[no definition available]
SERCA1;
SR Ca(2+)-ATPase 1;
EC 7.2.2.10;
Calcium pump 1;
Calcium-transporting ATPase sarcoplasmic reticulum type, fast twitch skeletal muscle isoform;
Endoplasmic reticulum class 1/2 Ca(2+) ATPase
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (16.67) | 29.6817 |
| 2010's | 2 (33.33) | 24.3611 |
| 2020's | 3 (50.00) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| 2-aminoethoxydiphenyl borate | Oryctolagus cuniculus (rabbit) | IC50 | 70.0000 | 1 | 1 |
| chlorocresol | Oryctolagus cuniculus (rabbit) | IC50 | 2,800.0000 | 1 | 1 |
| 4-nonylphenol | Oryctolagus cuniculus (rabbit) | IC50 | 0.3500 | 2 | 2 |
| 2,5-di-tert-butylhydroquinone | Oryctolagus cuniculus (rabbit) | IC50 | 2.0000 | 1 | 1 |
| cgp 37157 | Oryctolagus cuniculus (rabbit) | IC50 | 6.6000 | 1 | 1 |
| chelerythrine | Oryctolagus cuniculus (rabbit) | IC50 | 1.2000 | 1 | 1 |
| chlorpromazine | Oryctolagus cuniculus (rabbit) | IC50 | 23.0000 | 1 | 1 |
| clotrimazole | Oryctolagus cuniculus (rabbit) | Ki | 35.0000 | 1 | 1 |
| fluphenazine | Oryctolagus cuniculus (rabbit) | IC50 | 15.0000 | 1 | 1 |
| trifluoperazine | Oryctolagus cuniculus (rabbit) | IC50 | 45.0000 | 1 | 1 |
| tetrabromobisphenol a | Oryctolagus cuniculus (rabbit) | IC50 | 0.5000 | 1 | 1 |
| bisphenol a | Oryctolagus cuniculus (rabbit) | IC50 | 117.5000 | 2 | 2 |
| phenylhydroquinone | Oryctolagus cuniculus (rabbit) | IC50 | 2.2900 | 1 | 1 |
| 1,1'-methylenedi-2-naphthol | Oryctolagus cuniculus (rabbit) | IC50 | 15.0000 | 1 | 1 |
| epigallocatechin gallate | Oryctolagus cuniculus (rabbit) | IC50 | 12.0000 | 1 | 1 |
| paxilline | Oryctolagus cuniculus (rabbit) | IC50 | 5.0000 | 1 | 1 |
| thapsigargin | Oryctolagus cuniculus (rabbit) | IC50 | 0.0020 | 2 | 2 |
| diethylstilbestrol | Oryctolagus cuniculus (rabbit) | IC50 | 14.0000 | 1 | 1 |
| calmidazolium | Oryctolagus cuniculus (rabbit) | IC50 | 0.5000 | 1 | 1 |
| 3,6-dihydroxyflavone | Oryctolagus cuniculus (rabbit) | IC50 | 6.0000 | 1 | 1 |
| curcumin | Oryctolagus cuniculus (rabbit) | IC50 | 3.0000 | 1 | 1 |
| curcumin | Oryctolagus cuniculus (rabbit) | Ki | 5.8000 | 1 | 1 |
| quercetin | Oryctolagus cuniculus (rabbit) | IC50 | 9.0000 | 1 | 1 |
| galangin | Oryctolagus cuniculus (rabbit) | IC50 | 9.0000 | 1 | 1 |
| morusin | Oryctolagus cuniculus (rabbit) | IC50 | 43.5700 | 1 | 1 |
| cyclosporine | Oryctolagus cuniculus (rabbit) | IC50 | 62.0000 | 1 | 1 |
| sirolimus | Oryctolagus cuniculus (rabbit) | IC50 | 77.0000 | 1 | 1 |
| 22,23-dihydroavermectin b(1)a | Oryctolagus cuniculus (rabbit) | IC50 | 15.0000 | 1 | 1 |
| alisol b | Oryctolagus cuniculus (rabbit) | IC50 | 27.0000 | 1 | 1 |
| ethyl 2-amino-6-(3,5-dimethoxyphenyl)-4-(2-ethoxy-2-oxoethyl)-4h-chromene-3-carboxylate | Oryctolagus cuniculus (rabbit) | IC50 | 13.5000 | 1 | 1 |
| biselyngbyaside | Oryctolagus cuniculus (rabbit) | Ki | 0.0190 | 1 | 1 |
| alpha-cyclopiazonic acid | Oryctolagus cuniculus (rabbit) | IC50 | 0.0900 | 1 | 1 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| thapsigargin | Oryctolagus cuniculus (rabbit) | Kd | 0.0002 | 1 | 1 |