Page last updated: 2024-08-07 18:35:47

Solute carrier organic anion transporter family member 1A1

A solute carrier organic anion transporter family member 1A1 that is encoded in the genome of rat. [OMA:P46720, PRO:DNx]

Synonyms

Organic anion-transporting polypeptide 1;
OATP-1;
Sodium-independent organic anion transporter 1;
Solute carrier family 21 member 1

Research

Bioassay Publications (18)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's13 (72.22)18.2507
2000's5 (27.78)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (35)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ibuprofenRattus norvegicus (Norway rat)Ki126.000011
probenecidRattus norvegicus (Norway rat)Ki74.400011
corticosteroneRattus norvegicus (Norway rat)Ki5.300011
estriolRattus norvegicus (Norway rat)Ki9.800011
estroneRattus norvegicus (Norway rat)Ki15.700011
androsteroneRattus norvegicus (Norway rat)Ki10.600011
sulfobromophthalein sodiumRattus norvegicus (Norway rat)Ki1.980011
taurocholic acidRattus norvegicus (Norway rat)Ki21.400022
estradiol-3-sulfateRattus norvegicus (Norway rat)Ki1.100011
ethinyl estradiol-17-sulfateRattus norvegicus (Norway rat)Ki1.300011
testosterone 17-glucosiduronateRattus norvegicus (Norway rat)Ki3.800011
androsterone sulfateRattus norvegicus (Norway rat)Ki2.400011
corticosterone sulfateRattus norvegicus (Norway rat)Ki1.600011
estradiol-3-glucuronideRattus norvegicus (Norway rat)Ki9.700011
quinidineRattus norvegicus (Norway rat)Ki9.270011
estrone sulfateRattus norvegicus (Norway rat)Ki1.300011
quinineRattus norvegicus (Norway rat)Ki76.700011
rifamycin svRattus norvegicus (Norway rat)Ki6.600011
rifampinRattus norvegicus (Norway rat)Ki18.200011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
fexofenadineRattus norvegicus (Norway rat)Km32.000011
aldosteroneRattus norvegicus (Norway rat)Km0.015011
sulfobromophthalein sodiumRattus norvegicus (Norway rat)Km2.600032
taurocholic acidRattus norvegicus (Norway rat)Km36.520045
glycocholic acidRattus norvegicus (Norway rat)Km54.000011
dehydroepiandrosterone sulfateRattus norvegicus (Norway rat)Km5.000011
pravastatinRattus norvegicus (Norway rat)Km30.000011
taurochenodeoxycholic acidRattus norvegicus (Norway rat)Km5.950021
ouabainRattus norvegicus (Norway rat)Km2,350.000022
ochratoxin aRattus norvegicus (Norway rat)Km22.800022
temocaprilatRattus norvegicus (Norway rat)Km46.700011
bq 123Rattus norvegicus (Norway rat)Km600.000011
sodium taurodeoxycholateRattus norvegicus (Norway rat)Km3.500011
estrone sulfateRattus norvegicus (Norway rat)Km7.750022
estradiol-17 beta-glucuronideRattus norvegicus (Norway rat)Km7.911477
hyodeoxycholic acidRattus norvegicus (Norway rat)Km17.500011
enalaprilRattus norvegicus (Norway rat)Km252.000011
ursodoxicoltaurineRattus norvegicus (Norway rat)Km13.000011
deltorphin ii, ala(2)-Rattus norvegicus (Norway rat)Km137.000011