaphosphamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3,7-dimethyl-1-propargylxanthine | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
7,9-dimethyl-9aH-quinolizine-1,2,3,4-tetracarboxylic acid tetramethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
alphaxalone | Homo sapiens (human) | Potency | 6.3096 | 1 | 0 |
1-(2-methoxyphenyl)-4-(4-(2-phthalimido)butyl)piperazine | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
benzamil | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
vadimezan | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
methotrexate | Homo sapiens (human) | Potency | 19.6222 | 1 | 0 |
nsc-141549 | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
alpha-methylhistamine | Homo sapiens (human) | Potency | 63.0957 | 1 | 0 |
n-phthaloylglutamic acid | Homo sapiens (human) | Potency | 7.9433 | 1 | 0 |
3-cyano-7-ethoxycoumarin | Homo sapiens (human) | Potency | 21.8959 | 1 | 0 |
2-hexynyladenosine-5'-n-ethylcarboxamide | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
esatenolol | Homo sapiens (human) | Potency | 3.5481 | 1 | 0 |
migalastat | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
fr 122047 | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
6-methyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrile | Homo sapiens (human) | Potency | 42.8000 | 2 | 0 |
5-(3,4,5-trimethoxyphenyl)-3H-1,3,4-oxadiazol-2-one | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
2,6-diphenyl-1,7-dihydropyrazolo[3,4-b]pyridine-3,4-dione | Homo sapiens (human) | Potency | 3.1623 | 1 | 0 |
nsc606985 | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
2,5-bis(5-hydroxymethyl-2-thienyl)furan | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
N2-phenyl-5-methyl-4,5-dihydro-1,3-thiazol-2-amine | Homo sapiens (human) | Potency | 0.2239 | 1 | 0 |
1-methyl-3-phenylpyrazino[1,2-a]benzimidazole | Homo sapiens (human) | Potency | 35.7168 | 2 | 0 |
ritonavir | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ochratoxin a | Homo sapiens (human) | Potency | 27.7170 | 2 | 0 |
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol | Homo sapiens (human) | Potency | 32.8152 | 3 | 0 |
3-[di(propan-2-yl)phosphorylmethyl]benzonitrile | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
jp-1302 | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-furancarboxylic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] ester | Homo sapiens (human) | Potency | 3.5481 | 1 | 0 |
4,7-dimethoxy-2,3-dihydroinden-1-one | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1,3-dichloro-7-methyl-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrile | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-[6-(4-aminophenyl)-2-phenyl-4-pyrimidinyl]aniline | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
benzylideneacetone | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
xanthoangelol | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-imino-N,8-dimethyl-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamide | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
N-butan-2-yl-N-[2-[(4-methoxyphenyl)methylamino]-2-oxoethyl]-4-thiadiazolecarboxamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-(1-adamantyl)-3-[8-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]urea | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
3-(benzenesulfonyl)-2-imino-1-(2-oxolanylmethyl)-5-dipyrido[1,2-d-3',4'-f]pyrimidinone | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
1-[3-(4-morpholinyl)propyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-phenylurea | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-methoxy-3-[[2-oxolanylmethyl-[1-[1-(phenylmethyl)-5-tetrazolyl]propyl]amino]methyl]-1H-quinolin-2-one | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
8-[2-(4-methoxyphenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decane | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-methyl-4-[2-oxo-2-(2-phenylethylamino)ethyl]-5-thieno[3,2-b]pyrrolecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
1-[(3,4-dimethoxyphenyl)-[1-(2-methoxyethyl)-5-tetrazolyl]methyl]-2,3-dihydroindole | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
7-(2-methyl-2,3-dihydroindol-1-yl)-3-(phenylmethyl)triazolo[4,5-d]pyrimidine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
3-[1-azepanyl-[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl]-6,7-dimethoxy-1H-quinolin-2-one | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-(4-methoxyphenyl)-8-(6-methyl-2-phenyl-4-pyrimidinyl)-8-azabicyclo[3.2.1]octan-3-ol | Homo sapiens (human) | Potency | 7.9433 | 1 | 0 |
3-[[4-(1-benzotriazolyl)-1-piperidinyl]sulfonyl]-N-cyclopentylbenzenesulfonamide | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
N-[1,3-dimethyl-2-oxo-5-[[oxo(propoxy)methyl]amino]-4-imidazolidinyl]carbamic acid propyl ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-ethyl-6-methyl-5,8-dihydro-1H-thiopyrano[2,3]thieno[2,4-b]pyrimidine-2,4-dione | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
2-[(7-methyl-4-oxo-3-phenyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-2-yl)thio]acetic acid methyl ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
LSM-19776 | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
5-[10-(5-methoxy-1,5-dioxopentyl)-1,7-dioxa-4,10-diazacyclododec-4-yl]-5-oxopentanoic acid methyl ester | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
N-[5-[[2-(4-methylanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-2-(4-morpholinyl)acetamide | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
1-methyl-2-[(phenylthio)methyl]-3-indolecarbonitrile | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
6-cyclohexyl-3-furan-2-yl-(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazole | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-(1H-benzimidazol-2-ylmethylthio)-2-methylbenzofuro[3,2-d]pyrimidine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-(3-methylphenyl)sulfonyl-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetonitrile | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamine | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-2-pyridinecarboxamide | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl ester | Homo sapiens (human) | Potency | 0.3162 | 1 | 0 |
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanol | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
2-amino-4-(2-furanyl)-6-(2-pyridinyl)-3-pyridinecarbonitrile | Homo sapiens (human) | Potency | 36.4261 | 2 | 0 |
7-butyl-8-[[4-(3-chlorophenyl)-1-piperazinyl]methyl]-1,3-dimethylpurine-2,6-dione | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
5-[(2-chloro-6-fluorophenyl)methyl]-N-[2-[4-(4-methoxyphenyl)-1-piperazinyl]ethyl]-1,3,4-oxadiazole-2-carboxamide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
LSM-33283 | Homo sapiens (human) | Potency | 20.2676 | 2 | 0 |
ag-213 | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3',4'-dimethoxyflavone | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
caffeic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-[(dimethylamino)methyl]-4-methyl-6-(1-methylcyclohexyl)phenol | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-[[oxo(phenoxy)methyl]amino]benzene-1,4-dicarboxylic acid dimethyl ester | Homo sapiens (human) | Potency | 27.0050 | 2 | 0 |
2-thiophenecarboxylic acid 2-(1,3-dioxo-2-isoindolyl)ethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
7,7-dimethyl-2-(1-pyrrolidinyl)-5,8-dihydropyrano[4,3-b]pyridine-3-carbonitrile | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
2-methyl-N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)propanamide | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
1-(3-pyridinylmethyl)-3-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]urea | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-[[4-amino-2-(ethylamino)-5-thiazolyl]-phenylmethylidene]propanedinitrile | Homo sapiens (human) | Potency | 32.4648 | 2 | 0 |
(2'-(4-aminophenyl)-(2,5'-bi-1h-benzimidazol)-5-amine) | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
N-[[6-cyano-5-(ethylamino)-3-methyl-2-pyrazinyl]methyl]-N-phenylacetamide | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
4-(4-morpholinylmethyl)-3-quinolinol | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
5-(4-morpholinyl)-2-thiophen-2-yl-4-oxazolecarbonitrile | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
7-methoxy-2-oxo-1-benzopyran-3-carboxylic acid ethyl ester | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
7,8-dichloropyrido[1,2-a]benzimidazole | Homo sapiens (human) | Potency | 2.8184 | 1 | 0 |
7-acetoxycoumarin | Homo sapiens (human) | Potency | 31.8326 | 2 | 0 |
5-chloro-2-methoxy-N,N,4-trimethylbenzenesulfonamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
2-(2-fluorophenyl)-5-(4-methoxyanilino)-4-oxazolecarbonitrile | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
1-(4-methyl-2-oxo-1-benzopyran-7-yl)-3-(2-pyridinylmethyl)thiourea | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2,4-dimethyl-N-[4-(1-pyrrolidinyl)phenyl]benzamide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
2-[4-chloro-2-methyl-5-(2-pyridinylsulfamoyl)phenoxy]acetamide | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
2-[3-(4-methoxyphenyl)-1-benzo[f]quinolinyl]acetic acid ethyl ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
DND-167 dye | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
2-[methyl-(2,4,6-trimethylphenyl)sulfonylamino]-N-(2-pyridinylmethyl)acetamide | Homo sapiens (human) | Potency | 0.7943 | 1 | 0 |
2-(2,4,5-trimethoxyphenyl)-1,3-benzothiazole | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
ym-90709 | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
N-[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]-4-methylbenzamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3-(2-chloro-6-fluorophenyl)-N-(3-fluoro-4-methylphenyl)-5-methyl-4-isoxazolecarboxamide | Homo sapiens (human) | Potency | 1.2589 | 1 | 0 |
1-(3,4-dimethoxyphenyl)sulfonyl-4-(2-methoxyphenyl)piperazine | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
N-[4-[methyl(phenyl)sulfamoyl]phenyl]-2-thiophenecarboxamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
5-(2-amino-4-thiazolyl)-2,4-dimethyl-1H-pyrrole-3-carboxylic acid methyl ester | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
4-ethyl-5-methyl-N-[1-[(3-methylphenyl)methyl]-1,2,4-triazol-3-yl]-3-thiophenecarboxamide | Homo sapiens (human) | Potency | 63.0957 | 1 | 0 |
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamine | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
7-chloro-4-[4-(3,4-dimethylphenyl)sulfonyl-1-piperazinyl]quinoline | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-bromo-5-[[4-[hydroxy(diphenyl)methyl]-1-piperidinyl]-oxomethyl]-2-pyranone | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-(4-fluorophenyl)-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrile | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinone | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-tert-butyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrile | Homo sapiens (human) | Potency | 40.0748 | 2 | 0 |
2-(4-methylsulfonylphenyl)-6-imidazo[1,2-a]pyridinecarboxylic acid methyl ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
3-(5-chloro-1,3-benzoxazol-2-yl)-N-(phenylmethyl)-2-pyridinamine | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
N,N-dimethylcarbamic acid [4-[2-(4-fluorophenyl)sulfonyl-1-oxoethyl]-2,6-dimethylphenyl] ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
2-(4-chlorophenoxy)-4-(dimethylamino)-3-pyridinecarbonitrile | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
5-cyano-2-phenyl-6-[4-(2-pyridinyl)-1-piperazinyl]-3-pyridinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N2,N2-dimethyl-6-[[[1-(1-naphthalenyl)-5-tetrazolyl]thio]methyl]-1,3,5-triazine-2,4-diamine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
aurapten | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
6-(1,3-dioxo-2-isoindolyl)hexanoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
4-amino-2-[[4-amino-6-(4-fluoroanilino)-1,3,5-triazin-2-yl]methylthio]-5-pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-[(1,3-benzothiazol-2-ylthio)methyl]-4-triazolecarboxylic acid methyl ester | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
2-chloro-4,6-diphenyl-5-pyrimidinamine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
1-[2-[(3-chloro-4-methoxyphenyl)methylthio]ethyl]-3-phenylthiourea | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-amino-1-[2-(4-morpholinyl)ethyl]-N-prop-2-enyl-3-pyrrolo[3,2-b]quinoxalinecarboxamide | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
1-[2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl]-3-phenylurea | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-amino-N-(3-ethoxypropyl)-1-(4-sulfamoylphenyl)-3-pyrrolo[3,2-b]quinoxalinecarboxamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-(3,4-dimethoxyphenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
3-(1,3-benzothiazol-2-yl)propanoic acid (3,5-dimethyl-4-isoxazolyl)methyl ester | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
4-(2-oxo-1-pyrrolidinyl)benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
2-[2-furanyl(oxo)methyl]imino-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
4-[[(2-nitrophenyl)-oxomethyl]amino]benzoic acid propyl ester | Homo sapiens (human) | Potency | 6.3096 | 1 | 0 |
N-(4-chlorophenyl)-4-methyl-2-thiazolamine | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-(3-hydroxyphenyl)-1-(thiophen-2-ylmethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-phenyl-3-[2-(phenylmethylthio)ethyl]-1H-1,2,4-triazole-5-thione | Homo sapiens (human) | Potency | 0.1778 | 1 | 0 |
N-[2-[5-(1,3-benzothiazol-2-yl)-3-ethyl-1-phenyl-2-benzimidazol-3-iumyl]ethenyl]-N-methylaniline | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-methoxy-2-naphthalenecarboxylic acid [2-(4-morpholinyl)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
1-[1-(phenylmethyl)-4-piperidinyl]-3-(2-propan-2-ylphenyl)thiourea | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
1-(2-methoxyethyl)-7-thiophen-2-yl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione | Homo sapiens (human) | Potency | 35.7168 | 2 | 0 |
1-butyl-2,4-dioxo-7-thiophen-2-yl-5-pyrido[2,3-d]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-(2-furanylmethylamino)benzoic acid [2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl] ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3-methyl-2-thiophenecarboxylic acid [2-(4-morpholinyl)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 1.0000 | 1 | 0 |
2-(butylamino)benzoic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] ester | Homo sapiens (human) | Potency | 44.9647 | 2 | 0 |
5-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acid | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-[ethyl(phenyl)sulfamoyl]-4-methylbenzoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) ester | Homo sapiens (human) | Potency | 21.1699 | 2 | 0 |
digoxin | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
2-oxo-6-phenyl-4-(trifluoromethyl)-1H-pyridine-3-carbonitrile | Homo sapiens (human) | Potency | 22.0164 | 2 | 0 |
1-[[2-[5-[3,5-bis(trifluoromethyl)phenyl]-2-tetrazolyl]-1-oxoethyl]amino]-3-(4-chlorophenyl)thiourea | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-[bis(5-methyl-2-furanyl)methyl]-6-nitrophenol | Homo sapiens (human) | Potency | 5.6234 | 1 | 0 |
1-[(3-chlorophenyl)methyl]-3-[5-(methylthio)-1,3,4-oxadiazol-2-yl]-2-pyridinone | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-chlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] ester | Homo sapiens (human) | Potency | 24.0353 | 2 | 0 |
5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-amine | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
8-methoxy-4-oxo-1H-quinoline-2-carboxylic acid methyl ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
N-[1-(4-methyl-6-oxo-1-pyrimidinyl)-2-oxo-2-phenylethyl]benzamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrimidine | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
methyl-thiohydantoin-tryptophan | Homo sapiens (human) | Potency | 0.1122 | 1 | 0 |
3-(4-ethyl-1-piperazinyl)-5-methylpyridazino[3,4-b][1,4]benzoxazine | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
1-(2,6-dimethyl-1-piperidinyl)-2-phenylethanone | Homo sapiens (human) | Potency | 0.0631 | 1 | 0 |
1-(4-fluorophenyl)-3-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]pyrrolidine-2,5-dione | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
3-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) ester | Homo sapiens (human) | Potency | 30.3001 | 2 | 0 |
N-[(2-hydroxy-1-naphthalenyl)-(4-methoxyphenyl)methyl]-2-methylpropanamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-(3-hydroxyphenyl)-1-(2-oxolanylmethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
5-[(3,4-dimethoxyphenyl)methyl]-1-prop-2-enyl-1,3-diazinane-2,4,6-trione | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
5-(2-oxolanylmethylamino)-2-thiophen-2-yl-4-oxazolecarbonitrile | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-[[2-(2,3-dihydro-1,4-benzodioxin-3-yl)-1-oxoethyl]amino]benzoic acid ethyl ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamide | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
1-(4-morpholinyl)-2-(4-phenylphenoxy)-1-propanone | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazole | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-[5-(4-methylphenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acid | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-[5-(4-fluorophenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acid | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
[2-[(2,6-dimethyl-4-morpholinyl)-oxomethyl]phenyl]-(1H-imidazol-2-yl)methanone | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
2-(2-furanyl)-N-(2-oxolanylmethyl)-4-quinolinecarboxamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
N-[1-(1H-benzimidazol-2-yl)-2-phenylethyl]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxo-3-pyrrolidinecarboxamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-(4-methylphenyl)sulfonyl-1-(3-oxolanylmethyl)-2-pyrrolo[3,2-b]quinoxalinamine | Homo sapiens (human) | Potency | 35.7168 | 2 | 0 |
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
yl-109 | Homo sapiens (human) | Potency | 26.6320 | 2 | 0 |
LSM-24662 | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-[2-(tert-butylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2-oxolanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
N-[2-(cyclopentylamino)-2-oxoethyl]-4,7-dimethyl-N-(2-methylphenyl)-2-oxo-3H-pyrido[1,2-a]pyrimidine-4-carboxamide | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
3-[[2-(4-fluorophenoxy)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
7-(4-methoxyphenyl)-5-methyl-2-(methylthio)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
1-(4-methylphenyl)sulfonyl-3-methylsulfonylimidazolidine | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
4-[2-[(1'-acetyl-4-oxo-6-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]yl)oxy]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-[(3-oxo-2-propan-2-yl-2H-imidazo[1,2-c]quinazolin-5-yl)thio]-N-[2-(4-sulfamoylphenyl)ethyl]acetamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-[[(3-methoxyphenyl)-oxomethyl]amino]benzoic acid | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
1-[[4-[(4-fluorophenyl)methyl]-5-thieno[3,2-b]pyrrolyl]-oxomethyl]-N-(2-furanylmethyl)-4-piperidinecarboxamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2,4-dioxo-3-(2-oxolanylmethyl)-N-pentyl-1H-quinazoline-7-carboxamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
2-(2-methoxyethyl)-9-methyl-4-[(4-methyl-1-piperidinyl)-oxomethyl]-1-pyrido[3,4-b]indolone | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamide | Homo sapiens (human) | Potency | 40.0748 | 2 | 0 |
[1-(3-methylphenyl)-5-benzimidazolyl]-(1-piperidinyl)methanone | Homo sapiens (human) | Potency | 7.0795 | 1 | 0 |
4-[2-[[1-[(2-methylphenyl)methyl]-3-indolyl]sulfonyl]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
4-morpholinecarboxylic acid [3-(6-amino-5-cyano-3-propan-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
cyclobutyl-[5-[(2-ethyl-1-piperidinyl)sulfonyl]-2,3-dihydroindol-1-yl]methanone | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
2,5-dimethyl-N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-(2-naphthalenylamino)-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]-3-pyrazolecarboxamide | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
5-amino-2-(3-nitrophenyl)-1-phenyl-2H-pyrrole-3,3,4-tricarbonitrile | Homo sapiens (human) | Potency | 5.6234 | 1 | 0 |
2,3-dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
1-(3-ethoxypropyl)-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
N-[4-[2-(2-ethyl-1-oxobutyl)-3-phenyl-3,4-dihydropyrazol-5-yl]phenyl]methanesulfonamide | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
sodium dodecyl sulfate | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
2-[[2-(4-methoxyphenyl)-6-methyl-1-benzopyran-4-ylidene]amino]-4-methylpentanoic acid | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-butyl-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
2-benzoylimino-1-(2-furanylmethyl)-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-dimethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolamine | Homo sapiens (human) | Potency | 10.7362 | 2 | 0 |
obtusinin | Homo sapiens (human) | Potency | 42.8000 | 2 | 0 |
6-[2-(1-azepanyl)-2-oxoethoxy]-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-one | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-[[7-(4-methoxyphenyl)-5-phenyl-4-pyrrolo[2,3-d]pyrimidinyl]thio]propanoic acid ethyl ester | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
2-thiophen-2-yl-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) ester | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
5-(4-ethoxyphenyl)-1,3-diphenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dione | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
LSM-24581 | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
LSM-17147 | Homo sapiens (human) | Potency | 50.1187 | 2 | 0 |
N-(2-fluorophenyl)-6-(1,2,4-triazol-1-yl)-3-pyridinecarboxamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
LSM-31277 | Homo sapiens (human) | Potency | 22.0164 | 2 | 0 |
2-amino-4-(2-fluorophenyl)-6-(3-pyridinyl)-3-pyridinecarbonitrile | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
N-[4-[cyano-[3-[2-(4-morpholinyl)ethylamino]-2-quinoxalinyl]methyl]sulfonylphenyl]acetamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-1-nitro-9,10-dioxo-2-anthracenecarboxamide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-[4-[cyano-[3-(3-hydroxypropylamino)-2-quinoxalinyl]methyl]sulfonylphenyl]acetamide | Homo sapiens (human) | Potency | 30.3001 | 2 | 0 |
1-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-ethyl-1-(2-furanylmethyl)thiourea | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4-[4-diethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolyl]morpholine | Homo sapiens (human) | Potency | 25.2855 | 2 | 0 |
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
7-methoxy-N-(3-pyridinylmethyl)-2-furo[2,3-b]quinolinecarboxamide | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
5,5,7,7-tetramethyl-2-[[oxo-(4-propan-2-yloxyphenyl)methyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid methyl ester | Homo sapiens (human) | Potency | 42.8000 | 2 | 0 |
N-[4-(1H-benzimidazol-2-yl)phenyl]-3-(2,5-dioxo-1-pyrrolidinyl)benzamide | Homo sapiens (human) | Potency | 37.6460 | 2 | 0 |
LSM-27960 | Homo sapiens (human) | Potency | 3.5717 | 2 | 0 |
LSM-16446 | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
4-(9-acridinylamino)-1,5-dimethyl-2-phenyl-3-pyrazolone | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
6-chloro-2-[(phenylmethylthio)methyl]imidazo[1,2-a]pyridine | Homo sapiens (human) | Potency | 1.4125 | 1 | 0 |
LSM-31434 | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
3-(benzenesulfonyl)-1-cyclopropyl-2-pyrrolo[3,2-b]quinoxalinamine | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-dimethoxyphosphoryl-2-(1-naphthalenyl)-N-(phenylmethyl)-5-oxazolamine | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
2-(2,3-dihydroxypropylamino)-5-nitro-3-pyridinecarbonitrile | Homo sapiens (human) | Potency | 6.3096 | 1 | 0 |
1-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-[3-(dimethylamino)propyl]-1-ethylthiourea | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
LSM-24516 | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
LSM-28572 | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
5-(4-methylphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acid | Homo sapiens (human) | Potency | 17.0157 | 2 | 0 |
5-methyl-2-phenyl-4-propan-2-ylidene-3-pyrazolone | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
cgp 7930 | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-(3-oxo-2-benzo[f][1]benzopyranyl)acetamide | Homo sapiens (human) | Potency | 10.1578 | 2 | 0 |
N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]cyclohexanecarboxamide | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
4-tert-butyl-N-[3-[4-[3-[[(4-tert-butylphenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]benzamide | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
sphingosine | Homo sapiens (human) | Potency | 4.4668 | 1 | 0 |
luteolin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
scopoletin | Homo sapiens (human) | Potency | 30.2470 | 2 | 0 |
hymecromone | Homo sapiens (human) | Potency | 24.0682 | 2 | 0 |
gossypetin | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
fucoxanthin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
esculetin | Homo sapiens (human) | Potency | 27.8525 | 2 | 0 |
7-hydroxycoumarin | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
hyperoside | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
coumestrol | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
4',7-dihydroxyflavone | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
glyceryl 2-arachidonate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
n-oleoylethanolamine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
phenoxybenzamine hydrochloride | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
1-(3-amino-7-methoxy-1-pyrazolo[3,4-b]quinolinyl)-2-(2-methoxyphenyl)ethanone | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-(2,5-dimethoxyphenyl)-2-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methylsulfonyl]acetamide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
N-[2-(4-morpholinyl)ethyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamide | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
1-(4-tert-butylphenyl)sulfonyl-N-(2-pyridinylmethyl)-2-piperidinecarboxamide | Homo sapiens (human) | Potency | 3.5481 | 1 | 0 |
N-(1,3-benzodioxol-5-yl)-2-(5-methyl-2-furanyl)-3-imidazo[1,2-a]pyrazinamine | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
N-[3-(4-methyl-1-piperazinyl)propyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamide | Homo sapiens (human) | Potency | 27.7170 | 2 | 0 |
ml 10302 | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
psb 1115 | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
furazolidone | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
ag 556 | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
8-(3-chlorostyryl)caffeine | Homo sapiens (human) | Potency | 4.8022 | 1 | 0 |
nomifensine maleate | Homo sapiens (human) | Potency | 8.9125 | 1 | 0 |
7-hydroxy-4-methyl-1H-quinolin-2-one | Homo sapiens (human) | Potency | 35.4813 | 2 | 0 |
7-hydroxy-6-(4-morpholinylmethyl)-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-4-one | Homo sapiens (human) | Potency | 33.5520 | 2 | 0 |
sulindac sulfone | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
dithiazanine iodide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-fluoro-N-phenyl-1,3-benzothiazol-2-amine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-[3-(4-morpholinyl)propyl]-2,4-dioxo-3-(2-phenylethyl)-1H-quinazoline-7-carboxamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-(3,4-dimethylphenyl)-2,5-dioxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarbonitrile | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
1'-acetyl-6-[2-(4-ethyl-1-piperazinyl)-2-oxoethoxy]-4-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]one | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-(2-methoxyethyl)-2,4-dioxo-N-pentyl-1H-quinazoline-7-carboxamide | Homo sapiens (human) | Potency | 39.8107 | 2 | 0 |
ipamorelin | Homo sapiens (human) | Potency | 0.7943 | 1 | 0 |
2-(4'-methylaminophenyl)benzothiazole | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
lilly 78335 | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
fenoldopam hydrobromide | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
3-methoxytyramine hydrochloride | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
3-hydroxy-3-methyl-5-oxo-5-[[3,4,5-trihydroxy-6-[[6-methoxy-2-oxo-3-[(2-oxo-1-benzopyran-7-yl)oxy]-1-benzopyran-7-yl]oxy]-2-oxanyl]methoxy]pentanoic acid | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
N-(3-fluorophenyl)-2-(9-oxo-10-acridinyl)acetamide | Homo sapiens (human) | Potency | 4.4668 | 1 | 0 |
4-[3-(3-fluorophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
[5-Chloranyl-3-[(1E,3E)-3,5-dimethylhepta-1,3-dienyl]-7-methyl-6,8-bis(oxidanylidene)isochromen-7-yl] ethanoate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N'-butan-2-yl-N-[2-(3,5-dimethyl-1-piperidinyl)-4-methyl-6-quinolinyl]butanediamide | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
3-[[(3R,4S)-2-(4-bromophenyl)-5-(3-chlorophenyl)-4-(2-methoxyphenyl)-3,4-dihydropyrazol-3-yl]-oxomethyl]-2-oxazolidinone | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanone | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
N-(2-furanylmethyl)-2-[[4-oxo-3-[3-(1-pyrrolidinyl)propyl]-[1]benzothiolo[3,2-d]pyrimidin-2-yl]thio]acetamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-[3-[(6-methoxy-2-naphthalenyl)-oxomethyl]-1-piperidinyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)thio]ethanone | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
N-(5-chloro-2-pyridinyl)-4H-thieno[3,2-c][1]benzopyran-2-carboxamide | Homo sapiens (human) | Potency | 16.9036 | 2 | 0 |
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl ester | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
8-[1-[4-(dimethylamino)phenyl]-3-(3-methyl-1-piperidinyl)propyl]-5,7-dimethoxy-4-phenyl-1-benzopyran-2-one | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ampicillin sodium | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
phenytoin sodium | Homo sapiens (human) | Potency | 1.1220 | 1 | 0 |
l 817818 | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
4-hydroxy-6-methyl-2-pyrone | Homo sapiens (human) | Potency | 0.7943 | 1 | 0 |
mobic | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
ethyl 1-benzyl-3-hydroxy-2(5h)-oxopyrrole-4-carboxylate | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
folic acid | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
isoxanthopterin | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
5-amino-2-phenyl-3H-triazolo[4,5-d]pyrimidin-7-one | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
5,5-diethyl-2-(2-hydroxyethylamino)-1,6-dihydrobenzo[h]quinazolin-4-one | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |