Proteins > rac GTPase-activating protein 1 isoform a
Page last updated: 2024-08-08 00:31:57

rac GTPase-activating protein 1 isoform a

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (128)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
6-hydroxymelatoninHomo sapiens (human)IC5052.260010
mitoxantroneHomo sapiens (human)IC5014.460010
acriflavine chlorideHomo sapiens (human)IC5078.300010
phenidoneHomo sapiens (human)IC5046.480010
phenothiazineHomo sapiens (human)IC5018.500010
benzidineHomo sapiens (human)IC507.390010
3-hydroxydiphenylamineHomo sapiens (human)IC5062.550010
n,n,n',n'-tetramethyl-4,4'-methylenedianilineHomo sapiens (human)IC5073.150010
dianisidineHomo sapiens (human)IC509.000010
2-tolidineHomo sapiens (human)IC5012.160010
3-amino-9-ethylcarbazoleHomo sapiens (human)IC5064.100010
4,4'-thiodianilineHomo sapiens (human)IC5013.160010
sterogenolHomo sapiens (human)IC5061.090010
5H-dibenzo[b,f]azepineHomo sapiens (human)IC5014.900010
nitrophenideHomo sapiens (human)IC5053.920010
4,4'-diaminoazobenzeneHomo sapiens (human)IC5021.950010
2,2'-diaminodiphenyldisulfideHomo sapiens (human)IC5086.090010
4-hydroxyazobenzeneHomo sapiens (human)IC5070.940010
7-hydroxychlorpromazineHomo sapiens (human)IC5011.620010
ethyl violetHomo sapiens (human)IC5020.560010
3-aminofluorantheneHomo sapiens (human)IC5039.190010
2-hydroxy-7-nitrofluoreneHomo sapiens (human)IC5016.690010
(7S,9S)-7-[(4-amino-5-hydroxy-6-methyl-2-oxanyl)oxy]-6,9,11-trihydroxy-9-(2-hydroxy-1-oxoethyl)-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dioneHomo sapiens (human)IC5053.480010
NanaomycinHomo sapiens (human)IC5076.420010
3,3',5,5'-tetramethylbenzidineHomo sapiens (human)IC5010.830010
nsc 38280Homo sapiens (human)IC5035.800010
2-amino-7-naphtholHomo sapiens (human)IC5036.720010
harmolHomo sapiens (human)IC5044.910010
2-aminodiphenylamineHomo sapiens (human)IC5036.070010
epicatechinHomo sapiens (human)IC50205.620010
9-methoxyellipticineHomo sapiens (human)IC5028.760010
2,2'-((3,3'-dimethoxy(1,1'-biphenyl)-4,4'-diyl)diimino)bis-benzoic acidHomo sapiens (human)IC5041.420010
1-(10h-phenothiazin-2-yl)ethanoneHomo sapiens (human)IC5031.640010
n,n'-2-phenylenedimaleimideHomo sapiens (human)IC5062.160010
prochlorperazine edisylate saltHomo sapiens (human)IC5080.050010
4-chloro-3-(2,4-dihydroxyphenylazo)-2-hydroxybenzene-1-sulfonic acidHomo sapiens (human)IC5083.740010
n-acetylphenylalanine beta-naphthyl esterHomo sapiens (human)IC5039.710010
homoorientinHomo sapiens (human)IC5040.920010
n-(phenylthio)-epsilon-caprolactamHomo sapiens (human)IC5087.590010
c 1303Homo sapiens (human)IC5062.560010
moracin mHomo sapiens (human)IC5023.000010
2-[4-(4-methoxyphenyl)-1-piperazinyl]pyrimidineHomo sapiens (human)IC5082.850010
equilinHomo sapiens (human)IC5094.560010
4',6-dihydroxy-5,7-dimethoxyflavoneHomo sapiens (human)IC5018.200010
nsc 95397Homo sapiens (human)IC5032.490010
4,7-dimethoxy-2,3-dimethyl-1H-indoleHomo sapiens (human)IC5029.510010
nsc-260594Homo sapiens (human)IC5035.460010
TCMDC-138263Homo sapiens (human)IC5070.190010
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineHomo sapiens (human)IC5063.140010
epipinoresinolHomo sapiens (human)IC50171.320010
4-[4-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]-(3-pyridinyl)methyl]-1-piperazinyl]phenolHomo sapiens (human)IC5039.550010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-(2,6-dimethoxyphenyl)methanoneHomo sapiens (human)IC50248.370010
1-[4-[4-[(phenylmethyl)amino]phenyl]-1-piperazinyl]ethanoneHomo sapiens (human)IC5010.460010
2'-amino-5',6'-dimethoxy-1'-spiro[cyclopentane-1,3'-indene]carbonitrileHomo sapiens (human)IC5037.980010
3-[(4-methoxyanilino)methyl]-1H-quinolin-2-oneHomo sapiens (human)IC5094.720010
(4-chloro-5-hydroxy-3-benzofuranyl)-phenylmethanoneHomo sapiens (human)IC5075.430010
1-(3,4-dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanoneHomo sapiens (human)IC5030.610010
N-(4-anilinophenyl)cyclopropanecarboxamideHomo sapiens (human)IC5050.760010
N-[4-(diethylamino)phenyl]-N'-phenylureaHomo sapiens (human)IC5045.040010
1-[4-(4-aminophenyl)-1-piperazinyl]ethanoneHomo sapiens (human)IC5016.230010
2-(4-hydroxyanilino)-1,4-naphthoquinoneHomo sapiens (human)IC5023.720010
N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)-2-(1-pyrrolidinyl)acetamideHomo sapiens (human)IC50117.270010
N4,N4-dimethyl-N1-(4-nitro-1,1-dioxo-2,5-dihydrothiophen-3-yl)benzene-1,4-diamineHomo sapiens (human)IC5042.730010
N-[(2,3-dimethoxyphenyl)methyl]-4-(4-methyl-1-piperidinyl)anilineHomo sapiens (human)IC507.860010
6-amino-2-mercaptobenzothiazoleHomo sapiens (human)IC5030.430010
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-benzimidazolamineHomo sapiens (human)IC5092.060010
N-(4-anilinophenyl)-2-methylpropanamideHomo sapiens (human)IC5051.100010
3-amino-4-methoxy-1H-indole-2-carbohydrazideHomo sapiens (human)IC5099.390010
4-[2-(3-methoxyanilino)-4-thiazolyl]phenolHomo sapiens (human)IC5066.070010
4-[methyl-(4-thiophen-2-yl-2-thiazolyl)amino]phenolHomo sapiens (human)IC5070.450010
N-[(3-bromo-4,5-diethoxyphenyl)methyl]-4-(4-morpholinyl)anilineHomo sapiens (human)IC5019.590010
4-[[4-bromo-5-(4-morpholinyl)-2-furanyl]methylideneamino]phenolHomo sapiens (human)IC5042.010010
2-(1,3-benzodioxol-5-yl)-N-[(2-ethoxyphenyl)methyl]-N-(2-pyridinylmethyl)ethanamineHomo sapiens (human)IC50172.200010
6-ethyl-2-thieno[2,3-b]quinolinecarboxylic acidHomo sapiens (human)IC50121.980010
4-(4-anilinoanilino)-2-quinazolinecarboxylic acid ethyl esterHomo sapiens (human)IC50104.740010
1-[5-(5-chloro-2-methylphenyl)-2-furanyl]-N-[4-(4-morpholinyl)phenyl]methanimineHomo sapiens (human)IC5011.210010
2-[[5-(3-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneHomo sapiens (human)IC5079.460010
1-(3,4-dihydroxyphenyl)-2-[[5-(3-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneHomo sapiens (human)IC5077.720010
4-(4-chlorophenyl)sulfinyl-6-(methoxymethyl)-2-methylpyrimidineHomo sapiens (human)IC5087.820010
6-fluoro-2-phenyl-1,2-benzothiazol-3-oneHomo sapiens (human)IC5036.430010
4-[4-(3-chlorophenyl)-1-piperazinyl]anilineHomo sapiens (human)IC5021.000010
5-[(6-hydroxy-4-oxo-1-benzopyran-3-yl)methylidene]-1,3-diazinane-2,4,6-trioneHomo sapiens (human)IC50149.650010
N-[(2-furanylmethylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideHomo sapiens (human)IC5052.610010
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneHomo sapiens (human)IC50178.590010
3-[[(2,3-dimethylanilino)-sulfanylidenemethyl]amino]-1H-indole-2-carboxylic acid ethyl esterHomo sapiens (human)IC5095.400010
N-[[(5-hydroxy-1-naphthalenyl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)IC5032.300010
N-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)-2-furancarboxamideHomo sapiens (human)IC50102.440010
5-anilino-3-oxo-4-isothiazolecarbonitrileHomo sapiens (human)IC5079.500010
5-(4-chloroanilino)-3-oxo-4-isothiazolecarbonitrileHomo sapiens (human)IC5079.860010
xanthane hydrideHomo sapiens (human)IC50301.240010
2-(2-furanyl)-4-thiazolidinecarboxylic acidHomo sapiens (human)IC5070.620010
N-(4-anilinophenyl)-3-(hydroxymethyl)-1-piperidinecarbothioamideHomo sapiens (human)IC5041.760010
1-(2,4-dimethoxyphenyl)-3-[4-(4-morpholinyl)anilino]pyrrolidine-2,5-dioneHomo sapiens (human)IC50174.110010
2-(4-anilinophenoxy)acetic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)IC5077.440010
9-methoxy-n(2)-methylellipticinium iodideHomo sapiens (human)IC5024.740010
yl-109Homo sapiens (human)IC5016.150010
2-(4-ethoxy-3-methoxyphenyl)-4-mercapto-3-(4-methoxyphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileHomo sapiens (human)IC50133.680010
4-amino-2-nitrophenolHomo sapiens (human)IC5042.800010
N-[2-chloro-5-[ethyl(phenyl)sulfamoyl]phenyl]-2-[methyl-(1-methyl-4-piperidinyl)amino]acetamideHomo sapiens (human)IC5080.190010
quercetin 3-o-methyl etherHomo sapiens (human)IC5030.340010
kaempferolHomo sapiens (human)IC5044.490010
sulfuretinHomo sapiens (human)IC5020.560010
coumestrolHomo sapiens (human)IC5032.340010
daidzeinHomo sapiens (human)IC5091.260010
rosmarinic acidHomo sapiens (human)IC5035.000010
thunberginol aHomo sapiens (human)IC5019.650010
7,8-dihydroxy-4-methylcoumarinHomo sapiens (human)IC5025.950010
thunberginol bHomo sapiens (human)IC5020.440010
quinaldine redHomo sapiens (human)IC5046.580010
chloride of pseudoisocyanineHomo sapiens (human)IC5046.460010
1,5-anhydro-1-[2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-6-yl]hexitolHomo sapiens (human)IC5042.940010
4-[3-(3-methylanilino)-2-imidazo[1,2-a]pyrimidinyl]phenolHomo sapiens (human)IC5032.110010
1-(2-cyano-3,12-dioxooleana-1,9-dien-28-oyl) imidazoleHomo sapiens (human)IC5020.750010
2-(4-methoxyphenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC5034.450010
2-(4-chlorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC5034.690010
chlorhexidine hydrochlorideHomo sapiens (human)IC5042.330010
2-(3-chlorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC5033.910010
3,6-diamino-10-methylacridinium chloride hydrochlorideHomo sapiens (human)IC5097.470010
5-fluoro-2-phenyl-1,2-benzothiazol-3-oneHomo sapiens (human)IC5035.500010
2-(2-fluorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC5041.000010
2-(4-fluorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC5039.270010
1-[4-[4-(2-furanylmethylamino)phenyl]-1-piperazinyl]ethanoneHomo sapiens (human)IC5014.620010
1-[4-[4-[(3-methylphenyl)methylamino]phenyl]-1-piperazinyl]ethanoneHomo sapiens (human)IC509.890010
1-[4-[4-[(5-bromo-2-furanyl)methylamino]phenyl]-1-piperazinyl]ethanoneHomo sapiens (human)IC5013.740010
2,3-dimethoxy-N-[4-(1-piperidinyl)phenyl]anilineHomo sapiens (human)IC509.650010
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineHomo sapiens (human)IC5069.570010
2-(3-oxo-1,2-benzothiazol-2-yl)-N-phenylacetamideHomo sapiens (human)IC5073.110010
methacycline monohydrochlorideHomo sapiens (human)IC5066.850010