Page last updated: 2024-08-08 00:00:06
Histone deacetylase-like amidohydrolase
[no definition available]
Synonyms
HDAC-like amidohydrolase;
HDAH;
EC 3.5.1.-
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
entinostat | Alcaligenaceae bacterium FB188 | IC50 | 118.0000 | 1 | 1 |
entinostat | Alcaligenaceae bacterium FB188 | Ki | 100.0000 | 1 | 1 |
vorinostat | Alcaligenaceae bacterium FB188 | IC50 | 1.0000 | 1 | 1 |
vorinostat | Alcaligenaceae bacterium FB188 | Ki | 1.1500 | 2 | 2 |
trichostatin a | Alcaligenaceae bacterium FB188 | IC50 | 1.2000 | 1 | 1 |
trichostatin a | Alcaligenaceae bacterium FB188 | Ki | 0.7000 | 1 | 1 |
(3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone | Alcaligenaceae bacterium FB188 | Ki | 9.2000 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
vorinostat | Alcaligenaceae bacterium FB188 | Kd | 0.3000 | 1 | 1 |