Page last updated: 2024-08-07 17:15:03
Amine oxidase [flavin-containing] A
An amine oxidase [flavin-containing] A that is encoded in the genome of mouse. [OMA:Q64133, PRO:DNx]
Synonyms
EC 1.4.3.4;
Monoamine oxidase type A;
MAO-A
Research
Bioassay Publications (8)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 1 (12.50) | 18.7374 |
1990's | 1 (12.50) | 18.2507 |
2000's | 1 (12.50) | 29.6817 |
2010's | 4 (50.00) | 24.3611 |
2020's | 1 (12.50) | 2.80 |
Compounds (10)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
heliamine | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
u 0521 | Mus musculus (house mouse) | IC50 | 50.0000 | 1 | 1 |
piperine | Mus musculus (house mouse) | Ki | 19.0000 | 1 | 1 |
aurapten | Mus musculus (house mouse) | IC50 | 0.0000 | 1 | 1 |
6-methyl-2-(phenylethynyl)pyridine | Mus musculus (house mouse) | IC50 | 8.0000 | 1 | 1 |
formononetin | Mus musculus (house mouse) | IC50 | 21.2000 | 1 | 1 |
lacinartin | Mus musculus (house mouse) | IC50 | 5.7000 | 2 | 2 |
3-((2-methyl-1,3-thiazol-4-yl)ethynyl)piperidine | Mus musculus (house mouse) | IC50 | 30.0000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
selegiline | Mus musculus (house mouse) | Activity | 0.0010 | 2 | 6 |
desmethylselegiline | Mus musculus (house mouse) | Activity | 0.0012 | 2 | 3 |