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Cannabinoid receptor 2
A cannabinoid receptor 2 that is encoded in the genome of mouse. [OMA:P47936, PRO:DNx]
Synonyms
CB-2;
CB2;
mCB2
Research
Bioassay Publications (22)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (4.55) | 18.2507 |
| 2000's | 9 (40.91) | 29.6817 |
| 2010's | 11 (50.00) | 24.3611 |
| 2020's | 1 (4.55) | 2.80 |
Compounds (31)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
Drugs with Other Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| ly 255582 | Mus musculus (house mouse) | Kb | 0.0003 | 1 | 1 |
Oxa-adamantyl cannabinoids.Bioorganic & medicinal chemistry letters, , 04-15, Volume: 38, 2021
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential.Journal of medicinal chemistry, , 11-21, Volume: 61, Issue:22, 2018
2-Arylimino-5,6-dihydro-4H-1,3-thiazines as a new class of cannabinoid receptor agonists. Part 2: orally bioavailable compounds.Bioorganic & medicinal chemistry letters, , Jul-15, Volume: 17, Issue:14, 2007
Novel cannabinol probes for CB1 and CB2 cannabinoid receptors.Journal of medicinal chemistry, , Oct-05, Volume: 43, Issue:20, 2000
( R)- N-(1-Methyl-2-hydroxyethyl)-13-( S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes.Journal of medicinal chemistry, , 10-11, Volume: 61, Issue:19, 2018
Two new unsaturated fatty acid ethanolamides in brain that bind to the cannabinoid receptor.Journal of medicinal chemistry, , Oct-01, Volume: 36, Issue:20, 1993
Design, synthesis, and biological evaluation of (3R)-1,2,3,4-tetrahydro-7-hydroxy-N-[(1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl]-3-isoquinolinecarboxamide (JDTic) analogues: in vitro pharmacology and ADME profilJournal of medicinal chemistry, , Sep-11, Volume: 57, Issue:17, 2014