A dual specificity tyrosine-phosphorylation-regulated kinase 1A that is encoded in the genome of rat. [OMA:Q63470, PRO:DNx]
EC 2.7.12.1;
Dual specificity YAK1-related kinase;
Protein kinase minibrain homolog;
MNBH;
RP86
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (6.67) | 29.6817 |
| 2010's | 12 (80.00) | 24.3611 |
| 2020's | 2 (13.33) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| nsc 664704 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| staurosporine | Rattus norvegicus (Norway rat) | IC50 | 0.0120 | 1 | 1 |
| epigallocatechin gallate | Rattus norvegicus (Norway rat) | IC50 | 0.3300 | 1 | 1 |
| cercosporamide | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| cyc 202 | Rattus norvegicus (Norway rat) | IC50 | 11.0000 | 1 | 1 |
| paullone | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| meridianin g | Rattus norvegicus (Norway rat) | IC50 | 0.7000 | 1 | 1 |
| 6-bromoindirubin-3'-oxime | Rattus norvegicus (Norway rat) | IC50 | 1.1100 | 2 | 2 |
| harmine | Rattus norvegicus (Norway rat) | IC50 | 0.0397 | 3 | 3 |
| alvocidib | Rattus norvegicus (Norway rat) | IC50 | 0.3000 | 1 | 1 |
| leucettamine b | Rattus norvegicus (Norway rat) | IC50 | 1.5400 | 3 | 3 |
| ageladine a | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| meriolin 3 | Rattus norvegicus (Norway rat) | IC50 | 0.0290 | 1 | 1 |
| chr-6494 | Rattus norvegicus (Norway rat) | IC50 | 0.0130 | 1 | 1 |
| ((5z)5-(1,3-benzodioxol-5-yl)methylene-2-phenylamino-3,5-dihydro-4h-imidazol-4-one) | Rattus norvegicus (Norway rat) | IC50 | 0.0300 | 3 | 3 |
| 7-bromoindirubin-3'-oxime | Rattus norvegicus (Norway rat) | IC50 | 1.9000 | 1 | 1 |