Proteins > Glycoprotein hormones alpha chain
Page last updated: 2024-08-08 00:33:19

Glycoprotein hormones alpha chain

A glycoprotein hormones alpha chain that is encoded in the genome of human. [PRO:DNx, UniProtKB:P01215]

Synonyms

Anterior pituitary glycoprotein hormones common subunit alpha;
Choriogonadotropin alpha chain;
Chorionic gonadotrophin subunit alpha;
CG-alpha;
Follicle-stimulating hormone alpha chain;
FSH-alpha;
Follitropin alpha chain;
Lute

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (913)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ag 1295Homo sapiens (human)Potency2.238710
tyrphostin ag957Homo sapiens (human)Potency10.000010
azinphosmethylHomo sapiens (human)Potency31.622810
carbazilquinoneHomo sapiens (human)Potency3.981110
mitoxantroneHomo sapiens (human)Potency1.122010
pomiferinHomo sapiens (human)Potency11.220210
ppm 18Homo sapiens (human)Potency5.011910
aurinHomo sapiens (human)Potency5.011910
sulfaquinoxalineHomo sapiens (human)Potency28.183810
trifluoperazineHomo sapiens (human)Potency14.125410
trioxsalenHomo sapiens (human)Potency5.011910
methylene blueHomo sapiens (human)Potency0.501210
chlorquinaldolHomo sapiens (human)Potency3.162310
1-phenylazo-2-naphthylamineHomo sapiens (human)Potency28.183810
1-(2-pyridylazo)-2-naphtholHomo sapiens (human)Potency3.981110
salicylanilideHomo sapiens (human)Potency1.258910
pyronineHomo sapiens (human)Potency3.981110
fentichlorHomo sapiens (human)Potency10.000010
triclocarbanHomo sapiens (human)Potency11.220210
2,4-dihydroxybenzophenoneHomo sapiens (human)Potency2.818410
sterogenolHomo sapiens (human)Potency1.000010
5H-dibenzo[b,f]azepineHomo sapiens (human)Potency2.818410
dibromsalicilHomo sapiens (human)Potency28.183810
nitrophenideHomo sapiens (human)Potency28.183810
guaiacol carbonateHomo sapiens (human)Potency5.623410
diphenylamineHomo sapiens (human)Potency5.011910
c 137Homo sapiens (human)Potency1.584910
7-hydroxychlorpromazineHomo sapiens (human)Potency8.912510
fluorenone oximeHomo sapiens (human)Potency28.183810
mofebutazoneHomo sapiens (human)Potency5.623410
2-methoxy-1,4-naphthoquinoneHomo sapiens (human)Potency31.622810
1,3,5-triglycidyl-s-triazinetrioneHomo sapiens (human)Potency1.412510
1,2-benzisothiazoline-3-oneHomo sapiens (human)Potency1.995310
hydroxyphenytoinHomo sapiens (human)Potency12.589310
2-amino-3-chloro-1,4-naphthoquinoneHomo sapiens (human)Potency1.584910
nsc 3852Homo sapiens (human)Potency2.818410
Bis(2-furanylmethyl) disulfideHomo sapiens (human)Potency8.912510
oxycarboxinHomo sapiens (human)Potency22.387210
5-nitroindazoleHomo sapiens (human)Potency1.584910
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineHomo sapiens (human)Potency28.183810
marmesin, (r)-isomerHomo sapiens (human)Potency1.122010
3-methyl-2-quinoxalinolHomo sapiens (human)Potency22.387210
clioxanideHomo sapiens (human)Potency11.220210
n-(cyclohexylthio)phthalimideHomo sapiens (human)Potency31.622810
(7S,9S)-7-[(4-amino-5-hydroxy-6-methyl-2-oxanyl)oxy]-6,9,11-trihydroxy-9-(2-hydroxy-1-oxoethyl)-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dioneHomo sapiens (human)Potency0.316210
N-fluorenylacetamideHomo sapiens (human)Potency5.011910
isovelleralHomo sapiens (human)Potency12.589310
phenicaberanHomo sapiens (human)Potency28.183810
s-2678Homo sapiens (human)Potency6.309610
nsc 330770Homo sapiens (human)Potency14.125410
3-morpholinopropylamineHomo sapiens (human)Potency31.622810
2-Amino-5-(5-nitro-2-furyl)-1,3,4-thiadiazoleHomo sapiens (human)Potency10.000010
5-AminoacenaphtheneHomo sapiens (human)Potency19.952610
diacetylfluoresceinHomo sapiens (human)Potency11.220210
2,2'-dipyridyl disulfideHomo sapiens (human)Potency10.000010
n,n'-bis(salicyl)hydrazineHomo sapiens (human)Potency0.501210
n-acetylsulfamethoxypyridazineHomo sapiens (human)Potency3.981110
4,7-phenanthrolineHomo sapiens (human)Potency2.818410
dibenzthioneHomo sapiens (human)Potency0.446710
harmolHomo sapiens (human)Potency1.584910
oxiperomideHomo sapiens (human)Potency10.000010
1,2-bis(phenylsulfonyl)ethaneHomo sapiens (human)Potency7.943310
norcyclizineHomo sapiens (human)Potency4.466810
4-Formyl-antipyrineHomo sapiens (human)Potency0.631010
morphazinamideHomo sapiens (human)Potency4.466810
2,2',2''-terpyridineHomo sapiens (human)Potency10.000010
propipocaine monohydrochlorideHomo sapiens (human)Potency31.622810
9-methoxyellipticineHomo sapiens (human)Potency31.622810
2,2'-((3,3'-dimethoxy(1,1'-biphenyl)-4,4'-diyl)diimino)bis-benzoic acidHomo sapiens (human)Potency11.220210
coumarin 153Homo sapiens (human)Potency28.183810
methyl fluorone blackHomo sapiens (human)Potency28.183810
3-aminophenoxazoneHomo sapiens (human)Potency28.183810
2-phenyl-4,5-dichloro-3-pyridazinoneHomo sapiens (human)Potency2.511910
centazoloneHomo sapiens (human)Potency1.778310
methylene violetHomo sapiens (human)Potency10.000010
8-hydroxy-2-quinolinecarboxylic acidHomo sapiens (human)Potency5.623410
1-ethyl-2-benzo[cd]indoloneHomo sapiens (human)Potency28.183810
2-Amino-6-(benzylthio)purineHomo sapiens (human)Potency4.466810
7-bromo-5-phenyl-1,2-dihydro-2h-1,4-benzodiazepin-2-oneHomo sapiens (human)Potency3.981110
3,5-di-tert-butyl-1,2-benzoquinoneHomo sapiens (human)Potency1.258910
1-methyl-2-phenylindoleHomo sapiens (human)Potency1.000010
2-methyl-4-nitroquinoline 1-oxideHomo sapiens (human)Potency0.891310
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)Potency4.466810
n,n'-2-phenylenedimaleimideHomo sapiens (human)Potency11.220210
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dioneHomo sapiens (human)Potency11.220210
5-bromonicotinic acidHomo sapiens (human)Potency5.011910
5-benzyloxytryptamineHomo sapiens (human)Potency28.183810
streptovitacin aHomo sapiens (human)Potency0.501210
pyridabenHomo sapiens (human)Potency1.122010
coumarin 7Homo sapiens (human)Potency2.238710
1-piperonylpiperazineHomo sapiens (human)Potency28.183810
osajinHomo sapiens (human)Potency28.183810
9,10-phenanthrenequinone monoximeHomo sapiens (human)Potency5.623410
2-nitrobenzimidazoleHomo sapiens (human)Potency5.011910
1,3-diphenyl-2-propyn-1-oneHomo sapiens (human)Potency12.589310
3,3'-DihydroxyhexestrolHomo sapiens (human)Potency11.220210
wr 158122Homo sapiens (human)Potency1.000010
n-acetylphenylalanyl-phenylalanineHomo sapiens (human)Potency0.501210
difenpiramideHomo sapiens (human)Potency28.183810
diphyllinHomo sapiens (human)Potency5.011910
karanjinHomo sapiens (human)Potency17.782810
tanshinoneHomo sapiens (human)Potency5.011910
pirlindole hydrochlorideHomo sapiens (human)Potency7.943310
3-(1-piperidinyl)-1-(4-propan-2-yloxyphenyl)-1-propanoneHomo sapiens (human)Potency11.220210
1,3-dimethylbenzimidazoline-2-thioneHomo sapiens (human)Potency14.125410
3'-deamino-3'-hydroxydaunorubicinHomo sapiens (human)Potency3.162310
ly 188544Homo sapiens (human)Potency1.584910
omeprazole magnesiumHomo sapiens (human)Potency2.238710
n-(6-methoxy-8-quinolyl)-4-toluenesulfonamideHomo sapiens (human)Potency1.778310
umifenovirHomo sapiens (human)Potency28.183810
1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)-1-propanoneHomo sapiens (human)Potency5.623410
4,5-diphenyl-4-oxazolin-2-oneHomo sapiens (human)Potency5.011910
8-(methylsulfonylamino)quinolineHomo sapiens (human)Potency3.162310
1,4-di(2'-thienyl)-1,4-butadioneHomo sapiens (human)Potency14.125410
sch 45752Homo sapiens (human)Potency28.183810
2-chloroacetoacetanilideHomo sapiens (human)Potency28.183810
2-methyl-4-(phenylimino)naphth(2,3-d)oxazol-9-oneHomo sapiens (human)Potency1.412510
8-(4-benzenesulfonylamino)quinolineHomo sapiens (human)Potency12.589310
3,3-bis(4-hydroxy-3-methylphenyl)-1H-indol-2-oneHomo sapiens (human)Potency28.183810
2,4-dinitropyrimidinyl-2-thiophenolHomo sapiens (human)Potency3.162310
enniatin bHomo sapiens (human)Potency8.912510
2-phenyl-1,2-benzisothiazol-3-(2h)-oneHomo sapiens (human)Potency7.079510
4-butyl-4-(hydroxymethyl)-1,2-diphenylpyrazolidine-3,5-dioneHomo sapiens (human)Potency5.011910
2-(1,1,2,2-tetrafluoroethyl)benzimidazoleHomo sapiens (human)Potency3.162310
4-methoxy-1-vinylcarbolineHomo sapiens (human)Potency19.952610
2-[4-(4-methoxyphenyl)-1-piperazinyl]pyrimidineHomo sapiens (human)Potency28.183810
PhthalyltyrosineHomo sapiens (human)Potency5.011910
3-nitrotyrosineHomo sapiens (human)Potency3.548110
benzatropine methanesulfonateHomo sapiens (human)Potency28.183810
1',2'-dihydrorotenoneHomo sapiens (human)Potency4.466810
2-methyl-3-(phenylthio)pyrazineHomo sapiens (human)Potency2.818410
gant58Homo sapiens (human)Potency5.623410
coronopilinHomo sapiens (human)Potency0.891310
1,5-bis(2-methoxyphenyl)penta-1,4-dien-3-oneHomo sapiens (human)Potency2.238710
2-chloro-3-(4-methylanilino)naphthalene-1,4-dioneHomo sapiens (human)Potency8.912510
4-amino-1,2-dithiolane-4-carboxylic acidHomo sapiens (human)Potency1.995310
papaverinolHomo sapiens (human)Potency31.622810
dimethyl 2-(2-nitrobenzylidene)malonateHomo sapiens (human)Potency8.912510
nsc 154020Homo sapiens (human)Potency0.891310
4-chloro-1H-indazol-3-amineHomo sapiens (human)Potency28.183810
nsc228155Homo sapiens (human)Potency0.891310
2,2-bis(hydroxymethyl)-1-azabicyclo(2,2,2,)octan-3-oneHomo sapiens (human)Potency28.183810
CadabiciloneHomo sapiens (human)Potency7.943310
mitonafideHomo sapiens (human)Potency1.412510
pinafideHomo sapiens (human)Potency0.501210
rocaglamideHomo sapiens (human)Potency2.511910
2-[(4,4-dimethyl-2,6-dioxocyclohexyl)methyl]-5,5-dimethylcyclohexane-1,3-dioneHomo sapiens (human)Potency11.220210
6-dimethylaminopurine arabinosideHomo sapiens (human)Potency1.122010
nsc606985Homo sapiens (human)Potency0.446710
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneHomo sapiens (human)Potency0.501210
nsc668394Homo sapiens (human)Potency3.981110
nsc 680410Homo sapiens (human)Potency3.548110
nsc681152Homo sapiens (human)Potency7.943310
5,7-dimethoxy-4-methyl-1-benzopyran-2-oneHomo sapiens (human)Potency11.220210
nsc689857Homo sapiens (human)Potency4.466810
nsc697923Homo sapiens (human)Potency2.818410
4-(4-chlorophenyl)-1-methyl-2-(methylthio)-6-oxo-5-pyrimidinecarbonitrileHomo sapiens (human)Potency28.183810
nsc-134754Homo sapiens (human)Potency3.548110
N-[2-(dimethylamino)ethyl]-2,2-diphenylacetamideHomo sapiens (human)Potency5.011910
Destruxin BHomo sapiens (human)Potency1.412510
macbecin iiHomo sapiens (human)Potency5.623410
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency0.316210
6,8-diprenylgenisteinHomo sapiens (human)Potency28.183810
9,14-Dimethyl-5-methylidene-3,13-dioxatetracyclo[8.4.0.02,6.012,14]tetradec-9-ene-4,11-dioneHomo sapiens (human)Potency28.183810
2-sulfanylidene-1,3-dithiole-4,5-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency5.623410
2-chloro-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency1.000010
2-(2-phenoxyethylsulfonyl)-1H-benzimidazoleHomo sapiens (human)Potency2.238710
LSM-22807Homo sapiens (human)Potency11.220210
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineHomo sapiens (human)Potency10.000010
2-chlorothioxanthen-9-oneHomo sapiens (human)Potency5.011910
dibenzylidene acetoneHomo sapiens (human)Potency22.387210
cgp 60474Homo sapiens (human)Potency1.995310
2-(4-chlorophenoxy)-N-(2-pyridin-4-yl-1,3-benzoxazol-5-yl)acetamideHomo sapiens (human)Potency3.981110
4-(4-fluorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid 1,3-benzodioxol-5-ylmethyl esterHomo sapiens (human)Potency0.446710
7,8-dimethyl-1-[2-oxo-2-(1-pyrrolidinyl)ethyl]-4-phenyl-3H-1,5-benzodiazepin-2-oneHomo sapiens (human)Potency28.183810
3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazoleHomo sapiens (human)Potency3.548110
3-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclopentyl-5-tetrazolyl)methyl]amino]methyl]-6-ethyl-1H-quinolin-2-oneHomo sapiens (human)Potency28.183810
1-(3-chloro-4-methoxyphenyl)sulfonyl-N-(3-pyridinyl)-3-piperidinecarboxamideHomo sapiens (human)Potency10.000010
2-(4-bromophenyl)-5-(2-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency5.011910
5-(4-propylcyclohexyl)-3-(3-pyridinyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency4.466810
N-[2-[1,3-benzodioxol-5-yl-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-furancarboxamideHomo sapiens (human)Potency28.183810
N-[4-[4-[[1-oxo-2-(1-pyrrolidinyl)ethyl]amino]phenoxy]phenyl]-2-(1-pyrrolidinyl)acetamideHomo sapiens (human)Potency5.623410
N-tert-butyl-N-[2-(tert-butylamino)-2-oxoethyl]-3-(3,4-dihydro-2H-quinolin-1-yl)propanamideHomo sapiens (human)Potency5.011910
4-[4-[(5,6-dimethyl-1-benzimidazolyl)sulfonyl]phenyl]sulfonylmorpholineHomo sapiens (human)Potency4.466810
2-methoxy-N-(5-thiophen-2-yl-1,3,4-thiadiazol-2-yl)acetamideHomo sapiens (human)Potency11.220210
N-[1-[2-(2-chlorophenoxy)ethyl]-2-benzimidazolyl]acetamideHomo sapiens (human)Potency11.220210
N-[4-[(tert-butylamino)-oxomethyl]phenyl]-2,3-dihydro-1,4-benzodioxin-3-carboxamideHomo sapiens (human)Potency1.258910
3-(2,5-dimethyl-1-pyrrolyl)-4-methylanilineHomo sapiens (human)Potency10.000010
4-[[[[8-[(1-tert-butyl-5-tetrazolyl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]amino]-oxomethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency12.589310
N-(4-methylphenyl)-2-(3-oxo-5,6-dihydroimidazo[2,1-b]thiazol-2-yl)acetamideHomo sapiens (human)Potency19.952610
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency11.220210
1-[4-(2-methoxyphenyl)-1-piperazinyl]-2-[[5-(2-methyl-3-furanyl)-1,3,4-oxadiazol-2-yl]thio]ethanoneHomo sapiens (human)Potency28.183810
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[(2-hydroxyphenyl)methyl]-4-piperidinecarboxamideHomo sapiens (human)Potency8.912510
2-methoxy-N-methyl-N-[5-(5-methyl-2-pyrazinyl)-1,3,4-thiadiazol-2-yl]acetamideHomo sapiens (human)Potency15.848910
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency0.707910
2-[2-[[2-[[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterHomo sapiens (human)Potency11.220210
[4-[5-tert-butyl-3-[(2-chlorophenyl)methyl]-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency28.183810
N-[2-[2-[2-(4-methoxyanilino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency11.220210
9-oxo-N-(3-pyridinylmethyl)-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinoline-8-carboxamideHomo sapiens (human)Potency2.238710
(6-fluoro-2-methyl-3,4-dihydro-2H-quinolin-1-yl)-[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]methanoneHomo sapiens (human)Potency22.387210
5-[(2-fluoroanilino)methyl]-8-quinolinolHomo sapiens (human)Potency1.995310
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-2-methoxyphenolHomo sapiens (human)Potency14.125410
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideHomo sapiens (human)Potency28.183810
1-cyclohexyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-amineHomo sapiens (human)Potency28.183810
2'-amino-5',6'-dimethoxy-1'-spiro[cyclopentane-1,3'-indene]carbonitrileHomo sapiens (human)Potency4.466810
3-(4-butyl-3,5-dimethyl-1-pyrazolyl)-5-methyl-[1,2,4]triazino[5,6-b]indoleHomo sapiens (human)Potency2.511910
6-amino-4-(5-bromo-2-thiophenyl)-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileHomo sapiens (human)Potency14.125410
5-bromo-3-[[2-(4-cyclohexyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency3.548110
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideHomo sapiens (human)Potency2.818410
3-(5-cycloheptylidene-4-oxo-2-sulfanylidene-3-thiazolidinyl)propanoic acidHomo sapiens (human)Potency10.000010
1-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency31.622810
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency3.548110
2-(2-oxo-3H-1,4-benzoxazin-4-yl)acetic acid [2-(3-bromo-4-methoxyphenyl)-2-oxoethyl] esterHomo sapiens (human)Potency0.316210
2-[[5-cyano-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,3-thiazin-6-yl]thio]acetic acid ethyl esterHomo sapiens (human)Potency12.589310
1-(4-chlorophenyl)-N-(1-methoxypropan-2-yl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency5.011910
3-benzamido-5-bromo-2-benzofurancarboxylic acid methyl esterHomo sapiens (human)Potency3.548110
5-(2,4-dimethoxyphenyl)-7-(3,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency15.848910
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.000010
N-[3-(2-furanylmethylamino)-2-quinoxalinyl]-3-methylbenzenesulfonamideHomo sapiens (human)Potency5.011910
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneHomo sapiens (human)Potency8.912510
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterHomo sapiens (human)Potency31.622810
2-[(2,5-dimethyl-3-phenyl-7-pyrazolo[1,5-a]pyrimidinyl)thio]acetonitrileHomo sapiens (human)Potency8.912510
6-(3,4,5-triethoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency12.589310
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileHomo sapiens (human)Potency12.589310
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-bis(phenylmethyl)-2,4-dihydro-1,3,5-triazin-6-amineHomo sapiens (human)Potency6.309610
7-(3,4-dimethoxyphenyl)-4-methyl-2-[4-(phenylmethyl)-1-piperazinyl]-7,8-dihydro-6H-quinazolin-5-oneHomo sapiens (human)Potency10.000010
N-(3,4-dihydro-1H-[1,4]thiazino[4,3-a]benzimidazol-8-yl)pentanamideHomo sapiens (human)Potency5.011910
LSM-20899Homo sapiens (human)Potency14.125410
3,4,7-trimethyl-5-(3-oxobutan-2-yloxy)-1-benzopyran-2-oneHomo sapiens (human)Potency11.220210
4-(3-amino-2-imidazo[1,2-a]pyridinyl)-2-methoxyphenolHomo sapiens (human)Potency5.011910
N-(2-furanylmethyl)-4-(2-methyl-3-imidazo[1,2-a]pyridinyl)-2-thiazolamineHomo sapiens (human)Potency10.000010
2,6-dimethyl-N-(4-methylphenyl)-4-quinolinamineHomo sapiens (human)Potency3.548110
2-[(4-chloro-2-methylphenoxy)methyl]imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency1.995310
1-(2,4-dimethylphenyl)-4-(1-piperidinylsulfonyl)piperazineHomo sapiens (human)Potency5.011910
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency3.548110
N1-(6-bromo-4-quinazolinyl)-N4,N4-dimethylbenzene-1,4-diamineHomo sapiens (human)Potency10.000010
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency5.011910
2-mercaptobenzimidazoleHomo sapiens (human)Potency11.220210
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(4-oxo-3-quinazolinyl)acetamideHomo sapiens (human)Potency22.387210
2-methoxy-6-[[(1-methyl-2-benzimidazolyl)amino]methyl]phenolHomo sapiens (human)Potency3.548110
2-(3-oxo-2-phenyl-1H-pyrazol-5-yl)acetic acid methyl esterHomo sapiens (human)Potency3.981110
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileHomo sapiens (human)Potency31.622810
bemethylHomo sapiens (human)Potency2.818410
5-cyano-2-methyl-6-sulfanylidene-1H-pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency11.220210
1-cyclohexyl-3-[[oxo(thiophen-2-yl)methyl]amino]thioureaHomo sapiens (human)Potency28.183810
4,5-dimethylaminobenzylidene-2-thiobarbituric acidHomo sapiens (human)Potency12.589310
1-(4-chlorophenyl)-3-(4-sulfamoylphenyl)ureaHomo sapiens (human)Potency10.000010
N-[4-(diethylamino)phenyl]-N'-phenylureaHomo sapiens (human)Potency5.623410
N-[4-(4-ethylphenyl)-2-thiazolyl]carbamic acid phenyl esterHomo sapiens (human)Potency0.891310
1-benzoyl-4-phenyl-3-thiosemicarbazideHomo sapiens (human)Potency28.183810
2,4-Dimethyl-1,3-thiazole-5-carboxylic acidHomo sapiens (human)Potency3.981110
2-(4-hydroxyanilino)-1,4-naphthoquinoneHomo sapiens (human)Potency11.220210
1-(3,5-dichlorophenyl)-3-phenylureaHomo sapiens (human)Potency12.589310
3-(2,4-dioxo-6-methyl-5-pyrimidinyl)acrylic acidHomo sapiens (human)Potency5.011910
5,6-dimethyl-2-[2-(1-pyrrolidinyl)ethylthio]-1H-benzimidazoleHomo sapiens (human)Potency1.995310
nsc185058Homo sapiens (human)Potency14.125410
2-fluoro-N-phenacylbenzamideHomo sapiens (human)Potency17.782810
1-(3-pyridinylmethyl)-3-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]ureaHomo sapiens (human)Potency2.818410
3-(2,3-dimethyl-1H-indol-5-yl)-4-methyl-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency14.125410
2-(1,3-benzothiazol-2-ylmethoxy)phenolHomo sapiens (human)Potency5.011910
3-(8-methyl-2-imidazo[1,2-a]pyridinyl)-1-benzopyran-2-oneHomo sapiens (human)Potency31.622810
2-[[2-(5,6-dimethyl-1-benzimidazolyl)-1-oxoethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency7.079510
3-chloro-1-(3,4-dichlorophenyl)-4-(dimethylamino)pyrrole-2,5-dioneHomo sapiens (human)Potency5.011910
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-oneHomo sapiens (human)Potency7.943310
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazineHomo sapiens (human)Potency3.162310
1-spiro[2,4-dihydroisoquinoline-3,1'-cyclohexane]thioneHomo sapiens (human)Potency1.122010
4-(2-naphthalenylmethyl)-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency5.011910
4-tert-butyl-N-[2-(2-methoxyphenyl)ethyl]-1-cyclohexanamineHomo sapiens (human)Potency12.589310
N-(1-acetyl-2-chloro-3-indolyl)-2-chloroacetamideHomo sapiens (human)Potency0.501210
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-5-nitro-2-furancarboxamideHomo sapiens (human)Potency1.122010
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileHomo sapiens (human)Potency12.589310
N-[4-(1-azepanyl)phenyl]-2-chloroacetamideHomo sapiens (human)Potency1.412510
[4-(2-methylphenyl)-1-piperazinyl]-(4-nitrophenyl)methanethioneHomo sapiens (human)Potency14.125410
4-chloro-1-ethyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency5.011910
3-(3-nitrophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency3.162310
2,5-dimethyl-1-(phenylmethyl)pyrrole-3,4-dicarboxaldehydeHomo sapiens (human)Potency3.548110
3-(4-methoxyphenyl)-1H-pyrazole-5-carbohydrazideHomo sapiens (human)Potency0.794310
9-oxo-3-fluorenecarboxylic acid (phenylmethyl) esterHomo sapiens (human)Potency22.387210
1-(4-bromophenyl)-3-(2-phenylethyl)thioureaHomo sapiens (human)Potency8.912510
N-(1,3-benzothiazol-2-yl)-2-cyclohexylacetamideHomo sapiens (human)Potency14.125410
5-(3-chloro-4-methylphenyl)-3-pyridin-4-yl-1,2,4-oxadiazoleHomo sapiens (human)Potency0.501210
N-(4-fluorophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamideHomo sapiens (human)Potency31.622810
3-prop-2-enyl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency28.183810
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneHomo sapiens (human)Potency7.079510
7,8-dimethoxy-1,5-dimethyl-3-phenylpyrazolo[3,4-c]isoquinolineHomo sapiens (human)Potency5.011910
N-methyl-2-(4-methylphenyl)-N-(1-methylpiperidin-4-yl)quinazolin-4-amineHomo sapiens (human)Potency3.981110
N-[[(6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-4-phenylbenzamideHomo sapiens (human)Potency0.316210
N-(6-methyl-2-pyridinyl)-5-nitro-2-furancarboxamideHomo sapiens (human)Potency14.125410
1-(3-chlorophenyl)-3-(phenylmethyl)thioureaHomo sapiens (human)Potency7.943310
N-(3-phenyl-1,3-benzothiazol-2-ylidene)-2-propenamideHomo sapiens (human)Potency7.943310
2-[[4-(1-pyrrolidinylsulfonyl)phenyl]hydrazinylidene]propanedinitrileHomo sapiens (human)Potency11.220210
N-[3,4-dihydro-2H-quinolin-1-yl(sulfanylidene)methyl]-2-(3-methylphenoxy)acetamideHomo sapiens (human)Potency1.412510
N-[(2,3-dimethoxyphenyl)methyl]-4-(4-methyl-1-piperidinyl)anilineHomo sapiens (human)Potency8.912510
4-phenyl-N-(2-pyridinyl)butanamideHomo sapiens (human)Potency3.162310
3-[[(3-chloro-4-ethoxyphenyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency10.000010
N-(4-methyl-2-pyridinyl)-5-nitro-2-furancarboxamideHomo sapiens (human)Potency5.623410
2-methoxy-3-methyl-N-[4-(4-morpholinylmethyl)phenyl]benzamideHomo sapiens (human)Potency1.412510
2-chloro-N-[5-ethyl-3-[(4-methylphenyl)-oxomethyl]-2-thiophenyl]acetamideHomo sapiens (human)Potency3.981110
1-(2-methyl-6-propan-2-ylphenyl)-5-phenyltetrazoleHomo sapiens (human)Potency11.220210
5-(4-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamideHomo sapiens (human)Potency19.952610
N-(2-cyano-1-cyclopentenyl)-1-ethyl-3-pyrazolecarboxamideHomo sapiens (human)Potency5.011910
N-[(2-methoxyphenyl)methyl]-4-(1-piperidinyl)anilineHomo sapiens (human)Potency12.589310
N-(5-acetyl-4-methyl-2-thiazolyl)-5-bromo-2-furancarboxamideHomo sapiens (human)Potency1.412510
2-(2-methylphenoxy)-N-[2-(methylthio)phenyl]acetamideHomo sapiens (human)Potency5.011910
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency11.220210
2-methyl-4-phenyl-1H-pyrrole-3-carboxylic acid methyl esterHomo sapiens (human)Potency10.000010
2-(4-chlorophenyl)-4-propan-2-yloxyquinazolineHomo sapiens (human)Potency7.943310
N2-(4-fluorophenyl)-6-(3-methyl-2-benzofuranyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency6.309610
1-(4-methylphenyl)sulfonyl-4-phenyl-3-pyrazolamineHomo sapiens (human)Potency5.011910
5-hydroxy-7-(4-nitrophenyl)-1,3-benzoxathiol-2-oneHomo sapiens (human)Potency1.000010
3-[4-(2-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]-1H-pyridazin-6-oneHomo sapiens (human)Potency22.387210
1-methyl-5-(1-naphthalenyloxy)-4-nitroimidazoleHomo sapiens (human)Potency10.000010
3-[[(3-acetylanilino)-oxomethyl]amino]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency28.183810
N-(1,3-benzodioxol-5-yl)-4-(2-furanylmethyl)-1-piperazinecarbothioamideHomo sapiens (human)Potency5.011910
1-(4-acetylphenyl)-3-[2-(4-fluorophenyl)ethyl]thioureaHomo sapiens (human)Potency28.183810
6-hydroxy-2-(4-nitrophenyl)-3,1-benzoxazin-4-oneHomo sapiens (human)Potency5.011910
3-chloro-4-[(1-ethyl-2-benzimidazolyl)thio]anilineHomo sapiens (human)Potency2.818410
(2,3-dimethoxyphenyl)-(1-pyrrolidinyl)methanethioneHomo sapiens (human)Potency0.316210
1-(1-pyrrolidinyl)-2-(8-quinolinylthio)ethanoneHomo sapiens (human)Potency3.981110
1-[tert-butyl-[(3,5-dimethylphenyl)-oxomethyl]amino]-3-(4-chlorophenyl)ureaHomo sapiens (human)Potency14.125410
5-(4-bromophenyl)-N-[[(2-propyl-5-tetrazolyl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency5.011910
N-[3-chloro-2-(4-morpholinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency8.912510
6-chloro-4-phenyl-3-(1-phenyl-5-tetrazolyl)quinolineHomo sapiens (human)Potency12.589310
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency1.995310
1-(2,1,3-benzothiadiazol-5-yl)-3-[4-(4-morpholinyl)phenyl]ureaHomo sapiens (human)Potency5.011910
N-(1-tert-butyl-5-benzimidazolyl)-3,4,5-trimethoxybenzamideHomo sapiens (human)Potency28.183810
2-[[cyclohexyl(oxo)methyl]amino]-1,3-benzothiazole-6-carboxylic acid methyl esterHomo sapiens (human)Potency5.011910
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideHomo sapiens (human)Potency28.183810
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency10.000010
6-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]-N2-(4-methoxyphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency10.000010
N-[4-[(3,4-dimethoxyphenyl)sulfamoyl]phenyl]acetamideHomo sapiens (human)Potency25.118910
N'-methyl-N-[1-methyl-5-(4-methylphenyl)-2-imidazolyl]-N'-(phenylmethyl)butanediamideHomo sapiens (human)Potency10.000010
N2,N7-bis(2,5-dimethylphenyl)-9H-fluorene-2,7-disulfonamideHomo sapiens (human)Potency28.183810
LSM-16285Homo sapiens (human)Potency11.220210
5-nitro-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency1.778310
2-(3,4-dimethoxyphenyl)-8-methoxy-4,4-dimethyl-5H-isothiazolo[5,4-c]quinoline-1-thioneHomo sapiens (human)Potency1.778310
[4-(diphenylmethyl)-1-piperazinyl]-[5-thiophen-2-yl-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinyl]methanoneHomo sapiens (human)Potency5.011910
N-(4-Methoxybenzoyl)-2-{[4-methyl-5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}ethanehydrazonic acidHomo sapiens (human)Potency3.548110
3-[[2-[[6-fluoro-2-(4-fluorophenyl)-4-quinazolinyl]thio]-1-oxoethyl]amino]benzoic acidHomo sapiens (human)Potency2.818410
4,5-dimethoxy-2-[[1-oxo-2-[(3,5,8-trimethyl-2-quinolinyl)thio]ethyl]amino]benzoic acidHomo sapiens (human)Potency28.183810
3-pyridinecarboxylic acid [2-(2-furanyl)-4-oxo-1-benzopyran-3-yl] esterHomo sapiens (human)Potency7.079510
2-(4-methylphenyl)-N-[4-(4-morpholinyl)phenyl]-4-quinazolinamineHomo sapiens (human)Potency28.183810
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterHomo sapiens (human)Potency2.511910
5-(3,4-dimethoxyphenyl)-2-(4-methylphenyl)-4-thieno[2,3-d][1,3]oxazinoneHomo sapiens (human)Potency5.011910
9-(dimethylamino)-3-(4-methoxyphenyl)-4-pyrido[1,2]thieno[3,4-d]pyrimidinoneHomo sapiens (human)Potency31.622810
5-(4-fluorophenyl)sulfonyl-1-(2-methylpropyl)-4-nitro-2-propan-2-ylimidazoleHomo sapiens (human)Potency6.309610
N-[(4-ethylanilino)-sulfanylidenemethyl]-3-methylbutanamideHomo sapiens (human)Potency5.011910
N-(5-chloro-2-pyridinyl)-2-(3,5-dimethyl-4-nitro-1-pyrazolyl)acetamideHomo sapiens (human)Potency31.622810
5-methyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-isoxazolecarboxamideHomo sapiens (human)Potency7.079510
5-bromo-N-[2-(4-chlorophenyl)ethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency14.125410
N-[2-methoxy-5-(2-oxo-1-benzopyran-3-yl)phenyl]-5-nitro-2-furancarboxamideHomo sapiens (human)Potency1.000010
8-methoxy-6-nitro-3-[oxo-(2-phenyl-4,5-dihydroimidazol-1-yl)methyl]-1-benzopyran-2-oneHomo sapiens (human)Potency2.818410
2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(2-pyridinyl)acetamideHomo sapiens (human)Potency12.589310
N-(3,5-dichlorophenyl)-2-(methanesulfonamido)benzamideHomo sapiens (human)Potency14.125410
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(3-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency2.238710
[4-[(2-chlorophenyl)methyl]-1-piperazinyl]-(6,8-dimethyl-2-pyridin-4-yl-4-quinolinyl)methanoneHomo sapiens (human)Potency11.220210
N-(4-hydroxy-3,5-dimethylphenyl)-2,5-dimethyl-3-thiophenesulfonamideHomo sapiens (human)Potency28.183810
N-(2,4-dimethoxyphenyl)-2-(1-pyrrolidinyl)-4-quinazolinamineHomo sapiens (human)Potency22.387210
4-(2-methoxyphenoxy)-N-(3-pyridinyl)benzenesulfonamideHomo sapiens (human)Potency0.891310
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineHomo sapiens (human)Potency28.183810
4-methoxy-N-[2-[(4-nitrophenyl)methylthio]-4-oxo-3-quinazolinyl]benzamideHomo sapiens (human)Potency28.183810
2-(4-methoxyphenyl)-N-[4-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideHomo sapiens (human)Potency5.011910
N-(4-fluorophenyl)-3-([1,2,4]triazolo[4,3-a]quinolin-1-ylthio)propanamideHomo sapiens (human)Potency2.238710
3-[[2-[[4-ethyl-5-[(3-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]benzoic acidHomo sapiens (human)Potency14.125410
9-(3-bromo-4-hydroxyphenyl)-10-phenyl-3,4,5,6,7,9-hexahydro-2H-acridine-1,8-dioneHomo sapiens (human)Potency5.011910
2-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-N-(diphenylmethyl)acetamideHomo sapiens (human)Potency7.943310
8,9-dimethyl-N-(3-methylphenyl)-3-[2-(4-morpholinyl)ethyl]-4H-[1,3]thiazino[6,5-b]quinolin-2-imineHomo sapiens (human)Potency14.125410
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency8.912510
2-[(2-propyl-4-quinazolinyl)thio]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)Potency28.183810
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneHomo sapiens (human)Potency28.183810
3-amino-8-methyl-N-[4-(4-morpholinyl)phenyl]-2-thieno[2,3-b]quinolinecarboxamideHomo sapiens (human)Potency28.183810
N-(5-methyl-3-isoxazolyl)-2-[(2-propan-2-yl-4-quinazolinyl)thio]acetamideHomo sapiens (human)Potency7.079510
5-tert-butyl-N-[2-(cyclopentylamino)-2-oxoethyl]-N-(2,5-dimethylphenyl)-3-methyl-2-furancarboxamideHomo sapiens (human)Potency28.183810
4-tert-butyl-N-[2,5-dimethoxy-4-[[1-oxo-2-(1-piperidinyl)ethyl]amino]phenyl]benzamideHomo sapiens (human)Potency28.183810
4-chloro-N-(4-chloro-2-methylphenyl)-5-dithiazolimineHomo sapiens (human)Potency31.622810
2,5-dichloro-N-(1,5,6-trimethyl-4-benzimidazolyl)benzenesulfonamideHomo sapiens (human)Potency0.316210
4-[(3-methylphenyl)thio]-2-phenyl-5-pyrimidinecarboxylic acidHomo sapiens (human)Potency12.589310
4-(2-quinoxalinylamino)benzoic acid ethyl esterHomo sapiens (human)Potency28.183810
1-[[[1-(6-methyl-2-pyridinyl)-4-imidazolyl]-oxomethyl]amino]-3-phenylthioureaHomo sapiens (human)Potency12.589310
1,1-bis(4-chlorophenyl)-2-[(3-methoxyphenyl)methylamino]ethanolHomo sapiens (human)Potency28.183810
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.548110
2-(3,5-dimethyl-4-nitro-1-pyrazolyl)-N-[(2-methyl-4-quinolinyl)methyl]acetamideHomo sapiens (human)Potency12.589310
3-[(4-ethylsulfonyl-2-nitrophenyl)thio]-4-methyl-1,2,4-triazoleHomo sapiens (human)Potency10.000010
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency2.511910
4-chloro-N-(3,4-dimethoxyphenyl)-1-ethyl-3-pyrazolecarboxamideHomo sapiens (human)Potency28.183810
5-[(4-methyl-1-piperidinyl)methyl]-1-[4-(1-pyrrolyl)-1,2,5-oxadiazol-3-yl]-4-triazolecarboxylic acid ethyl esterHomo sapiens (human)Potency7.943310
2-chloro-1-[1-(2-furanylmethyl)-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)Potency10.000010
N-[2-[(phenylmethyl)amino]-1,3-benzodioxol-2-yl]carbamic acid ethyl esterHomo sapiens (human)Potency10.000010
2-[(4-cyano-1-methyl-5,6,7,8-tetrahydroisoquinolin-3-yl)thio]-N-(3-ethoxyphenyl)acetamideHomo sapiens (human)Potency10.000010
11-[2-(diethylamino)ethylamino]-7,8,9,10-tetrahydrobenzimidazolo[1,2-b]isoquinoline-6-carbonitrileHomo sapiens (human)Potency28.183810
N-(4-methoxyphenyl)-2-(3-methylphenoxy)-N-(4-methylphenyl)sulfonylacetamideHomo sapiens (human)Potency19.952610
cyqualonHomo sapiens (human)Potency11.220210
1-amino-3-[3-(2-sulfanylidene-3H-1,3,4-oxadiazol-5-yl)phenyl]thioureaHomo sapiens (human)Potency10.000010
2-chloro-N-heptyl-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency3.162310
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneHomo sapiens (human)Potency5.623410
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideHomo sapiens (human)Potency19.952610
5-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxymethyl]-2-furancarboxylic acidHomo sapiens (human)Potency28.183810
N-cyano-N'-(2-fluorophenyl)carbamimidothioic acid [2-(tert-butylamino)-2-oxoethyl] esterHomo sapiens (human)Potency10.000010
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(3,4-dimethoxyphenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency2.818410
N-(5-chloro-2-methoxyphenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineHomo sapiens (human)Potency1.995310
5-bromo-3-[[3-(3,3-dimethyl-1-piperidinyl)-1-oxopropyl]amino]-1H-indole-2-carboxylic acid ethyl esterHomo sapiens (human)Potency14.125410
N-[[(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideHomo sapiens (human)Potency2.818410
N-bis(2-fluorophenoxy)phosphoryl-3,4-dimethylanilineHomo sapiens (human)Potency0.501210
2-[6-bromo-4-(2-chlorophenyl)-2-oxo-1H-quinolin-3-yl]acetic acidHomo sapiens (human)Potency0.446710
2-[5-(4-chlorophenyl)-1,3,5-dithiazinan-2-ylidene]-2-diethoxyphosphorylacetonitrileHomo sapiens (human)Potency11.220210
LSM-20401Homo sapiens (human)Potency28.183810
5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineHomo sapiens (human)Potency11.220210
6-(2-chloro-1-oxoethyl)-3H-1,3-benzoxazol-2-oneHomo sapiens (human)Potency7.079510
N,N-dimethyl-3-[(2-phenyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)thio]-1-propanamineHomo sapiens (human)Potency28.183810
N-[2-(3,4-dimethoxyphenyl)ethyl]-8-ethoxy-5H-pyrimido[5,4-b]indol-4-amineHomo sapiens (human)Potency1.000010
1-[1-naphthalenyl(oxo)methyl]-3-indolecarboxylic acid methyl esterHomo sapiens (human)Potency5.011910
N-[3-(2-methoxyphenyl)-1-methyl-4-oxo-2-quinolinyl]-2-methylpropanamideHomo sapiens (human)Potency8.912510
4-(4-chlorophenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency11.220210
3,4,5-trimethoxy-N-(3-methyl-1,3-benzothiazol-2-ylidene)benzamideHomo sapiens (human)Potency14.125410
benzotriptHomo sapiens (human)Potency15.848910
2-(2-bromophenyl)-5-[(7-nitro-4-quinazolinyl)oxymethyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency11.220210
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)thio]ethanoneHomo sapiens (human)Potency14.125410
N-(3-cyano-2-thiophenyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]acetamideHomo sapiens (human)Potency12.589310
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideHomo sapiens (human)Potency28.183810
2-chloro-1-[2,5-dimethyl-1-(5-methyl-3-isoxazolyl)-3-pyrrolyl]ethanoneHomo sapiens (human)Potency10.000010
2-chloro-N-[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]acetamideHomo sapiens (human)Potency3.981110
N-(2-methyl-1,3-benzothiazol-6-yl)-2,3-dihydro-1,4-benzodioxin-6-sulfonamideHomo sapiens (human)Potency2.511910
3-(4-methoxyphenyl)-1-phenyl-4-pyrazolamineHomo sapiens (human)Potency0.446710
1-[4-(1H-benzimidazol-2-yl)phenyl]-3-[3-(4-morpholinyl)propyl]thioureaHomo sapiens (human)Potency10.000010
2-(1H-benzimidazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneHomo sapiens (human)Potency28.183810
1-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]-2-(2-methyl-4-thiazolyl)ethanoneHomo sapiens (human)Potency3.981110
2-chloro-N-(2-phenyl-5-propyl-3-pyrazolyl)acetamideHomo sapiens (human)Potency4.466810
N-(1H-benzimidazol-2-yl)-3-[methyl-(4-methylphenyl)sulfamoyl]benzamideHomo sapiens (human)Potency28.183810
N-[(2S)-1-(1H-benzimidazol-2-ylamino)-3-methyl-1-oxobutan-2-yl]-3,5-dimethoxybenzamideHomo sapiens (human)Potency12.589310
N-(3-acetyl-2-methyl-5-benzofuranyl)-N-(8-quinolinylsulfonyl)acetamideHomo sapiens (human)Potency7.079510
4-[2-[[3-(4-methylphenyl)-5-triazolo[1,5-a]quinazolinyl]amino]ethyl]benzenesulfonamideHomo sapiens (human)Potency5.011910
N-(4-fluoro-3-methyl-1,3-benzothiazol-2-ylidene)-2-nitrobenzamideHomo sapiens (human)Potency11.220210
(4-tert-butylphenyl)-[2-(4-fluorophenyl)-8-methyl-3-sulfanylidene-1,4,8-triazaspiro[4.5]dec-1-en-4-yl]methanoneHomo sapiens (human)Potency7.079510
3-(1H-indol-3-yl)-N-[4-(2-pyrimidinylsulfamoyl)phenyl]propanamideHomo sapiens (human)Potency12.589310
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterHomo sapiens (human)Potency15.848910
mcb-613Homo sapiens (human)Potency2.238710
6-bromo-3-[4-nitro-3-(trifluoromethyl)phenyl]-2-propyl-4-quinazolinoneHomo sapiens (human)Potency28.183810
4-[(2,4-dichlorophenoxy)methyl]-N-[2-(dimethylamino)ethyl]benzamideHomo sapiens (human)Potency11.220210
N-[4-(1H-benzimidazol-2-yl)phenyl]-2,3,4,5,6-pentafluorobenzamideHomo sapiens (human)Potency28.183810
2,5-dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) esterHomo sapiens (human)Potency7.079510
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterHomo sapiens (human)Potency11.220210
1-[[(5-bromo-2-furanyl)-oxomethyl]amino]-3-[(4-chlorophenyl)methyl]thioureaHomo sapiens (human)Potency10.000010
1-[[(4-bromo-2-methyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxy-5-methylphenyl)thioureaHomo sapiens (human)Potency12.589310
5-[(2-chlorophenyl)methylsulfonyl]-1-(2,6-dimethylphenyl)tetrazoleHomo sapiens (human)Potency10.000010
N-[(3-ethoxy-2-prop-2-enoxyphenyl)methyl]-2-thiazolamineHomo sapiens (human)Potency22.387210
6-bromo-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency22.387210
N-(2-naphthalenyl)-2-[[6-[[[2-(2-naphthalenylamino)-2-oxoethyl]thio]methyl]-2-pyridinyl]methylthio]acetamideHomo sapiens (human)Potency2.818410
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-dibenzofuransulfonamideHomo sapiens (human)Potency25.118910
N-(2-fluorophenyl)-4-methoxy-2,5-dimethylbenzenesulfonamideHomo sapiens (human)Potency15.848910
1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(5,7-diphenyl-2-pyrazolo[1,5-a]pyrimidinyl)methanoneHomo sapiens (human)Potency2.818410
2-[benzenesulfonyl-(phenylmethyl)amino]-N-ethylacetamideHomo sapiens (human)Potency19.952610
2-[2-[[3-(1,3-benzoxazol-2-yl)anilino]-oxomethyl]phenyl]benzoic acidHomo sapiens (human)Potency1.778310
N-[3-[[diethylamino(sulfanylidene)methyl]thio]-1-oxopropyl]carbamic acid (4-propan-2-ylphenyl) esterHomo sapiens (human)Potency10.000010
3,4-dimethoxy-N-[4-(2,2,3,3-tetrafluoropropoxy)-3-(trifluoromethyl)phenyl]benzamideHomo sapiens (human)Potency11.220210
1-[(7-chloro-4-quinolinyl)amino]-3-(2,4-dichlorophenyl)thioureaHomo sapiens (human)Potency28.183810
1-[2-[3-(1-methylethenyl)phenyl]propan-2-yl]-3-(4-methyl-2-pyridinyl)ureaHomo sapiens (human)Potency4.466810
2-(1,3-benzothiazol-2-yl)-5-methyl-3-pyrazolamineHomo sapiens (human)Potency2.818410
N-(1H-benzimidazol-2-yl)-4-(dimethylsulfamoyl)benzamideHomo sapiens (human)Potency8.912510
N-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethenyl]-4-morpholinecarboxamideHomo sapiens (human)Potency5.623410
3-[2-(4-fluorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineHomo sapiens (human)Potency10.000010
N-[[2-(diethylamino)ethylamino]-sulfanylidenemethyl]-3-(4-methoxyphenyl)-1-phenyl-4-pyrazolecarboxamideHomo sapiens (human)Potency0.501210
1,2,3,4-tetrahydroacridine-9-carboxylic acid [2-(3-chloro-4-methoxyanilino)-2-oxoethyl] esterHomo sapiens (human)Potency22.387210
3-methyl-5-[[1-oxo-2-(2-pyridinylmethylamino)ethyl]amino]thiophene-2,4-dicarboxylic acid diethyl esterHomo sapiens (human)Potency5.011910
N-[[2-(1-cyclohexenyl)ethylamino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency2.818410
2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-[4-[4-(2-methylbutan-2-yl)phenoxy]anilino]-2-oxoethyl] esterHomo sapiens (human)Potency17.782810
N,N-diethyl-2-[(4-fluorophenyl)methylthio]-1,3-benzoxazole-5-sulfonamideHomo sapiens (human)Potency28.183810
2-[(1-oxido-2-pyridin-1-iumyl)thio]-1-(4-phenylphenyl)ethanoneHomo sapiens (human)Potency2.818410
4-(4-methoxyanilino)-2,5-dimethyl-6-thieno[2,3-d]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency2.818410
N-[(1-adamantylamino)-oxomethyl]-2-chloroacetamideHomo sapiens (human)Potency1.000010
4-methoxy-3-[2-phenylethyl-(phenylmethyl)sulfamoyl]benzoic acidHomo sapiens (human)Potency1.995310
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideHomo sapiens (human)Potency0.707910
2-[5-(1-pyrrolidinylsulfonyl)-2-thiophenyl]-N-[2-(4-sulfamoylphenyl)ethyl]acetamideHomo sapiens (human)Potency5.011910
2-hydroxy-4-methylbenzoic acid [2-(2-chloroanilino)-2-oxoethyl] esterHomo sapiens (human)Potency3.548110
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideHomo sapiens (human)Potency2.238710
2-(1-benzimidazolyl)acetic acid [2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency6.309610
2,5-dimethyl-1-(3-methylphenyl)-N-(4-methylphenyl)-3-pyrrolecarboxamideHomo sapiens (human)Potency28.183810
5-bromo-2-furancarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency28.183810
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4-methyl-5-phenyl-2-thiazolyl)-N-prop-2-enylacetamideHomo sapiens (human)Potency14.125410
4-[(1-methyl-5-tetrazolyl)thio]-5-phenylthieno[2,3-d]pyrimidineHomo sapiens (human)Potency1.995310
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)Potency3.981110
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideHomo sapiens (human)Potency0.891310
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideHomo sapiens (human)Potency0.891310
2-chloro-1-[4-[(3-methylphenyl)methyl]-1-piperazinyl]ethanoneHomo sapiens (human)Potency1.412510
2-(2,3-dichlorophenoxy)-N-(2,3-dihydro-1H-inden-5-yl)acetamideHomo sapiens (human)Potency1.412510
4-methyl-N-[1-methyl-2-oxo-6-(trifluoromethyl)-3-pyridinyl]benzamideHomo sapiens (human)Potency5.011910
3,4-dimethoxy-N-(2-methyl-1,3-benzothiazol-6-yl)benzamideHomo sapiens (human)Potency5.011910
2-chloro-N-[(5-chloro-2-thiophenyl)methyl]-N-methylacetamideHomo sapiens (human)Potency1.000010
2-(2,4-dichlorophenoxy)-N-[2-(methylthio)phenyl]acetamideHomo sapiens (human)Potency0.316210
N'-(4-quinazolinyl)acetohydrazideHomo sapiens (human)Potency10.000010
N-[2-(1-cyclohexenyl)ethyl]-1-phenyl-5-tetrazolamineHomo sapiens (human)Potency11.220210
1-[4-(3-chloro-2,4,6-trifluorophenyl)sulfonyl-1-piperazinyl]ethanoneHomo sapiens (human)Potency2.818410
3-(diethylsulfamoyl)benzoic acid [2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl] esterHomo sapiens (human)Potency28.183810
2-chloro-N-(2-chloro-5-methylsulfonylphenyl)acetamideHomo sapiens (human)Potency22.387210
5,6-dimethyl-N-[2-methyl-2-(4-morpholinyl)propyl]-4-thieno[2,3-d]pyrimidinamineHomo sapiens (human)Potency3.548110
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneHomo sapiens (human)Potency1.778310
N-[3-(4-morpholinyl)propyl]-3-(3-pyridinyl)-7,8-dihydro-6H-cyclopenta[4,5]thieno[1,2-c]pyrimidin-1-amineHomo sapiens (human)Potency22.387210
2-[(3-butyl-4-oxo-2-quinazolinyl)thio]-N-cyclopropylacetamideHomo sapiens (human)Potency12.589310
N-[5-chloro-2-(4-methyl-1-piperazinyl)phenyl]-3-(dimethylsulfamoyl)benzamideHomo sapiens (human)Potency6.309610
2-(1-piperidinyl)-6-thiophen-2-yl-4-(trifluoromethyl)-3-pyridinecarbonitrileHomo sapiens (human)Potency7.079510
5-(2-chloroanilino)-3-oxo-4-isothiazolecarbonitrileHomo sapiens (human)Potency31.622810
N-benzyl-N'-methyl-N-(pyridin-3-ylmethyl)thioureaHomo sapiens (human)Potency5.011910
5-Methyl-6-(2-thienyl)-2,3,4,5-tetrahydropyridazin-3-oneHomo sapiens (human)Potency3.981110
3-(4-Chloroanilino)propanoic acidHomo sapiens (human)Potency28.183810
2-phenyl-N-(2-piperidin-1-ylethyl)quinolin-4-amineHomo sapiens (human)Potency28.183810
6-cyclohex-3-enyl-5-nitropiperidin-2-oneHomo sapiens (human)Potency1.995310
3-(tert-butyl)-1-methyl-4,5-dihydro-1H-pyrazol-5-oneHomo sapiens (human)Potency3.162310
2,2-dimethyl-N-pyridin-4-yl-3H-benzofuran-7-carboxamideHomo sapiens (human)Potency1.412510
N,N-diethyl-5-thiophen-2-yl-2-thiophenecarboxamideHomo sapiens (human)Potency5.011910
3-(tert-butylsulfamoyl)-4-phenyl-5-(trifluoromethyl)-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency10.000010
4-(2-fluorophenyl)-N-(2-methylbut-3-yn-2-yl)benzamideHomo sapiens (human)Potency10.000010
N'-[(4-chlorophenyl)-oxomethyl]-2-methyl-4-thiazolecarbohydrazideHomo sapiens (human)Potency28.183810
N-(4-chlorophenyl)-2-[[4-methyl-5-[4-methyl-2-(5-methyl-3-isoxazolyl)-5-thiazolyl]-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency5.011910
N-(2-chlorophenyl)-2-[[5-[5-(trifluoromethyl)-2-pyridinyl]-1,3,4-oxadiazol-2-yl]thio]acetamideHomo sapiens (human)Potency11.220210
N-(6-methoxy-3-pyridinyl)-2-thiophenecarboxamideHomo sapiens (human)Potency28.183810
3-[[(2,4-dichlorophenyl)methylthio]methyl]-4-propan-2-yl-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency11.220210
2,6-dichlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] esterHomo sapiens (human)Potency28.183810
3-(2,4-dichlorophenyl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazoleHomo sapiens (human)Potency4.466810
2-(2-Thienyl)-1,3-thiazole-4-carboxylic acidHomo sapiens (human)Potency11.220210
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineHomo sapiens (human)Potency1.995310
3-[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]propanoic acid ethyl esterHomo sapiens (human)Potency11.220210
N-[amino(1-pyrrolidinyl)methylidene]-3-(2,6-dichlorophenyl)-5-methyl-4-isoxazolecarboxamideHomo sapiens (human)Potency1.122010
2,6-dimethoxy-N-(1-methyl-1H-pyrazol-5-yl)benzamideHomo sapiens (human)Potency2.818410
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamideHomo sapiens (human)Potency7.943310
5-[[[5-(4-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esterHomo sapiens (human)Potency8.912510
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(4-fluorophenyl)sulfonylethylthio]-1H-1,2,4-triazol-5-oneHomo sapiens (human)Potency2.238710
N'-(3-chloro-4-methylphenyl)-5-isoxazolecarbohydrazideHomo sapiens (human)Potency1.584910
2-(1,3-dimethyl-1H-pyrazol-5-yl)-1H-isoindole-1,3(2H)-dioneHomo sapiens (human)Potency5.011910
2-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency5.011910
N-{5-[(dimethylamino)sulfonyl]-2-methylphenyl}cyclohexanecarboxamideHomo sapiens (human)Potency3.981110
LSM-28486Homo sapiens (human)Potency2.818410
3,3-dimethyl-5-oxo-5-[(3-phenyl-1H-pyrazol-5-yl)amino]pentanoic acidHomo sapiens (human)Potency28.183810
2-amino-4-(2-chlorophenyl)-6-[(4-chlorophenyl)thio]pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency2.238710
2-[5-[(3-chlorophenyl)thio]-2-thiophenyl]pyridineHomo sapiens (human)Potency2.511910
8-methylsulfinyl-4,5-dihydrothieno[3,4-g][2,1]benzoxazole-6-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-[4-(2-methylpropyl)phenyl]propanoic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
3,3,3-trifluoro-2-hydroxy-2-[4-[methoxycarbonyl(methyl)amino]phenyl]propanoic acid methyl esterHomo sapiens (human)Potency5.011910
3-[[sulfanylidene-[[2,2,2-trichloro-1-[[(3-nitrophenyl)-oxomethyl]amino]ethyl]amino]methyl]amino]benzoic acidHomo sapiens (human)Potency5.011910
4,6-dimorpholino-n-(4-nitrophenyl)-1,3,5-triazin-2-amineHomo sapiens (human)Potency10.000010
(4-chlorophenyl)-[6,7-dichloro-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-3-benzofuranyl]methanoneHomo sapiens (human)Potency0.446710
N-[2-(1-methyl-2-pyrrolidinyl)ethyl]-2-adamantanamineHomo sapiens (human)Potency8.912510
N-[2-(4-chlorophenoxy)ethyl]-5-(3,5-dimethyl-1-piperazinyl)-2-nitroanilineHomo sapiens (human)Potency5.623410
2-(4,6,7-Trimethyl-2-quinazolinyl)guanidineHomo sapiens (human)Potency12.589310
4-ethyl-2-methoxy-3-phenyl-3,3a,9,9a-tetrahydropyrrolo[2,3-b]quinoxalineHomo sapiens (human)Potency11.220210
4-(4-hydroxy-3-methoxyphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid (4-methoxyphenyl)methyl esterHomo sapiens (human)Potency15.848910
2-[[2-methyl-5-nitro-3-(phenylmethyl)-4-imidazolyl]thio]-6-nitro-1H-benzimidazoleHomo sapiens (human)Potency5.011910
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamideHomo sapiens (human)Potency3.981110
N-(3-bicyclo[2.2.1]heptanyl)-4-chlorobenzenesulfonamideHomo sapiens (human)Potency3.162310
N-[4-methyl-5-[2-(3-nitroanilino)-4-thiazolyl]-2-thiazolyl]acetamideHomo sapiens (human)Potency11.220210
N-(4-fluorophenyl)-4-(4-nitrophenyl)-1-piperazinecarbothioamideHomo sapiens (human)Potency3.162310
4-chloro-3-(diethylsulfamoyl)-N-(2-nitrophenyl)benzamideHomo sapiens (human)Potency11.220210
2-[(4-chlorophenyl)thio]-N-[4-[(2,4-dimethylphenyl)sulfamoyl]phenyl]propanamideHomo sapiens (human)Potency31.622810
1-butyl-3-(2-hydroxyethylamino)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrileHomo sapiens (human)Potency5.011910
4-methylbenzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-methoxyphenyl] esterHomo sapiens (human)Potency5.011910
(3-amino-5-nitro-2-benzofuranyl)-phenylmethanoneHomo sapiens (human)Potency28.183810
3-acetamidobenzoic acid [2-(4-methylphenyl)-2-oxo-1-phenylethyl] esterHomo sapiens (human)Potency28.183810
1-(3,4-dimethylphenyl)-3-(2-pyrimidinylthio)pyrrolidine-2,5-dioneHomo sapiens (human)Potency3.548110
N-(3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-9H-xanthene-9-carboxamideHomo sapiens (human)Potency5.011910
4-ethoxy-N-(3-quinolinyl)benzenesulfonamideHomo sapiens (human)Potency11.220210
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Potency28.183810
N-[4-(butylsulfamoyl)phenyl]-2-phenyl-2-(phenylthio)acetamideHomo sapiens (human)Potency10.000010
1-[4-(3,4-dihydroxyphenyl)-6-phenyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidin-5-yl]ethanoneHomo sapiens (human)Potency8.912510
importazoleHomo sapiens (human)Potency11.220210
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamideHomo sapiens (human)Potency28.183810
N-[amino-[2-(1H-indol-3-yl)ethylimino]methyl]-4-chlorobenzamideHomo sapiens (human)Potency28.183810
2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-N-(2-methoxy-3-dibenzofuranyl)acetamideHomo sapiens (human)Potency31.622810
1-[2-(hydroxymethyl)-1-benzimidazolyl]-3-(1-indolyl)-2-propanolHomo sapiens (human)Potency28.183810
1-[3-[4-(2-chloro-5-methoxyphenyl)-1-piperazinyl]propyl]-3-(4-methylphenyl)ureaHomo sapiens (human)Potency17.782810
2-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-3-hydroxy-3-phenyl-1-isoindoloneHomo sapiens (human)Potency5.011910
1-(4-methoxy-2-nitrophenyl)-4-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)piperazineHomo sapiens (human)Potency6.309610
cb 7969312Homo sapiens (human)Potency5.623410
4H-[1,3]thiazino[3,2-a]benzimidazol-4-olHomo sapiens (human)Potency10.000010
2-[1-(4-chlorophenyl)-5-oxo-3-(2-pyridin-4-ylethyl)-2-sulfanylidene-4-imidazolidinyl]-N-(4-fluorophenyl)acetamideHomo sapiens (human)Potency28.183810
N-[4-[(3-acetylphenyl)sulfamoyl]phenyl]-1-piperidinecarboxamideHomo sapiens (human)Potency28.183810
1-(1,3-benzodioxol-5-yl)-3-[4-(4-hydroxyphenyl)-1-piperazinyl]pyrrolidine-2,5-dioneHomo sapiens (human)Potency5.011910
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[[1-(2-methylpropyl)-2-benzimidazolyl]thio]ethanoneHomo sapiens (human)Potency28.183810
1-[2-hydroxy-3-[4-(2-methylbutan-2-yl)phenoxy]propyl]-4-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency19.952610
3-[[5,5-dimethyl-3-(4-morpholinyl)-1-cyclohex-2-enylidene]amino]-N,N-dimethylanilineHomo sapiens (human)Potency14.125410
N-[1-oxo-1-[[4-(2-pyridinyl)-2-thiazolyl]amino]propan-2-yl]-2-furancarboxamideHomo sapiens (human)Potency11.220210
N-[1-(1H-benzimidazol-2-yl)-2-phenylethyl]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxo-3-pyrrolidinecarboxamideHomo sapiens (human)Potency2.818410
3-chloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideHomo sapiens (human)Potency28.183810
2-[8-(6-amino-1H-benzimidazol-2-yl)octyl]-3H-benzimidazol-5-amineHomo sapiens (human)Potency22.387210
N-methyl-5-nitro-N-(phenylmethyl)-2-furancarboxamideHomo sapiens (human)Potency2.511910
2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterHomo sapiens (human)Potency11.220210
N-[3-(1,3-benzothiazol-2-ylthio)-5-nitrophenyl]-2-fluorobenzamideHomo sapiens (human)Potency14.125410
phenyl-(2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)methanoneHomo sapiens (human)Potency10.000010
2-[(prop-2-enylthio)-(4,5,6,7-tetrahydro-1H-indol-2-yl)methylidene]propanedinitrileHomo sapiens (human)Potency0.891310
N'-[(2-nitrophenyl)-oxomethyl]-2-pyridinecarbohydrazideHomo sapiens (human)Potency5.011910
N-[[5-[(4-chlorophenyl)methylthio]-4-phenyl-1,2,4-triazol-3-yl]methyl]-4-ethoxyanilineHomo sapiens (human)Potency10.000010
3-nitro-N-(pyridin-4-ylmethyl)benzenesulfonamideHomo sapiens (human)Potency2.511910
1-[3-(benzenesulfonyl)-2-(1-piperidinyl)propyl]piperidineHomo sapiens (human)Potency4.466810
6-amino-5,7,7-tricyano-8-pyridin-4-yl-1,3,8,8a-tetrahydroisoquinoline-2-carboxylic acid (phenylmethyl) esterHomo sapiens (human)Potency15.848910
5-methyl-1-[3-(2-methylphenoxy)propyl]indole-2,3-dioneHomo sapiens (human)Potency10.000010
N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency28.183810
2-chloro-N-(3-ethyl-2-oxo-1,3-benzoxazol-6-yl)acetamideHomo sapiens (human)Potency1.122010
N-[2-[1-methyl-5-[[(4-methylphenyl)-oxomethyl]amino]-2-benzimidazolyl]ethyl]-2-furancarboxamideHomo sapiens (human)Potency2.818410
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency1.778310
4-amino-N5-(4-butoxyphenyl)-N5-[2-(cyclohexylamino)-2-oxoethyl]isothiazole-3,5-dicarboxamideHomo sapiens (human)Potency28.183810
N-[2-(tert-butylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2-oxolanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideHomo sapiens (human)Potency1.000010
1-[2-(diethylamino)ethyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-(2-oxolanylmethyl)thioureaHomo sapiens (human)Potency3.162310
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-5-methyl-N-(thiophen-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamideHomo sapiens (human)Potency5.011910
4-(2-azaspiro[5.5]undecan-2-ylsulfonyl)-N-butan-2-ylbenzenesulfonamideHomo sapiens (human)Potency1.122010
2-[(3,6-dimethyl-2-quinolinyl)thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency12.589310
3-(2,4-dimethoxyphenyl)-1-[(1-ethyl-2-pyrrolidinyl)methyl]-1-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]thioureaHomo sapiens (human)Potency14.125410
CID 3192987Homo sapiens (human)Potency3.981110
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency28.183810
2-[2-[[2-[[1-(2,4-dimethylphenyl)-5-tetrazolyl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterHomo sapiens (human)Potency10.000010
N-(4-Butan-2-ylphenyl)-N-[2-(cyclopentylamino)-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamideHomo sapiens (human)Potency7.943310
2-[2-methoxyethyl-(1-oxo-2-thiophen-2-ylethyl)amino]-N-[(4-methoxyphenyl)methyl]-2-(4-propan-2-ylphenyl)acetamideHomo sapiens (human)Potency3.162310
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency5.011910
1-[9-[(4-fluorophenyl)methyl]-9-azabicyclo[3.3.1]nonan-3-yl]-3-(2-phenylphenyl)ureaHomo sapiens (human)Potency3.162310
1-(9-cyclopentyl-9-azabicyclo[3.3.1]nonan-3-yl)-3-(3,5-dimethylphenyl)thioureaHomo sapiens (human)Potency28.183810
N1-cyclohexyl-N2-cyclopropylpyrrolidine-1,2-dicarboxamideHomo sapiens (human)Potency5.011910
1-[2-[(3-cyano-5,7-dimethyl-2-quinolinyl)amino]ethyl]-3-(3-methoxypropyl)thioureaHomo sapiens (human)Potency3.162310
[4-[5-tert-butyl-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency28.183810
N-[2-(3-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-N',N'-dimethylpropane-1,3-diamineHomo sapiens (human)Potency22.387210
1-[(4-fluorophenyl)methyl]-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-oxo-3H-benzimidazole-5-carboxamideHomo sapiens (human)Potency11.220210
2-[(6-fluoro-1,3-benzothiazol-2-yl)amino]-4-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
2-[(3-methoxyphenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency7.079510
N-[3-(diethylamino)propyl]-6-(4-fluorophenyl)-3-methyl-2-imidazo[2,1-b]thiazolecarboxamideHomo sapiens (human)Potency31.622810
4-[[2-(4-methoxyphenyl)-6-imidazo[2,1-b][1,3]benzothiazolyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency0.707910
4-[(1-methyl-2-oxo-4-quinolinyl)oxy]-N-(4-methyl-2-pyridinyl)butanamideHomo sapiens (human)Potency28.183810
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolHomo sapiens (human)Potency1.000010
N-(2,3-dihydro-1H-inden-5-yl)-2-[(4-hydroxy-6-oxo-1H-pyrimidin-2-yl)thio]acetamideHomo sapiens (human)Potency5.011910
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
3-chloro-4-ethoxy-N-[3-(2-oxazolo[5,4-b]pyridinyl)phenyl]benzamideHomo sapiens (human)Potency3.548110
3,7-dimethyl-2-(methylthio)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency35.481310
5-methyl-N-(5-methyl-2-phenyl-3-pyrazolyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency14.125410
1-[[2-(4-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-N-[2-(dipropylamino)ethyl]-4-piperidinecarboxamideHomo sapiens (human)Potency2.511910
N-[4-methyl-2-(4-methyl-1-piperazinyl)-6-quinolinyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency28.183810
2-[[2-(3,4-dimethoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-[3-(1-pyrrolidinyl)propyl]acetamideHomo sapiens (human)Potency3.548110
6-[(2-ethylphenyl)sulfamoyl]-N-(2-furanylmethyl)-4-oxo-1H-quinoline-3-carboxamideHomo sapiens (human)Potency31.622810
2-amino-4-[5-methyl-2-(methylthio)-3-thiophenyl]-5-oxo-1-(3-pyridinyl)-4,6,7,8-tetrahydroquinoline-3-carbonitrileHomo sapiens (human)Potency7.943310
N-(3,4-dimethylphenyl)-3-[(4-fluorophenyl)methyl]-1,3-diazinane-1-carboxamideHomo sapiens (human)Potency8.912510
2-[[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-thieno[3,2-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency7.079510
4-[dimethylamino(oxo)methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl esterHomo sapiens (human)Potency28.183810
2-[3-[3-(2-furanylmethylamino)-3-oxopropyl]-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetic acid (phenylmethyl) esterHomo sapiens (human)Potency3.162310
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-1-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methyl]-4-piperidinecarboxamideHomo sapiens (human)Potency1.778310
N-butan-2-yl-6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-1H-quinoline-3-carboxamideHomo sapiens (human)Potency5.011910
3-methyl-5-(4-morpholinylsulfonyl)-N-(2-pyridinylmethyl)-2-benzofurancarboxamideHomo sapiens (human)Potency0.501210
4-[3-(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)-1-oxopropyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency31.622810
4-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-3-nitrobenzenesulfonamideHomo sapiens (human)Potency3.548110
2-(6-amino-5-cyano-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)benzoic acidHomo sapiens (human)Potency2.818410
4-[[(4-methylphenyl)sulfonylamino]methyl]-N-[2-[(phenylmethyl)-propan-2-ylamino]ethyl]benzamideHomo sapiens (human)Potency3.981110
N-[4-(difluoromethoxy)phenyl]-4-(phenylmethyl)-1-piperazinecarbothioamideHomo sapiens (human)Potency1.122010
N4-(1,1-dioxo-3-thiolanyl)-5-nitropyrimidine-4,6-diamineHomo sapiens (human)Potency2.511910
2-amino-7,7-dimethyl-5-oxo-4-[1-phenyl-3-(4-propan-2-ylphenyl)-4-pyrazolyl]-6,8-dihydro-4H-1-benzopyran-3-carbonitrileHomo sapiens (human)Potency19.952610
N-[4-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency3.548110
2-(2-methoxyphenyl)-1-methyl-3,5-dinitro-2H-pyridineHomo sapiens (human)Potency1.778310
N-[(4-methoxyphenyl)methyl]-2-(phenylmethyl)-4-thiazolecarboxamideHomo sapiens (human)Potency3.162310
5-(diethylsulfamoyl)-2-hydroxybenzoic acid [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] esterHomo sapiens (human)Potency5.011910
1-(3-methoxyphenyl)-3-[5-(2-methyl-1-piperidinyl)-1,3,4-thiadiazol-2-yl]ureaHomo sapiens (human)Potency28.183810
1-(3,4-dichlorophenyl)-3-[1-(4-morpholinyl)-1-phenylpropan-2-yl]ureaHomo sapiens (human)Potency4.466810
N,N-dimethylcarbamodithioic acid (1-acetamido-2,2,2-trichloroethyl) esterHomo sapiens (human)Potency3.162310
LSM-16990Homo sapiens (human)Potency11.220210
6-amino-5-cyano-4-(2-fluorophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyridine-3-carboxamideHomo sapiens (human)Potency3.548110
2-benzoylimino-1-(2-furanylmethyl)-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency31.622810
N-[5-ethyl-3-[(4-fluorophenyl)-(4-morpholinyl)methyl]-2-thiophenyl]benzamideHomo sapiens (human)Potency10.000010
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olHomo sapiens (human)Potency1.000010
1-(4-butylphenyl)-3-[4-chloro-3-(dimethylsulfamoyl)phenyl]thioureaHomo sapiens (human)Potency12.589310
2-[[2-[3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]thio]acetic acid butyl esterHomo sapiens (human)Potency15.848910
N-[[4-[[4-(4-fluorophenyl)-1-piperazinyl]-oxomethyl]cyclohexyl]methyl]-2-thiophenesulfonamideHomo sapiens (human)Potency22.387210
N'-[(3-nitrophenyl)-oxomethyl]-2-pyridinecarbohydrazideHomo sapiens (human)Potency0.501210
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)-5-(4-morpholinylsulfonyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)Potency1.995310
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideHomo sapiens (human)Potency0.501210
3-[(4-ethylphenoxy)methyl]-4-(6-methylheptan-2-yl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency8.912510
ML162Homo sapiens (human)Potency0.501210
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency0.501210
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency0.354810
2-(cyclohexylamino)-N-[(diphenylmethylene)amino]propanamideHomo sapiens (human)Potency3.162310
5-[3-[[(4-methylphenyl)-oxomethyl]hydrazo]-2,5-dioxo-1-pyrrolidinyl]benzene-1,3-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency5.623410
4-chloro-N-(2-methoxy-1-phenazinyl)benzamideHomo sapiens (human)Potency28.183810
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency28.183810
LSM-1924Homo sapiens (human)Potency28.183810
2-[1-(2-methylphenyl)-3-oxo-3-thiophen-2-ylpropyl]propanedinitrileHomo sapiens (human)Potency11.220210
N4-(3-fluorophenyl)-N2-[3-(4-morpholinyl)propyl]-5-nitropyrimidine-2,4,6-triamineHomo sapiens (human)Potency8.912510
2-(4-chlorophenyl)-5-methyl-4-oxo-2,3-dihydro-1H-thieno[3,4-d]pyrimidine-7-carboxylic acid ethyl esterHomo sapiens (human)Potency3.548110
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamideHomo sapiens (human)Potency1.258910
4-(2-methylcyclohexyl)-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency10.000010
1-bromo-3-(5,5-dimethyl-3-phenyl-4H-pyrazolo[4,3-a]carbazol-10-yl)-2-propanolHomo sapiens (human)Potency22.387210
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency10.000010
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneHomo sapiens (human)Potency0.562310
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamideHomo sapiens (human)Potency3.162310
1-(4-chlorophenyl)-3-[2-(2-furanylmethyl)cyclohexyl]ureaHomo sapiens (human)Potency28.183810
4-[(2-hydroxy-3-nitrophenyl)-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)methyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneHomo sapiens (human)Potency28.183810
1-[4-(3-chlorophenyl)-1-piperazinyl]-2-phenyl-1-butanoneHomo sapiens (human)Potency31.622810
2-furanyl-[4-(4-propan-2-ylphenyl)sulfonyl-1-piperazinyl]methanoneHomo sapiens (human)Potency11.220210
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleHomo sapiens (human)Potency31.622810
6-nitro-3-phenyl-1H-benzimidazole-2-thioneHomo sapiens (human)Potency28.183810
LSM-22738Homo sapiens (human)Potency25.118910
fg 9041Homo sapiens (human)Potency0.316210
N-(3,5-dichloro-2-pyridinyl)-2-[(4-methyl-2-quinolinyl)thio]propanamideHomo sapiens (human)Potency3.548110
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineHomo sapiens (human)Potency4.466810
2-(1H-benzimidazol-2-yl)-5-methyl-4-(phenylmethyl)-4H-pyrazol-3-oneHomo sapiens (human)Potency5.011910
N-(1,1-dioxo-3-thiolanyl)-N-ethyl-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)acetamideHomo sapiens (human)Potency19.952610
4-tert-butylbenzoic acid [2-[(2-methoxy-3-dibenzofuranyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency2.238710
N-[3-(dimethylsulfamoyl)-4-methylphenyl]-2-quinolinecarboxamideHomo sapiens (human)Potency5.011910
4-oxo-4-thiophen-2-ylbutanoic acid [2-(ethylamino)-2-oxoethyl] esterHomo sapiens (human)Potency2.818410
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-1-nitro-9,10-dioxo-2-anthracenecarboxamideHomo sapiens (human)Potency11.220210
1-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-ethyl-1-(2-furanylmethyl)thioureaHomo sapiens (human)Potency28.183810
[4-[(2-chlorophenyl)methylsulfonyl]-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency28.183810
2-amino-4-(3,4-dimethoxyphenyl)-7,7-dimethyl-5-oxo-1-(3-pyridinyl)-6,8-dihydro-4H-quinoline-3-carbonitrileHomo sapiens (human)Potency14.125410
7-chloro-4-[(2-fluorophenyl)-oxomethyl]-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-oneHomo sapiens (human)Potency1.778310
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamideHomo sapiens (human)Potency12.589310
2-(5-bromo-2-thiophenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency19.952610
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency28.183810
2-methoxy-N-(5-phenyl-1,2,4-thiadiazol-3-yl)benzamideHomo sapiens (human)Potency2.818410
7-(1-azepanyl)-3-(2-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency28.183810
LSM-16386Homo sapiens (human)Potency5.011910
2-(4-methoxyphenyl)sulfonylquinoxalineHomo sapiens (human)Potency14.125410
N-[1-(1H-benzimidazol-2-yl)ethyl]-3-(dimethylsulfamoyl)benzamideHomo sapiens (human)Potency28.183810
2-(hexylamino)-1-[4-(phenylmethyl)-1-piperidinyl]ethanoneHomo sapiens (human)Potency1.778310
5-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineHomo sapiens (human)Potency5.011910
N-[3-(N-(2-chloro-1-oxoethyl)-4-nitroanilino)propyl]-2,2,2-trifluoroacetamideHomo sapiens (human)Potency1.122010
1-[(2,4-dichlorophenyl)methyl]-4-(methylthio)-2-oxo-6-phenyl-3-pyridinecarbonitrileHomo sapiens (human)Potency28.183810
6-benzoyl-2-phenyl-5-(trifluoromethyl)-3-pyridazinoneHomo sapiens (human)Potency2.238710
N-[3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxo-1-pyrrolidinyl)benzamideHomo sapiens (human)Potency5.011910
4-(3-chlorophenyl)sulfonyl-N-cyclohexyl-N-methyl-3-nitrobenzamideHomo sapiens (human)Potency0.891310
6-(2-methyl-1-piperidinyl)-5-nitro-4-pyrimidinamineHomo sapiens (human)Potency4.466810
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]-4-methylbenzamideHomo sapiens (human)Potency28.183810
N-(3-methoxyphenyl)-1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolecarboxamideHomo sapiens (human)Potency3.981110
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency1.000010
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency0.891310
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency0.316210
4-(2,5-dioxo-1-pyrrolidinyl)-N-[4-(4-methoxyphenyl)-2-thiazolyl]benzamideHomo sapiens (human)Potency12.589310
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaHomo sapiens (human)Potency11.220210
5-nitro-2-furancarboxylic acid [2-oxo-2-[3-(1-piperidinylsulfonyl)anilino]ethyl] esterHomo sapiens (human)Potency1.995310
3-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethyl]-1,1-bis(phenylmethyl)ureaHomo sapiens (human)Potency15.848910
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideHomo sapiens (human)Potency12.589310
4-bromo-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency2.818410
N-(3-chlorophenyl)-2-[4-oxo-2-phenylimino-3-(2-pyridinylmethyl)-5-thiazolidinyl]acetamideHomo sapiens (human)Potency28.183810
2-chloro-N-(1,2-diphenylethyl)acetamideHomo sapiens (human)Potency1.258910
1-(2-methoxy-3-dibenzofuranyl)-3-(3-methylphenyl)thioureaHomo sapiens (human)Potency31.622810
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneHomo sapiens (human)Potency11.220210
N-(1-dibutoxyphosphoryl-4-oxo-1-naphthalenyl)benzenesulfonamideHomo sapiens (human)Potency10.000010
2-chloro-N-(2,6-dimethylphenyl)-3-oxo-3-phenylpropanamideHomo sapiens (human)Potency28.183810
N-[3-(1-azepanylsulfonyl)phenyl]-4-oxo-1-benzopyran-2-carboxamideHomo sapiens (human)Potency8.912510
8-[4-(4-fluorophenoxy)-3-nitrophenyl]-7-(2-hydroxyethyl)-3-(phenylmethyl)purine-2,6-dioneHomo sapiens (human)Potency28.183810
2-bromo-6-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneHomo sapiens (human)Potency2.818410
1-(3-chlorophenyl)-3-pyridin-4-ylureaHomo sapiens (human)Potency12.589310
2-(4-bromophenyl)-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)Potency28.183810
4-(1-azepanylsulfonyl)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-hydroxyphenyl]benzamideHomo sapiens (human)Potency19.952610
4-chloro-N-[3-(N-methylanilino)-1,4-dioxo-2-naphthalenyl]benzamideHomo sapiens (human)Potency10.000010
4-(5-methyl-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)benzoic acid 8-quinolinyl esterHomo sapiens (human)Potency1.995310
8-nitro-5-[3-(trifluoromethyl)-1-piperidinyl]isoquinolineHomo sapiens (human)Potency28.183810
N-[(4-ethoxy-3-methoxyphenyl)methyl]-N-methyl-2-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency1.778310
7-chloro-N-(phenylmethyl)-4-quinolinamineHomo sapiens (human)Potency8.912510
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaHomo sapiens (human)Potency17.782810
1-[2-(trifluoromethyl)phenyl]sulfonyl-4-piperidinecarboxylic acid [2-[(4-fluorophenyl)methylamino]-2-oxoethyl] esterHomo sapiens (human)Potency28.183810
N-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxolanylmethoxy)benzamideHomo sapiens (human)Potency28.183810
2-phenyl-N-[1-(phenylmethyl)-4-piperidinyl]-4-quinazolinamineHomo sapiens (human)Potency10.000010
1-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-[3-(dimethylamino)propyl]-1-ethylthioureaHomo sapiens (human)Potency10.000010
1-[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-[3-(dimethylamino)propyl]thioureaHomo sapiens (human)Potency28.183810
4-[4-(4-acetylphenyl)-1-piperazinyl]-N-[3-(dimethylamino)propyl]-3-nitrobenzenesulfonamideHomo sapiens (human)Potency2.511910
2-[[4-(2-methoxyphenyl)sulfonyl-1-piperazinyl]sulfonyl]benzonitrileHomo sapiens (human)Potency3.548110
LSM-24516Homo sapiens (human)Potency28.183810
2-(Chloroacetyl)-N,2-diphenylhydrazinecarboxamideHomo sapiens (human)Potency4.466810
2-chloro-1-[1-(3-isoxazolyl)-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)Potency19.952610
N-(1-benzylpiperidin-4-yl)-2-(pyridin-3-yl)quinazolin-4-amineHomo sapiens (human)Potency11.220210
N-(3-chloro-4-fluorophenyl)-2-[5-(dimethylsulfamoyl)-2-(ethylamino)anilino]acetamideHomo sapiens (human)Potency7.943310
5-[(3-nitro-2-pyridinyl)thio]-N-prop-2-enyl-1,3,4-thiadiazol-2-amineHomo sapiens (human)Potency5.011910
LSM-24595Homo sapiens (human)Potency10.000010
N-(4-Nitro-1,2,5-oxadiazol-3-yl)-2-pyridin-2-ylsulfanylacetamideHomo sapiens (human)Potency6.309610
[5-(4-fluorophenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[2-(3-pyridinyl)-1-piperidinyl]methanoneHomo sapiens (human)Potency10.000010
2-(4-methylphenoxy)-N-[2-[oxo(1-piperidinyl)methyl]phenyl]acetamideHomo sapiens (human)Potency11.220210
2-Chloro-1-[5-(furan-2-yl)-3-(5-methylfuran-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneHomo sapiens (human)Potency3.981110
2-(2-chloro-1-oxoethyl)-3,4-dihydro-1H-isoquinoline-3-carboxylic acid methyl esterHomo sapiens (human)Potency1.000010
5-carbamoyl-4-methyl-2-[[1-oxo-2-(1,2,3,4-tetrahydronaphthalen-1-ylamino)ethyl]amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
N-[(4-chlorophenyl)methyl]-2-[[[(2-fluorophenyl)methyl-(phenylmethyl)amino]-sulfanylidenemethyl]amino]acetamideHomo sapiens (human)Potency7.943310
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thioureaHomo sapiens (human)Potency10.000010
alsterpaulloneHomo sapiens (human)Potency0.794310
5-[(5-bromo-2-hydroxyphenyl)-oxomethyl]-1-cyclohexyl-2-oxo-3-pyridinecarbonitrileHomo sapiens (human)Potency11.220210
LSM-25964Homo sapiens (human)Potency17.782810
N-[2-chloro-5-[ethyl(phenyl)sulfamoyl]phenyl]-2-[methyl-(1-methyl-4-piperidinyl)amino]acetamideHomo sapiens (human)Potency28.183810
2-(4-fluoro-3-nitrophenyl)-4,4-dimethyl-5H-oxazoleHomo sapiens (human)Potency1.258910
1-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-3-phenylureaHomo sapiens (human)Potency8.912510
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideHomo sapiens (human)Potency28.183810
4-[3-(2-chloro-1-oxoethyl)-2,5-dimethyl-1-pyrrolyl]-1,5-dimethyl-2-phenyl-3-pyrazoloneHomo sapiens (human)Potency1.122010
4-tert-butyl-N-[3-[4-[3-[[(4-tert-butylphenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]benzamideHomo sapiens (human)Potency12.589310
N,N-diethylcarbamodithioic acid (2,2,2-trichloro-1-formamidoethyl) esterHomo sapiens (human)Potency12.589310
5-benzoyl-6-methyl-4-[4-(4-morpholinyl)phenyl]-3,4-dihydro-1H-pyrimidin-2-oneHomo sapiens (human)Potency3.162310
N-(5-acetyl-4-methyl-2-thiazolyl)-2-(2,4-dichlorophenoxy)acetamideHomo sapiens (human)Potency1.000010
Euparotin acetateHomo sapiens (human)Potency3.162310
astragalinHomo sapiens (human)Potency5.011910
fenretinideHomo sapiens (human)Potency15.848910
N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamideHomo sapiens (human)Potency28.183810
2-(2-furanylmethyl)-3-[[2-(3-pyridinyl)-3H-benzimidazol-5-yl]amino]-3H-isoindol-1-oneHomo sapiens (human)Potency7.079510
2-[[4-methyl-5-[(2-oxo-1,3-benzothiazol-3-yl)methyl]-1,2,4-triazol-3-yl]thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency28.183810
3-(4-chlorophenyl)-1-methyl-N-[3-(1-pyrrolidinyl)propyl]-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency10.000010
3-[3-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]propyl]-1H-benzimidazol-2-oneHomo sapiens (human)Potency1.122010
(2e)-3-phenyl-1-(2,3,4,5-tetrahydro-1,6-benzodioxocin-8-yl)prop-2-en-1-oneHomo sapiens (human)Potency11.220210
BucharaineHomo sapiens (human)Potency10.000010
serratinHomo sapiens (human)Potency1.000010
3,3'-diethylthiatricarbocyanine iodide, 3h-labeledHomo sapiens (human)Potency1.000010
5233705 compoundHomo sapiens (human)Potency1.412510
10-hydroxy-3-methyl-8-pentyl-2,4-dihydro-1H-[1]benzopyrano[3,4-c]pyridin-5-oneHomo sapiens (human)Potency28.183810
[4-(3-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency12.589310
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazineHomo sapiens (human)Potency6.309610
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-1-(4-methoxyphenyl)ethanoneHomo sapiens (human)Potency2.818410
4-hydroxyderricinHomo sapiens (human)Potency28.183810
kolavenic acidHomo sapiens (human)Potency0.316210
1-(2-methoxy-5-methylphenyl)-3-pyridin-4-ylureaHomo sapiens (human)Potency28.183810
2-chloro-N-(1-methyl-3-pyrazolyl)acetamideHomo sapiens (human)Potency3.981110
(3S)-2-(2-chloro-1-oxoethyl)-1,1-dimethyl-4,9-dihydro-3H-pyrido[3,4-b]indole-3-carboxylic acid methyl esterHomo sapiens (human)Potency1.000010
N-(5-carbamoyl-2-methoxyphenyl)-3-(2,4-dimethoxyphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamideHomo sapiens (human)Potency3.981110
N-[(2-chlorophenyl)methyl]-2-[7-oxo-3-(phenylmethyl)-6-triazolo[4,5-d]pyrimidinyl]acetamideHomo sapiens (human)Potency1.584910
N-cyclohexyl-2-[[6-(4-ethoxyphenyl)-3-pyridazinyl]thio]acetamideHomo sapiens (human)Potency1.778310
3-(ethylthio)-6-(2-furanyl)pyridazineHomo sapiens (human)Potency28.183810
N-[3-(dimethylamino)propyl]-N-(6-methyl-1,3-benzothiazol-2-yl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency28.183810
n-(4-methylthiazol-2-yl)-2-(6-phenylpyridazin-3-ylthio)acetamideHomo sapiens (human)Potency28.183810
4-[3-(3-methylanilino)-2-imidazo[1,2-a]pyrimidinyl]phenolHomo sapiens (human)Potency3.162310
N-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-quinoline-6-sulfonamideHomo sapiens (human)Potency1.000010
2-(2,5-dichlorophenyl)sulfonyl-N-methyl-N-[(2-methylphenyl)methyl]ethanamineHomo sapiens (human)Potency5.623410
N-[2-(2-methoxyphenoxy)ethyl]-2,3-dihydro-1H-indene-5-carboxamideHomo sapiens (human)Potency28.183810
3-(diphenylmethylene)-1-[4-(4-phenyl-1-piperazinyl)butyl]pyrrolidine-2,5-dioneHomo sapiens (human)Potency28.183810
alpha-solanineHomo sapiens (human)Potency28.183810
N-[4-(1-adamantylsulfamoyl)phenyl]-4-bromo-1-methyl-3-pyrazolecarboxamideHomo sapiens (human)Potency12.589310
N-[3-(4-morpholinyl)propyl]-2,4-dioxo-3-(2-phenylethyl)-1H-quinazoline-7-carboxamideHomo sapiens (human)Potency12.589310
1-(3,5-dimethylphenyl)-3-(4-methyl-3-oxo-1,4-benzothiazin-6-yl)ureaHomo sapiens (human)Potency3.981110
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency28.183810
n-phenacylthiazolium bromideHomo sapiens (human)Potency28.183810
lissamine rhodamine bHomo sapiens (human)Potency31.622810
1-(2-cyano-3,12-dioxooleana-1,9-dien-28-oyl) imidazoleHomo sapiens (human)Potency0.316210
a 443654Homo sapiens (human)Potency2.511910
garcinone eHomo sapiens (human)Potency3.981110
2-(4-methoxyphenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency11.220210
2-(4-chlorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency14.125410
ditryptophenalineHomo sapiens (human)Potency0.446710
[4-(2-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(phenylmethyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency3.548110
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency0.562310
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency0.316210
2-[(2-chloro-1-oxoethyl)-(2,2-dimethoxyethyl)amino]-2-(4-chlorophenyl)-N-cyclohexylacetamideHomo sapiens (human)Potency5.011910
2-[2-fluoro-5-(4-methyl-1-piperazinyl)-4-nitrophenyl]-3,4-dihydro-1H-isoquinolineHomo sapiens (human)Potency11.220210
4-[3-(2-furanyl)-4-(3-nitrophenyl)-6-oxo-2,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoic acid ethyl esterHomo sapiens (human)Potency10.000010
N-butyl-3-[1-[(2,5-dimethylphenyl)methyl]-2,4-dioxo-3-quinazolinyl]propanamideHomo sapiens (human)Potency5.011910
5-(1,3-benzodioxol-5-ylmethyl)-4-methyl-2-[[1-naphthalenyl(oxo)methyl]amino]-3-thiophenecarboxamideHomo sapiens (human)Potency31.622810
4-(4-chlorophenyl)sulfonyl-5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-ethylsulfonylthiazoleHomo sapiens (human)Potency1.122010
[9-(benzenesulfonyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinolin-8-yl]-(4-methylphenyl)methanoneHomo sapiens (human)Potency3.548110
2-(3-chlorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency8.912510
ortho-topolin ribosideHomo sapiens (human)Potency0.707910
dehydrocurvularinHomo sapiens (human)Potency28.183810
malyngamide AHomo sapiens (human)Potency0.501210
3-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-2,4-dioxo-1H-quinazoline-7-carboxamideHomo sapiens (human)Potency3.548110
4-chloro-N-[3-(3-methyl-1-piperidinyl)propyl]-2-thieno[3,2-c]quinolinecarboxamideHomo sapiens (human)Potency3.162310
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)Potency3.981110
(3-propan-2-yloxyphenyl)-[1-[(1-propan-2-yl-4-pyrazolyl)methyl]-3-piperidinyl]methanoneHomo sapiens (human)Potency1.995310
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[3-(4-fluorophenyl)-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetamideHomo sapiens (human)Potency31.622810
8-methyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-5H-thieno[3,2-c]quinoline-2-carboxamideHomo sapiens (human)Potency28.183810
1-(1-piperidinyl)-3-[4-[[2-[4-(trifluoromethyl)phenyl]ethylamino]methyl]phenoxy]-2-propanolHomo sapiens (human)Potency0.891310
[3-(1-methyl-2-pyrrolyl)-1H-pyrazol-5-yl]-[1-(2-pyridinyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methanoneHomo sapiens (human)Potency7.079510
N-(2-furanylmethyl)-2-[[4-oxo-3-[3-(1-pyrrolidinyl)propyl]-[1]benzothiolo[3,2-d]pyrimidin-2-yl]thio]acetamideHomo sapiens (human)Potency10.000010
2-(3,5-dimethyl-1-pyrazolyl)-1-[3-[oxo-(3-propan-2-yloxyphenyl)methyl]-1-piperidinyl]ethanoneHomo sapiens (human)Potency28.183810
1-[[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-4-pyrazolyl]methyl]-4-methoxypiperidineHomo sapiens (human)Potency5.011910
N-[[3-(3-methylphenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-3-(1-pyrazolyl)-1-propanamineHomo sapiens (human)Potency15.848910
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)Potency28.183810
[1-[(6-chloro-2H-1-benzopyran-3-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)Potency1.778310
[1-[(1,2-dimethyl-3-indolyl)methyl]-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolHomo sapiens (human)Potency8.912510
1-(5-isoquinolinylmethyl)-4-[(3-methoxyphenyl)methyl]-4-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency28.183810
5-[[1-(2-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methyl]-2-methylthiazoleHomo sapiens (human)Potency3.981110
[1-[[1-(5-chloro-2-pyridinyl)-2-pyrrolyl]methyl]-3-piperidinyl]-(2,4-dimethoxyphenyl)methanoneHomo sapiens (human)Potency14.125410
1-[[3-(2-fluorophenyl)-1-methyl-4-pyrazolyl]methyl]-3-propoxypiperidineHomo sapiens (human)Potency5.011910
1-(2-chloro-4-methylphenyl)-3-[[1-[(3-chlorophenyl)methyl]-4-piperidinyl]methyl]ureaHomo sapiens (human)Potency28.183810
N-[3-(1-azepanyl)propyl]-3-[(4-methoxyphenyl)methyl]-2,4-dioxo-1H-quinazoline-7-carboxamideHomo sapiens (human)Potency12.589310
4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidineHomo sapiens (human)Potency28.183810
N-(4-ethoxyphenyl)-2-[4-[2-(methylthio)ethyl]-2,5-dioxo-1-imidazolidinyl]acetamideHomo sapiens (human)Potency10.000010
2-[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)amino]-1-(4-nitrophenyl)ethanolHomo sapiens (human)Potency12.589310
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideHomo sapiens (human)Potency10.000010
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideHomo sapiens (human)Potency28.183810
(5S)-1-(4-cyclohexylbutyl)-5-phenyl-4,5-dihydroimidazol-2-amineHomo sapiens (human)Potency11.220210
(5R)-1-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]-5-butyl-4,5-dihydroimidazol-2-amineHomo sapiens (human)Potency7.943310
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterHomo sapiens (human)Potency8.912510
1-[1-(4-butan-2-ylphenyl)ethyl]-3-[(4-fluorophenyl)methyl]thioureaHomo sapiens (human)Potency10.000010
N-butyl-4-(phenylmethyl)-1-piperidinecarbothioamideHomo sapiens (human)Potency5.011910
2-(2,5-dichlorophenoxy)-1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-butanoneHomo sapiens (human)Potency2.818410
1-[(4-fluorophenyl)methyl]-3-[1-(4-propan-2-ylphenyl)propyl]thioureaHomo sapiens (human)Potency28.183810
1-(3-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)thioureaHomo sapiens (human)Potency5.011910
N-[2-(2,5-dimethoxyphenyl)ethyl]-4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazine-6-carboxamideHomo sapiens (human)Potency5.011910
5-fluoro-2-phenyl-1,2-benzothiazol-3-oneHomo sapiens (human)Potency12.589310
2-(2-fluorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency8.912510
3-[1-[[1-(4-methylphenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneHomo sapiens (human)Potency3.162310
fractalsHomo sapiens (human)Potency3.162310
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency28.183810
4-(1-((5-((2,6-dimethylphenoxy)methyl)-3-isoxazolyl)carbonyl)-4-piperidinyl)pyridineHomo sapiens (human)Potency11.220210
1-[(2,3-dimethyl-4-imidazolyl)methyl]-N-[4-(2-furanyl)phenyl]-3-piperidinecarboxamideHomo sapiens (human)Potency7.943310
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideHomo sapiens (human)Potency0.707910
(2R)-N2-[2-(4-bicyclo[2.2.1]heptanyl)ethyl]-N1-[(2R,3R)-3-methyl-1-(methylamino)pentan-2-yl]hexane-1,2-diamineHomo sapiens (human)Potency3.162310
4-[(2S)-2-[2-(4-ethoxyphenyl)ethylamino]-3-[[(2S)-1-(methylamino)hexan-2-yl]amino]propyl]phenolHomo sapiens (human)Potency7.943310
(2R)-3-[[(2S)-1-cyclohexyl-3-(methylamino)propan-2-yl]amino]-2-[2-[3-(trifluoromethyl)phenyl]ethylamino]-1-propanolHomo sapiens (human)Potency3.981110
N-[2-[1-[(4-methoxy-3-methylphenyl)methyl]-4-piperidinyl]-3-pyrazolyl]-4-phenylbutanamideHomo sapiens (human)Potency1.778310
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamideHomo sapiens (human)Potency2.238710
[2-(2-methoxyethyl)-1-piperidinyl]-[5-[[4-(1,2,4-triazol-1-yl)phenoxy]methyl]-3-isoxazolyl]methanoneHomo sapiens (human)Potency1.778310
N-methyl-N-(3-pyridinylmethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-yloxymethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency31.622810
1-[(1-ethyl-3-methyl-4-pyrazolyl)methyl]-N-[4-(2-fluorophenoxy)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency8.912510
2-[[[4-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterHomo sapiens (human)Potency11.220210
5-[(3,4-dimethylphenoxy)methyl]-N-methyl-N-(4-oxanylmethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency2.818410
2-(2,6-dimethylphenoxy)-N-[2-(1-piperidinyl)phenyl]acetamideHomo sapiens (human)Potency6.309610
(5S)-1-heptyl-5-(2-methylpropyl)-N-phenyl-4,5-dihydroimidazol-2-amineHomo sapiens (human)Potency12.589310
4-(4-acetyloxyphenyl)benzoic acid [2-[[2-(2-chloroanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] esterHomo sapiens (human)Potency28.183810
2-(3-oxo-1,2-benzothiazol-2-yl)-N-phenylacetamideHomo sapiens (human)Potency10.000010
3-furanyl-[4-[5-(2-furanyl)-2-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]methanoneHomo sapiens (human)Potency28.183810
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamideHomo sapiens (human)Potency14.125410
3-benzyl-4-hydroxyquinolin-2(1H)-oneHomo sapiens (human)Potency28.183810
kf38789Homo sapiens (human)Potency1.995310
6-[5-[[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]methyl]-2-oxo-1,3-dihydroimidazol-4-yl]-6-oxohexanoic acid ethyl esterHomo sapiens (human)Potency11.220210
azaguanineHomo sapiens (human)Potency2.818410
N-tert-butyl-3-(3-tert-butyl-1-methyl-7-oxo-4H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxybenzenesulfonamideHomo sapiens (human)Potency15.848910
salicylaldehyde thiosemicarbazoneHomo sapiens (human)Potency0.891310
7-methyl-2-[(4-methyl-6-phenyl-2-pyrimidinyl)amino]-1H-quinazolin-4-oneHomo sapiens (human)Potency1.000010
N-[4-[2-[3-(dimethylsulfamoyl)anilino]-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideHomo sapiens (human)Potency28.183810
1-[4-[[oxo-(7-oxo-4H-isothiazolo[4,3-d]pyrimidin-3-yl)methyl]amino]phenyl]-3-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency5.011910
pyridoxal 4-methoxybenzoyl hydrazoneHomo sapiens (human)Potency5.011910
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency28.183810
2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]acetamideHomo sapiens (human)Potency12.589310
5-(4-chlorophenyl)-3-(4-nitrophenyl)-1H-pyrazoleHomo sapiens (human)Potency28.183810

Enables

This protein enables 3 target(s):

TargetCategoryDefinition
hormone activitymolecular functionThe action characteristic of a hormone, any substance formed in very small amounts in one specialized organ or group of cells and carried (sometimes in the bloodstream) to another organ or group of cells in the same organism, upon which it has a specific regulatory action. The term was originally applied to agents with a stimulatory physiological action in vertebrate animals (as opposed to a chalone, which has a depressant action). Usage is now extended to regulatory compounds in lower animals and plants, and to synthetic substances having comparable effects; all bind receptors and trigger some biological process. [GOC:dph, GOC:mah, ISBN:0198506732]
protein bindingmolecular functionBinding to a protein. [GOC:go_curators]
follicle-stimulating hormone activitymolecular functionThe action characteristic of follicle-stimulating hormone (FSH), a gonadotrophic glycoprotein hormone secreted, in mammals, by the anterior pituitary gland. Upon receptor binding, FSH stimulates growth of Graafian follicles in the ovaries in females, and stimulates the epithelium of the seminiferous tubules to increase spermatogenesis. [ISBN:0198547684]

Located In

This protein is located in 3 target(s):

TargetCategoryDefinition
extracellular regioncellular componentThe space external to the outermost structure of a cell. For cells without external protective or external encapsulating structures this refers to space outside of the plasma membrane. This term covers the host cell environment outside an intracellular parasite. [GOC:go_curators]
extracellular spacecellular componentThat part of a multicellular organism outside the cells proper, usually taken to be outside the plasma membranes, and occupied by fluid. [ISBN:0198547684]
Golgi lumencellular componentThe volume enclosed by the membranes of any cisterna or subcompartment of the Golgi apparatus, including the cis- and trans-Golgi networks. [GOC:mah]

Active In

This protein is active in 1 target(s):

TargetCategoryDefinition
extracellular spacecellular componentThat part of a multicellular organism outside the cells proper, usually taken to be outside the plasma membranes, and occupied by fluid. [ISBN:0198547684]

Part Of

This protein is part of 2 target(s):

TargetCategoryDefinition
follicle-stimulating hormone complexcellular componentA gonadotrophic glycoprotein hormone secreted, in mammals, by the anterior pituitary gland; consists of alpha and beta subunits, the latter of which confers hormonal specificity. [ISBN:0198547684]
pituitary gonadotropin complexcellular componentA protein complex that is a protein hormone secreted by gonadotrope cells of the anterior pituitary of vertebrates. capable of regulating normal growth, sexual development, and reproductive function. [GOC:dph, PMID:11420129]

Involved In

This protein is involved in 14 target(s):

TargetCategoryDefinition
G protein-coupled receptor signaling pathwaybiological processThe series of molecular signals initiated by a ligand binding to its receptor, in which the activated receptor promotes the exchange of GDP for GTP on the alpha-subunit of an associated heterotrimeric G-protein complex. The GTP-bound activated alpha-G-protein then dissociates from the beta- and gamma-subunits to further transmit the signal within the cell. The pathway begins with receptor-ligand interaction, and ends with regulation of a downstream cellular process. The pathway can start from the plasma membrane, Golgi or nuclear membrane. [GOC:bf, GOC:mah, PMID:16902576, PMID:24568158, Wikipedia:G_protein-coupled_receptor]
positive regulation of cell population proliferationbiological processAny process that activates or increases the rate or extent of cell proliferation. [GOC:go_curators]
hormone-mediated signaling pathwaybiological processThe series of molecular signals mediated by the detection of a hormone. [GOC:sm]
regulation of signaling receptor activitybiological processAny process that modulates the frequency, rate or extent of a signaling receptor activity. Receptor activity is when a molecule combines with an extracellular or intracellular messenger to initiate a change in cell activity. [GOC:dph, GOC:tb]
positive regulation of steroid biosynthetic processbiological processAny process that increases the frequency, rate or extent of the chemical reactions and pathways resulting in the formation of steroids, compounds with a 1,2,cyclopentanoperhydrophenanthrene nucleus. [GOC:tb]
positive regulation of cell migrationbiological processAny process that activates or increases the frequency, rate or extent of cell migration. [GOC:go_curators]
thyroid gland developmentbiological processThe process whose specific outcome is the progression of the thyroid gland over time, from its formation to the mature structure. The thyroid gland is an endoderm-derived gland that produces thyroid hormone. [GOC:dgh]
luteinizing hormone secretionbiological processThe regulated release of luteinizing hormone, a gonadotropic glycoprotein hormone secreted by the anterior pituitary. [ISBN:0198506732]
organ growthbiological processThe increase in size or mass of an organ. Organs are commonly observed as visibly distinct structures, but may also exist as loosely associated clusters of cells that function together as to perform a specific function. [GOC:bf, ISBN:0471245208, ISBN:0721662544]
follicle-stimulating hormone signaling pathwaybiological processA G protein-coupled receptor signaling pathway initiated by follicle-stimulating hormone binding to its receptor on the surface of a target cell, and ending with the regulation of a downstream cellular process. [GOC:dph]
positive regulation of transcription by RNA polymerase IIbiological processAny process that activates or increases the frequency, rate or extent of transcription from an RNA polymerase II promoter. [GOC:go_curators, GOC:txnOH]
negative regulation of organ growthbiological processAny process that stops, prevents, or reduces the frequency, rate or extent of growth of an organ of an organism. [GOC:bf, GOC:tb]
follicle-stimulating hormone secretionbiological processThe regulated release of follicle-stimulating hormone, a gonadotropic glycoprotein hormone secreted by the anterior pituitary. [ISBN:0198506732]
thyroid hormone generationbiological processThe formation of either of the compounds secreted by the thyroid gland, mainly thyroxine and triiodothyronine. This is achieved by the iodination and joining of tyrosine molecules to form the precursor thyroglobin, proteolysis of this precursor gives rise to the thyroid hormones. [GOC:jl, ISBN:0716720094]