Page last updated: 2024-08-07 19:29:44
Beta-1 adrenergic receptor
A beta-1 adrenergic receptor that is encoded in the genome of mouse. [OMA:P34971, PRO:DNx]
Synonyms
Beta-1 adrenoreceptor;
Beta-1 adrenoceptor
Research
Bioassay Publications (4)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 1 (25.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 3 (75.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (8)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
bisoprolol | Mus musculus (house mouse) | Ki | 0.0053 | 1 | 1 |
cgp 20712a | Mus musculus (house mouse) | Ki | 0.0014 | 1 | 1 |
isoproterenol | Mus musculus (house mouse) | Ki | 0.2200 | 1 | 1 |
metoprolol | Mus musculus (house mouse) | Ki | 0.0490 | 1 | 1 |
propranolol | Mus musculus (house mouse) | Ki | 0.0024 | 1 | 1 |
salmeterol xinafoate | Mus musculus (house mouse) | Ki | 0.5500 | 1 | 1 |
carazolol | Mus musculus (house mouse) | Ki | 0.0001 | 1 | 1 |
L-isoprenaline | Mus musculus (house mouse) | Ki | 0.2200 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
isoproterenol | Mus musculus (house mouse) | EC50 | 0.9800 | 1 | 1 |