[no definition available]
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0) | 18.7374 |
1990's | 0 (0) | 18.2507 |
2000's | 0 (0) | 29.6817 |
2010's | 0 (0) | 24.3611 |
2020's | 0 (0) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
aspirin | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
celecoxib | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
indirubin-3'-monoxime | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
ketoprofen | Homo sapiens (human) | EC50 | 15.1885 | 2 | 0 |
indirubin | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
6-methoxy-2-naphthylacetic acid | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
dexibuprofen | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
1,3-diphenyl-2-propyn-1-one | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
valdecoxib | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
2-(2-phenylethylthio)-3-pyridinecarboxylic acid | Homo sapiens (human) | EC50 | 0.1185 | 2 | 0 |
2-[[benzamido(sulfanylidene)methyl]amino]-5,5-dimethyl-4,7-dihydrothieno[2,3-c]pyran-3-carboxylic acid | Homo sapiens (human) | EC50 | 0.0849 | 8 | 0 |
sulindac | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
2-[(2-bromophenyl)methoxy]benzoic acid | Homo sapiens (human) | EC50 | 0.1090 | 1 | 0 |
sulindac sulfide | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
1-[2-(2,5-dimethylphenoxy)ethyl]-3-indolecarboxylic acid | Homo sapiens (human) | EC50 | 0.1950 | 1 | 0 |
4-[3-(4-methylphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamide | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
naproxen sodium | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
4-[3-(3-methylphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamide | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
4-[3-(3-bromophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamide | Homo sapiens (human) | EC50 | 30.0000 | 2 | 0 |
7-bromoindirubin-3'-oxime | Homo sapiens (human) | EC50 | 33.7485 | 2 | 0 |
2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-N-phenylacetamide | Homo sapiens (human) | EC50 | 1.9660 | 1 | 0 |