Page last updated: 2024-08-07 12:21:30

Chain A, Putative fructose-1,6-bisphosphate aldolase

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (1194)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
gallic acidGiardia intestinalisPotency8.832620
deoxycytidineGiardia intestinalisPotency10.000010
indol-3-yl pyruvic acidGiardia intestinalisPotency15.811410
dihydroxyphenylalanineGiardia intestinalisPotency15.811410
kynurenineGiardia intestinalisPotency17.740710
n-acetylserotoninGiardia intestinalisPotency4.456310
pyrazinoic acidGiardia intestinalisPotency17.740710
quinolinic acidGiardia intestinalisPotency8.220410
catechinGiardia intestinalisPotency9.976310
2,4-methanoglutamateGiardia intestinalisPotency5.610110
vanilmandelic acidGiardia intestinalisPotency22.334210
5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)-3,4-dihydro-2H-chromen-3-yl 3,4,5-trihydroxybenzoateGiardia intestinalisPotency9.976310
1,10-phenanthrolineGiardia intestinalisPotency14.299610
2,2'-dipyridylGiardia intestinalisPotency44.562510
2,4,5-trichlorophenoxyacetic acidGiardia intestinalisPotency17.740710
2-methyl-5-htGiardia intestinalisPotency11.193610
p-chloromercuribenzoic acidGiardia intestinalisPotency19.905410
chlorocresolGiardia intestinalisPotency15.811410
phenytoinGiardia intestinalisPotency19.905410
6-hydroxymelatoninGiardia intestinalisPotency7.062710
7,8-dihydroxyflavoneGiardia intestinalisPotency7.924510
oxyquinolineGiardia intestinalisPotency31.622810
aa 861Giardia intestinalisPotency16.776110
acemetacinGiardia intestinalisPotency15.811410
beta-aminoethyl isothioureaGiardia intestinalisPotency25.059410
ag 127Giardia intestinalisPotency17.740710
tyrphostin a23Giardia intestinalisPotency14.091910
tyrphostin 25Giardia intestinalisPotency15.811410
5-aminoisoquinolinoneGiardia intestinalisPotency11.193610
amlexanoxGiardia intestinalisPotency22.334210
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolGiardia intestinalisPotency7.623720
aristolochic acid iGiardia intestinalisPotency22.334210
aurintricarboxylic acidGiardia intestinalisPotency35.397310
azinphosmethylGiardia intestinalisPotency22.334210
benzbromaroneGiardia intestinalisPotency17.740710
benzothiazideGiardia intestinalisPotency15.811410
berberineGiardia intestinalisPotency6.565610
2,5-di-tert-butylhydroquinoneGiardia intestinalisPotency4.456310
bay h 4502Giardia intestinalisPotency25.059410
brimonidineGiardia intestinalisPotency14.467210
carbidopaGiardia intestinalisPotency15.811410
carbonyl cyanide m-chlorophenyl hydrazoneGiardia intestinalisPotency35.397310
3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-7-[[1-oxo-2-(1-tetrazolyl)ethyl]amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidGiardia intestinalisPotency15.848910
chelerythrineGiardia intestinalisPotency11.370410
chloroxineGiardia intestinalisPotency11.530110
chloroxylenolGiardia intestinalisPotency15.811410
cisplatinGiardia intestinalisPotency19.905410
amberlite cg 400Giardia intestinalisPotency8.891410
2,3-dimethoxy-5-methyl-6-decyl-1,4-benzoquinoneGiardia intestinalisPotency2.233410
deferiproneGiardia intestinalisPotency6.190410
pentetic acidGiardia intestinalisPotency21.797030
diflunisalGiardia intestinalisPotency21.964210
disulfiramGiardia intestinalisPotency18.823110
ebselenGiardia intestinalisPotency22.665530
embelinGiardia intestinalisPotency25.059410
erythrosineGiardia intestinalisPotency15.811410
ethacrynic acidGiardia intestinalisPotency17.740710
ethoxyquinGiardia intestinalisPotency17.740710
flufenamic acidGiardia intestinalisPotency15.811410
flumequineGiardia intestinalisPotency25.059410
fusaric acidGiardia intestinalisPotency11.559710
gliclazideGiardia intestinalisPotency8.912510
glimepirideGiardia intestinalisPotency18.823110
glyburideGiardia intestinalisPotency19.072810
gossypolGiardia intestinalisPotency19.350310
gyki 52466Giardia intestinalisPotency39.716410
2,2',3,3',4,4'-hexahydroxy-1,1'-biphenyl-6,6'-dimethanol dimethyl etherGiardia intestinalisPotency3.971610
beta-thujaplicinGiardia intestinalisPotency14.091910
ethidiumGiardia intestinalisPotency0.561010
hydralazineGiardia intestinalisPotency12.559410
idebenoneGiardia intestinalisPotency4.456310
amrinoneGiardia intestinalisPotency3.095110
indigotindisulfonateGiardia intestinalisPotency17.740710
indomethacinGiardia intestinalisPotency25.157410
iodoacetamideGiardia intestinalisPotency31.547910
jugloneGiardia intestinalisPotency4.574910
lansoprazoleGiardia intestinalisPotency18.711610
lapacholGiardia intestinalisPotency1.446810
beta-lapachoneGiardia intestinalisPotency1.785810
lavendustin bGiardia intestinalisPotency19.905410
nordefrinGiardia intestinalisPotency4.456310
ly 171883Giardia intestinalisPotency22.334210
vitamin k 3Giardia intestinalisPotency2.733820
mesalamineGiardia intestinalisPotency3.539710
3-Hydroxy-alpha-methyl-DL-tyrosineGiardia intestinalisPotency11.193610
3,7-bis(dimethylamino)phenothiazin-5-iumGiardia intestinalisPotency17.740710
etoposide phosphateGiardia intestinalisPotency12.559410
nifedipineGiardia intestinalisPotency12.741510
nimesulideGiardia intestinalisPotency15.811410
masoprocolGiardia intestinalisPotency22.334210
omeprazoleGiardia intestinalisPotency24.049220
oxidopamineGiardia intestinalisPotency5.610110
pd 153035Giardia intestinalisPotency25.059410
pd 158780Giardia intestinalisPotency0.315510
1,3a,8-Trimethyl-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-yl methylcarbamateGiardia intestinalisPotency50.000010
probenecidGiardia intestinalisPotency19.905410
prochlorperazineGiardia intestinalisPotency15.811410
protopineGiardia intestinalisPotency7.062710
protoporphyrin ixGiardia intestinalisPotency11.193610
1,2,5,8-tetrahydroxy anthraquinoneGiardia intestinalisPotency1.000010
hydrochlorothiazideGiardia intestinalisPotency12.893810
ro 31-8220Giardia intestinalisPotency17.740710
sanguinarineGiardia intestinalisPotency6.294610
sb 220025Giardia intestinalisPotency15.811410
streptonigrinGiardia intestinalisPotency0.315510
sulfobromophthaleinGiardia intestinalisPotency15.811410
tetrahydroxy-1,4-quinoneGiardia intestinalisPotency12.559410
thiramGiardia intestinalisPotency22.750630
tinoridineGiardia intestinalisPotency17.740710
tolazamideGiardia intestinalisPotency17.740710
trigonellineGiardia intestinalisPotency35.397310
trimetrexateGiardia intestinalisPotency5.610110
vincaGiardia intestinalisPotency7.062710
pirinixic acidGiardia intestinalisPotency25.059410
xanthurenic acidGiardia intestinalisPotency9.976310
alloxanGiardia intestinalisPotency15.811410
procaine hydrochlorideGiardia intestinalisPotency14.125410
isoproterenol hydrochlorideGiardia intestinalisPotency6.319020
penicillamineGiardia intestinalisPotency12.559410
racepinephrine hydrochlorideGiardia intestinalisPotency1.990510
cystamine dihydrochlorideGiardia intestinalisPotency15.811410
physostigmineGiardia intestinalisPotency15.811410
apomorphineGiardia intestinalisPotency22.334210
cephalothinGiardia intestinalisPotency28.117110
carbostyrilGiardia intestinalisPotency15.811410
thiamineGiardia intestinalisPotency7.943310
papaverine hydrochlorideGiardia intestinalisPotency9.121010
methylene blueGiardia intestinalisPotency22.334210
egtazic acidGiardia intestinalisPotency31.547910
gliotoxinGiardia intestinalisPotency22.334210
quinacrine monohydrochlorideGiardia intestinalisPotency15.811410
chlorpromazine hydrochlorideGiardia intestinalisPotency17.740710
purpurinGiardia intestinalisPotency17.740710
acenaphthenequinoneGiardia intestinalisPotency2.233410
lawsoneGiardia intestinalisPotency15.811410
7,8-dimethyl-10-[(2R,3R,4S)-2,3,4,5-tetrahydroxypentyl]benzo[g]pteridine-2,4-dioneGiardia intestinalisPotency7.924510
9,10-phenanthrenequinoneGiardia intestinalisPotency4.617430
acriflavine chlorideGiardia intestinalisPotency2.233410
sulfaethidoleGiardia intestinalisPotency15.848910
diethyl ketoneGiardia intestinalisPotency14.091910
tetramethylthiuram monosulfideGiardia intestinalisPotency15.811410
methyl gallateGiardia intestinalisPotency15.811410
barbanGiardia intestinalisPotency7.062710
4-phenylenediamineGiardia intestinalisPotency4.917110
diethylenetriamineGiardia intestinalisPotency17.740710
1-amino-4-hydroxyanthraquinoneGiardia intestinalisPotency15.811410
chloranilGiardia intestinalisPotency0.561010
dextrothyroxineGiardia intestinalisPotency19.905410
amprolium hydrochlorideGiardia intestinalisPotency17.740710
chelidamic acidGiardia intestinalisPotency17.740710
protocatechualdehydeGiardia intestinalisPotency7.924510
cysteamine hydrochlorideGiardia intestinalisPotency15.811410
chlormadinone acetateGiardia intestinalisPotency17.740710
hydralazine hydrochlorideGiardia intestinalisPotency15.029710
lithocholic acidGiardia intestinalisPotency15.811410
glycyrrhetinic acidGiardia intestinalisPotency15.811410
glaucineGiardia intestinalisPotency0.177410
rheinGiardia intestinalisPotency22.334210
plumbaginGiardia intestinalisPotency0.111910
imperatorinGiardia intestinalisPotency16.776110
dihydralazineGiardia intestinalisPotency17.740710
2,4-pyridinedicarboxylic acidGiardia intestinalisPotency1.774110
dipicolinic acidGiardia intestinalisPotency28.183810
hematoxylinGiardia intestinalisPotency13.100010
1,2-naphthoquinoneGiardia intestinalisPotency3.539710
chlormethiazoleGiardia intestinalisPotency31.547910
gentian violetGiardia intestinalisPotency15.811410
amitriptyline hydrochlorideGiardia intestinalisPotency17.740710
6-aminoquinolineGiardia intestinalisPotency2.233410
Berberine chloride (TN)Giardia intestinalisPotency4.456310
phosmetGiardia intestinalisPotency19.905410
carbophenothionGiardia intestinalisPotency15.811410
malononitrile dimerGiardia intestinalisPotency3.154810
diphenyl disulfideGiardia intestinalisPotency19.905410
3-methoxycatecholGiardia intestinalisPotency17.740710
2,2'-diaminodiphenyldisulfideGiardia intestinalisPotency15.811410
ethidium bromideGiardia intestinalisPotency1.258910
carmineGiardia intestinalisPotency20.037410
tribromsalanGiardia intestinalisPotency19.905410
methylene diphosphonateGiardia intestinalisPotency6.294610
dienochlorGiardia intestinalisPotency17.740710
quinomethionateGiardia intestinalisPotency5.610110
pontamine sky blueGiardia intestinalisPotency11.193610
cyclacillinGiardia intestinalisPotency11.193610
palmatineGiardia intestinalisPotency12.559410
nsc 3852Giardia intestinalisPotency12.351410
todralazineGiardia intestinalisPotency11.193610
nitroxolineGiardia intestinalisPotency19.905410
2-hydroxyjugloneGiardia intestinalisPotency6.294610
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineGiardia intestinalisPotency5.000010
4-(4-dimethylaminophenylazo)benzoic acidGiardia intestinalisPotency25.118910
isoetharine mesylateGiardia intestinalisPotency5.851610
hydroxyzine pamoateGiardia intestinalisPotency16.776110
diacereinGiardia intestinalisPotency22.334210
benserazide hydrochlorideGiardia intestinalisPotency7.572410
cephalexinGiardia intestinalisPotency11.876510
metergolineGiardia intestinalisPotency7.924510
1-(trimethylsilyl)-1h-imidazoleGiardia intestinalisPotency22.387210
daunorubicinGiardia intestinalisPotency18.213010
ergocristineGiardia intestinalisPotency3.154810
cefazolinGiardia intestinalisPotency17.740710
oxcarbazepineGiardia intestinalisPotency16.776110
carbidopaGiardia intestinalisPotency17.740710
prothiophosGiardia intestinalisPotency12.559410
10-carboxymethyl-9-acridanoneGiardia intestinalisPotency31.622810
ticrynafenGiardia intestinalisPotency19.905410
methyldopaGiardia intestinalisPotency14.342110
nitazoxanideGiardia intestinalisPotency14.091910
s-2678Giardia intestinalisPotency12.559410
terazosin hydrochloride anhydrousGiardia intestinalisPotency15.811410
triclabendazoleGiardia intestinalisPotency15.811410
cefaclor anhydrousGiardia intestinalisPotency11.205610
mitoxantrone hydrochlorideGiardia intestinalisPotency17.740710
dazoxiben hydrochlorideGiardia intestinalisPotency17.740710
lovastatinGiardia intestinalisPotency15.811410
chaetochrominGiardia intestinalisPotency6.294610
imazaquinGiardia intestinalisPotency6.294610
daunorubicin hydrochlorideGiardia intestinalisPotency12.559410
desferrioxamine b mesylateGiardia intestinalisPotency0.445610
meclizine monohydrochlorideGiardia intestinalisPotency19.905410
epigallocatechin gallateGiardia intestinalisPotency14.091910
salvinGiardia intestinalisPotency9.976310
neocuproineGiardia intestinalisPotency35.481310
ticlopidine hydrochlorideGiardia intestinalisPotency35.397310
glutathione disulfideGiardia intestinalisPotency1.990510
benzydamine hydrochlorideGiardia intestinalisPotency28.183810
physodic acidGiardia intestinalisPotency25.059410
pazufloxacinGiardia intestinalisPotency19.905410
repaglinideGiardia intestinalisPotency17.740710
toxoflavinGiardia intestinalisPotency5.417230
n(4)-acetylsulfamerazineGiardia intestinalisPotency35.481310
N(4)-acetylsulfathiazoleGiardia intestinalisPotency19.952610
dimidium bromideGiardia intestinalisPotency1.584910
2,6-dimethoxy-1,4-benzoquinoneGiardia intestinalisPotency7.062710
prazosin hydrochlorideGiardia intestinalisPotency17.740710
mianserin hydrochlorideGiardia intestinalisPotency9.976310
plasmenylserineGiardia intestinalisPotency39.716410
n-acetylhistamineGiardia intestinalisPotency28.183810
2-chloro-1,4-benzoquinoneGiardia intestinalisPotency44.562510
5-fluoroorotic acidGiardia intestinalisPotency19.905410
4-aminobenzo-2,1,3-thiadiazoleGiardia intestinalisPotency17.740710
3-methylxanthineGiardia intestinalisPotency15.811410
5-aminoisoquinolineGiardia intestinalisPotency4.456310
4-hexyloxybenzoic acidGiardia intestinalisPotency17.740710
2,2',2''-terpyridineGiardia intestinalisPotency29.021620
bicinchoninic acidGiardia intestinalisPotency2.511910
masoprocolGiardia intestinalisPotency12.559410
jatrorrhizineGiardia intestinalisPotency19.905410
tetrahydroalstonineGiardia intestinalisPotency5.000010
9-aminocamptothecinGiardia intestinalisPotency1.409210
2,2'-((3,3'-dimethoxy(1,1'-biphenyl)-4,4'-diyl)diimino)bis-benzoic acidGiardia intestinalisPotency35.397310
methyl fluorone blackGiardia intestinalisPotency11.437110
9-hydroxyphenylfluoronGiardia intestinalisPotency9.025020
3-aminophenoxazoneGiardia intestinalisPotency18.846620
5-nitro-1,10-phenanthrolineGiardia intestinalisPotency22.334210
ergocornineGiardia intestinalisPotency1.990510
tryptanthrineGiardia intestinalisPotency7.093910
8-hydroxy-2-quinolinecarboxylic acidGiardia intestinalisPotency22.159230
1-ethyl-2-benzo[cd]indoloneGiardia intestinalisPotency17.740710
4-(2-thiazolylazo)resorcinolGiardia intestinalisPotency5.000010
4,4'-dipyridyl disulfideGiardia intestinalisPotency25.118910
3,5-di-tert-butyl-1,2-benzoquinoneGiardia intestinalisPotency7.062710
2,4,6-tripyridyl-s-triazineGiardia intestinalisPotency15.811410
4-phenyl-1,2,4-triazoline-3,5-dioneGiardia intestinalisPotency17.782810
2-methyl-4-nitroquinoline 1-oxideGiardia intestinalisPotency22.334210
6-aminoindazoleGiardia intestinalisPotency7.924510
5-chloroindole-2-carboxylateGiardia intestinalisPotency15.916310
5-aminoindazoleGiardia intestinalisPotency3.539710
4,5-dimethoxy-2-nitrobenzaldehydeGiardia intestinalisPotency5.000010
1,8-bis(dimethylamino)naphthaleneGiardia intestinalisPotency3.154810
prochlorperazine edisylate saltGiardia intestinalisPotency35.397310
gliquidoneGiardia intestinalisPotency17.740710
D-dopaGiardia intestinalisPotency15.811410
meclizine hydrochlorideGiardia intestinalisPotency17.740710
tarenflurbilGiardia intestinalisPotency35.397310
1-(2-thiazolylazo)-2-naphtholGiardia intestinalisPotency18.839220
3-(n-salicyloyl)amino-1,2,4-triazoleGiardia intestinalisPotency19.905410
2-(4-hydroxyphenyl)-5,6,7,8-tetrahydroxy-4H-1-benzopyran-4-oneGiardia intestinalisPotency13.434820
2,3-bis(2-pyridinyl)quinoxalineGiardia intestinalisPotency19.905410
oxoglaucineGiardia intestinalisPotency3.539710
phellopterinGiardia intestinalisPotency17.740710
6,6'-methylene bis(2,2,4-trimethyl-1,2-dihydroquinoline)Giardia intestinalisPotency28.183810
4-methoxydalbergioneGiardia intestinalisPotency19.905410
n-acetyldopamineGiardia intestinalisPotency9.976310
3-chloro-6-hydrazino-pyridazineGiardia intestinalisPotency19.905410
1,2-bis(2-aminophenoxy)ethane-n,n,n',n'-tetraacetic acidGiardia intestinalisPotency3.971610
sudan yellow 3gGiardia intestinalisPotency17.740710
awd 19166Giardia intestinalisPotency7.943310
homoorientinGiardia intestinalisPotency17.740710
tanshinoneGiardia intestinalisPotency1.255910
3,4-dimethoxydalbergioneGiardia intestinalisPotency22.334210
eserolineGiardia intestinalisPotency4.456310
roemerineGiardia intestinalisPotency2.233410
medica 16Giardia intestinalisPotency17.740710
ly 255283Giardia intestinalisPotency17.740710
pd 81723Giardia intestinalisPotency25.059410
loe 908Giardia intestinalisPotency15.811410
a 68930Giardia intestinalisPotency25.059410
nsc 607097Giardia intestinalisPotency1.258910
cp 93129Giardia intestinalisPotency25.059410
2,2'-pyridylisatogen tosylateGiardia intestinalisPotency14.091910
3-hydroxyphenazepamGiardia intestinalisPotency15.811410
sdz 220-581Giardia intestinalisPotency13.858510
omeprazole magnesiumGiardia intestinalisPotency12.589310
n-(6-methoxy-8-quinolyl)-4-toluenesulfonamideGiardia intestinalisPotency14.951610
pyrophenGiardia intestinalisPotency19.905410
isoteolinGiardia intestinalisPotency3.971610
3',4'-dihydroxyflavoneGiardia intestinalisPotency15.811410
n-methylserotoninGiardia intestinalisPotency25.059410
12-phenyllauric acidGiardia intestinalisPotency15.811410
2-benzenesulfonamidopyrimidineGiardia intestinalisPotency28.183810
nefopam hydrochlorideGiardia intestinalisPotency10.000010
oxidopamine hydrochlorideGiardia intestinalisPotency6.294610
cryptotanshinoneGiardia intestinalisPotency13.484010
Serotonin hydrochlorideGiardia intestinalisPotency3.539710
epiberberineGiardia intestinalisPotency1.990510
8-(4-benzenesulfonylamino)quinolineGiardia intestinalisPotency28.775710
stephenanthrineGiardia intestinalisPotency7.062710
tanshinone ii aGiardia intestinalisPotency12.401710
corbadrineGiardia intestinalisPotency7.062710
2-phenyl-1,2-benzisothiazol-3-(2h)-oneGiardia intestinalisPotency12.559410
n-methylpapaverineGiardia intestinalisPotency19.905410
cystamine hydrochlorideGiardia intestinalisPotency19.905410
1-benzylimidazole-4,5-dicarboxylic acidGiardia intestinalisPotency7.933920
carboline-3-carboxylic acidGiardia intestinalisPotency12.589310
2,10,11-trihydroxy-n-n-propylnoraporphineGiardia intestinalisPotency12.559410
sb 216763Giardia intestinalisPotency15.848910
chrysene-1,4-dioneGiardia intestinalisPotency14.091910
fonsecinGiardia intestinalisPotency1.255910
brazilinGiardia intestinalisPotency17.740710
nsc13345Giardia intestinalisPotency15.848910
gossypol acetic acidGiardia intestinalisPotency15.811410
(R)-RoemerineGiardia intestinalisPotency0.251210
3-nitrotyrosineGiardia intestinalisPotency17.740710
2-pentan-3-yl-1H-imidazoleGiardia intestinalisPotency35.481310
PorfiromycineGiardia intestinalisPotency17.740710
2-hydroxyestradiolGiardia intestinalisPotency9.896220
1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diolGiardia intestinalisPotency12.639110
4-[(1,3-dimethyl-2,6-dioxo-7H-purin-8-yl)methylamino]benzoic acidGiardia intestinalisPotency19.952610
n-methylserotonin oxalate saltGiardia intestinalisPotency1.990510
nsc 95397Giardia intestinalisPotency9.570430
2-chloro-3-(4-methylanilino)naphthalene-1,4-dioneGiardia intestinalisPotency1.581110
methylnaphthazarinGiardia intestinalisPotency8.891410
papaverinolGiardia intestinalisPotency15.811410
2-glycineamide-5-chlorophenyl-2-pyrryl ketoneGiardia intestinalisPotency22.334210
oxopurpureineGiardia intestinalisPotency19.905410
5-(4-methylphenyl)-2H-tetrazoleGiardia intestinalisPotency35.481310
2-(4-aminophenyl)quinolineGiardia intestinalisPotency22.334210
2-quinolinecarboxylic acid (4-nitrophenyl) esterGiardia intestinalisPotency25.118910
nafronyloxalateGiardia intestinalisPotency16.797110
nsc228155Giardia intestinalisPotency2.886330
dicentrineGiardia intestinalisPotency0.500010
hematoxylinGiardia intestinalisPotency19.905410
N-(4-fluorophenyl)carbamic acid (2-oxo-1H-pyridin-3-yl) esterGiardia intestinalisPotency0.934920
3-(prop-2-enylthio)-5-thiophen-2-yl-1H-1,2,4-triazoleGiardia intestinalisPotency12.589310
5-aminonicotinic acidGiardia intestinalisPotency16.776110
4,5,7-trihydroxy-9,10-dioxo-2-anthracenecarboxylic acidGiardia intestinalisPotency17.740710
7-hydroxy-5-methyl-2-(2-oxopropyl)-8-[3,4,5-trihydroxy-6-(hydroxymethyl)-2-oxanyl]-1-benzopyran-4-oneGiardia intestinalisPotency17.740710
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneGiardia intestinalisPotency1.255910
7-benzoyl-3-chloroindolizine-1,2-dicarboxylic acid dimethyl esterGiardia intestinalisPotency15.811410
8-anilino-1,3-dimethyl-7H-purine-2,6-dioneGiardia intestinalisPotency22.334210
2,3-diaminophenazineGiardia intestinalisPotency0.445610
carboplatinGiardia intestinalisPotency14.091910
5-hydroxytryptophanGiardia intestinalisPotency5.000010
raubasineGiardia intestinalisPotency5.610110
hematoxylinGiardia intestinalisPotency14.091910
GirgensonineGiardia intestinalisPotency9.976310
L-isoprenalineGiardia intestinalisPotency6.974010
Saphenic acid methyl esterGiardia intestinalisPotency19.905410
carubicinGiardia intestinalisPotency12.559410
doxorubicin hydrochlorideGiardia intestinalisPotency22.334210
dihydroergocristine monomesylateGiardia intestinalisPotency14.091910
aconitic acidGiardia intestinalisPotency12.559410
hts 466284Giardia intestinalisPotency15.811410
dactinomycinGiardia intestinalisPotency7.062710
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneGiardia intestinalisPotency4.496520
menadione sodium bisulfite, trihydrateGiardia intestinalisPotency8.912510
jp-1302Giardia intestinalisPotency15.811410
4-(4-chloro-2-methylphenoxy)-n-hydroxybutanamideGiardia intestinalisPotency15.811410
1-(4-methylphenyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneGiardia intestinalisPotency28.183810
8-prop-2-enylsulfonylquinolineGiardia intestinalisPotency15.811410
6-nitro-1,3-benzodioxol-5-amineGiardia intestinalisPotency12.559410
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimineGiardia intestinalisPotency22.334210
tolfenamic acidGiardia intestinalisPotency15.811410
4-[[bis(2-hydroxyethyl)amino]methyl]-2,6-ditert-butylphenolGiardia intestinalisPotency17.740710
2,4-bis(4-methoxyphenyl)-4-methyl-1,2,3,5-tetrahydro-1,5-benzodiazepineGiardia intestinalisPotency15.811410
4-methyl-2-[(5-methyl-2-thiophenyl)methylideneamino]phenolGiardia intestinalisPotency15.811410
6-amino-2-methyl-8-phenyl-1,6,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileGiardia intestinalisPotency17.740710
2-[[5-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-1,2,4-triazol-3-yl]thio]-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamideGiardia intestinalisPotency3.548110
3-[(1-cyclopentyl-5-tetrazolyl)-(3,4-dihydro-1H-isoquinolin-2-yl)methyl]-7-methoxy-1H-quinolin-2-oneGiardia intestinalisPotency14.091910
LSM-34798Giardia intestinalisPotency19.952610
N-butan-2-yl-N-[2-[(4-methoxyphenyl)methylamino]-2-oxoethyl]-4-thiadiazolecarboxamideGiardia intestinalisPotency6.309610
N-[1-[(4-methylphenyl)methyl]-2-benzimidazolyl]-2-furancarboxamideGiardia intestinalisPotency25.059410
N-[2,5-diethoxy-4-[[2-(3-methoxyphenyl)-1-oxoethyl]amino]phenyl]-2-furancarboxamideGiardia intestinalisPotency17.740710
N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-cyclohexyl-2-furancarboxamideGiardia intestinalisPotency14.091910
3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazoleGiardia intestinalisPotency11.193610
2-(1,3-benzodioxol-5-ylamino)-N-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetamideGiardia intestinalisPotency17.740710
4-methoxy-1,3-dimethyl-6-thiophen-2-yl-8-cyclohepta[c]furanoneGiardia intestinalisPotency15.811410
6-amino-4-[4-(2-amino-2-oxoethoxy)-2-chloro-5-methoxyphenyl]-5-cyano-2-methyl-4H-pyran-3-carboxylic acid methyl esterGiardia intestinalisPotency15.811410
4-[2-[[4-(dimethylamino)phenyl]methylamino]ethyl]-2,2-dimethyl-4-oxanolGiardia intestinalisPotency12.559410
1-[1-[oxo(1-pyrrolidinyl)methyl]cyclohexyl]-3-(phenylmethyl)ureaGiardia intestinalisPotency3.548110
N-[2-[1,3-benzodioxol-5-yl-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-furancarboxamideGiardia intestinalisPotency19.905410
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-(2,6-dimethoxyphenyl)methanoneGiardia intestinalisPotency15.848910
3-[(1-cyclopentyl-5-tetrazolyl)-[4-(2-methoxyphenyl)-1-piperazinyl]methyl]-7-methyl-1H-quinolin-2-oneGiardia intestinalisPotency28.183810
6-amino-4-(2,3-dimethoxyphenyl)-3-methyl-1-phenyl-4H-pyrano[2,3-c]pyrazole-5-carbonitrileGiardia intestinalisPotency2.818410
9,10-dimethoxy-2,4,6,7-tetrahydro-[1,3]oxazino[4,3-a]isoquinoline-1-carbonitrileGiardia intestinalisPotency25.118910
6,7-dimethoxy-2-[[2-[4-(4-methoxyphenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-quinolinecarbonitrileGiardia intestinalisPotency12.559410
1-(1-piperidinyl)-2-[[4-(prop-2-enylamino)-1-phthalazinyl]thio]ethanoneGiardia intestinalisPotency14.125410
3-(2,5-dimethyl-1-pyrrolyl)-4-methylanilineGiardia intestinalisPotency25.059410
6-hydroxy-1-(3-hydroxypropyl)-4-methyl-2-oxo-5-(1-piperidinylmethyl)-3-pyridinecarbonitrileGiardia intestinalisPotency7.062710
6-(3,4-dimethoxyphenyl)-4-methoxy-1,3-dimethyl-8-cyclohepta[c]furanoneGiardia intestinalisPotency11.220210
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-methyl-1H-quinolin-2-oneGiardia intestinalisPotency17.740710
3-[[1-(1,3-benzodioxol-5-ylmethyl)-5-tetrazolyl]-(1-pyrrolidinyl)methyl]-8-methyl-1H-quinolin-2-oneGiardia intestinalisPotency19.952610
5,8-dimethoxy-4-(4-methyl-1-piperazinyl)-2-(trifluoromethyl)quinolineGiardia intestinalisPotency15.811410
N-[2-[1,3-benzodioxol-5-yl-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-furancarboxamideGiardia intestinalisPotency19.905410
N-[2,5-dimethoxy-4-[[2-(4-morpholinyl)-1-oxoethyl]amino]phenyl]benzamideGiardia intestinalisPotency25.059410
2-[(5-methyl-1H-1,2,4-triazol-3-yl)thio]-1-phenylethanoneGiardia intestinalisPotency12.589310
3-[[4-(1-benzotriazolyl)-1-piperidinyl]sulfonyl]-N-cyclopentylbenzenesulfonamideGiardia intestinalisPotency17.740710
2-[[5-[[2-(3-chloroanilino)-4-thiazolyl]methyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]thio]acetic acid methyl esterGiardia intestinalisPotency14.091910
5-(2-furanyl)-N-(4-methylphenyl)-3-isoxazolecarboxamideGiardia intestinalisPotency25.059410
propylthiouracilGiardia intestinalisPotency17.740710
1-cyclohexyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-amineGiardia intestinalisPotency22.334210
2'-amino-5',6'-dimethoxy-1'-spiro[cyclopentane-1,3'-indene]carbonitrileGiardia intestinalisPotency17.740710
2-[2-hydroxy-6,7-dimethoxy-4-(4-morpholinyl)-1-naphthalenyl]-N-phenylacetamideGiardia intestinalisPotency25.118910
LSM-19776Giardia intestinalisPotency22.334210
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideGiardia intestinalisPotency20.037410
1-[(1,3-benzothiazol-2-ylthio)methyl]-2-azepanoneGiardia intestinalisPotency17.740710
4-amino-3-(2-furyl)-5-mercapto-1,2,4-triazoleGiardia intestinalisPotency6.294610
2-cyano-N-(2-furanylmethyl)-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetamideGiardia intestinalisPotency22.334210
1-(4-hydroxyphenyl)-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaGiardia intestinalisPotency15.811410
2-cyano-2-[3-[4-(phenylmethyl)-1-piperazinyl]-2-quinoxalinyl]acetic acid 2-methoxyethyl esterGiardia intestinalisPotency0.397210
2-[[5-cyano-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,3-thiazin-6-yl]thio]acetic acid ethyl esterGiardia intestinalisPotency44.562510
3-(6-methyl-4-oxo-2-sulfanylidene-1H-pyrimidin-5-yl)propanoic acid methyl esterGiardia intestinalisPotency19.905410
1,3-dimethyl-6-(1-naphthalenyl)pyrrolo[3,4-d]pyrimidine-2,4-dioneGiardia intestinalisPotency12.559410
2-amino-4-(2-ethoxyphenyl)-7-methyl-5-oxo-6-(2-pyridinylmethyl)-4H-pyrano[3,2-c]pyridine-3-carbonitrileGiardia intestinalisPotency17.740710
N-(3-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideGiardia intestinalisPotency3.539710
2-[[4-amino-5-(4-tert-butylphenyl)-1,2,4-triazol-3-yl]thio]acetic acid propan-2-yl esterGiardia intestinalisPotency22.334210
LSM-32147Giardia intestinalisPotency17.740710
3-[(4-methoxyanilino)methyl]-1H-quinolin-2-oneGiardia intestinalisPotency11.193610
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-(dimethylamino)-4-oxazolecarbonitrileGiardia intestinalisPotency31.547910
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneGiardia intestinalisPotency20.063920
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-propyl-2-pyridinecarboxamideGiardia intestinalisPotency15.811410
1-(3,4-dihydroxyphenyl)-2-[[5-(2-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneGiardia intestinalisPotency6.033620
LSM-28489Giardia intestinalisPotency17.740710
N5,N5-dimethyl-2,1,3-benzoxadiazole-4,5-diamineGiardia intestinalisPotency12.559410
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileGiardia intestinalisPotency4.466810
2-amino-6-[3-(1-imidazolyl)propyl]-4-(2-methoxyphenyl)-7-methyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carbonitrileGiardia intestinalisPotency17.740710
3-(2-furanylmethyl)-8-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileGiardia intestinalisPotency0.445610
5-(1,3-benzodioxol-5-ylmethylamino)-2-(4-morpholinyl)benzoic acid methyl esterGiardia intestinalisPotency15.811410
7-chloro-5-(4-morpholinyl)-2,1,3-benzoxadiazol-4-amineGiardia intestinalisPotency3.539710
mercaptopurineGiardia intestinalisPotency17.788020
methylthiouracilGiardia intestinalisPotency15.811410
dexketoprofenGiardia intestinalisPotency25.059410
ag-213Giardia intestinalisPotency14.091910
3,3',4,5'-tetrahydroxystilbeneGiardia intestinalisPotency15.811410
2-mercaptonicotinic acidGiardia intestinalisPotency4.456310
7,8,3'-trihydroxyflavoneGiardia intestinalisPotency19.905410
6-methyl-2-(trifluoromethyl)-3,5-dihydroimidazo[4,5-f]benzimidazoleGiardia intestinalisPotency3.154810
benzylthiouracilGiardia intestinalisPotency15.811410
3',4'-dimethoxyflavoneGiardia intestinalisPotency21.702920
caffeic acidGiardia intestinalisPotency21.230010
4-(4-propan-2-yl-1-piperazinyl)phenolGiardia intestinalisPotency7.924510
4-(3-amino-2-imidazo[1,2-a]pyridinyl)-2-methoxyphenolGiardia intestinalisPotency25.118910
2-(8-quinolinylthio)acetic acidGiardia intestinalisPotency17.740710
N-(2-furanylmethyl)-4-(2-methyl-3-imidazo[1,2-a]pyridinyl)-2-thiazolamineGiardia intestinalisPotency11.193610
ondansetron, (s)-isomerGiardia intestinalisPotency17.782810
N-[(4-pyrimidinylthio)methyl]benzamideGiardia intestinalisPotency15.811410
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-oneGiardia intestinalisPotency12.559410
2-methyl-5-(1,4,5,7-tetramethyl-6-pyrrolo[3,4-d]pyridazinyl)anilineGiardia intestinalisPotency15.811410
4-(3-chlorophenyl)thiosemicarbazideGiardia intestinalisPotency17.740710
N-[(3-nitroanilino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency15.811410
5-bromo-N-(5-methyl-2-pyridinyl)-2-thiophenesulfonamideGiardia intestinalisPotency7.924510
1-(3,4-dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanoneGiardia intestinalisPotency11.220210
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileGiardia intestinalisPotency15.811410
4-chloro-N-(3,4,5-trimethoxyphenyl)-5-dithiazolimineGiardia intestinalisPotency19.905410
N-(2-chlorophenyl)hydrazine-1-carbothioamideGiardia intestinalisPotency15.811410
phenylthiazolylthioureaGiardia intestinalisPotency0.631010
5-amino-3-(4-methoxyphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterGiardia intestinalisPotency0.561010
2-anilino-N-(4-fluorophenyl)acetamideGiardia intestinalisPotency19.905410
2-(3-nitrophenyl)-2,3-dihydro-1H-perimidineGiardia intestinalisPotency19.905410
5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineGiardia intestinalisPotency35.397310
2-(thiophen-2-ylmethylidene)indene-1,3-dioneGiardia intestinalisPotency1.581110
1-(2,5-dimethoxyphenyl)-3-phenylthioureaGiardia intestinalisPotency39.810710
pseudoginsenoside f11Giardia intestinalisPotency5.610110
5-phenyl-1,3,4-oxadiazole-2-thiolGiardia intestinalisPotency7.062710
5-amino-3-(4-methoxyphenyl)-7-methyl-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid methyl esterGiardia intestinalisPotency1.990510
2-amino-4-(2-furanyl)-3-thiophenecarboxylic acid ethyl esterGiardia intestinalisPotency9.976310
N-[(3,5-dimethoxyphenyl)methyl]-1-[4-(methylthio)phenyl]methanamineGiardia intestinalisPotency15.811410
2-(4-hydroxyanilino)-1,4-naphthoquinoneGiardia intestinalisPotency7.062710
3-[(6-methyl-4-phenyl-2-quinazolinyl)amino]propanoic acidGiardia intestinalisPotency17.740710
4-[(2-methoxy-1-naphthalenyl)methyl]thiomorpholineGiardia intestinalisPotency15.848910
1-(cyclohexylmethyl)-4-phenylpiperazineGiardia intestinalisPotency28.183810
2-(2,3-dihydroindol-1-yl)-N,N-dimethylethanamineGiardia intestinalisPotency25.118910
4-pyridin-4-yl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrileGiardia intestinalisPotency2.505910
3,4,5-trimethoxybenzoic acid [(3,5-dimethyl-4-oxo-1-cyclohexa-2,5-dienylidene)amino] esterGiardia intestinalisPotency5.610110
4-(2,5-dimethylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency19.905410
N-(4-methoxyphenyl)carbamic acid (9-fluorenylideneamino) esterGiardia intestinalisPotency4.456310
nsc185058Giardia intestinalisPotency14.058620
2,2,2-trifluoro-N-(2-methyl-8-quinolinyl)acetamideGiardia intestinalisPotency15.811410
1-(2-chloro-6-fluorophenyl)-[1,2,4]triazolo[4,3-a]quinolineGiardia intestinalisPotency15.811410
N'-[(4-chlorophenyl)-oxomethyl]-2-pyrazinecarbohydrazideGiardia intestinalisPotency12.559410
4-(2-furanylmethyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency2.811710
2-[4-[(3-fluorophenyl)methyl]-1-piperazinyl]pyrimidineGiardia intestinalisPotency15.811410
1-[(3,4-dimethoxyphenyl)methyl]-4-(2,3-dimethylphenyl)piperazineGiardia intestinalisPotency19.905410
2-(2-phenylethyl)-1,3-benzoxazol-5-amineGiardia intestinalisPotency44.562510
N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)-2-(1-pyrrolidinyl)acetamideGiardia intestinalisPotency17.782810
4-(4-chlorophenyl)-3-[(4-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency14.125410
4-(3-fluorophenyl)-2-thiazolamineGiardia intestinalisPotency11.193610
1-(1,3-benzodioxol-5-ylmethyl)-3-(2,1,3-benzothiadiazol-5-yl)thioureaGiardia intestinalisPotency11.193610
3,5,5-trimethyl-4H-pyrazole-1-carbothioamideGiardia intestinalisPotency11.193610
thiopyrineGiardia intestinalisPotency15.811410
4-(2-naphthalenylmethyl)-1-piperazinecarboxylic acid ethyl esterGiardia intestinalisPotency25.118910
2-[(3-fluorophenyl)methyl-(phenylmethyl)amino]ethanolGiardia intestinalisPotency15.811410
6-(4-morpholinyl)naphthalene-2,3-dicarbonitrileGiardia intestinalisPotency3.154810
2-(1,4,5,7-tetramethyl-6-pyrrolo[3,4-d]pyridazinyl)anilineGiardia intestinalisPotency3.154810
4-(4-morpholinyl)-N-(pyridin-4-ylmethyl)anilineGiardia intestinalisPotency19.905410
2-(3-cyano-4,5,6-trimethyl-1H-pyridin-2-ylidene)propanedinitrileGiardia intestinalisPotency7.062710
2-methoxy-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-6-nitrophenolGiardia intestinalisPotency17.782810
N-[[(4,6-dimethyl-2-pyrimidinyl)amino]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency19.952610
9-ethyl-1,2,4,5-tetrazaspiro[5.5]undecane-3-thioneGiardia intestinalisPotency12.559410
4-tert-butyl-N-(1,4-dioxo-2,3-dihydrophthalazin-5-yl)benzamideGiardia intestinalisPotency17.877220
6-(1,4,5,7-tetramethyl-6-pyrrolo[3,4-d]pyridazinyl)quinolineGiardia intestinalisPotency7.924510
4-(5-methoxy-1,2-dimethyl-3-indolyl)-2-thiazolamineGiardia intestinalisPotency17.782810
2-[2-[[benzamido(sulfanylidene)methyl]amino]-4-thiazolyl]acetic acid ethyl esterGiardia intestinalisPotency1.990510
5-[(5-acetyl-2-propan-2-yloxyphenyl)methyl]-6-hydroxy-2-sulfanylidene-1H-pyrimidin-4-oneGiardia intestinalisPotency14.091910
6-[amino(methyl)amino]-N2,N4-diethyl-1,3,5-triazine-2,4-diamineGiardia intestinalisPotency44.562510
2-[[(3-methylphenyl)-oxomethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acidGiardia intestinalisPotency15.811410
N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideGiardia intestinalisPotency28.117110
N-[(2,3-dimethoxyphenyl)methyl]-4-(4-methyl-1-piperidinyl)anilineGiardia intestinalisPotency4.456310
3-ethoxy-N-[(3-pyridinylamino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency7.924510
3-(1,3-dimethyl-4-pyrazolyl)-4-(2-methoxyphenyl)-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency7.924510
N'-[(4-chlorophenyl)-oxomethyl]-2-hydroxy-3-methylbenzohydrazideGiardia intestinalisPotency11.193610
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideGiardia intestinalisPotency12.559410
N-[[(6-methyl-4-pyrimidinyl)thio]methyl]benzamideGiardia intestinalisPotency14.091910
1-(2-methyl-6-propan-2-ylphenyl)-5-phenyltetrazoleGiardia intestinalisPotency15.811410
N-[[(6-methoxy-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency4.456310
4-sulfanylidene-1,6,7,8,9,10-hexahydropyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileGiardia intestinalisPotency17.740710
3-acetyl-2-methylbenzo[f]benzofuran-4,9-dioneGiardia intestinalisPotency0.397210
N-[(2,1,3-benzothiadiazol-4-ylamino)-sulfanylidenemethyl]-4-methylbenzamideGiardia intestinalisPotency3.971610
N-[(3-acetylanilino)-sulfanylidenemethyl]-3-chlorobenzamideGiardia intestinalisPotency7.924510
5-acetyloxy-2-[[cyclohexyl(oxo)methyl]amino]benzoic acidGiardia intestinalisPotency17.740710
1-propylsulfonyl-4-(2-pyridinyl)piperazineGiardia intestinalisPotency31.547910
1-cyclopropyl-3-(4-sulfamoylphenyl)thioureaGiardia intestinalisPotency19.905410
N-[(2-methoxyphenyl)methyl]-4-(1-piperidinyl)anilineGiardia intestinalisPotency14.091910
5-amino-3-(2-methylphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterGiardia intestinalisPotency1.119410
1-(4-methoxyphenyl)-1-methyl-3-(1-methyl-5-benzotriazolyl)ureaGiardia intestinalisPotency15.811410
1-(2-hydroxyphenyl)-2-(2H-tetrazol-5-yl)ethanoneGiardia intestinalisPotency5.000010
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneGiardia intestinalisPotency12.559410
3-amino-2-(4-methoxyphenyl)-7-nitro-1-oxo-4-isoquinolinecarbonitrileGiardia intestinalisPotency5.610110
fluromidineGiardia intestinalisPotency15.811410
1-(2-methyl-1H-indol-3-yl)-2-(2-thiazolylamino)ethanoneGiardia intestinalisPotency39.810710
1-ethyl-3-(4-methylphenyl)sulfonylthioureaGiardia intestinalisPotency3.539710
2-(2-cyclohexylidenehydrazinyl)-1-cyclohepta-2,4,6-trienoneGiardia intestinalisPotency12.559410
4-(4-methylphenyl)-3-(2-pyrazinyl)-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency15.811410
2-mercaptonaphth(2,3)imidazoleGiardia intestinalisPotency7.062710
2-(4-ethoxyanilino)-3-methoxynaphthalene-1,4-dioneGiardia intestinalisPotency7.062710
3-[4-(2-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]-1H-pyridazin-6-oneGiardia intestinalisPotency6.294610
6-methoxy-3-[(3-methylanilino)methyl]-1H-quinolin-2-oneGiardia intestinalisPotency14.091910
3-[(2,5-dimethylanilino)methyl]-6-methoxy-1H-quinolin-2-oneGiardia intestinalisPotency15.811410
terazosinGiardia intestinalisPotency5.011910
curcuminGiardia intestinalisPotency17.740710
4-(2-methylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency11.193610
1-(4-methoxyphenyl)-3-(6-quinoxalinyl)thioureaGiardia intestinalisPotency3.971610
4-mercapto-5-(4-methoxyphenyl)-2-oxo-1,5-diazaspiro[5.5]undec-3-ene-3-carbonitrileGiardia intestinalisPotency14.091910
1-(3-chloro-4-methoxyphenyl)-3-[2-(4-methyl-1-piperidinyl)ethyl]thioureaGiardia intestinalisPotency14.091910
2,4-dimethyl-N-[4-(1-pyrrolidinyl)phenyl]benzamideGiardia intestinalisPotency35.397310
N-[(3-bromo-4-ethoxy-5-methoxyphenyl)methyl]-2,3-dihydro-1,4-benzodioxin-6-amineGiardia intestinalisPotency19.905410
3-methyl-7-[(4-methylphenyl)methyl]-8-[2-(1-piperidinyl)ethylthio]purine-2,6-dioneGiardia intestinalisPotency31.547910
umi-77Giardia intestinalisPotency7.079510
1-[[[2-(difluoromethoxy)phenyl]-oxomethyl]amino]-3-(3-methylphenyl)thioureaGiardia intestinalisPotency17.740710
5-(4-bromophenyl)-N-[[(2-propyl-5-tetrazolyl)amino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency11.193610
N-[4-[(2,6-dimethoxy-4-pyrimidinyl)sulfamoyl]phenyl]butanamideGiardia intestinalisPotency39.810710
N-[(3-acetylanilino)-sulfanylidenemethyl]-5-bromo-3-pyridinecarboxamideGiardia intestinalisPotency12.589310
4-[4-[[(3,4-dimethylphenyl)-oxomethyl]amino]phenoxy]phthalic acidGiardia intestinalisPotency12.559410
4-[[4-bromo-5-(4-morpholinyl)-2-furanyl]methylideneamino]phenolGiardia intestinalisPotency1.990510
(4-anilino-1,1-dioxo-2H-1$l^{6},2-benzothiazin-3-yl)-phenylmethanoneGiardia intestinalisPotency6.294610
1-(2-fluorophenyl)-4-[(6-nitro-1,3-benzodioxol-5-yl)methyl]piperazineGiardia intestinalisPotency25.118910
pyridine-2-carboxylic acid thiazol-2-ylamideGiardia intestinalisPotency40.418220
4-[[[2,3-bis(2-pyridinyl)-6-quinoxalinyl]amino]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterGiardia intestinalisPotency15.811410
5-amino-4-[anilino(oxo)methyl]-3-methyl-2-thiophenecarboxylic acid ethyl esterGiardia intestinalisPotency17.740710
4,5-dichloro-2-[oxo-(8-quinolinylamino)methyl]benzoic acidGiardia intestinalisPotency19.905410
3-amino-N-tert-butyl-6-methyl-7,8-dihydro-5H-thieno[2,3-b][1,6]naphthyridine-2-carboxamideGiardia intestinalisPotency31.547910
1-methyl-2-oxo-N-(2-pyridinyl)-6-benzo[cd]indolesulfonamideGiardia intestinalisPotency17.740710
4-chloro-2-[[(1-methyl-5-phenyl-2-imidazolyl)amino]methyl]phenolGiardia intestinalisPotency31.622810
LSM-16285Giardia intestinalisPotency1.774110
4-chloro-N-[3-chloro-4-(4-morpholinyl)phenyl]benzamideGiardia intestinalisPotency23.038030
2-(1,3-benzodioxol-5-yl)-N-[(2-ethoxyphenyl)methyl]-N-(2-pyridinylmethyl)ethanamineGiardia intestinalisPotency19.905410
N-(2-furanylmethyl)-4-(1-pyrrolidinylsulfonyl)benzenesulfonamideGiardia intestinalisPotency3.971610
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acidGiardia intestinalisPotency19.905410
4-(4-methylphenyl)-2-[[3-(4-morpholinyl)-1-oxopropyl]amino]-3-thiophenecarboxylic acid ethyl esterGiardia intestinalisPotency22.334210
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterGiardia intestinalisPotency9.976310
rhodanineGiardia intestinalisPotency7.943310
3-methoxy-4-(2-methoxy-3-methoxycarbonyl-1-naphthalenyl)-2-naphthalenecarboxylic acid methyl esterGiardia intestinalisPotency19.905410
1-[1-ethyl-4-[4-(4-methoxyphenyl)-1-piperazinyl]-6-methyl-2-sulfanylidene-5-pyrimidinyl]ethanoneGiardia intestinalisPotency14.091910
2-[[(2,3-dimethoxyphenyl)-oxomethyl]amino]-5-propan-2-yl-3-thiophenecarboxamideGiardia intestinalisPotency19.905410
N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-pyridinecarboxamideGiardia intestinalisPotency17.740710
3-[[[4-(4-methoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]methyl]benzoic acidGiardia intestinalisPotency17.740710
5-(2,3-dihydroindol-1-ylsulfonyl)-1,3-diethyl-2-benzimidazoloneGiardia intestinalisPotency15.811410
2-(3-bromophenyl)-6-methyl-N-(1,2,4-triazol-4-yl)-4-quinolinecarboxamideGiardia intestinalisPotency15.811410
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(2-pyridinyl)-4-quinolinecarboxamideGiardia intestinalisPotency22.334210
thiouracilGiardia intestinalisPotency15.811410
N-[[2-methyl-5-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency3.971610
5-[(5-tert-butyl-2,3-dimethylphenyl)sulfonylamino]-2-hydroxybenzoic acidGiardia intestinalisPotency15.811410
5-bromo-N-[[(3-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideGiardia intestinalisPotency9.976310
5-bromo-N-[(2-carbamoylanilino)-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency17.740710
1-[2,3-bis(2-furanyl)-6-quinoxalinyl]-3-[4-(4-morpholinyl)phenyl]thioureaGiardia intestinalisPotency0.561010
N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamideGiardia intestinalisPotency14.091910
1-[1-ethyl-6-methyl-4-(4-phenyl-1-piperazinyl)-2-sulfanylidene-5-pyrimidinyl]ethanoneGiardia intestinalisPotency17.740710
4-(dimethylsulfamoyl)-N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideGiardia intestinalisPotency19.905410
N-[[3-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency15.811410
3-[[3-(4-morpholinyl)-1,4-dioxo-2-naphthalenyl]amino]benzoic acidGiardia intestinalisPotency7.062710
6-amino-5-(4-chlorophenyl)sulfonyl-2-oxo-1H-pyridine-3-carbonitrileGiardia intestinalisPotency22.334210
4-chloro-N-(4-chloro-2-methylphenyl)-5-dithiazolimineGiardia intestinalisPotency15.811410
2-[2-[2-(3-fluorophenyl)-4-thiazolyl]ethyl]isoindole-1,3-dioneGiardia intestinalisPotency17.740710
4-[(3-methylphenyl)thio]-2-phenyl-5-pyrimidinecarboxylic acidGiardia intestinalisPotency17.740710
6-(4-methyl-1-piperazinyl)-2-(3,4,5-trimethoxyphenyl)-1H-benzimidazoleGiardia intestinalisPotency19.905410
7,8-dimethoxy-1,3-dihydro-3-benzazepin-2-oneGiardia intestinalisPotency44.562510
N-[1-[(3,4-dichlorophenyl)methyl]-6-oxo-3-pyridinyl]benzenesulfonamideGiardia intestinalisPotency7.062710
2-(5-methyl-3-oxo-1H-pyrazol-2-yl)-6-oxo-1H-pyrimidine-5-carboxylic acid ethyl esterGiardia intestinalisPotency12.559410
2-(benzenesulfonylmethyl)-5-(4-chlorophenyl)cyclohexane-1,3-dioneGiardia intestinalisPotency15.811410
2-(6-chloro-3-pyridinyl)-1H-benzimidazoleGiardia intestinalisPotency22.334210
(2-methylanilino)thioureaGiardia intestinalisPotency15.811410
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneGiardia intestinalisPotency11.193610
1-[[2-[[4-(4-chlorophenyl)-5-phenyl-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-3-phenylthioureaGiardia intestinalisPotency22.334210
epalrestatGiardia intestinalisPotency19.905410
1,4-benzoquinone guanylhydrazone thiosemicarbazoneGiardia intestinalisPotency20.811420
1-[[2-(1,3-benzothiazol-2-ylthio)-1-oxoethyl]amino]-3-phenylthioureaGiardia intestinalisPotency15.811410
ac 55649Giardia intestinalisPotency16.776110
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneGiardia intestinalisPotency1.000010
3-(5,8-dinitro-1,3-dioxo-2-benzo[de]isoquinolinyl)benzoic acidGiardia intestinalisPotency17.782810
N-[4-[(4,6-dimethyl-2-pyrimidinyl)sulfamoyl]phenyl]-2-nitrobenzamideGiardia intestinalisPotency15.848910
N-[3-(dimethylamino)propyl]-9H-carbazole-3-carboxamideGiardia intestinalisPotency7.062710
N-[[[2-(2-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency17.740710
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency5.610110
2-methyl-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency15.811410
4-chloro-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency8.891410
5-(methylamino)-3H-1,3,4-thiadiazole-2-thioneGiardia intestinalisPotency17.740710
5,5-diethyl-1-[oxo(1-piperidinyl)methyl]-6H-pyrrolo[2,1-a]isoquinoline-2,3-dioneGiardia intestinalisPotency3.539710
N-[[(5-chloro-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency5.610110
2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylamino]phenolGiardia intestinalisPotency15.811410
3-chloro-6-(3,5-dimethyl-1h-pyrazol-1-yl)picolinic acidGiardia intestinalisPotency15.811410
N-[2-[tert-butyl(methyl)amino]ethyl]-N-methyl-2,2-diphenylacetamideGiardia intestinalisPotency17.740710
4-[[3-[(2-methoxyanilino)-oxomethyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidGiardia intestinalisPotency44.562510
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamideGiardia intestinalisPotency2.233410
1-(6-methyl-2-pyridinyl)-3-(2-phenylethyl)thioureaGiardia intestinalisPotency15.811410
2-[5-(4-chlorophenyl)-1,3,5-dithiazinan-2-ylidene]-2-diethoxyphosphorylacetonitrileGiardia intestinalisPotency39.810710
6-(bromomethyl)-1,3-dimethyl-5-[(4-nitrophenyl)-oxomethyl]pyrimidine-2,4-dioneGiardia intestinalisPotency22.334210
3-methoxy-N-[[(2-oxo-1-benzopyran-6-yl)amino]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency9.976310
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)thio]acetamideGiardia intestinalisPotency7.924510
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(4-methyl-1-piperidinyl)sulfonyl]benzamideGiardia intestinalisPotency35.481310
4-(4-morpholinylsulfonyl)-N-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)benzamideGiardia intestinalisPotency14.091910
benzotriptGiardia intestinalisPotency22.334210
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)thio]ethanoneGiardia intestinalisPotency15.811410
N-[(tert-butylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideGiardia intestinalisPotency15.811410
4-(6-fluoro-3-methyl-4-oxo-1-benzopyran-2-yl)-2-methyl-1-phthalazinoneGiardia intestinalisPotency5.000010
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneGiardia intestinalisPotency1.255910
1-[4-(1H-benzimidazol-2-yl)phenyl]-3-[3-(4-morpholinyl)propyl]thioureaGiardia intestinalisPotency22.334210
3-[(4-acetyl-1-piperazinyl)sulfonyl]-N-(1H-benzimidazol-2-yl)benzamideGiardia intestinalisPotency17.740710
3-[(3-hydroxy-5-benzotriazolyl)sulfonylamino]benzoic acidGiardia intestinalisPotency17.740710
2-methyl-3-[oxo(thiophen-2-yl)methyl]-1-indolizinecarboxaldehydeGiardia intestinalisPotency15.811410
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideGiardia intestinalisPotency0.397210
6-propan-2-yl-2-sulfanylidene-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-oneGiardia intestinalisPotency44.562510
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[methyl(phenyl)sulfamoyl]benzamideGiardia intestinalisPotency7.924510
4-[butyl(methyl)sulfamoyl]-N-[5-[(methylthio)methyl]-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency35.397310
4-[ethyl-(phenylmethyl)sulfamoyl]-N-(5-methyl-1,3,4-oxadiazol-2-yl)benzamideGiardia intestinalisPotency17.782810
4-[ethyl-(phenylmethyl)sulfamoyl]-N-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency17.740710
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency14.091910
1-[2,3-bis(2-pyridinyl)-6-quinoxalinyl]-3-propylthioureaGiardia intestinalisPotency1.774110
3-[4-[(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]-3-(2-oxo-1-benzopyran-3-yl)-1-pyrazolyl]propanoic acidGiardia intestinalisPotency17.740710
5-bromo-N-[[(4-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideGiardia intestinalisPotency3.539710
1-(2,3-dimethyl-6-quinoxalinyl)-3-(3-hydroxypropyl)thioureaGiardia intestinalisPotency3.971610
2-[(3-cyano-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)thio]-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]acetamideGiardia intestinalisPotency17.740710
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterGiardia intestinalisPotency14.091910
4-[[[(2-methoxy-1-oxoethyl)hydrazo]-sulfanylidenemethyl]amino]benzoic acid ethyl esterGiardia intestinalisPotency25.059410
4-[2-(3,4-dimethoxyphenyl)ethyl]-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency19.905410
1-[[(4-bromo-2-methyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxy-5-methylphenyl)thioureaGiardia intestinalisPotency15.811410
N-[[[2-(2-bromo-4-propan-2-ylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency28.183810
N-[4-[(3-bromo-5-methoxy-4-prop-2-enoxyphenyl)methylamino]-2-methoxyphenyl]-2-methylpropanamideGiardia intestinalisPotency7.924510
3-chloro-N-[3-(4-morpholinyl)propyl]-6-nitro-1-benzothiophene-2-carboxamideGiardia intestinalisPotency2.505910
N-[[(5-hydroxy-1-naphthalenyl)amino]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency22.387210
5-(2-ethoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneGiardia intestinalisPotency17.740710
N-[(3,5-dimethoxyphenyl)methyl]-1-(2,3,4-trimethoxyphenyl)methanamineGiardia intestinalisPotency19.905410
N-(2,1,3-benzothiadiazol-4-yl)-5-(3-chlorophenyl)-2-furancarboxamideGiardia intestinalisPotency17.740710
4E2RCatGiardia intestinalisPotency19.905410
2-chloro-N-[(2-pyrimidinylamino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency24.104020
2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-oneGiardia intestinalisPotency9.976310
1-(5-isoquinolinyl)-3-(2-phenylethyl)thioureaGiardia intestinalisPotency14.091910
2-[5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl(oxo)methyl]-1,1-dioxo-1,2-benzothiazol-3-oneGiardia intestinalisPotency17.740710
1-[3-(2-bromo-4-chlorophenoxy)propyl]-4-methylpiperidineGiardia intestinalisPotency14.091910
5-[2-(4-ethoxy-2-hydroxyphenyl)-2-oxoethyl]-2-benzofurancarboxylic acidGiardia intestinalisPotency19.905410
2,8-dimercapto-6-hydroxypurineGiardia intestinalisPotency12.559410
N4-(2-methoxyphenyl)benzene-1,4-diamineGiardia intestinalisPotency17.740710
2-(5H-[1,2,4]triazolo[5,1-a]isoindol-2-yl)ethanethioamideGiardia intestinalisPotency14.091910
4-methyl-N-[sulfanylidene-(1,2,4-triazol-4-ylamino)methyl]benzamideGiardia intestinalisPotency15.811410
N-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)-2-furancarboxamideGiardia intestinalisPotency23.445120
1-(4-ethoxyphenyl)-3-(5-isoquinolinyl)thioureaGiardia intestinalisPotency1.774110
2-[(1-oxido-2-pyridin-1-iumyl)thio]-1-(4-phenylphenyl)ethanoneGiardia intestinalisPotency17.740710
4-methoxy-3-[2-phenylethyl-(phenylmethyl)sulfamoyl]benzoic acidGiardia intestinalisPotency17.740710
1-(2-furanyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneGiardia intestinalisPotency22.334210
2,5-dimethyl-1-(3-methylphenyl)-N-(4-methylphenyl)-3-pyrrolecarboxamideGiardia intestinalisPotency15.811410
2-[(2-hydroxy-1-naphthalenyl)methyl-methylamino]-N-[4-(4-morpholinyl)phenyl]acetamideGiardia intestinalisPotency15.811410
1-[4-(4-hydroxyphenyl)-1-piperazinyl]-3-(1H-indol-3-yl)-1-propanoneGiardia intestinalisPotency35.397310
N-[5-[(2,6-dichlorophenyl)methylthio]-1,3,4-thiadiazol-2-yl]-5-methyl-2-pyrazinecarboxamideGiardia intestinalisPotency17.740710
N-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideGiardia intestinalisPotency19.905410
N-[2-(2,3-dimethylanilino)-2-oxoethyl]-3-(3-methylphenoxy)propanamideGiardia intestinalisPotency15.811410
N-[[2-cyanoethyl(methyl)amino]-sulfanylidenemethyl]-4-(4-morpholinylsulfonyl)benzamideGiardia intestinalisPotency15.811410
N-(1H-benzimidazol-2-yl)-2-methylsulfonylbenzamideGiardia intestinalisPotency15.811410
[1-(4-fluorophenyl)sulfonyl-4-piperidinyl]-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methanoneGiardia intestinalisPotency15.811410
N-(3-pyridinylmethyl)-1,3-benzodioxol-5-amineGiardia intestinalisPotency9.976310
4-[[6-[(2-methyl-5-thieno[2,3-e][1,3]benzothiazolyl)oxy]-3-pyridinyl]sulfonyl]morpholineGiardia intestinalisPotency19.905410
5-(3-fluorophenoxy)-8-nitroisoquinolineGiardia intestinalisPotency15.811410
1-(2-chlorophenyl)-3-(2-oxo-1,3-dihydrobenzimidazol-5-yl)thioureaGiardia intestinalisPotency35.397310
4-(diethylsulfamoyl)benzoic acid 1,3-benzodioxol-5-yl esterGiardia intestinalisPotency5.000010
thioguanine anhydrousGiardia intestinalisPotency3.154810
4-amino-5-hydrazino-1,2,4-triazole-3-thiolGiardia intestinalisPotency9.058720
2-oxo-6-phenyl-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileGiardia intestinalisPotency17.740710
N-(7-methoxy-4,5-dihydrobenzo[e][1,3]benzothiazol-2-yl)-2-furancarboxamideGiardia intestinalisPotency15.811410
1,4-dihydroxy-4a,5,6,7,8,8a-hexahydroquinoxaline-2,3-dioneGiardia intestinalisPotency14.091910
1-[[2-[5-[3,5-bis(trifluoromethyl)phenyl]-2-tetrazolyl]-1-oxoethyl]amino]-3-(4-chlorophenyl)thioureaGiardia intestinalisPotency12.559410
1-anilino-3-ethylthioureaGiardia intestinalisPotency11.193610
mecysteine hydrochlorideGiardia intestinalisPotency15.811410
capsazepineGiardia intestinalisPotency25.059410
3-(tert-butyl)-1-methyl-4,5-dihydro-1H-pyrazol-5-oneGiardia intestinalisPotency0.561010
2-[1-[2-oxo-2-[(4-thiophen-2-ylphenyl)methylamino]ethyl]cyclohexyl]acetic acidGiardia intestinalisPotency15.811410
N'-[(4-chlorophenyl)-oxomethyl]-2-methyl-4-thiazolecarbohydrazideGiardia intestinalisPotency31.204620
5-cyano-2-(methoxymethyl)-6-sulfanylidene-1H-pyridine-3-carboxylic acid methyl esterGiardia intestinalisPotency15.811410
N-(2-chlorophenyl)-2-[[5-[5-(trifluoromethyl)-2-pyridinyl]-1,3,4-oxadiazol-2-yl]thio]acetamideGiardia intestinalisPotency17.740710
4-(2-furanyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterGiardia intestinalisPotency25.059410
3-(2,2-dimethoxyethyl)-4-phenyl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency15.811410
2-chloro-N-[(methylcarbamoylamino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency12.559410
2-(benzenesulfonylmethyl)-5-(4-methoxyphenyl)cyclohexane-1,3-dioneGiardia intestinalisPotency19.905410
1H-benzimidazole-5,6-diamineGiardia intestinalisPotency0.445610
5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-amineGiardia intestinalisPotency15.811410
3-[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]propanoic acid ethyl esterGiardia intestinalisPotency15.811410
2-[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]butanedioic acidGiardia intestinalisPotency18.532820
1-(4-hydroxyphenyl)-3-(3-methoxyphenyl)thioureaGiardia intestinalisPotency17.740710
2-[3-(4-pyridyl)-1H-1,2,4-triazol-5-yl]pyridineGiardia intestinalisPotency3.539710
N-[amino(1-pyrrolidinyl)methylidene]-3-(2,6-dichlorophenyl)-5-methyl-4-isoxazolecarboxamideGiardia intestinalisPotency22.334210
2-({[2-acetyl-5-(tert-butyl)-3-thienyl]amino}carbonyl)benzoic acidGiardia intestinalisPotency17.740710
2,3-dichloro-N'-[4-(trifluoromethyl)-2-pyrimidinyl]benzenesulfonohydrazideGiardia intestinalisPotency19.099320
3-[[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)thio]methyl]-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency2.233410
3-oxo-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)thio]butanoic acid ethyl esterGiardia intestinalisPotency44.562510
5-[[(4-methoxyanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid ethyl esterGiardia intestinalisPotency15.811410
5-(methoxymethyl)-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-oneGiardia intestinalisPotency15.811410
3-chloro-4-propan-2-ylsulfonyl-2-thiophenecarbohydrazideGiardia intestinalisPotency14.091910
8-methylsulfinyl-4,5-dihydrothieno[3,4-g][2,1]benzoxazole-6-carboxylic acid ethyl esterGiardia intestinalisPotency22.334210
N'-benzoyl-2-(3-pyridinyl)-4-thiazolecarbohydrazideGiardia intestinalisPotency31.547910
1-tert-butyl-3-[(4-methylphenyl)sulfonylamino]thioureaGiardia intestinalisPotency68.542820
(4-chloro-2-methylanilino)thioureaGiardia intestinalisPotency15.811410
2-(2-furanyl)-4-thiazolidinecarboxylic acidGiardia intestinalisPotency15.811410
2-amino-4-(4,5-dimethoxy-2-nitrophenyl)-7,7-dimethyl-5-oxo-6,8-dihydro-4H-1-benzopyran-3-carbonitrileGiardia intestinalisPotency7.062710
4-[[4-(3-methylanilino)-3,5-dinitrophenyl]-oxomethyl]-1,3-dihydroquinoxalin-2-oneGiardia intestinalisPotency14.091910
(4-chlorophenyl)-[6,7-dichloro-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-3-benzofuranyl]methanoneGiardia intestinalisPotency25.118910
2-amino-7-methyl-5-oxo-4-(2,4,5-trimethoxyphenyl)-4,6,7,8-tetrahydro-1-benzopyran-3-carbonitrileGiardia intestinalisPotency15.811410
1-(4-tert-butylphenoxy)-3-(1H-1,2,4-triazol-5-ylthio)-2-propanolGiardia intestinalisPotency12.559410
5-cyclopentylidene-2-sulfanylidene-4-thiazolidinoneGiardia intestinalisPotency19.905410
N-(2-methoxycyclohexyl)-2,5-dimethylanilineGiardia intestinalisPotency19.905410
N-(2-methoxycyclohexyl)-3,4-dimethylanilineGiardia intestinalisPotency19.905410
3-ethyl-N-(2H-tetrazol-5-yl)-1-adamantanecarboxamideGiardia intestinalisPotency8.891410
3-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propylthio]propanoic acidGiardia intestinalisPotency19.905410
4-ethyl-2-methoxy-3-phenyl-3,3a,9,9a-tetrahydropyrrolo[2,3-b]quinoxalineGiardia intestinalisPotency17.740710
N-(4-methylphenyl)-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]amineGiardia intestinalisPotency14.091910
N-cyclohexyl-1-hydroxy-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]imineGiardia intestinalisPotency7.062710
3,4-dimethyl-6-(6-nitro-1,3-benzodioxol-5-yl)-2-oxo-1,6-dihydropyrimidine-5-carboxylic acid propyl esterGiardia intestinalisPotency5.610110
6-amino-5-cyano-4-(2,4-dimethoxyphenyl)-2-(2-ethoxy-2-oxoethyl)-4H-pyran-3-carboxylic acid ethyl esterGiardia intestinalisPotency15.811410
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamideGiardia intestinalisPotency3.154810
1-(3-nitrophenyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneGiardia intestinalisPotency25.059410
2-methoxy-N-(2-pyridinylmethyl)-3-dibenzofuranamineGiardia intestinalisPotency19.905410
[(2S)-1,3-dimethyl-3'-nitro-1'-spiro[cyclohepta[d]imidazol-3-ium-2,4'-cyclohexa-2,5-diene]ylidene]-dioxidoammoniumGiardia intestinalisPotency7.062710
1-(4-methylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneGiardia intestinalisPotency17.740710
1-(3,5-dimethylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneGiardia intestinalisPotency19.905410
4-[(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)amino]-4-oxobutanoic acidGiardia intestinalisPotency15.811410
4-(3-methoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thioneGiardia intestinalisPotency15.811410
4-[5-(3-chloro-2-methylphenyl)-2-furanyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterGiardia intestinalisPotency31.547910
N-(1-butyl-2-benzimidazolyl)cyclohexanecarboxamideGiardia intestinalisPotency19.905410
2-(2-hydroxyethylamino)-3-(4-methoxyanilino)naphthalene-1,4-dioneGiardia intestinalisPotency4.456310
5-(4-ethylsulfonyl-1-piperazinyl)-2-nitro-N-(3-pyridinylmethyl)anilineGiardia intestinalisPotency17.740710
5-[(3,4-dimethoxyphenyl)methyl]-1-prop-2-enyl-1,3-diazinane-2,4,6-trioneGiardia intestinalisPotency15.811410
5-[(3-ethoxycarbonyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-5-oxopentanoic acidGiardia intestinalisPotency15.811410
6-hydroxy-5-[(6-hydroxy-1-methyl-4-oxo-2-sulfanylidene-5-pyrimidinyl)-(2-pyridinyl)methyl]-1-methyl-2-sulfanylidene-4-pyrimidinoneGiardia intestinalisPotency17.740710
4-[[1-[(3,4-dichlorophenyl)methyl]-3-indolyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneGiardia intestinalisPotency12.559410
N-[3-(4-chlorophenyl)-5-oxo-4-pyrazolidinyl]-3-methylbenzamideGiardia intestinalisPotency35.397310
2-methyl-3-[(2-methyl-1H-indol-3-yl)-(2-pyridinyl)methyl]-1H-indoleGiardia intestinalisPotency3.971610
N-(4-chloro-2,5-dimethoxyphenyl)-3-methyl-1-piperidinecarbothioamideGiardia intestinalisPotency19.905410
2-(2-oxo-1-benzo[cd]indolyl)-N-(2-oxolanylmethyl)acetamideGiardia intestinalisPotency15.811410
1-[4-(4-morpholinyl)-2,1,3-benzoxadiazol-7-yl]-3-(4-nitrophenyl)ureaGiardia intestinalisPotency15.811410
N-[(4-sulfamoylanilino)-sulfanylidenemethyl]-1,3-benzodioxole-5-carboxamideGiardia intestinalisPotency15.811410
3-[(2-chloro-6-fluorophenyl)methyl]-5-fluoro-1-(2-oxolanyl)pyrimidine-2,4-dioneGiardia intestinalisPotency44.668410
N-cycloheptyl-2-(cyclohexylamino)-2-sulfanylideneacetamideGiardia intestinalisPotency40.418220
cb 7969312Giardia intestinalisPotency31.547910
7-ethyl-7-methyl-2-sulfanylidene-6,9-dihydro-1H-pyrano[2,3]thieno[2,4-b]pyrimidin-4-oneGiardia intestinalisPotency7.924510
2-[1-[[[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid methyl esterGiardia intestinalisPotency15.811410
1-(3-chlorophenyl)-3-[[1-[(2,5-dimethoxyphenyl)methyl]-4-piperidinyl]methyl]ureaGiardia intestinalisPotency44.562510
2-[3-oxo-1-[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]-2-piperazinyl]acetic acid propan-2-yl esterGiardia intestinalisPotency5.610110
3-methyl-N-[[(2-methyl-5-quinolinyl)amino]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency14.125410
1-(1,3-benzodioxol-5-yl)-3-[4-(4-hydroxyphenyl)-1-piperazinyl]pyrrolidine-2,5-dioneGiardia intestinalisPotency15.811410
4-[(1-ethyl-6-methyl-4-pyrazolo[3,4-b]pyridinyl)oxymethyl]benzonitrileGiardia intestinalisPotency15.811410
2-[(2-furanylmethylthio)methyl]-5-methylimidazo[1,2-a]pyridineGiardia intestinalisPotency19.952610
nsc 727447Giardia intestinalisPotency17.740710
7-[[[1-(3-methylphenyl)-2-benzimidazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneGiardia intestinalisPotency25.059410
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[[4-methyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanoneGiardia intestinalisPotency15.811410
3-(4-chlorophenyl)sulfonyl-N-[2,5-diethoxy-4-(4-morpholinyl)phenyl]propanamideGiardia intestinalisPotency14.091910
4,5-dimethyl-3-(2-oxolanylmethyl)-1H-imidazole-2-thioneGiardia intestinalisPotency12.559410
2-benzoyl-N-(6-methoxy-3-pyridinyl)-3,4-dihydro-1H-isoquinoline-3-carboxamideGiardia intestinalisPotency19.905410
6-mercapto-9-(tetrahydro-2-furyl)purineGiardia intestinalisPotency2.505910
2-amino-9-pentyl-3H-purine-6-thioneGiardia intestinalisPotency2.811710
1,4-dimethoxy-10H-acridine-9-thioneGiardia intestinalisPotency25.059410
thiophanateGiardia intestinalisPotency15.811410
burimamideGiardia intestinalisPotency11.193610
racloprideGiardia intestinalisPotency44.562510
9-cyclopentyl-3H-purine-6-thioneGiardia intestinalisPotency3.971610
9-(n-butyl)-6-thioguanineGiardia intestinalisPotency7.062710
1,3-dimethyl-8-[2-(1-pyrrolidinyl)ethylthio]-6-sulfanylidene-7H-purin-2-oneGiardia intestinalisPotency11.220210
acth (11-24)Giardia intestinalisPotency6.294610
homoquinolinic acidGiardia intestinalisPotency12.589310
asterric acidGiardia intestinalisPotency15.811410
2,2-dimethyl-N-[2,2,2-trichloro-1-(2-pyrimidinylthio)ethyl]propanamideGiardia intestinalisPotency6.294610
2,2,3,3-tetrafluoro-N-(1H-1,2,4-triazol-5-yl)propanamideGiardia intestinalisPotency15.811410
2-[8-(6-amino-1H-benzimidazol-2-yl)octyl]-3H-benzimidazol-5-amineGiardia intestinalisPotency19.905410
2-(2,3,3-trichloro-1-nitroprop-2-enylidene)-1,3-dihydrobenzimidazoleGiardia intestinalisPotency17.740710
N-tert-butyl-2-[[(3-nitrophenyl)-oxomethyl]hydrazo]-2-oxoacetamideGiardia intestinalisPotency15.811410
5-acetyl-2-amino-6-methyl-4-(3-nitrophenyl)-4h-pyran-3-carbonitrileGiardia intestinalisPotency17.740710
N'-[(2-nitrophenyl)-oxomethyl]-2-pyridinecarbohydrazideGiardia intestinalisPotency15.811410
N-[[[2-(2-methylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-nitrobenzamideGiardia intestinalisPotency17.740710
2-[2-[(4-acetamidophenyl)sulfonylamino]-4-thiazolyl]acetic acid ethyl esterGiardia intestinalisPotency14.125410
1-(3,4-dihydroxyphenyl)-2-[(4-methyl-1,2,4-triazol-3-yl)thio]ethanoneGiardia intestinalisPotency15.811410
3-[5-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl esterGiardia intestinalisPotency14.091910
4-mercapto-6-oxo-3-phenyl-2-thiophen-2-yl-1,2-dihydropyrimidine-5-carbonitrileGiardia intestinalisPotency6.309610
2-methyl-N-[1-(4-prop-2-enyl-5-sulfanylidene-1H-1,2,4-triazol-3-yl)ethyl]benzamideGiardia intestinalisPotency5.000010
2-(4-ethoxy-3-methoxyphenyl)-4-mercapto-3-(4-methoxyphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileGiardia intestinalisPotency9.976310
2-chloro-5-[[1-oxo-2-[(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)thio]ethyl]amino]benzoic acidGiardia intestinalisPotency28.183810
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneGiardia intestinalisPotency5.000010
1-[2-(diethylamino)ethyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-(2-oxolanylmethyl)thioureaGiardia intestinalisPotency7.924510
3-(2,4-dimethoxyphenyl)-1-[(1-ethyl-2-pyrrolidinyl)methyl]-1-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]thioureaGiardia intestinalisPotency15.811410
4-[4-[[1-(2-methylbutan-2-yl)-5-tetrazolyl]-(6-quinolinyl)methyl]-1-piperazinyl]phenolGiardia intestinalisPotency15.811410
N'-(1,3-benzodioxol-5-ylmethyl)-N'-[2-(cyclopentylamino)-2-oxoethyl]-N-(5-methyl-3-isoxazolyl)butanediamideGiardia intestinalisPotency17.740710
N-[2-[butyl-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-thiophenecarboxamideGiardia intestinalisPotency22.334210
N-(1,3-benzodioxol-5-ylmethyl)-N-[2-(cyclohexylamino)-2-oxo-1-pyridin-4-ylethyl]-2,2,2-trifluoroacetamideGiardia intestinalisPotency28.117110
4-[4-[(1-tert-butyl-5-tetrazolyl)-pyridin-4-ylmethyl]-1-piperazinyl]phenolGiardia intestinalisPotency14.091910
4-[butan-2-yl-[(3,4-dichloroanilino)-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterGiardia intestinalisPotency15.811410
N-[3-(1-azepanyl)propyl]-1-[(4-methoxyphenyl)methyl]-5-oxo-3-pyrrolidinecarboxamideGiardia intestinalisPotency31.547910
1-(4-methyl-2-prop-2-enylphenoxy)-3-(4-phenyl-1-piperazinyl)-2-propanolGiardia intestinalisPotency19.905410
N-[[1-(4-methoxyphenyl)-3-pyrrolidinyl]methyl]-3-(trifluoromethyl)benzenesulfonamideGiardia intestinalisPotency6.294610
1-(4-chlorophenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-4-pyrazolecarboxylic acidGiardia intestinalisPotency15.811410
3-[4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-4-oxobutyl]-6,7-diethoxy-2-sulfanylidene-1H-quinazolin-4-oneGiardia intestinalisPotency15.811410
1-[[1-(2-methoxyanilino)-4-isoquinolinyl]-oxomethyl]-4-piperidinecarboxamideGiardia intestinalisPotency17.740710
LSM-18934Giardia intestinalisPotency4.456310
N-[4-[[4-(2-fluorophenyl)-1-piperazinyl]-oxomethyl]-1-oxo-2-isoquinolinyl]-2-pyrazinecarboxamideGiardia intestinalisPotency35.397310
6,7-diethoxy-3-[3-(2-oxo-1-pyrrolidinyl)propyl]-2-sulfanylidene-1H-quinazolin-4-oneGiardia intestinalisPotency17.740710
N-[3-(1-azepanyl)propyl]-5-oxo-1-(2-phenylethyl)-3-pyrrolidinecarboxamideGiardia intestinalisPotency19.905410
N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-2-(3-oxo-1,4-benzoxazin-4-yl)acetamideGiardia intestinalisPotency19.905410
5-[2-(1-cyclohexenyl)ethylsulfamoyl]-3-methyl-2-benzofurancarboxylic acidGiardia intestinalisPotency17.740710
2-[[3-oxo-2-[3-oxo-3-(4-phenyl-1-piperazinyl)propyl]-2H-imidazo[1,2-c]quinazolin-5-yl]thio]acetonitrileGiardia intestinalisPotency17.740710
N-[3-(1-azepanyl)propyl]-2-(4-morpholinyl)-3-oxo-4H-1,4-benzothiazine-6-carboxamideGiardia intestinalisPotency22.334210
2-amino-4-[5-methyl-2-(methylthio)-3-thiophenyl]-5-oxo-1-(3-pyridinyl)-4,6,7,8-tetrahydroquinoline-3-carbonitrileGiardia intestinalisPotency17.740710
3-(2-furanylmethyl)-5-(2-methoxyethyl)-1,3,5-thiadiazinane-2-thioneGiardia intestinalisPotency22.334210
N-butyl-2-[[6-(4-morpholinyl)-4-oxo-3-(2-phenylethyl)-2-quinazolinyl]thio]acetamideGiardia intestinalisPotency1.774110
1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-ethylphenyl)ureaGiardia intestinalisPotency19.905410
7-(5-chloro-2-methoxyanilino)-6-[(4-methoxyphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-oneGiardia intestinalisPotency28.183810
4-[dimethylamino(oxo)methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl esterGiardia intestinalisPotency31.547910
2-(2-methoxyethyl)-9-methyl-1-oxo-N-(thiophen-2-ylmethyl)-4-pyrido[3,4-b]indolecarboxamideGiardia intestinalisPotency15.811410
2-amino-4-[4-(methylthio)phenyl]-5-oxo-1-phenyl-4,6,7,8-tetrahydroquinoline-3-carbonitrileGiardia intestinalisPotency12.559410
2,5-dimethyl-4-(4-methyl-1-piperidinyl)-6-thieno[2,3-d]pyrimidinecarboxylic acidGiardia intestinalisPotency19.905410
N-[3-(1-azepanyl)propyl]-1-ethylsulfonyl-4-piperidinecarboxamideGiardia intestinalisPotency28.183810
N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideGiardia intestinalisPotency31.622810
4-oxo-4-[5-(1,2,3,4-tetrahydronaphthalen-1-ylsulfamoyl)-2,3-dihydroindol-1-yl]butanoic acidGiardia intestinalisPotency31.547910
mannonateGiardia intestinalisPotency14.091910
sb 258585Giardia intestinalisPotency19.905410
2,3-dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxalineGiardia intestinalisPotency21.119810
4-bromo-N-(2-phenazinyl)benzamideGiardia intestinalisPotency8.891410
4-methyl-N-[2,4,6-trioxo-1-phenyl-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzenesulfonamideGiardia intestinalisPotency15.811410
8-[(1-ethyl-3-piperidinyl)thio]-1,3-dimethyl-6-sulfanylidene-7H-purin-2-oneGiardia intestinalisPotency7.924510
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl esterGiardia intestinalisPotency7.062710
2-amino-7-methyl-4-(5-nitro-2-furanyl)-5-oxo-4H-pyrano[3,2-c]pyran-3-carbonitrileGiardia intestinalisPotency4.456310
1-(4-fluorophenyl)-N-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbothioamideGiardia intestinalisPotency15.811410
1-[2-(dimethylamino)ethyl]-3-(2,4-dimethylphenyl)-1-(thiophen-2-ylmethyl)thioureaGiardia intestinalisPotency14.091910
3,3,3-trifluoro-2-[[(4-hydroxyanilino)-oxomethyl]amino]-2-phenylpropanoic acid ethyl esterGiardia intestinalisPotency12.559410
5-[3,4-dihydro-1H-isoquinolin-2-yl(phenyl)methyl]-6-thiazolo[3,2-b][1,2,4]triazololGiardia intestinalisPotency35.397310
2-fluoro-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)benzamideGiardia intestinalisPotency19.905410
N-[3-[4-(4-fluorophenyl)-1-piperazinyl]-1,4-dioxo-2-naphthalenyl]benzenesulfonamideGiardia intestinalisPotency8.891410
7-[[2-(4-chloro-3-methyl-1-pyrazolyl)-1-oxopropyl]amino]-3-[[(1-methyl-5-tetrazolyl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidGiardia intestinalisPotency15.811410
4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)-N-(5-ethyl-1,3,4-oxadiazol-2-yl)benzamideGiardia intestinalisPotency19.905410
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolGiardia intestinalisPotency15.811410
6-amino-5-cyano-4-(2-fluorophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyridine-3-carboxamideGiardia intestinalisPotency19.905410
2-amino-4-(2-ethoxyphenyl)-6,7-dimethyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carbonitrileGiardia intestinalisPotency12.589310
N-(4-ethoxyphenyl)sulfonyl-N-(2-oxo-5-benzo[g][1,3]benzoxathiolyl)-2-furancarboxamideGiardia intestinalisPotency17.740710
4-chloro-N-[1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-methylpropan-2-yl]benzenesulfonamideGiardia intestinalisPotency31.547910
N-[[[(2-chlorophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-nitrobenzamideGiardia intestinalisPotency19.905410
N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-(3-oxo-1,4-benzoxazin-4-yl)propanamideGiardia intestinalisPotency28.117110
nsc 105827Giardia intestinalisPotency14.091910
7-(2-chloro-6-fluorophenyl)-5-methyl-6,7-dihydro-1H-1,4-diazepine-2,3-dicarbonitrileGiardia intestinalisPotency14.091910
N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]-5-nitro-2-thiophenecarboxamideGiardia intestinalisPotency35.481310
3-(1,3-benzothiazol-2-ylhydrazo)-1-(4-ethylphenyl)pyrrolidine-2,5-dioneGiardia intestinalisPotency14.091910
N-butyl-1-hydroxy-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]imineGiardia intestinalisPotency4.456310
2-[(5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]acetic acidGiardia intestinalisPotency15.811410
N'-[(3-nitrophenyl)-oxomethyl]-2-pyridinecarbohydrazideGiardia intestinalisPotency12.912620
4-[1-oxo-6-(4-oxo-2-sulfanylidene-1H-thieno[3,2-d]pyrimidin-3-yl)hexyl]-1-piperazinecarboxylic acid ethyl esterGiardia intestinalisPotency22.334210
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]-1,4-dioxo-2-naphthalenyl]-2-thiophenesulfonamideGiardia intestinalisPotency5.000010
3-(3-bromoanilino)-2-oxo-1H-indole-3-carbonitrileGiardia intestinalisPotency15.811410
2-[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]propanoic acid methyl esterGiardia intestinalisPotency15.811410
N-tert-butyl-1-hydroxy-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]imineGiardia intestinalisPotency3.154810
4-(4-methylphenyl)sulfonyl-3-phenyl-2,3-dihydro-1,4-benzoxazineGiardia intestinalisPotency17.740710
N-[3-(4-methyl-1-piperazinyl)-1,4-dioxo-2-naphthalenyl]benzenesulfonamideGiardia intestinalisPotency3.162310
N-(2,2,4-trimethyl-3H-benzofuran-7-yl)benzenesulfonamideGiardia intestinalisPotency19.905410
2-amino-5-(1-benzotriazolyl)-6-methyl-4-phenyl-4H-pyran-3-carbonitrileGiardia intestinalisPotency7.924510
3-methyl-N-[[[(4-nitrophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]butanamideGiardia intestinalisPotency17.740710
4-fluoro-N-[[2-(3-pyridinyl)-1-piperidinyl]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency7.943310
4-chloro-N-[3-(3-methyl-1-piperidinyl)-1,4-dioxo-2-naphthalenyl]benzenesulfonamideGiardia intestinalisPotency5.610110
6-(5,6-Dihydroxy-4-oxo-2-phenylchromen-7-yl)oxy-3,4,5-trihydroxyoxane-2-carboxylic acidGiardia intestinalisPotency15.811410
N-[(5-quinolinylamino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency17.740710
(2,5-dimethylanilino)thioureaGiardia intestinalisPotency15.811410
N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideGiardia intestinalisPotency4.456310
4-[[(2-methyl-5-nitro-1H-imidazol-4-yl)thio]methyl]-2-nitrophenolGiardia intestinalisPotency17.740710
5-amino-2-(diethylamino)-N-(2-methoxyphenyl)benzenesulfonamideGiardia intestinalisPotency15.811410
7-[(3-hydroxy-3,4-dihydro-2H-benzo[h]quinolin-1-yl)methyl]-5-thiazolo[3,2-a]pyrimidinoneGiardia intestinalisPotency17.740710
2-[(4-hydroxy-3-nitrophenyl)sulfonylamino]benzoic acid [2-(4-methoxyphenyl)-2-oxoethyl] esterGiardia intestinalisPotency15.811410
2-(1H-benzimidazol-2-yl)-5-methyl-4-(phenylmethyl)-4H-pyrazol-3-oneGiardia intestinalisPotency17.740710
2,5-dihydroxy-4-methoxybenzophenoneGiardia intestinalisPotency3.539710
N-[(3-hydroxyanilino)-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency15.811410
4-[(3-methyl-5-nitro-4-imidazolyl)amino]phenolGiardia intestinalisPotency22.334210
2-amino-4-(3,4-dimethoxyphenyl)-7,7-dimethyl-5-oxo-1-(3-pyridinyl)-6,8-dihydro-4H-quinoline-3-carbonitrileGiardia intestinalisPotency14.091910
5-bromo-N-[(1,2-dimethyl-5-indolyl)methyl]-2-furancarboxamideGiardia intestinalisPotency15.811410
4-chloro-N-[(4-ethoxy-2-nitroanilino)-sulfanylidenemethyl]-2,5-dimethyl-3-pyrazolecarboxamideGiardia intestinalisPotency14.091910
2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-6,7,8,8a-tetrahydro-5H-imidazo[1,5-a]pyridine-1,3-dioneGiardia intestinalisPotency17.782810
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidGiardia intestinalisPotency12.589310
5-[2-furanyl(4-morpholinyl)methyl]-6-thiazolo[3,2-b][1,2,4]triazololGiardia intestinalisPotency14.091910
3-hydroxy-6-(hydroxymethyl)-2-[(3-methoxyphenyl)-(2-pyridinylamino)methyl]-4-pyranoneGiardia intestinalisPotency19.905410
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamideGiardia intestinalisPotency15.811410
3-nitro-N-[(3-sulfamoylanilino)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency17.740710
1-[[2-(2,4-dichlorophenoxy)-1-oxoethyl]amino]-3-(4-methoxyphenyl)thioureaGiardia intestinalisPotency17.740710
1,8-dimethoxyphenazineGiardia intestinalisPotency1.409210
2-pyridinecarboxylic acid [2-[2-(difluoromethoxy)anilino]-2-oxoethyl] esterGiardia intestinalisPotency19.905410
N-(1,3-diphenylpropan-2-ylideneamino)-2-hydroxybenzamideGiardia intestinalisPotency7.924510
2-[(3-fluorophenyl)-(2-pyridinylamino)methyl]-3-hydroxy-6-(hydroxymethyl)-4-pyranoneGiardia intestinalisPotency14.091910
1-(1-adamantyl)-2-[(1-oxido-2-pyridin-1-iumyl)thio]ethanoneGiardia intestinalisPotency31.547910
3-(1,5-dimethyl-3-pyrazolyl)-4-phenyl-1H-1,2,4-triazole-5-thioneGiardia intestinalisPotency7.062710
sb 415286Giardia intestinalisPotency29.572420
2-(hexylamino)-1-[4-(phenylmethyl)-1-piperidinyl]ethanoneGiardia intestinalisPotency25.118910
1-(2,6-dimethylphenyl)-3-[[1-(4-methoxyphenyl)-3-pyrrolidinyl]methyl]thioureaGiardia intestinalisPotency15.811410
3-chloro-N-[5-(3-pyridinyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency17.740710
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-oneGiardia intestinalisPotency5.610110
4-methylene-2-octyl-5-oxo-3-oxolanecarboxylic acidGiardia intestinalisPotency15.811410
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methyl-1-piperidinyl)sulfonyl]benzamideGiardia intestinalisPotency31.622810
2-[[2-(3,4-dimethoxyanilino)-2-oxoethyl]thio]-3-pyridinecarboxylic acid propan-2-yl esterGiardia intestinalisPotency31.547910
7-[[2-[5-cyclopropyl-3-(difluoromethyl)-1-pyrazolyl]-1-oxoethyl]amino]-3-[[(1-methyl-5-tetrazolyl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidGiardia intestinalisPotency17.740710
7-[[2-(4-chloro-3,5-dimethyl-1-pyrazolyl)-1-oxoethyl]amino]-3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidGiardia intestinalisPotency39.284120
2-[(5-methyl-4-phenyl-2-thiazolyl)methyl]-4-thiazololGiardia intestinalisPotency22.334210
5-bromo-N-[2-(2-methyl-1-indolyl)ethyl]-2-furancarboxamideGiardia intestinalisPotency17.740710
N-[3-[(2,4-dimethylphenyl)sulfamoyl]-4-methylphenyl]-3-oxo-4H-1,4-benzothiazine-6-carboxamideGiardia intestinalisPotency15.811410
1-(5-nitro-2-thiophenyl)piperidineGiardia intestinalisPotency35.397310
N-[2-(2,4,6-trinitrophenyl)ethyl]anilineGiardia intestinalisPotency15.811410
3-(3-chloro-4-methoxyphenyl)-1-(2-methoxyethyl)-1-(1-propan-2-yl-4-piperidinyl)thioureaGiardia intestinalisPotency9.136620
1-[(2-fluorophenyl)methyl]-4-pyrazolamineGiardia intestinalisPotency17.740710
pd 407824Giardia intestinalisPotency25.059410
1-[3-(dimethylsulfamoyl)phenyl]-3-(2-furanylmethyl)thioureaGiardia intestinalisPotency44.562510
2-chloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency15.811410
5-nitro-2-furancarboxylic acid [2-oxo-2-[3-(1-piperidinylsulfonyl)anilino]ethyl] esterGiardia intestinalisPotency15.811410
4-bromo-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideGiardia intestinalisPotency12.362020
4-[1-(4-fluorophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneGiardia intestinalisPotency1.774110
6-amino-4-(3,5-dimethyl-1-phenyl-4-pyrazolyl)-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileGiardia intestinalisPotency14.091910
N-[5-(phenylmethyl)-2-thiazolyl]-4,5-dihydro-1H-imidazole-2-carboxamideGiardia intestinalisPotency17.740710
N-(2-ethoxyphenyl)-2,1,3-benzothiadiazole-4-sulfonamideGiardia intestinalisPotency17.740710
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamideGiardia intestinalisPotency17.740710
N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[(phenylmethyl)amino]acetamideGiardia intestinalisPotency25.118910
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-[(2-methyl-1-piperidinyl)sulfonyl]benzamideGiardia intestinalisPotency28.183810
1-[3-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-4-methoxyphenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acidGiardia intestinalisPotency3.971610
N-[(3,5-dimethyl-1-piperidinyl)-sulfanylidenemethyl]-2-methyl-5-(4-morpholinylsulfonyl)benzamideGiardia intestinalisPotency15.811410
N-(2-methoxyethyl)-4-oxo-3-[3-(2-oxo-1-pyrrolidinyl)propyl]-2-sulfanylidene-1H-quinazoline-7-carboxamideGiardia intestinalisPotency15.811410
4-(4-propan-2-ylphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazolin-2-oneGiardia intestinalisPotency17.740710
1-amino-3-(4-chloro-2-methoxy-5-methylphenyl)thioureaGiardia intestinalisPotency54.515220
2,4-dichloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency19.905410
4-[bis(2-methoxyethyl)sulfamoyl]-N-[5-(methoxymethyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency22.334210
2-(2-furanyl)-4-mercapto-3-(4-methylphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileGiardia intestinalisPotency15.811410
5-bromo-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-2-thiophenecarboxamideGiardia intestinalisPotency31.547910
4-(1-azepanylsulfonyl)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-hydroxyphenyl]benzamideGiardia intestinalisPotency7.062710
4-chloro-N-[3-(N-methylanilino)-1,4-dioxo-2-naphthalenyl]benzamideGiardia intestinalisPotency1.409210
4-(5-methyl-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)benzoic acid 8-quinolinyl esterGiardia intestinalisPotency17.740710
8-nitro-5-[3-(trifluoromethyl)-1-piperidinyl]isoquinolineGiardia intestinalisPotency22.387210
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaGiardia intestinalisPotency2.818410
3-[4-(4-butan-2-ylphenyl)sulfonyl-1-piperazinyl]butanoic acidGiardia intestinalisPotency17.740710
2-(5-chloro-2,4-dimethoxyanilino)-1-(4-ethyl-1-piperazinyl)-1-propanoneGiardia intestinalisPotency5.000010
N-[(1,5-dimethyl-2-pyrrolyl)methyl]-1-(4-methylphenyl)-5-oxo-3-pyrrolidinecarboxamideGiardia intestinalisPotency11.193610
2-[2,5-diethoxy-4-(4-morpholinyl)anilino]-1-(4-methyl-1-piperidinyl)-1-propanoneGiardia intestinalisPotency3.539710
N-(4-bromo-2-fluorophenyl)-2-(2,4-dimethoxyanilino)acetamideGiardia intestinalisPotency3.154810
N-[[[2-(2-naphthalenyloxy)-1-oxopropyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideGiardia intestinalisPotency17.740710
3-(2-methoxyphenyl)-4-phenyl-1H-imidazole-2-thioneGiardia intestinalisPotency19.905410
diclofenac sodiumGiardia intestinalisPotency19.905410
N-[2-chloro-5-[ethyl(phenyl)sulfamoyl]phenyl]-2-[methyl-(1-methyl-4-piperidinyl)amino]acetamideGiardia intestinalisPotency19.905410
N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzenesulfonamideGiardia intestinalisPotency19.605420
5-[2-furanyl-[4-(phenylmethyl)-1-piperidinyl]methyl]-6-thiazolo[3,2-b][1,2,4]triazololGiardia intestinalisPotency12.559410
[4-[bis(4-morpholinyl)phosphoryl]-1-methyl-2-pyrrolyl]-bis(4-morpholinyl)-sulfanylidenephosphoraneGiardia intestinalisPotency25.059410
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-(1-pyrrolidinylsulfonyl)benzamideGiardia intestinalisPotency5.000010
4-(dimethylsulfamoyl)-N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency6.294610
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideGiardia intestinalisPotency15.811410
N-(4-methoxyphenyl)sulfonyl-N-(2-oxo-5-benzo[g][1,3]benzoxathiolyl)-2-furancarboxamideGiardia intestinalisPotency17.740710
2-(2-methoxyanilino)-2-(2-phenylmethoxyphenyl)acetonitrileGiardia intestinalisPotency15.811410
3,7-dibutyl-3,7-dimethyl-2,6-dihydro-[1,2,4]triazolo[1,2-a][1,2,4]triazole-1,5-dithioneGiardia intestinalisPotency15.811410
2-(4-acetyl-1-piperazinyl)-6-amino-4-(cyanomethyl)pyridine-3,5-dicarbonitrileGiardia intestinalisPotency15.811410
(3,5-dichloroanilino)thioureaGiardia intestinalisPotency7.924510
6-(4-methoxyphenyl)-N,3-dimethyl-2-imidazo[2,1-b]thiazolecarboxamideGiardia intestinalisPotency11.193610
2-[[3-butyl-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideGiardia intestinalisPotency1.774110
fraxetinGiardia intestinalisPotency22.482410
geranylgeranic acidGiardia intestinalisPotency22.334210
quercetinGiardia intestinalisPotency15.811410
bilirubinGiardia intestinalisPotency14.091910
apigeninGiardia intestinalisPotency6.294610
daphnetinGiardia intestinalisPotency9.976310
gossypetinGiardia intestinalisPotency7.062710
rutinGiardia intestinalisPotency22.334210
pyrantel pamoateGiardia intestinalisPotency25.059410
methysergide maleateGiardia intestinalisPotency1.255910
chartreusinGiardia intestinalisPotency7.062710
esculetinGiardia intestinalisPotency13.538310
baicaleinGiardia intestinalisPotency7.633610
fisetinGiardia intestinalisPotency25.059410
hyperosideGiardia intestinalisPotency7.924510
myricetinGiardia intestinalisPotency10.950110
myricitrinGiardia intestinalisPotency10.405710
robinetinGiardia intestinalisPotency11.193610
caffeic acid phenethyl esterGiardia intestinalisPotency16.776110
rosmarinic acidGiardia intestinalisPotency17.740710
wedelolactoneGiardia intestinalisPotency19.905410
ellagic acidGiardia intestinalisPotency9.998220
ginkgolic acidGiardia intestinalisPotency15.811410
flupenthixolGiardia intestinalisPotency15.811410
arachidonyl dopamineGiardia intestinalisPotency15.811410
domoic acidGiardia intestinalisPotency17.740710
4-hydroxyestradiolGiardia intestinalisPotency12.559410
menatetrenoneGiardia intestinalisPotency15.811410
prostaglandin f2 methyl esterGiardia intestinalisPotency17.740710
2-bromoergocryptine mesylateGiardia intestinalisPotency17.740710
geldanamycinGiardia intestinalisPotency3.539710
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidGiardia intestinalisPotency25.059410
4-(3,4-dihydroxyphenyl)-6-[(4-fluoro-3-methylphenyl)sulfonylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterGiardia intestinalisPotency15.811410
5-[(2-fluorophenyl)methyl]-6,11-dioxo-3-benzo[b][1,4]benzothiazepinecarboxylic acidGiardia intestinalisPotency17.740710
N-[[4-(dimethylamino)phenyl]methyl]-2-[methyl(8-quinolinylsulfonyl)amino]acetamideGiardia intestinalisPotency28.117110
N-(6-methyl-1,3-benzothiazol-2-yl)-2-(5,6,7,8-tetrahydro-4H-cyclohepta[c]pyrazol-2-yl)acetamideGiardia intestinalisPotency17.740710
4-[3-oxo-1-(3,4,5-trimethoxyanilino)-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterGiardia intestinalisPotency15.811410
N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineGiardia intestinalisPotency28.117110
8-(2-chlorophenyl)-3-(4-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileGiardia intestinalisPotency3.154810
rosmarinic acidGiardia intestinalisPotency12.186110
fumarprotocetraric acidGiardia intestinalisPotency19.905410
baicalein-7-o-glucosideGiardia intestinalisPotency22.334210
salazinic acidGiardia intestinalisPotency17.740710
erbstatinGiardia intestinalisPotency14.091910
ag 99Giardia intestinalisPotency25.059410
tyrphostin ag 555Giardia intestinalisPotency23.005510
tyrphostin ag-494Giardia intestinalisPotency25.059410
nifuroxazideGiardia intestinalisPotency14.091910
bay 11-7082Giardia intestinalisPotency15.811410
7,8-dihydroxy-4-methylcoumarinGiardia intestinalisPotency7.062710
styrylquinolineGiardia intestinalisPotency22.334210
norstictic acidGiardia intestinalisPotency15.811410
5,6-dichloro-1H-imidazo[4,5-b]pyrazine-2-carboxylic acidGiardia intestinalisPotency12.589310
phentolamineGiardia intestinalisPotency17.740710
dithiazanine iodideGiardia intestinalisPotency15.811410
3,3'-diethylthiatricarbocyanine iodide, 3h-labeledGiardia intestinalisPotency35.481310
5-(4-methyl-1-naphthalenyl)-N-phenyl-2-furancarboxamideGiardia intestinalisPotency19.905410
HTS 01037Giardia intestinalisPotency15.811410
3',4'-dihydroxyauroneGiardia intestinalisPotency17.740710
obtusaquinoneGiardia intestinalisPotency22.334210
nf023Giardia intestinalisPotency19.905410
3,5-di-tert-butylchalcone 4'-carboxylic acidGiardia intestinalisPotency17.740710
4-methyl-N-prop-2-enyl-1-phthalazinamineGiardia intestinalisPotency11.220210
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-1-(4-methoxyphenyl)ethanoneGiardia intestinalisPotency17.740710
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-N-(3-methylphenyl)acetamideGiardia intestinalisPotency17.740710
N-methyl-6-phenyl-3-(2-pyridinyl)-1,2,4-triazin-5-amineGiardia intestinalisPotency19.905410
N'1-(6-methylpyridazin-3-yl)-4-chlorobenzene-1-carbohydrazideGiardia intestinalisPotency17.740710
ubp 302Giardia intestinalisPotency19.905410
1,5-anhydro-1-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-6-yl]hexitolGiardia intestinalisPotency22.334210
thermozymocidinGiardia intestinalisPotency15.811410
mareinGiardia intestinalisPotency17.740710
N-(1,3-benzothiazol-2-yl)-2-(2,6-dimethyl-4-morpholinyl)acetamideGiardia intestinalisPotency14.125410
3,4,5-trimethoxy-N-[[[oxo-[(1S,2S)-2-phenylcyclopropyl]methyl]hydrazo]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency22.334210
a 77636Giardia intestinalisPotency44.562510
nitrofurantoinGiardia intestinalisPotency25.059410
azetidine-2,4-dicarboxylic acidGiardia intestinalisPotency39.716410
bay-k-8644Giardia intestinalisPotency7.924510
bvt.948Giardia intestinalisPotency5.709730
N-(5-carbamoyl-2-methoxyphenyl)-3-(2,4-dimethoxyphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamideGiardia intestinalisPotency10.000010
(2R,4R)-4-(1-acetyl-3-indolyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamideGiardia intestinalisPotency17.740710
epinephrine bitartrateGiardia intestinalisPotency5.778710
LSM-6455Giardia intestinalisPotency2.233410
3-(2-pyridinyl)-6-(2-pyridinylmethylthio)pyridazineGiardia intestinalisPotency31.547910
2-[[6-(2-furanyl)-3-pyridazinyl]thio]-1-(1-piperidinyl)ethanoneGiardia intestinalisPotency12.559410
N-cyclohexyl-2-[[6-(2-pyridinyl)-3-pyridazinyl]thio]acetamideGiardia intestinalisPotency22.334210
(3aR,6aR)-5-(3-methoxyphenyl)-3-[oxo(2-pyrazinyl)methyl]-3a,6a-dihydro-1H-pyrrolo[3,4-c]pyrazole-4,6-dioneGiardia intestinalisPotency15.811410
3-(diphenylmethylene)-1-[4-(4-phenyl-1-piperazinyl)butyl]pyrrolidine-2,5-dioneGiardia intestinalisPotency15.811410
3-hydroxy-2-methyl-1-(phenylmethyl)-4-pyridinoneGiardia intestinalisPotency9.976310
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-2-(1-methyl-3-indolyl)ethanoneGiardia intestinalisPotency31.547910
levodopa methyl ester hydrochloride, (dl)-isomerGiardia intestinalisPotency17.740710
thioacetazoneGiardia intestinalisPotency15.811410
cefotaxime sodiumGiardia intestinalisPotency14.091910
impentamineGiardia intestinalisPotency25.059410
bn82002Giardia intestinalisPotency7.924510
a-317491Giardia intestinalisPotency17.740710
lissamine rhodamine bGiardia intestinalisPotency28.183810
trimetazidine dihydrochlorideGiardia intestinalisPotency22.387210
ps1145Giardia intestinalisPotency15.811410
NNC 55-0396 (free base)Giardia intestinalisPotency19.905410
levodopa methyl ester hydrochlorideGiardia intestinalisPotency6.294610
1-(2,4-dichlorophenyl)-6-methyl-N-(1-piperidinyl)-4H-indeno[1,2-c]pyrazole-3-carboxamideGiardia intestinalisPotency17.740710
garcinone eGiardia intestinalisPotency17.740710
ws-5995 cGiardia intestinalisPotency15.811410
Dihydrotanshinone IGiardia intestinalisPotency7.062710
2-methylene-3-hexylbutanedioic acidGiardia intestinalisPotency15.811410
losartan potassiumGiardia intestinalisPotency26.200020
gw9508Giardia intestinalisPotency15.811410
(1S,2R)-2-[[4-[(2,4-dimethylphenyl)sulfamoyl]anilino]-oxomethyl]-1-cyclohexanecarboxylic acidGiardia intestinalisPotency17.740710
N-(2-methoxyethyl)-2-[[3-[(4-methoxyphenyl)methyl]-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideGiardia intestinalisPotency3.971610
R-(-)-actinodaphnineGiardia intestinalisPotency8.891410
6-fluoronorepinephrine monohydrochloride, (+-)-isomerGiardia intestinalisPotency5.610110
calcimycinGiardia intestinalisPotency17.740710
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideGiardia intestinalisPotency17.740710
dehydrocurvularinGiardia intestinalisPotency15.811410
rabeprazole sodiumGiardia intestinalisPotency32.545520
4-chloro-N-[1-[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-3-methyl-1-oxobutan-2-yl]benzamideGiardia intestinalisPotency17.740710
1-hydroxy-5-nitro-N-(2-phenylethyl)-4-spiro[benzimidazole-2,1'-cyclohexane]imineGiardia intestinalisPotency1.774110
3-bromo-N-[5-(4-morpholinylsulfonyl)-1,3,4-thiadiazol-2-yl]benzamideGiardia intestinalisPotency28.183810
GS4012Giardia intestinalisPotency15.811410
1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-nitrophenyl)ureaGiardia intestinalisPotency19.905410
2-[[6-(4-morpholinyl)-4-oxo-3-(2-phenylethyl)-2-quinazolinyl]thio]-N-(2-oxolanylmethyl)acetamideGiardia intestinalisPotency8.891410
2-(1,3-benzodioxol-5-ylmethyl)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolineGiardia intestinalisPotency15.811410
1-[3-[(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-6-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]-3,4-dihydro-2H-pyran-4-yl]-1-indolyl]ethanoneGiardia intestinalisPotency15.811410
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid tert-butyl esterGiardia intestinalisPotency15.811410
(2S)-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]-3-phenylpropanoic acid (phenylmethyl) esterGiardia intestinalisPotency15.811410
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid (phenylmethyl) esterGiardia intestinalisPotency17.740710
(2S)-4-methyl-2-[[[5-(methylcarbamoyl)-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterGiardia intestinalisPotency19.905410
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterGiardia intestinalisPotency17.740710
(2S)-2-[[[5-[[methyl-(phenylmethyl)amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterGiardia intestinalisPotency17.740710
violaceol IIGiardia intestinalisPotency15.811410
(3aR,4S,9aR,9bS)-N-(4-chlorophenyl)-2-(4-fluorophenyl)-1,3-dioxo-3a,4,9a,9b-tetrahydropyrrolo[1,2]pyrrolo[3,5-b]pyridazine-4-carboxamideGiardia intestinalisPotency17.740710
phenylmercuric acetateGiardia intestinalisPotency17.740710
phentin acetateGiardia intestinalisPotency1.990510
thimerosalGiardia intestinalisPotency12.559410
3-phenylpropanoic acid [3-(4-cyanophenyl)-2-cyclohexyl-7-methyl-6,8-dioxo-7-isoquinolinyl] esterGiardia intestinalisPotency0.903210
3-phenylpropanoic acid [3-(4-cyanophenyl)-7-methyl-6,8-dioxo-2-[2-(2-pyridinyl)ethyl]-7-isoquinolinyl] esterGiardia intestinalisPotency1.990510
3-(1,3-benzodioxol-5-yl)-3-(2-hydroxy-4,6-dimethoxyphenyl)-1-(3-methyl-1-piperidinyl)-1-propanoneGiardia intestinalisPotency17.740710
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterGiardia intestinalisPotency56.100910
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterGiardia intestinalisPotency25.059410
2,3,4,10-tetrahydro-7,10-dimethyl-2,4-dioxobenzo(g)pteridineGiardia intestinalisPotency0.125610
N-[4-[[[6-(3,5-dimethyl-4-isoxazolyl)-4-quinazolinyl]amino]methyl]phenyl]acetamideGiardia intestinalisPotency31.547910
4-(phenylmethyl)-N-prop-2-enyl-1-piperidinecarbothioamideGiardia intestinalisPotency3.548110
1-(3-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)thioureaGiardia intestinalisPotency19.952610
N-[1,4-dimethyl-2,3-dioxo-7-(1-piperidinyl)-6-quinoxalinyl]-4-ethylbenzenesulfonamideGiardia intestinalisPotency19.952610
ampicillin sodiumGiardia intestinalisPotency12.559410
cefoxitin sodiumGiardia intestinalisPotency15.811410
cefamandole nafateGiardia intestinalisPotency15.811410
estrone sulfate, potassium saltGiardia intestinalisPotency19.905410
sodium cephalothinGiardia intestinalisPotency15.811410
cefazolin sodiumGiardia intestinalisPotency15.811410
N-[5-Bromo-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chlorideGiardia intestinalisPotency17.782810
hcl(s)-isomer of tetrahydropalmatineGiardia intestinalisPotency28.183810
N-[5-Fluoro-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chlorideGiardia intestinalisPotency25.118910
4-(4-chloro-3-nitrophenyl)-N-[2-(5,6-dichloro-1-propyl-2-benzimidazolyl)ethyl]-2-thiazolamineGiardia intestinalisPotency15.848910
2-[[[4-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterGiardia intestinalisPotency28.183810
4-[(6-chloro-1H-benzimidazol-2-yl)amino]benzoic acidGiardia intestinalisPotency19.952610
4-[[3-(4-chlorophenyl)-5-isoxazolyl]methyl]-1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinecarboxylic acidGiardia intestinalisPotency39.810710
oxytetracycline, anhydrousGiardia intestinalisPotency4.456310
mobiflexGiardia intestinalisPotency14.951610
warfarinGiardia intestinalisPotency17.740710
LSM-23865Giardia intestinalisPotency5.000010
3-benzyl-4-hydroxyquinolin-2(1H)-oneGiardia intestinalisPotency15.811410
citrininGiardia intestinalisPotency12.559410
antimycinGiardia intestinalisPotency11.193610
methacycline monohydrochlorideGiardia intestinalisPotency17.740710
mysteclin fGiardia intestinalisPotency14.125410
demeclocycline hydrochlorideGiardia intestinalisPotency14.091910
vulpinic acidGiardia intestinalisPotency17.740710
1-ethyl-4-hydroxy-2-oxo-N-(3-pyridinylmethyl)-3-quinolinecarboxamideGiardia intestinalisPotency44.562510
4-hydroxy-2-oxo-1-pentyl-N-(2-pyridinylmethyl)-3-quinolinecarboxamideGiardia intestinalisPotency31.547910
stf 083010Giardia intestinalisPotency22.334210
hypoxanthineGiardia intestinalisPotency19.905410
folic acidGiardia intestinalisPotency39.810710
suptopin 2Giardia intestinalisPotency17.188620
azaguanineGiardia intestinalisPotency7.943310
hemateinGiardia intestinalisPotency13.502510
1-hydroxyphenazineGiardia intestinalisPotency10.126320
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-6-methyl-1H-pyrimidin-4-oneGiardia intestinalisPotency15.811410
6-methyl-3-sulfanylidene-1,2-dihydro-[1,2,4]triazolo[4,3-b][1,2,4]triazin-7-oneGiardia intestinalisPotency11.193610
5-(4-methoxyphenyl)-6-sulfanylidene-1,2-dihydropyrazolo[3,4-d]pyrimidin-4-oneGiardia intestinalisPotency17.740710
adenalleneGiardia intestinalisPotency8.912510
N-carbamoyl-2-[4-oxo-2-[(2-oxo-5H-thiazol-4-yl)hydrazo]-5-thiazolyl]acetamideGiardia intestinalisPotency12.559410
2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]acetamideGiardia intestinalisPotency17.740710
6-amino-2-[[2-(3,4-dimethylphenyl)-2-oxoethyl]thio]-1H-pyrimidin-4-oneGiardia intestinalisPotency39.810710
6,7-dimethoxy-2-[[methyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]methyl]-1H-quinazolin-4-oneGiardia intestinalisPotency5.000010
galloflavinGiardia intestinalisPotency2.811710
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-[2-(methylthio)phenyl]acetamideGiardia intestinalisPotency3.539710
5,5-diethyl-2-hydrazinyl-1,6-dihydrobenzo[h]quinazolin-4-oneGiardia intestinalisPotency25.059410
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-(3-fluorophenyl)acetamideGiardia intestinalisPotency6.294610
N-[(cyclohexylamino)-oxomethyl]-2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]acetamideGiardia intestinalisPotency5.000010
2-[[2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]-4-methylpentanoic acid methyl esterGiardia intestinalisPotency22.334210
2-(butylthio)-4-oxo-1H-pyrimidine-6-carboxylic acidGiardia intestinalisPotency17.740710
N-[6-amino-2-[[2-(4-methyl-1-piperidinyl)-2-oxoethyl]thio]-4-oxo-1H-pyrimidin-5-yl]benzamideGiardia intestinalisPotency28.183810