Page last updated: 2024-08-07 13:13:54

Vasopressin V2 receptor

A vasopressin V2 receptor that is encoded in the genome of pig. [OMA:P32307, PRO:DNx]

Synonyms

V2R;
AVPR V2;
Antidiuretic hormone receptor;
Renal-type arginine vasopressin receptor

Research

Bioassay Publications (3)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (6)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
relcovaptanSus scrofa (pig)Ki0.285011
opc 21268Sus scrofa (pig)Ki10.000011
l 371257Sus scrofa (pig)Ki37.000011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
1,3-dipropyl-8-cyclopentylxanthineSus scrofa (pig)Kb0.140011
theophyllineSus scrofa (pig)Kb14.000011
caffeineSus scrofa (pig)Kb30.000011