Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
ellipticine | Homo sapiens (human) | EC50 | 3.9900 | 1 | 0 |
naftopidil | Homo sapiens (human) | EC50 | 3.7200 | 1 | 0 |
oxatomide | Homo sapiens (human) | EC50 | 5.1500 | 1 | 0 |
antazoline hydrochloride | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
coumarin 7 | Homo sapiens (human) | EC50 | 0.4340 | 1 | 0 |
6-methyl-2-[(4-nitrophenyl)methylthio]-1H-benzimidazole | Homo sapiens (human) | EC50 | 4.4100 | 1 | 0 |
1-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-4-(2,3-dimethylphenyl)piperazine | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
1-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-3,4-dihydro-2H-quinoline | Homo sapiens (human) | EC50 | 8.8800 | 1 | 0 |
N-(3,4-dimethylphenyl)-2-[[5-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]acetamide | Homo sapiens (human) | EC50 | 4.0500 | 1 | 0 |
5-(2,4-dichlorophenyl)-N-(2-methylphenyl)-2-furancarboxamide | Homo sapiens (human) | EC50 | 7.9600 | 1 | 0 |
N-[4-chloro-3-(trifluoromethyl)phenyl]-3-methoxybenzamide | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
5-[(2,4-dichlorophenoxy)methyl]-N-[1-[(2-fluorophenyl)methyl]-3-pyrazolyl]-2-furancarboxamide | Homo sapiens (human) | EC50 | 10.3000 | 1 | 0 |
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamide | Homo sapiens (human) | EC50 | 2.3070 | 2 | 0 |
5-(3-chlorophenyl)-N-(2-propyl-5-tetrazolyl)-2-furancarboxamide | Homo sapiens (human) | EC50 | 6.8100 | 1 | 0 |
[4-(diphenylmethyl)-1-piperazinyl]-[5-thiophen-2-yl-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinyl]methanone | Homo sapiens (human) | EC50 | 6.7500 | 1 | 0 |
3-(2-chloro-6-fluorophenyl)-N-(3-fluoro-4-methylphenyl)-5-methyl-4-isoxazolecarboxamide | Homo sapiens (human) | EC50 | 5.6900 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-4-methyl-3-(1-piperidinylsulfonyl)benzamide | Homo sapiens (human) | EC50 | 5.2300 | 1 | 0 |
N-[2-(4-acetyl-1-piperazinyl)phenyl]-2-(5-methyl-2-propan-2-ylphenoxy)acetamide | Homo sapiens (human) | EC50 | 3.6700 | 1 | 0 |
3-phenyl-5-[[[4-phenyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-1,2,4-oxadiazole | Homo sapiens (human) | EC50 | 4.1600 | 1 | 0 |
N-[3-[[2-(2-bromo-4,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamide | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
2-[2-(2,4-dichloro-5-propan-2-yloxyanilino)-2-oxoethyl]sulfinyl-N-[3-(trifluoromethyl)phenyl]acetamide | Homo sapiens (human) | EC50 | 3.2300 | 1 | 0 |
5-bromo-N-(2-phenylphenyl)-2-furancarboxamide | Homo sapiens (human) | EC50 | 7.4700 | 1 | 0 |
N-[2-[(2-methylphenyl)methylthio]ethyl]-3-[(4-methylphenyl)thio]propanamide | Homo sapiens (human) | EC50 | 2.8700 | 1 | 0 |
N-[3-[[2-(2,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamide | Homo sapiens (human) | EC50 | 6.7800 | 1 | 0 |
2-(1H-benzimidazol-2-ylthio)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamide | Homo sapiens (human) | EC50 | 13.3000 | 1 | 0 |
2-(2,4-dichlorophenyl)-3-(phenylmethyl)-1,2-dihydroquinazolin-4-one | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
5-[[(1-cyclohexyl-5-tetrazolyl)thio]methyl]-3-phenyl-1,2,4-oxadiazole | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
N-(5-chloro-2-pyridinyl)-2-[(1-phenyl-5-tetrazolyl)thio]propanamide | Homo sapiens (human) | EC50 | 6.1400 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamide | Homo sapiens (human) | EC50 | 7.9700 | 1 | 0 |
4-diphenylacetoxy-n-methylpiperidine methiodide | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
2-[7-oxo-7-(3-phenyl-1-pyrrolidinyl)heptyl]isoindole-1,3-dione | Homo sapiens (human) | EC50 | 1.2170 | 2 | 0 |
3,4-dihydro-2H-quinolin-1-yl-[4-(phenylmethyl)-5-thieno[3,2-b]pyrrolyl]methanone | Homo sapiens (human) | EC50 | 5.9800 | 1 | 0 |
1-(2-methyl-2,3-dihydroindol-1-yl)-2-[4-[5-(trifluoromethyl)-1-benzotriazolyl]-1-piperidinyl]ethanone | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
1-(1-tert-butyl-5-tetrazolyl)-N-[(4-fluorophenyl)methyl]-N-(2-furanylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamine | Homo sapiens (human) | EC50 | 2.8400 | 1 | 0 |
1-(4-methyl-2-prop-2-enylphenoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol | Homo sapiens (human) | EC50 | 8.3300 | 1 | 0 |
5-ethyl-N-[2-(2-phenyl-4-thiazolyl)ethyl]-2-thiophenesulfonamide | Homo sapiens (human) | EC50 | 4.2200 | 1 | 0 |
3,5-dimethyl-N-(2-phenylethyl)-N-(phenylmethyl)-4-isoxazolesulfonamide | Homo sapiens (human) | EC50 | 0.0000 | 1 | 0 |
1-[bis(prop-2-enyl)amino]-3-(9-carbazolyl)-2-propanol | Homo sapiens (human) | EC50 | 9.0600 | 1 | 0 |
N-[3-(cyclohexylthio)propyl]-2-[[5-methyl-2-(3-methylphenyl)-4-oxazolyl]methylsulfinyl]acetamide | Homo sapiens (human) | EC50 | 3.9400 | 1 | 0 |
N-ethyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(phenylmethyl)propanamide | Homo sapiens (human) | EC50 | 4.8000 | 1 | 0 |
2-phenoxy-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamide | Homo sapiens (human) | EC50 | 2.1085 | 2 | 0 |
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-(2-methoxyphenyl)-1-piperazinyl]acetamide | Homo sapiens (human) | EC50 | 4.0800 | 1 | 0 |
2-(4-chlorophenoxy)-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamide | Homo sapiens (human) | EC50 | 2.8000 | 1 | 0 |
N-(3,4-dimethylphenyl)-2-[[1-(phenylmethyl)-2-imidazolyl]thio]acetamide | Homo sapiens (human) | EC50 | 2.7400 | 1 | 0 |
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamide | Homo sapiens (human) | EC50 | 10.8000 | 1 | 0 |
N-(3,5-dimethylphenyl)-2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamide | Homo sapiens (human) | EC50 | 2.0100 | 1 | 0 |
N-(5-bromo-2-thiazolyl)-3-phenyl-2-(1-pyrrolyl)propanamide | Homo sapiens (human) | EC50 | 1.3300 | 1 | 0 |
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanone | Homo sapiens (human) | EC50 | 2.2100 | 1 | 0 |
3-(diphenylmethylene)-1-[4-(4-phenyl-1-piperazinyl)butyl]pyrrolidine-2,5-dione | Homo sapiens (human) | EC50 | 3.7700 | 1 | 0 |
3-(1H-benzimidazol-2-yl)-1-[4-(2,4-dimethylphenyl)-1-piperazinyl]-1-propanone | Homo sapiens (human) | EC50 | 3.2700 | 1 | 0 |