Page last updated: 2024-08-07 19:27:55

Calcium/calmodulin-dependent protein kinase type II subunit alpha

A calcium/calmodulin-dependent protein kinase type II subunit alpha that is encoded in the genome of rat. [OMA:P11275, PRO:DNx]

Synonyms

CaM kinase II subunit alpha;
CaMK-II subunit alpha;
EC 2.7.11.17

Research

Bioassay Publications (6)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's0 (0.00)24.3611
2020's2 (33.33)2.80

Compounds (10)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
diclofenacRattus norvegicus (Norway rat)Ki5.100011
4-hydroxybutyric acidRattus norvegicus (Norway rat)Ki19.433333
2-hydroxyphenylacetic acidRattus norvegicus (Norway rat)IC500.002111
2-hydroxyphenylacetic acidRattus norvegicus (Norway rat)Ki1.995311
3-hydroxybenzeneacetic acidRattus norvegicus (Norway rat)IC500.000111
3-hydroxybenzeneacetic acidRattus norvegicus (Norway rat)Ki0.125911
staurosporineRattus norvegicus (Norway rat)IC500.059011
5-hydroxydiclofenacRattus norvegicus (Norway rat)Ki0.510345
kn 93Rattus norvegicus (Norway rat)IC508.400011
arcyriaflavin aRattus norvegicus (Norway rat)IC500.639428
jnj-7706621Rattus norvegicus (Norway rat)IC5034.0700113
3-hydroxycyclopent-1-enecarboxylic acidRattus norvegicus (Norway rat)Ki0.696733