Page last updated: 2024-08-07 17:31:50

Transient receptor potential cation channel subfamily V member 2

A transient receptor potential cation channel TRPV2 that is encoded in the genome of rat. [OMA:Q9WUD2, PRO:DNx]

Synonyms

TrpV2;
Osm-9-like TRP channel 2;
OTRPC2;
Stretch-activated channel 2B;
Vanilloid receptor-like protein 1;
VRL-1

Research

Bioassay Publications (13)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's3 (23.08)18.2507
2000's5 (38.46)29.6817
2010's4 (30.77)24.3611
2020's1 (7.69)2.80

Compounds (30)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
palmitic acidRattus norvegicus (Norway rat)IC5010.000022
clemizoleRattus norvegicus (Norway rat)IC5020.000011
haloperidolRattus norvegicus (Norway rat)Ki0.005011
palmidrolRattus norvegicus (Norway rat)IC5010.000022
arachidic acidRattus norvegicus (Norway rat)IC5010.000022
stearoylethanolamideRattus norvegicus (Norway rat)IC5010.000022
hexadecanamideRattus norvegicus (Norway rat)IC5010.000022
arachidonic acidRattus norvegicus (Norway rat)IC5010.000022
oleic acidRattus norvegicus (Norway rat)IC5010.000022
cannabidiolRattus norvegicus (Norway rat)IC501.100011
capsazepineRattus norvegicus (Norway rat)IC50162.975044
erucic acidRattus norvegicus (Norway rat)IC5010.000022
anandamideRattus norvegicus (Norway rat)IC504.780022
oleylamideRattus norvegicus (Norway rat)IC502.100022
linoleoyl ethanolamideRattus norvegicus (Norway rat)IC501.025022
N-(4Z,7Z,10Z,13Z,16Z,19Z)-docosahexaenoylethanolamineRattus norvegicus (Norway rat)IC505.815022
n-oleoylethanolamineRattus norvegicus (Norway rat)IC503.600022
olvanilRattus norvegicus (Norway rat)IC500.930022
cannabigerolRattus norvegicus (Norway rat)IC501.500011
erucyl amideRattus norvegicus (Norway rat)IC503.885022
iodoresiniferatoxinRattus norvegicus (Norway rat)IC504.000011
linoleamideRattus norvegicus (Norway rat)IC501.700022
kjm 429Rattus norvegicus (Norway rat)IC500.110022
jyl 1421Rattus norvegicus (Norway rat)IC500.037011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
cannabinolRattus norvegicus (Norway rat)EC5019.000011
nonivamideRattus norvegicus (Norway rat)EC500.550022
dihydrocapsaicinRattus norvegicus (Norway rat)EC500.190011
cannabidiolRattus norvegicus (Norway rat)EC501.200011
capsaicinRattus norvegicus (Norway rat)EC500.246045
capsazepineRattus norvegicus (Norway rat)EC50100.000011
N-octylhomovanillamideRattus norvegicus (Norway rat)EC500.300011
olvanilRattus norvegicus (Norway rat)EC500.170022
cannabigerolRattus norvegicus (Norway rat)EC501.700011
ne 21610Rattus norvegicus (Norway rat)EC500.250011