angiogenesis inhibitor

An agent and endogenous substances that antagonize or inhibit the development of new blood vessels.

ChEBI ID: 48422

Members (56)

Member	Definition	Class
2-methyl-1,4-hydroquinone	A member of the class of hydroquinones that is hydroquinone in which one of the benzene hydrogens has been replaced by a methyl group.	toluquinol
3-(3-pyridinyl)-1-(4-pyridinyl)-2-propen-1-one	A member of the class of pyridines that is pyridine substituted by a 3-oxo-3-(pyridin-4-yl)prop-1-en-1-yl group at position 3. An inhibitor of PFKFB3 kinase, an enzyme with a key role in glycolysis.	3PO
abt 869	A member of the class of phenylureas that is urea in which one of the nitrogens is substituted by a 2-fluoro-5-methylphenyl group, while the other is substituted by a p-(3-amino-1H-indazol-4-yl)phenyl group. It is a potent, selective inhibitor of vascular endothelial growth factor and platelet-derived growth factor receptor tyrosine kinases.	linifanib
acetopyrrothine	A dithiolopyrrolone antibiotic that is 4,5-dihydro[1,2]dithiolo[4,3-b]pyrrole in which the hydrogens at positions 4,5 and 6 have been replaced by methyl, oxo and acetamido groups, respectively. It is a potent inhibitor of RNA polymerases, inhibits the angiogenesis of human umbilical vein endothelial cells, and also inhibits JAMM metalloproteases.	thiolutin
aee 788	A 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-N-(1-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine which adopts an R-configuration. It is a potent inhibitor of human EGFR, VEGFR and HER2 receptor tyrosine kinases and exhibits anticancer and antiangiogenic activity.	AEE788
ageladine a	An imidazopyridine that is 1H-imidazo[4,5-c]pyridin-2-amine substituted by a 4,5-dibromo-1H-pyrrol-2-yl group at position 4. It is an alkaloid isolated from a marine sponge Agelas nakamurai and acts as an inhibitor of the matrix metalloproteinases, the key enzymes involved in tumour growth, migration, angiogenesis, invasion and metastasis.	ageladine A
amentoflavone	A biflavonoid that is obtained by oxidative coupling of two molecules of apigenin resulting in a bond between positions C-3 of the hydroxyphenyl ring and C-8 of the chromene ring. A natural product found particularly in Ginkgo biloba and Hypericum perforatum.	amentoflavone
antofine	An organic heteropentacyclic compound that is (13aR)-9,11,12,13,13a,14-hexahydrodibenzo[f,h]pyrrolo[1,2-b]isoquinoline substituted at positions 2, 3 and 6 by methoxy groups. It is an alkaloid produced by relatives of the milkweed family and exhibits antiviral, anti-inflammatory, antiadipogenic and antitumorigenic activities.	(-)-antofine
ascochlorin	A dihydroxybenzaldehyde that is 2,4-dihydroxybenzaldehyde which is substituted by a (1E,3E)-3-methyl-1-[(1R,2R,6R)-1,2,6-trimethyl-3-oxocyclohexyl]penta-1,3-dien-5-yl group at position 3, chlorine at position 5, and a methyl group at position 6. A meroterpenoid produced by several fungi including Ascochyta viciae . It exhibits anticancer, antifungal and antiprotozoal activities.	ascochlorin
ascofuranone	A dihydroxybenzaldehyde that is 2,4-dihydroxybenzaldehyde which is substituted by a (2E,6E)-7-[(2S)-5,5-dimethyl-4-oxotetrahydrofuran-2-yl]-3-methylocta-2,6-dien-1-yl group at position 3, chlorine at position 5, and a methyl group at position 6. A meroterpenoid produced by the soil fungus, Acremonium sclerotigenum. It is a promising drug candidate against the tropical disease, African trypanosomiasis.	ascofuranone
aureothricin	A dithiolopyrrolone antibiotic that is 4,5-dihydro[1,2]dithiolo[4,3-b]pyrrole in which the hydrogens at positions 4,5 and 6 have been replaced by methyl, oxo and propanoylamino groups, respectively. It is a moderate antimicrobial by-product of the thiolutin fermentation in various Streptomyces species.	aureothricin
baicalein	A trihydroxyflavone with the hydroxy groups at positions C-5, -6 and -7.	baicalein
batimastat	A secondary carboxamide resulting from the formal condensation of the carboxy group of (2S,3R)-5-methyl-3-{[(2S)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]carbamoyl}-2-[(thiophen-2-ylsulfanyl)methyl]hexanoic acid with the amino group of hydroxylamine. It a broad-spectrum matrix metalloprotease inhibitor.	batimastat
bms 387032	A secondary carboxamide resulting from the formal condensation of the carboxy group of piperidine-4-carboxylic acid with the amino group of 5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-amine. It is an ATP-competitive inhibitor of CDK2, CDK7 and CDK9 kinases and exhibits anti-cancer properties.	N-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide
brivanib	A secondary alcohol resulting from the hydrolysis of the carboxylic ester group of brivanib alaninate. It is a dual VEGFR-2/FGFR-1 kinase inhibitor whose alanine prodrug, brivanib alaninate is currently under development as an oral agent for the treatment of cancer.	(2R)-1-[[4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methyl-6-pyrrolo[2,1-f][1,2,4]triazinyl]oxy]-2-propanol; brivanib
cafestol	An organic heteropentacyclic compound and furan diterpenoid with formula C20H28O3 obtained from the unsaponifiable fraction of coffee oil (a lipid fraction obtained from coffee beans by organic solvent extraction).	cafestol
can 508	A member of the class of pyrazoles that is 1H-pyrazole substituted by amino, (4-hydroxyphenyl)diazenyl, and amino groups at positions 3, 4 and 5, respectively. It is a CDK9 inhibitor (IC50 = 0.35 muM) with 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes.	CAN-508
capsiate	A carboxylic ester obtained by formal condensation of the carboxy group of (6E)-8-methylnon-6-enoic acid with the benzylic hydroxy group of vanillyl alcohol. A non-pungent analogue of capsaicin with a similar biological profile.	capsiate
crenolanib	A member of the class of benzimidazoles that is 1H-benzimidazole which is substituted by a 8-(4-aminopiperidin-1-yl)quinolin-2-yl group at position 1 and by a (3-methyloxetan-3-yl)methoxy group at position 5. It is an inhibitor of type III tyrosine kinases, PDGFRalpha/beta and FLT3 (IC50 of 11, 3.2, and 4 nM). Currently under clinical development for the treatment of acute myeloid leukemia.	crenolanib
deguelin	A rotenone that is 13,13a-dihydro-3H-chromeno[3,4-b]pyrano[2,3-h]chromen-7(7aH)-one substituted by methoxy groups at positions 9 and 10, and by two methyl groups at position 3 (the 7aS,13aS-stereoisomer). It exists in abundant quantities in the bark, roots, and leaves of the Leguminosae family of plants and reported to exert anti-tumour effects in various cancers.	deguelin
diosmetin	A monomethoxyflavone that is the 4'-methyl ether derivative of luteolin. It is a natural product isolated from citrus fruits which exhibits a range of pharmacological activities.	diosmetin
disulfiram	An organic disulfide that results from the formal oxidative dimerisation of N,N-diethyldithiocarbamic acid. A multi-enzyme inhibitor that is used in alcohol aversion therapy and also exhibits anticancer properties.	disulfiram
EG00229	A member of the class of thiophenes that is thiophene substituted by a carbonyl-L-arginine and (2,1,3-benzothiadiazole-4-sulfonyl)amino groups at positions 2 and 3. It is an inhibitor of the neuropilin-1 and VEGF-A interaction and a potential anti-cancer agent.	EG00229
fumagillin	A meroterpenoid resulting from the formal condensation of the hydroxy group of fumagillol with the carboxylic acid group of (all-E)-deca-2,4,6,8-tetraenedioic acid. Originally isolated from the fungus Aspergillus fumigatus, it is used for the control of Nosema infection in honey bees.	fumagillin
herbacetin	A pentahydroxyflavone that is kaempferol substituted by a hydroxy group at position 8. It is a natural flavonoid from flaxseed which exerts antioxidant, anti-inflammatory and anticancer activities.	herbacetin
jq1 compound	A member of the class of thienotriazolodiazepines that is the tert-butyl ester of [(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetic acid. An inhibitor of bromodomain-containing protein 4 that exhibits anti-cancer and cardioprotective properties.	JQ1
kahweol	A diterpenoid with formula C20H26O3, isolated from the beans of Coffea arabica. It exhibits antioxidant, anti-inflammatory, anti-angiogenesis and anti-proliferative properties.	kahweol
lenalidomide	A dicarboximide that consists of 1-oxoisoindoline bearing an amino substituent at position 4 and a 2,6-dioxopiperidin-3-yl group at position 2. Inhibits the secretion of TNF-alpha.	lenalidomide
lupulon	A beta-bitter acid in which the acyl group is specified as 3-methylbutanoyl.	lupulone
luteolin	A tetrahydroxyflavone in which the four hydroxy groups are located at positions 3', 4', 5 and 7. It is thought to play an important role in the human body as an antioxidant, a free radical scavenger, an anti-inflammatory agent and an immune system modulator as well as being active against several cancers.	luteolin
matairesinol	A lignan that is gamma-butyrolactone in which the 3 and 4 positions are substituted by 4-hydroxy-3-methoxybenzyl groups (the 3R,4R-diastereomer).	(-)-matairesinol
n-(3-(aminomethyl)benzyl)acetamidine	An aralkylamine that is Nbenzylacetamidine substituted at position 3 on the benzene ring by an aminomethyl group. An inhibitor of nitric oxide synthase.	N-[3-(aminomethyl)benzyl]acetamidine
nnc 55-0396	The dihydrochloride salt of NNC 55-0396. It is a stable analogue of mibefradil and a highly selective T-type calcium channel blocker.	NNC 55-0396 dihydrochloride
NNC 55-0396 (free base)		NNC 55-0396 (free base)
npi 2358	A member of the class of 2,5-diketopiperazines that is piperazine-2,5-dione substituted by benzylidene and (5-tert-butyl-1H-imidazol-4-yl)methylidene groups at positions 3 and 6, respectively. It is a vascular disrupting agent and a microtubule destabalising agent which was in clinical trials (now discontinued) for the treatment of non-small cell lung cancer.	plinabulin
o-(chloroacetylcarbamoyl)fumagillol	A carbamate ester that is fumagillol in which the hydroxy group has been converted to the corresponding N-(chloroacetyl)carbamate derivative.	O-(chloroacetylcarbamoyl)fumagillol
oridonin	An organic heteropentacyclic compound and ent-kaurane diterpenoid with formula C20H28O6 isolated from the leaves of the medicinal herb Rabdosia rubescens.	oridonin
pd 166866	A member of the class of pyridopyrimidines that is pyrido[2,3-d]pyrimidine substituted by an amino group at position 2, 3,5-dimethoxyphenyl group at position 6, and by a (tert-butylcarbamoyl)nitrilo group at position 7. It is a selective ATP competitive inhibitor of the human fibroblast growth factor-1 receptor (FGFR1) tyrosine kinase with an IC50 of 52.4 nM.	PD-166866
pj-34	A member of the class of phenanthridines that is 5,6-dihydrophenanthridine substituted at positions 2 and 6 by (N,N-dimethylglycyl)amino and oxo groups, respectively. It is a potent inhibitor of poly(ADP-ribose) polymerases PARP1 and PARP2 (IC50 of 110 nM and 86 nM, respectively) and exhibits anti-cancer, cardioprotective and neuroprotective properties.	PJ34
pomalidomide	An aromatic amine that is thalidomide substituted at position 4 on the isoindole ring system by an amino group. Used for the treatment of multiple myeloma in patients who failed to respond to previous therapies.	pomalidomide
ptk 787	A succinate salt obtained by combining vatalanib with one molar equivalent of succinic acid. It is a multi-targeted tyrosine kinase inhibitor for all isoforms of VEGFR, PDGFR and c-Kit.	vatalanib succinate
quininib	A styrylquinoline that is trans-2-styrylquinoline in which the the phenyl group has been substituted at position 2 by a hydroxy group. It is an anti-angiogenic compound that exerts a dose-dependent antagonism of the cysteinyl leukotriene pathway, preferentially antagonising cysteinyl leukotriene receptor 1. The major species at pH 7.3	quininib
rhapontin	A rhaponticin in which the double bond adopts a trans-configuration. It possesses a range of pharmacological activities including antitumour, antiinflammatory, antilipemic and neuroprotective activities.	trans-rhaponticin
rifampin	A member of the class of rifamycins that is a a semisynthetic antibiotic derived from Amycolatopsis rifamycinica (previously known as Amycolatopsis mediterranei and Streptomyces mediterranei).	rifampicin zwitterion; rifampicin
sb 220025	Am member of the class of imidazoles carrying piperidin-4-yl, 4-fluophenyl and 2-aminopyrimidin-4-yl substituents at posiitons 1, 4 and 5 respectively.	SB220025
sorafenib	A member of the class of phenylureas that is urea in which one of the nitrogens is substituted by a 4-chloro-3-trifluorophenyl group while the other is substituted by a phenyl group which, in turn, is substituted at the para position by a [2-(methylcarbamoyl)pyridin-4-yl]oxy group.	sorafenib
su 11248		sunitinib
suramin	A member of the class of phenylureas that is urea in which each of the amino groups has been substituted by a 3-({2-methyl-5-[(4,6,8-trisulfo-1-naphthyl)carbamoyl]phenyl}carbamoyl)phenyl group. An activator of both the rabbit skeletal muscle RyR1 and sheep cardiac RyR2 isoform ryanodine receptor channels, it has been used for the treatment of human African trypanosomiasis for over 100 years.	suramin
suramin sodium	An organic sodium salt that is the hexasodium salt of suramin. It is an FDA approved drug for African sleeping sickness and river blindness.	suramin sodium
tamoxifen		tamoxifen
tamoxifen citrate		tamoxifen citrate
vatalanib	A member of the class of phthalazines that is phthalazine in which the hydrogens at positions 1 and 4have been replaced by a p-chlorophenylamino group and a pyridin-4-ylmethyl group, respectively. It is a multi-targeted tyrosine kinase inhibitor for all isoforms of VEGFR, PDGFR and c-Kit.	vatalanib
ver 52296	A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 5-(2,4-dihydroxy-5-isopropylphenyl)-4-[4-(morpholin-4-ylmethyl)phenyl]-1,2-oxazole-3-carboxylic acid with the amino group of ethylamine.	luminespib
vitamin k 3	A member of the class of 1,4-naphthoquinones that is 1,4-naphthoquinone which is substituted at position 2 by a methyl group. It is used as a nutritional supplement and for the treatment of hypoprothrombinemia.	menadione
voacamine	A monoterpenoid indole alkaloid with formula C22H28N2O3, isolated from several plant species.	(-)-voacangine
wogonin	A dihydroxy- and monomethoxy-flavone in which the hydroxy groups are positioned at C-5 and C-7 and the methoxy group is at C-8.	wogonin

Research

Studies (66,885)

Timeframe	Studies, Drugs with This Role(%)	All Drugs %
pre-1990	11,449 (17.12)	18.7374
1990's	8,930 (13.35)	18.2507
2000's	14,553 (21.76)	29.6817
2010's	23,859 (35.67)	24.3611
2020's	8,094 (12.10)	2.80

Study Types

Publication Type	Studies, Drugs with this Role (%)	All Drugs (%)
Trials	6,302 (8.70%)	5.53%
Reviews	7,569 (10.45%)	6.00%
Case Studies	6,353 (8.78%)	4.05%
Observational	298 (0.41%)	0.25%
Other	51,874 (71.65%)	84.16%

Protein Targets (1,248)

Potency Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1	Homo sapiens (human)	Potency	10.9165	1	11
15-lipoxygenase, partial	Homo sapiens (human)	Potency	5.5253	1	7
67.9K protein	Vaccinia virus	Potency	13.3499	2	9
acetylcholinesterase	Homo sapiens (human)	Potency	58.5840	4	18
acid sphingomyelinase	Homo sapiens (human)	Potency	89.1251	1	1
activating transcription factor 6	Homo sapiens (human)	Potency	32.6305	2	16
aldehyde dehydrogenase 1 family, member A1	Homo sapiens (human)	Potency	14.9990	1	16
alpha-galactosidase	Homo sapiens (human)	Potency	50.1187	1	1
Alpha-synuclein	Homo sapiens (human)	Potency	16.3696	1	5
Amyloid-beta precursor protein	Homo sapiens (human)	Potency	5.1735	1	1
apical membrane antigen 1, AMA1	Plasmodium falciparum 3D7	Potency	28.3627	1	3
AR protein	Homo sapiens (human)	Potency	26.3833	10	80
aryl hydrocarbon receptor	Homo sapiens (human)	Potency	30.4024	3	11
arylsulfatase A	Homo sapiens (human)	Potency	5.3582	1	1
ATAD5 protein, partial	Homo sapiens (human)	Potency	11.1375	4	8
Ataxin-2	Homo sapiens (human)	Potency	40.6377	2	12
ATP-dependent phosphofructokinase	Trypanosoma brucei brucei TREU927	Potency	15.3454	5	11
ATPase family AAA domain-containing protein 5	Homo sapiens (human)	Potency	44.9017	2	15
atrial natriuretic peptide receptor 1 precursor	Homo sapiens (human)	Potency	2.3934	1	1
atrial natriuretic peptide receptor 2 precursor	Homo sapiens (human)	Potency	5.2119	1	1
beta-2 adrenergic receptor	Homo sapiens (human)	Potency	10.6238	1	2
Bloom syndrome protein isoform 1	Homo sapiens (human)	Potency	11.6943	3	10
BRCA1	Homo sapiens (human)	Potency	18.7570	1	4
bromodomain adjacent to zinc finger domain 2B	Homo sapiens (human)	Potency	42.3956	1	4
caspase 7, apoptosis-related cysteine protease	Homo sapiens (human)	Potency	35.0310	1	9
caspase-1 isoform alpha precursor	Homo sapiens (human)	Potency	39.8107	1	1
caspase-3	Cricetulus griseus (Chinese hamster)	Potency	31.3341	1	6
caspase-3	Homo sapiens (human)	Potency	35.0310	1	9
Caspase-7	Cricetulus griseus (Chinese hamster)	Potency	31.3341	1	6
Cellular tumor antigen p53	Homo sapiens (human)	Potency	43.1928	3	26
cellular tumor antigen p53 isoform a	Homo sapiens (human)	Potency	15.3659	2	17
Chain A, 2-oxoglutarate Oxygenase	Homo sapiens (human)	Potency	12.0057	1	8
Chain A, ATP-DEPENDENT DNA HELICASE Q1	Homo sapiens (human)	Potency	17.5505	4	14
Chain A, Beta-lactamase	Escherichia coli K-12	Potency	32.7114	2	6
Chain A, Breast cancer type 1 susceptibility protein	Homo sapiens (human)	Potency	14.2191	1	2
Chain A, Cruzipain	Trypanosoma cruzi	Potency	16.9329	2	13
Chain A, Ferritin light chain	Equus caballus (horse)	Potency	27.7928	2	4
Chain A, HADH2 protein	Homo sapiens (human)	Potency	12.7718	2	14
Chain A, JmjC domain-containing histone demethylation protein 3A	Homo sapiens (human)	Potency	54.3177	1	6
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE	Homo sapiens (human)	Potency	7.2337	3	18
Chain A, Putative fructose-1,6-bisphosphate aldolase	Giardia intestinalis	Potency	10.4465	2	10
Chain A, TYROSYL-DNA PHOSPHODIESTERASE	Homo sapiens (human)	Potency	15.1259	2	12
Chain B, HADH2 protein	Homo sapiens (human)	Potency	12.7718	2	14
chromobox protein homolog 1	Homo sapiens (human)	Potency	24.4517	2	5
core-binding factor subunit beta isoform 2	Homo sapiens (human)	Potency	17.6943	3	5
cytochrome P450 2C19 precursor	Homo sapiens (human)	Potency	7.9113	1	8
cytochrome P450 2C9 precursor	Homo sapiens (human)	Potency	12.9128	1	6
cytochrome P450 2C9, partial	Homo sapiens (human)	Potency	16.4462	1	11
cytochrome P450 2D6	Homo sapiens (human)	Potency	14.4115	1	7
cytochrome P450 2D6 isoform 1	Homo sapiens (human)	Potency	21.0124	1	7
cytochrome P450 3A4 isoform 1	Homo sapiens (human)	Potency	17.5388	2	28
cytochrome P450 family 3 subfamily A polypeptide 4	Homo sapiens (human)	Potency	13.9527	2	11
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a	Homo sapiens (human)	Potency	13.2008	1	12
D(1A) dopamine receptor	Homo sapiens (human)	Potency	5.1014	2	3
D(1A) dopamine receptor	Sus scrofa (pig)	Potency	14.6892	1	1
Disintegrin and metalloproteinase domain-containing protein 17	Homo sapiens (human)	Potency	3.4703	1	2
DNA dC->dU-editing enzyme APOBEC-3G isoform 1	Homo sapiens (human)	Potency	27.9428	2	2
DNA polymerase beta	Homo sapiens (human)	Potency	3.9854	1	2
DNA polymerase eta isoform 1	Homo sapiens (human)	Potency	23.1951	2	7
DNA polymerase III, partial	Bacillus subtilis	Potency	29.9349	1	1
DNA polymerase iota isoform a (long)	Homo sapiens (human)	Potency	36.6778	2	9
DNA polymerase kappa isoform 1	Homo sapiens (human)	Potency	13.2029	1	16
endonuclease IV	Escherichia coli	Potency	17.8010	2	4
estrogen nuclear receptor alpha	Homo sapiens (human)	Potency	20.5990	11	104
estrogen receptor 2 (ER beta)	Homo sapiens (human)	Potency	36.7051	3	23
estrogen-related nuclear receptor alpha	Homo sapiens (human)	Potency	23.5576	10	86
euchromatic histone-lysine N-methyltransferase 2	Homo sapiens (human)	Potency	13.0388	1	21
EWS/FLI fusion protein	Homo sapiens (human)	Potency	11.9376	4	56
farnesoid X nuclear receptor	Homo sapiens (human)	Potency	36.0896	5	24
flap endonuclease 1	Homo sapiens (human)	Potency	43.9639	2	9
fructose-bisphosphate aldolase A	Oryctolagus cuniculus (rabbit)	Potency	6.3096	1	1
Fumarate hydratase	Homo sapiens (human)	Potency	26.0872	1	16
G	Vesicular stomatitis virus	Potency	16.4462	1	11
GABA theta subunit	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
galactokinase	Homo sapiens (human)	Potency	32.5259	2	2
GALC protein	Homo sapiens (human)	Potency	0.6310	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Potency	17.5388	1	14
geminin	Homo sapiens (human)	Potency	12.2316	4	24
GLI family zinc finger 3	Homo sapiens (human)	Potency	15.6191	3	27
glp-1 receptor, partial	Homo sapiens (human)	Potency	16.6351	1	3
GLS protein	Homo sapiens (human)	Potency	24.3396	2	10
glucocerebrosidase	Homo sapiens (human)	Potency	26.1355	1	11
glucocorticoid receptor [Homo sapiens]	Homo sapiens (human)	Potency	34.7278	4	23
Glutamate receptor 1	Rattus norvegicus (Norway rat)	Potency	4.7718	1	2
Glutamate receptor 2	Rattus norvegicus (Norway rat)	Potency	12.7124	2	15
Glutamate receptor 3	Rattus norvegicus (Norway rat)	Potency	4.7718	1	2
Glutamate receptor 4	Rattus norvegicus (Norway rat)	Potency	4.7718	1	2
glyceraldehyde-3-phosphate dehydrogenase isoform 1	Homo sapiens (human)	Potency	10.0000	1	1
GTP-binding nuclear protein Ran isoform 1	Homo sapiens (human)	Potency	27.6461	1	2
Guanine nucleotide-binding protein G	Homo sapiens (human)	Potency	4.4668	1	1
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)	Homo sapiens (human)	Potency	12.5893	1	1
heat shock protein beta-1	Homo sapiens (human)	Potency	26.2698	2	20
hemoglobin subunit beta	Homo sapiens (human)	Potency	22.1060	2	2
Histamine H2 receptor	Cavia porcellus (domestic guinea pig)	Potency	11.1962	2	48
histone acetyltransferase KAT2A isoform 1	Homo sapiens (human)	Potency	31.3838	1	3
histone deacetylase 9 isoform 3	Homo sapiens (human)	Potency	17.7310	1	2
Histone H2A.x	Cricetulus griseus (Chinese hamster)	Potency	39.5267	2	21
histone-lysine N-methyltransferase 2A isoform 2 precursor	Homo sapiens (human)	Potency	39.1539	1	5
HLA class I histocompatibility antigen, B alpha chain	Homo sapiens (human)	Potency	16.4462	1	11
huntingtin isoform 2	Homo sapiens (human)	Potency	23.9190	1	3
hypothetical protein, conserved	Trypanosoma brucei	Potency	15.0506	2	5
hypoxia-inducible factor 1 alpha subunit	Homo sapiens (human)	Potency	27.8007	2	20
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)	Homo sapiens (human)	Potency	16.2246	3	9
IDH1	Homo sapiens (human)	Potency	10.9111	1	3
importin subunit beta-1 isoform 1	Homo sapiens (human)	Potency	33.3202	2	3
Inositol hexakisphosphate kinase 1	Homo sapiens (human)	Potency	16.4462	1	22
Inositol monophosphatase 1	Rattus norvegicus (Norway rat)	Potency	7.0348	1	4
Integrin alpha-IIb	Homo sapiens (human)	Potency	16.7946	1	9
Integrin beta-3	Homo sapiens (human)	Potency	16.7946	1	9
Interferon beta	Homo sapiens (human)	Potency	14.4472	3	55
interleukin 8	Homo sapiens (human)	Potency	66.8242	1	1
lamin isoform A-delta10	Homo sapiens (human)	Potency	11.2702	3	14
lethal factor (plasmid)	Bacillus anthracis str. A2012	Potency	18.4528	1	11
lethal(3)malignant brain tumor-like protein 1 isoform I	Homo sapiens (human)	Potency	27.8298	1	2
Luciferase	Photinus pyralis (common eastern firefly)	Potency	18.3626	4	11
lysosomal alpha-glucosidase preproprotein	Homo sapiens (human)	Potency	45.8624	3	3
M-phase phosphoprotein 8	Homo sapiens (human)	Potency	14.4719	1	4
Microtubule-associated protein tau	Homo sapiens (human)	Potency	17.4592	2	35
mitogen-activated protein kinase 1	Homo sapiens (human)	Potency	13.4067	1	3
muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	Potency	5.5620	1	3
muscleblind-like protein 1 isoform 1	Homo sapiens (human)	Potency	23.9063	1	3
Neuronal acetylcholine receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	56.2341	1	1
Neuronal acetylcholine receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	56.2341	1	1
neuropeptide S receptor isoform A	Homo sapiens (human)	Potency	19.7830	1	2
NFKB1 protein, partial	Homo sapiens (human)	Potency	4.7427	2	8
nonstructural protein 1	Influenza A virus (A/WSN/1933(H1N1))	Potency	10.4356	1	4
NPC intracellular cholesterol transporter 1 precursor	Homo sapiens (human)	Potency	58.0479	1	1
nuclear factor erythroid 2-related factor 2 isoform 1	Homo sapiens (human)	Potency	26.6298	4	31
nuclear factor erythroid 2-related factor 2 isoform 2	Homo sapiens (human)	Potency	20.5962	1	1
nuclear factor NF-kappa-B p105 subunit isoform 1	Homo sapiens (human)	Potency	47.3936	1	2
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a	Homo sapiens (human)	Potency	27.7047	2	17
Nuclear receptor ROR-gamma	Homo sapiens (human)	Potency	29.8493	1	1
nuclear receptor ROR-gamma isoform 1	Mus musculus (house mouse)	Potency	42.2402	2	39
nuclear receptor subfamily 1, group I, member 3	Homo sapiens (human)	Potency	29.6917	3	32
Ornithine decarboxylase	Rattus norvegicus (Norway rat)	Potency	28.3708	1	2
P53	Homo sapiens (human)	Potency	39.1512	1	2
parathyroid hormone/parathyroid hormone-related peptide receptor precursor	Homo sapiens (human)	Potency	125.8920	1	1
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1	Homo sapiens (human)	Potency	54.1162	1	4
peripheral myelin protein 22	Rattus norvegicus (Norway rat)	Potency	20.9168	2	9
peripheral myelin protein 22 isoform 1	Homo sapiens (human)	Potency	21.0634	1	2
peroxisome proliferator activated receptor gamma	Homo sapiens (human)	Potency	34.2171	5	29
Peroxisome proliferator-activated receptor alpha	Homo sapiens (human)	Potency	50.1187	1	2
peroxisome proliferator-activated receptor delta	Homo sapiens (human)	Potency	33.3517	5	24
phosphoglycerate kinase	Trypanosoma brucei brucei TREU927	Potency	28.1838	1	1
phosphopantetheinyl transferase	Bacillus subtilis	Potency	34.8307	2	19
plasminogen precursor	Mus musculus (house mouse)	Potency	10.1775	1	3
Platelet-activating factor receptor	Homo sapiens (human)	Potency	14.2191	1	2
polyprotein	Zika virus	Potency	26.0872	1	16
polypyrimidine tract-binding protein 1 isoform a	Homo sapiens (human)	Potency	14.5500	2	2
polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	Potency	8.5438	1	8
Polyunsaturated fatty acid lipoxygenase ALOX15B	Homo sapiens (human)	Potency	10.1662	1	15
potassium voltage-gated channel subfamily H member 2 isoform d	Homo sapiens (human)	Potency	9.5352	1	6
PPM1D protein	Homo sapiens (human)	Potency	13.1893	1	28
pregnane X nuclear receptor	Homo sapiens (human)	Potency	18.4450	3	20
pregnane X receptor	Rattus norvegicus (Norway rat)	Potency	79.4328	1	1
progesterone receptor	Homo sapiens (human)	Potency	44.6219	3	22
pyruvate kinase	Leishmania mexicana mexicana	Potency	8.3216	2	4
pyruvate kinase PKM isoform a	Homo sapiens (human)	Potency	15.8489	2	2
pyruvate kinase PKM isoform b	Homo sapiens (human)	Potency	28.3708	2	4
Rap guanine nucleotide exchange factor 3	Homo sapiens (human)	Potency	59.6193	2	5
RAR-related orphan receptor gamma	Mus musculus (house mouse)	Potency	20.6003	2	26
ras-related protein Rab-9A	Homo sapiens (human)	Potency	91.9997	1	1
regulator of G-protein signaling 4	Homo sapiens (human)	Potency	5.7764	1	4
retinoic acid nuclear receptor alpha variant 1	Homo sapiens (human)	Potency	32.6123	3	34
retinoid X nuclear receptor alpha	Homo sapiens (human)	Potency	20.8661	4	25
runt-related transcription factor 1 isoform AML1b	Homo sapiens (human)	Potency	17.6943	3	5
serine-protein kinase ATM isoform a	Homo sapiens (human)	Potency	39.8107	1	1
serine/threonine-protein kinase mTOR isoform 1	Homo sapiens (human)	Potency	11.8094	5	8
serine/threonine-protein kinase PLK1	Homo sapiens (human)	Potency	11.0180	1	2
SMAD family member 2	Homo sapiens (human)	Potency	47.1852	3	13
SMAD family member 3	Homo sapiens (human)	Potency	47.1852	3	13
Smad3	Homo sapiens (human)	Potency	17.2863	1	8
snurportin-1	Homo sapiens (human)	Potency	33.3202	2	3
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	Potency	29.0691	1	5
survival motor neuron protein isoform d	Homo sapiens (human)	Potency	14.2728	1	6
TAR DNA-binding protein 43	Homo sapiens (human)	Potency	3.3998	1	2
TDP1 protein	Homo sapiens (human)	Potency	15.1954	2	48
thioredoxin glutathione reductase	Schistosoma mansoni	Potency	26.6514	1	2
thioredoxin reductase	Rattus norvegicus (Norway rat)	Potency	21.6856	2	5
Thrombopoietin	Homo sapiens (human)	Potency	4.7931	2	6
thyroid hormone receptor beta isoform 2	Rattus norvegicus (Norway rat)	Potency	13.9030	3	33
thyroid hormone receptor beta isoform a	Homo sapiens (human)	Potency	40.9168	4	7
thyroid stimulating hormone receptor	Homo sapiens (human)	Potency	39.0962	6	34
thyrotropin-releasing hormone receptor	Homo sapiens (human)	Potency	27.1740	2	10
transcriptional regulator ERG isoform 3	Homo sapiens (human)	Potency	11.2202	1	1
tyrosine-protein kinase Yes	Homo sapiens (human)	Potency	14.4834	2	11
ubiquitin carboxyl-terminal hydrolase 2 isoform a	Homo sapiens (human)	Potency	3.4703	1	2
urokinase plasminogen activator surface receptor precursor	Mus musculus (house mouse)	Potency	10.1775	1	3
urokinase-type plasminogen activator precursor	Mus musculus (house mouse)	Potency	10.1775	1	3
USP1 protein, partial	Homo sapiens (human)	Potency	38.6476	2	16
v-jun sarcoma virus 17 oncogene homolog (avian)	Homo sapiens (human)	Potency	16.4073	2	24
vitamin D (1,25- dihydroxyvitamin D3) receptor	Homo sapiens (human)	Potency	26.2985	5	28
vitamin D3 receptor isoform VDRA	Homo sapiens (human)	Potency	26.2830	1	13
Voltage-dependent calcium channel gamma-2 subunit	Mus musculus (house mouse)	Potency	13.9340	1	13
Vpr	Human immunodeficiency virus 1	Potency	26.2000	1	2
WRN	Homo sapiens (human)	Potency	17.1205	2	4

Inhibition Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a	Homo sapiens (human)	IC50	6.4860	2	4
1-deoxy-D-xylulose 5-phosphate reductoisomerase	Escherichia coli K-12	IC50	2.8000	1	2
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1	Bos taurus (cattle)	IC50	29.0000	1	1
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1	Homo sapiens (human)	IC50	29.0000	1	1
10 kDa chaperonin	Escherichia coli	IC50	52.8750	4	4
10 kDa heat shock protein, mitochondrial	Homo sapiens (human)	IC50	57.5000	2	2
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase	Homo sapiens (human)	IC50	0.0120	1	1
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase	Homo sapiens (human)	Ki	0.0050	1	1
3-oxoacyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	4.0000	1	1
3-oxoacyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	Ki	1.3000	2	2
4-aminobutyrate aminotransferase, mitochondrial	Homo sapiens (human)	IC50	12,800.0000	1	1
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	IC50	26.0800	2	2
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	Ki	1.1810	1	1
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	Ki	6.9490	1	1
5-hydroxytryptamine receptor 1B	Rattus norvegicus (Norway rat)	IC50	26.0800	2	2
5-hydroxytryptamine receptor 1B	Rattus norvegicus (Norway rat)	Ki	6.9490	1	1
5-hydroxytryptamine receptor 1D	Rattus norvegicus (Norway rat)	IC50	40.0000	1	1
5-hydroxytryptamine receptor 1D	Sus scrofa (pig)	Ki	4.0940	1	1
5-hydroxytryptamine receptor 1F	Rattus norvegicus (Norway rat)	IC50	40.0000	1	1
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	IC50	4.8010	1	1
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	Ki	1.6655	2	2
5-hydroxytryptamine receptor 2B	Homo sapiens (human)	IC50	18.3155	1	2
5-hydroxytryptamine receptor 2B	Homo sapiens (human)	Ki	7.7887	2	3
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	IC50	0.4600	1	1
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	Ki	1.0710	3	3
5-hydroxytryptamine receptor 3A	Homo sapiens (human)	IC50	0.0250	1	1
5-hydroxytryptamine receptor 3B	Homo sapiens (human)	IC50	0.0250	1	1
5-hydroxytryptamine receptor 3C	Homo sapiens (human)	IC50	0.0250	1	1
5-hydroxytryptamine receptor 3D	Homo sapiens (human)	IC50	0.0250	1	1
5-hydroxytryptamine receptor 3E	Homo sapiens (human)	IC50	0.0250	1	1
5-hydroxytryptamine receptor 4	Cavia porcellus (domestic guinea pig)	IC50	0.4600	1	1
5-hydroxytryptamine receptor 4	Cavia porcellus (domestic guinea pig)	Ki	0.2410	1	1
5-hydroxytryptamine receptor 5A	Homo sapiens (human)	Ki	3.2960	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	IC50	9.3400	1	2
5-hydroxytryptamine receptor 6	Homo sapiens (human)	Ki	3.9818	3	4
5-hydroxytryptamine receptor 7	Homo sapiens (human)	IC50	350.0000	1	2
5-hydroxytryptamine receptor 7	Homo sapiens (human)	Ki	7.0710	1	1
5'-AMP-activated protein kinase catalytic subunit alpha-1	Homo sapiens (human)	IC50	0.1580	1	1
5'-AMP-activated protein kinase catalytic subunit alpha-2	Homo sapiens (human)	IC50	0.0617	1	1
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3	Homo sapiens (human)	IC50	49.3000	3	3
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3	Homo sapiens (human)	Ki	25.1000	1	1
60 kDa chaperonin	Escherichia coli K-12	IC50	250.0000	1	1
60 kDa chaperonin	Escherichia coli	IC50	52.8750	4	4
60 kDa heat shock protein, mitochondrial	Homo sapiens (human)	IC50	57.5000	2	2
7-dehydrocholesterol reductase	Homo sapiens (human)	IC50	0.0120	1	1
72 kDa type IV collagenase	Homo sapiens (human)	IC50	4.1597	9	9
Acetylcholinesterase	Electrophorus electricus (electric eel)	IC50	4.4000	1	1
Acetylcholinesterase	Homo sapiens (human)	IC50	66.2850	2	2
Acetylcholinesterase	Homo sapiens (human)	Ki	65.8000	1	1
Adenosine receptor A1	Homo sapiens (human)	IC50	23.7670	1	1
Adenosine receptor A1	Homo sapiens (human)	Ki	13.8640	1	1
Adenosine receptor A2a	Homo sapiens (human)	IC50	7.0990	1	1
Adenosine receptor A2a	Homo sapiens (human)	Ki	3.9850	1	1
Adenosine receptor A3	Homo sapiens (human)	IC50	2.0285	1	2
Adenosine receptor A3	Homo sapiens (human)	Ki	1.1465	1	2
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1	Homo sapiens (human)	IC50	8.2000	1	1
Aldehyde dehydrogenase, mitochondrial	Homo sapiens (human)	IC50	3.4000	1	1
Aldehyde oxidase	Homo sapiens (human)	IC50	0.2000	1	1
Aldehyde oxidase 1	Macaca fascicularis (crab-eating macaque)	IC50	0.1100	1	1
Aldehyde oxidase 1	Mus musculus (house mouse)	IC50	0.1500	1	1
Aldehyde oxidase 1	Oryctolagus cuniculus (rabbit)	IC50	2.0000	1	1
Aldehyde oxidase 1	Cavia porcellus (domestic guinea pig)	Ki	7.2300	1	1
Aldehyde oxidase 1	Rattus norvegicus (Norway rat)	IC50	0.1900	1	1
Aldo-keto reductase family 1 member B1	Bos taurus (cattle)	IC50	5.1620	2	2
Aldo-keto reductase family 1 member B1	Homo sapiens (human)	IC50	1.9000	2	2
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	IC50	24.4607	2	3
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	Ki	35.6355	1	2
Aldo-keto reductase family 1 member B10	Homo sapiens (human)	IC50	58.5000	2	2
ALK tyrosine kinase receptor	Homo sapiens (human)	IC50	1.1773	2	2
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	2.0285	1	2
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	1.1465	1	2
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	2.0285	1	2
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	1.1465	1	2
Alpha-1D adrenergic receptor	Homo sapiens (human)	IC50	4.9820	1	1
Alpha-1D adrenergic receptor	Homo sapiens (human)	Ki	2.4490	1	1
Alpha-2A adrenergic receptor	Homo sapiens (human)	IC50	3.4195	1	2
Alpha-2A adrenergic receptor	Homo sapiens (human)	Ki	1.2825	1	2
Alpha-2B adrenergic receptor	Homo sapiens (human)	IC50	3.3680	1	2
Alpha-2B adrenergic receptor	Homo sapiens (human)	Ki	1.5375	1	2
Alpha-amylase 1A	Homo sapiens (human)	IC50	18.4000	2	2
Alpha-synuclein	Homo sapiens (human)	IC50	20.9000	3	5
Alternative oxidase, mitochondrial	Trypanosoma brucei brucei	IC50	0.0020	1	1
Alternative oxidase, mitochondrial	Trypanosoma brucei brucei	Ki	0.0001	1	1
Amine oxidase [flavin-containing] A	Homo sapiens (human)	IC50	7.9635	3	4
Amine oxidase [flavin-containing] A	Homo sapiens (human)	Ki	26.0000	1	1
Amine oxidase [flavin-containing] B	Homo sapiens (human)	IC50	59.7000	1	1
Amine oxidase [flavin-containing] B	Homo sapiens (human)	Ki	0.4000	1	1
Amyloid-beta precursor protein	Homo sapiens (human)	IC50	5.6000	2	2
Androgen receptor	Rattus norvegicus (Norway rat)	IC50	17.3423	2	2
Androgen receptor	Rattus norvegicus (Norway rat)	Ki	15.1080	1	1
Angiopoietin-1 receptor	Homo sapiens (human)	IC50	0.7468	9	14
Angiotensin-converting enzyme	Oryctolagus cuniculus (rabbit)	IC50	193.6557	3	3
Angiotensin-converting enzyme	Oryctolagus cuniculus (rabbit)	Ki	0.7922	1	1
Angiotensin-converting enzyme 2	Homo sapiens (human)	IC50	8.8250	1	2
AP2-associated protein kinase 1	Homo sapiens (human)	IC50	0.0462	2	2
apelin receptor	Homo sapiens (human)	IC50	2.6300	1	1
Aromatase	Homo sapiens (human)	IC50	0.0826	3	14
Arylacetamide deacetylase	Homo sapiens (human)	Ki	300.0000	1	1
ATP-binding cassette sub-family C member 3	Homo sapiens (human)	IC50	117.0000	1	4
ATP-dependent 6-phosphofructokinase	Trypanosoma brucei brucei	IC50	3.0000	1	1
ATP-dependent translocase ABCB1	Homo sapiens (human)	IC50	23.2500	6	6
ATP-dependent translocase ABCB1	Homo sapiens (human)	Ki	0.1000	1	1
Aurora kinase A	Homo sapiens (human)	IC50	2.4146	5	8
Aurora kinase B	Homo sapiens (human)	IC50	3.3250	2	4
B2 bradykinin receptor	Homo sapiens (human)	IC50	20.3560	1	1
B2 bradykinin receptor	Homo sapiens (human)	Ki	12.0480	1	1
Beta-1 adrenergic receptor	Homo sapiens (human)	IC50	17.2890	1	1
Beta-1 adrenergic receptor	Homo sapiens (human)	Ki	9.9840	1	1
Beta-3 adrenergic receptor	Homo sapiens (human)	IC50	7.7030	1	1
Beta-3 adrenergic receptor	Homo sapiens (human)	Ki	5.7780	1	1
Beta-adrenergic receptor kinase 1	Bos taurus (cattle)	IC50	130.0000	1	1
Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein)	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	5.0000	1	1
Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein)	Plasmodium falciparum (malaria parasite P. falciparum)	Ki	11.5000	1	1
Beta-secretase 1	Homo sapiens (human)	IC50	1.5400	1	1
Bifunctional epoxide hydrolase 2	Homo sapiens (human)	IC50	5.0060	1	2
bifunctional UDP-N-acetylglucosamine pyrophosphorylase/glucosamine-1-phosphate N-acetyltransferase	Mycobacterium tuberculosis H37Rv	IC50	85.0300	1	1
Bile salt export pump	Homo sapiens (human)	IC50	44.4182	8	17
Bile salt export pump	Rattus norvegicus (Norway rat)	IC50	34.7000	1	1
Bile salt export pump	Rattus norvegicus (Norway rat)	Ki	11.9000	1	1
Breakpoint cluster region protein	Homo sapiens (human)	GI50	7.3000	1	1
Broad substrate specificity ATP-binding cassette transporter ABCG2	Homo sapiens (human)	IC50	17.7500	3	4
Bromodomain testis-specific protein	Homo sapiens (human)	IC50	0.1902	13	13
Bromodomain-containing protein 1	Homo sapiens (human)	IC50	44.5000	1	1
Bromodomain-containing protein 2	Homo sapiens (human)	IC50	0.0959	22	22
Bromodomain-containing protein 2	Homo sapiens (human)	Ki	0.0128	4	4
Bromodomain-containing protein 3	Homo sapiens (human)	IC50	0.0573	18	18
Bromodomain-containing protein 3	Homo sapiens (human)	Ki	0.0078	4	4
Bromodomain-containing protein 4	Homo sapiens (human)	IC50	0.8621	120	120
Bromodomain-containing protein 4	Homo sapiens (human)	Ki	0.0193	8	8
C-8 sterol isomerase	Saccharomyces cerevisiae S288C	Ki	1.5000	1	1
C-C chemokine receptor type 2	Homo sapiens (human)	IC50	2.4680	1	1
C-C chemokine receptor type 2	Homo sapiens (human)	Ki	0.9540	1	1
C-C chemokine receptor type 4	Homo sapiens (human)	IC50	8.3950	1	1
C-C chemokine receptor type 4	Homo sapiens (human)	Ki	4.3970	1	1
C-C chemokine receptor type 5	Homo sapiens (human)	IC50	23.6610	1	1
C-C chemokine receptor type 5	Homo sapiens (human)	Ki	18.2840	1	1
C-X-C chemokine receptor type 2	Homo sapiens (human)	IC50	6.0130	1	1
C-X-C chemokine receptor type 2	Homo sapiens (human)	Ki	4.2090	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	IC50	10.0000	1	1
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	IC50	10.0000	1	1
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	IC50	10.0000	1	1
Canalicular multispecific organic anion transporter 1	Homo sapiens (human)	IC50	100.4000	2	5
Cannabinoid receptor 2	Mus musculus (house mouse)	IC50	50.0310	2	2
Carbamate kinase	Giardia intestinalis	IC50	0.6000	1	1
Carbonic anhydrase 1	Homo sapiens (human)	Ki	5.4567	3	6
Carbonic anhydrase 12	Homo sapiens (human)	Ki	0.0603	1	1
Carbonic anhydrase 2	Homo sapiens (human)	Ki	4.4053	3	6
Carbonic anhydrase 3	Bos taurus (cattle)	Ki	3.1850	1	4
Carbonic anhydrase 4	Homo sapiens (human)	Ki	2.6066	2	5
Carbonic anhydrase 7	Homo sapiens (human)	Ki	4.0706	2	2
Carbonic anhydrase 9	Homo sapiens (human)	Ki	10.0000	1	1
Casein kinase I isoform alpha	Homo sapiens (human)	IC50	0.1255	1	2
Casein kinase I isoform alpha	Sus scrofa (pig)	IC50	50.0000	1	1
Casein kinase II subunit alpha	Homo sapiens (human)	IC50	3.8333	2	3
Casein kinase II subunit alpha 3	Homo sapiens (human)	IC50	5.2500	1	2
Casein kinase II subunit alpha'	Homo sapiens (human)	IC50	3.1250	3	4
Casein kinase II subunit beta	Homo sapiens (human)	IC50	3.1250	3	4
Caspase-1	Homo sapiens (human)	IC50	5.0595	2	2
Cathepsin B	Homo sapiens (human)	IC50	30.0000	1	1
Cationic trypsin	Bos taurus (cattle)	IC50	35.3000	1	1
CDK-activating kinase assembly factor MAT1	Homo sapiens (human)	IC50	3.1520	4	4
Cereblon isoform 4	Magnetospirillum gryphiswaldense	Ki	1.9500	1	2
Chain A, Casein kinase II subunit alpha	Zea mays	IC50	0.3500	1	3
Chain A, CES1 protein	Homo sapiens (human)	Ki	15.2000	1	1
Chain A, Cyclin-dependent kinase 9	Homo sapiens (human)	IC50	0.7400	1	1
Chain A, Exotoxin A	Pseudomonas aeruginosa	Ki	0.1400	1	1
Chain A, Extracellular Regulated Kinase 2	Rattus norvegicus (Norway rat)	IC50	9.0095	1	4
Chain A, MAP KINASE P38	Homo sapiens (human)	IC50	9.0095	1	2
Chain A, PROTEIN (MAP KINASE P38)	Homo sapiens (human)	IC50	9.0095	1	6
Chain A, RNA-directed RNA polymerase NS5	Dengue virus 2 16681-PDK53	IC50	35.0600	1	1
Chain A, VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	Homo sapiens (human)	Ki	0.0005	1	5
Chemotaxis protein CheA	Escherichia coli K-12	IC50	111.0000	1	1
Collagenase 3	Homo sapiens (human)	IC50	5.0275	2	2
CREB-binding protein	Homo sapiens (human)	IC50	9.7153	3	3
Cruzipain	Trypanosoma cruzi	IC50	91.5000	2	2
Cyclin homolog	Herpesvirus saimiri (strain 11)	IC50	77.7000	1	4
Cyclin-A1	Homo sapiens (human)	IC50	34.5105	2	2
Cyclin-A1	Homo sapiens (human)	Ki	69.0000	1	1
Cyclin-A2	Homo sapiens (human)	IC50	21.3782	7	12
Cyclin-A2	Homo sapiens (human)	Ki	69.0000	1	1
Cyclin-C	Homo sapiens (human)	IC50	2.0108	3	3
Cyclin-dependent kinase 1	Homo sapiens (human)	IC50	16.1804	17	26
Cyclin-dependent kinase 1	Oryzias latipes (Japanese medaka)	IC50	77.7000	1	4
Cyclin-dependent kinase 1	Homo sapiens (human)	Ki	0.4800	1	1
Cyclin-dependent kinase 19	Homo sapiens (human)	IC50	0.1150	1	2
Cyclin-dependent kinase 2	Homo sapiens (human)	IC50	20.9140	27	37
Cyclin-dependent kinase 2	Homo sapiens (human)	Ki	27.4460	3	3
Cyclin-dependent kinase 4	Homo sapiens (human)	IC50	15.6734	11	20
Cyclin-dependent kinase 4	Homo sapiens (human)	Ki	0.9250	1	1
Cyclin-dependent kinase 5 activator 1	Homo sapiens (human)	IC50	45.0400	4	7
Cyclin-dependent kinase 6	Homo sapiens (human)	IC50	101.8217	3	6
Cyclin-dependent kinase 7	Homo sapiens (human)	IC50	15.5281	13	22
Cyclin-dependent kinase 8	Homo sapiens (human)	IC50	2.3242	11	14
Cyclin-dependent kinase 9	Homo sapiens (human)	IC50	9.3365	21	30
Cyclin-dependent kinase 9	Homo sapiens (human)	Ki	0.1770	2	2
Cyclin-dependent-like kinase 5	Homo sapiens (human)	IC50	45.0400	4	7
Cyclin-H	Homo sapiens (human)	IC50	15.8429	10	15
Cyclin-T1	Homo sapiens (human)	IC50	9.1942	14	19
Cyclin-T1	Homo sapiens (human)	Ki	0.3500	1	1
Cytochrome P450 11B1, mitochondrial	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Cytochrome P450 1A1	Homo sapiens (human)	IC50	0.6945	1	2
Cytochrome P450 1A1	Homo sapiens (human)	Ki	1.3998	2	5
Cytochrome P450 1A2	Homo sapiens (human)	IC50	10.1254	4	5
Cytochrome P450 1B1	Homo sapiens (human)	IC50	0.1560	2	3
Cytochrome P450 1B1	Homo sapiens (human)	Ki	0.5496	3	5
Cytochrome P450 2B6	Homo sapiens (human)	Ki	0.9000	1	1
Cytochrome P450 2C19	Homo sapiens (human)	IC50	20.0040	2	2
Cytochrome P450 2C9	Homo sapiens (human)	IC50	19.4270	3	4
Cytochrome P450 2D6	Homo sapiens (human)	IC50	40.0000	1	1
Cytochrome P450 3A4	Homo sapiens (human)	IC50	11.9167	8	8
Cytochrome P450 3A4	Homo sapiens (human)	Ki	0.2000	1	1
Cytosol aminopeptidase	Sus scrofa (pig)	IC50	49.6000	1	1
Cytosolic phospholipase A2	Homo sapiens (human)	IC50	100.0000	1	1
D(1A) dopamine receptor	Homo sapiens (human)	IC50	5.3300	1	2
D(1A) dopamine receptor	Homo sapiens (human)	Ki	2.6650	1	2
D(2) dopamine receptor	Homo sapiens (human)	IC50	18.4515	1	2
D(2) dopamine receptor	Homo sapiens (human)	Ki	6.1505	1	2
D(3) dopamine receptor	Homo sapiens (human)	IC50	1.0780	1	2
D(3) dopamine receptor	Rattus norvegicus (Norway rat)	IC50	18.1000	1	1
D(3) dopamine receptor	Homo sapiens (human)	Ki	0.6577	2	3
D(4) dopamine receptor	Homo sapiens (human)	IC50	7.1555	1	2
D(4) dopamine receptor	Homo sapiens (human)	Ki	2.5090	1	2
Death-associated protein kinase 1	Homo sapiens (human)	IC50	70.5000	1	2
Delta-type opioid receptor	Homo sapiens (human)	IC50	13.3390	1	1
Delta-type opioid receptor	Homo sapiens (human)	Ki	1.5915	3	3
Delta-type opioid receptor	Sus scrofa (pig)	Ki	0.0365	1	1
Dihydroorotate dehydrogenase (quinone), mitochondrial	Homo sapiens (human)	IC50	3.3500	1	2
Dipeptidyl peptidase 3	Homo sapiens (human)	IC50	22.0000	1	1
Dipeptidyl peptidase 4	Homo sapiens (human)	IC50	100.0600	2	2
Discoidin domain-containing receptor 2	Homo sapiens (human)	IC50	0.0215	2	2
Disintegrin and metalloproteinase domain-containing protein 17	Homo sapiens (human)	IC50	0.0149	1	1
DNA damage-binding protein 1	Homo sapiens (human)	IC50	1.7972	3	5
DNA gyrase subunit A	Mycobacterium tuberculosis H37Rv	IC50	150.0000	3	3
DNA gyrase subunit B	Mycobacterium tuberculosis H37Rv	IC50	125.0000	2	2
DNA primase	Mycobacterium tuberculosis CDC1551	IC50	8.2000	1	1
DNA topoisomerase 1	Rattus norvegicus (Norway rat)	IC50	2.8300	2	2
DNA-dependent protein kinase catalytic subunit	Homo sapiens (human)	IC50	33.9000	2	3
DNA-directed RNA polymerase subunit beta	Escherichia coli O127:H6 str. E2348/69	IC50	511.3333	3	3
DNA-directed RNA polymerase subunit beta	Mycobacterium tuberculosis H37Rv	IC50	0.0100	1	1
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	IC50	3.3000	1	1
Dual specificity protein phosphatase 1	Mus musculus (house mouse)	IC50	24.0000	1	1
Dual specificity protein phosphatase 5	Homo sapiens (human)	Ki	0.0250	1	1
Dual specificity protein phosphatase 6	Rattus norvegicus (Norway rat)	IC50	20.5000	1	1
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Rattus norvegicus (Norway rat)	IC50	30.0000	1	1
Ectonucleoside triphosphate diphosphohydrolase 1	Rattus norvegicus (Norway rat)	Ki	300.0000	2	2
Ectonucleoside triphosphate diphosphohydrolase 2	Rattus norvegicus (Norway rat)	Ki	65.4000	2	2
Ectonucleoside triphosphate diphosphohydrolase 3	Rattus norvegicus (Norway rat)	Ki	12.7000	1	1
Ectonucleoside triphosphate diphosphohydrolase 8	Homo sapiens (human)	Ki	100.0000	1	1
Emopamil-binding protein-like	Homo sapiens (human)	Ki	0.0028	1	1
Endoplasmin	Canis lupus familiaris (dog)	IC50	0.0120	1	1
Endoplasmin	Homo sapiens (human)	IC50	0.0850	1	1
Endoplasmin	Homo sapiens (human)	Ki	0.0040	1	1
Endothelin-converting enzyme 2	Homo sapiens (human)	IC50	6.4200	1	1
Enoyl-[acyl-carrier-protein] reductase [NADH]	Mycobacterium tuberculosis H37Rv	IC50	0.0300	1	1
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI	Escherichia coli K-12	Ki	7.0500	1	1
Enoyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	2.0000	2	2
Enoyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	Ki	2.1000	1	1
Ephrin type-B receptor 4	Homo sapiens (human)	IC50	6.7262	6	8
Epidermal growth factor receptor	Homo sapiens (human)	IC50	35.3205	33	37
Estrogen receptor	Homo sapiens (human)	IC50	1.1920	42	42
Estrogen receptor	Homo sapiens (human)	Ki	0.0586	4	4
Estrogen receptor beta	Homo sapiens (human)	IC50	1.2236	23	23
Estrogen receptor beta	Homo sapiens (human)	Ki	0.0510	4	4
Estrogen-related receptor gamma	Homo sapiens (human)	IC50	0.0622	1	1
Fatty acid synthase	Gallus gallus (chicken)	IC50	62.5000	1	1
Fatty acid synthase	Homo sapiens (human)	IC50	62.5000	1	1
Fatty-acid amide hydrolase 1	Homo sapiens (human)	IC50	363.0780	1	1
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	IC50	6.1000	1	1
Fibroblast growth factor receptor 1	Homo sapiens (human)	IC50	4.9864	22	32
Fibroblast growth factor receptor 2	Homo sapiens (human)	IC50	3.1700	4	4
Fibroblast growth factor receptor 3	Homo sapiens (human)	IC50	3.1700	4	4
Fibroblast growth factor receptor 4	Homo sapiens (human)	IC50	3.1700	4	4
Focal adhesion kinase 1	Homo sapiens (human)	IC50	20.8000	2	2
Fructose-1,6-bisphosphatase 1	Homo sapiens (human)	IC50	87.5067	11	12
G protein-coupled receptor kinase 5	Homo sapiens (human)	IC50	0.8300	1	1
G protein-coupled receptor kinase 6	Homo sapiens (human)	IC50	8.7000	1	1
G-protein coupled receptor 35	Homo sapiens (human)	IC50	23.4000	1	2
G1/S-specific cyclin-D1	Homo sapiens (human)	IC50	17.1354	7	12
G1/S-specific cyclin-D2	Homo sapiens (human)	IC50	0.9250	1	1
G1/S-specific cyclin-D3	Homo sapiens (human)	IC50	0.9250	1	1
G1/S-specific cyclin-E1	Homo sapiens (human)	IC50	17.7863	11	16
G1/S-specific cyclin-E1	Homo sapiens (human)	Ki	13.3000	1	1
G1/S-specific cyclin-E2	Homo sapiens (human)	IC50	17.8870	4	4
G1/S-specific cyclin-E2	Homo sapiens (human)	Ki	13.3000	1	1
G2/mitotic-specific cyclin-B	Marthasterias glacialis (spiny starfish)	IC50	77.7000	1	4
G2/mitotic-specific cyclin-B1	Homo sapiens (human)	IC50	16.8565	12	17
G2/mitotic-specific cyclin-B2	Homo sapiens (human)	IC50	16.8933	3	3
G2/mitotic-specific cyclin-B3	Homo sapiens (human)	IC50	16.8933	3	3
GABA theta subunit	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Homo sapiens (human)	IC50	281,838.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-2	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-3	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-4	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-5	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit alpha-6	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit beta-1	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit beta-2	Homo sapiens (human)	IC50	281,838.0000	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit beta-3	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit delta	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit epsilon	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit gamma-1	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit gamma-2	Homo sapiens (human)	IC50	281,838.0000	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit gamma-3	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	IC50	0.0149	1	1
Gamma-aminobutyric acid receptor subunit pi	Homo sapiens (human)	Ki	1.9193	3	4
Gamma-aminobutyric acid receptor subunit theta	Homo sapiens (human)	Ki	1.9193	3	4
Gasdermin-D	Homo sapiens (human)	IC50	0.4000	1	1
Gasdermin-D	Mus musculus (house mouse)	IC50	0.4000	1	1
Gastrin/cholecystokinin type B receptor	Rattus norvegicus (Norway rat)	IC50	50.0000	2	2
Genome polyprotein	Zika virus	IC50	53.0000	1	1
Glucocorticoid receptor	Homo sapiens (human)	IC50	19.0000	1	1
glucose-6-phosphate 1-dehydrogenase isoform b	Homo sapiens (human)	IC50	80.0000	1	1
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase	Plasmodium berghei	IC50	56.7000	3	3
Glutathione reductase, mitochondrial	Homo sapiens (human)	Ki	14.1000	2	2
Glutathione S-transferase omega-1	Homo sapiens (human)	IC50	75.0000	1	1
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	IC50	0.8000	1	1
Glycogen synthase kinase-3 beta	Homo sapiens (human)	IC50	10.1500	4	5
Glycogen synthase kinase-3 beta	Rattus norvegicus (Norway rat)	IC50	77.7000	1	4
Group 10 secretory phospholipase A2	Homo sapiens (human)	IC50	100.0000	1	1
Heat shock protein 75 kDa, mitochondrial	Homo sapiens (human)	IC50	0.3577	3	3
Heat shock protein 75 kDa, mitochondrial	Homo sapiens (human)	Ki	0.0160	1	1
Heat shock protein HSP 90-alpha	Homo sapiens (human)	IC50	2.8407	16	16
Heat shock protein HSP 90-alpha	Homo sapiens (human)	Ki	0.0055	2	2
Heat shock protein HSP 90-beta	Homo sapiens (human)	IC50	0.0657	12	12
Heat shock protein HSP 90-beta	Homo sapiens (human)	Ki	0.0026	4	4
Hepatocyte growth factor receptor	Homo sapiens (human)	IC50	7.2188	8	8
Histamine H2 receptor	Homo sapiens (human)	IC50	9.3960	1	1
Histamine H2 receptor	Homo sapiens (human)	Ki	9.2400	1	1
Histidine kinase	Caulobacter vibrioides	IC50	7.3000	1	1
histidine kinase	Streptococcus pneumoniae TIGR4	IC50	216.0000	1	1
Histone acetyltransferase p300	Homo sapiens (human)	IC50	19.4000	1	1
Histone deacetylase 1	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 11	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 2	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 3	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 4	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 5	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 6	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 7	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 8	Homo sapiens (human)	IC50	0.2910	1	1
Histone deacetylase 9	Homo sapiens (human)	IC50	0.2910	1	1
Histone-lysine N-methyltransferase EHMT1	Homo sapiens (human)	IC50	1.6000	1	1
Histone-lysine N-methyltransferase EHMT2	Homo sapiens (human)	IC50	0.6000	1	1
Histone-lysine N-methyltransferase SETD7	Homo sapiens (human)	IC50	6.0800	1	1
Homeobox protein Nkx-2.5	Mus musculus (house mouse)	IC50	22.0000	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	IC50	0.1000	1	1
Homeodomain-interacting protein kinase 2	Homo sapiens (human)	IC50	0.1000	1	1
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	IC50	0.1000	1	1
Homeodomain-interacting protein kinase 4	Homo sapiens (human)	IC50	0.0515	2	2
hypothetical protein SA1422	Staphylococcus aureus subsp. aureus N315	IC50	19.3900	2	2
Indoleamine 2,3-dioxygenase 1	Homo sapiens (human)	IC50	0.8925	4	4
Inositol hexakisphosphate kinase 2	Homo sapiens (human)	IC50	1.1000	1	2
Inositol polyphosphate multikinase	Homo sapiens (human)	IC50	6.3500	1	2
Insulin receptor	Homo sapiens (human)	IC50	19.5000	2	3
Insulin-like growth factor 1 receptor	Homo sapiens (human)	IC50	15.0000	3	3
Integrase	Human immunodeficiency virus 1	IC50	10.3730	5	10
integrase, partial	Human immunodeficiency virus 1	IC50	7.8945	2	2
Interstitial collagenase	Homo sapiens (human)	IC50	0.6551	8	8
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	0.6600	1	1
Kappa-type opioid receptor	Homo sapiens (human)	IC50	10.8660	1	2
Kappa-type opioid receptor	Homo sapiens (human)	Ki	4.3465	1	2
Lactoylglutathione lyase	Homo sapiens (human)	IC50	9.3500	1	2
Lanosterol 14-alpha demethylase	Homo sapiens (human)	IC50	30.0000	1	1
large T antigen	Betapolyomavirus macacae	IC50	11.3150	1	2
lens epithelium-derived growth factor p75	Homo sapiens (human)	IC50	7.8945	2	2
Leucine-rich repeat serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.0215	2	2
Linoleate 9S-lipoxygenase-4	Glycine max (soybean)	IC50	22.0000	1	1
Low affinity immunoglobulin epsilon Fc receptor	Homo sapiens (human)	IC50	0.1000	2	2
Lysine-specific demethylase 4E	Homo sapiens (human)	IC50	3.0000	1	1
Lysine-specific demethylase 4E	Homo sapiens (human)	Ki	4.3300	1	1
Lysine-specific demethylase 5A	Homo sapiens (human)	IC50	10.0000	1	1
Lysine-specific histone demethylase 1A	Homo sapiens (human)	IC50	16.4233	2	3
Lysosomal alpha-glucosidase	Homo sapiens (human)	IC50	500.0000	1	1
Lysyl oxidase homolog 2	Homo sapiens (human)	IC50	0.1500	1	1
Lysyl oxidase homolog 3	Homo sapiens (human)	IC50	0.0930	1	1
Lysyl oxidase homolog 4	Homo sapiens (human)	IC50	0.0590	1	1
M-phase inducer phosphatase 1	Homo sapiens (human)	IC50	4.5500	2	2
M-phase inducer phosphatase 2	Homo sapiens (human)	IC50	3.1600	3	3
M-phase inducer phosphatase 3	Homo sapiens (human)	IC50	18.9000	2	2
M1-family alanyl aminopeptidase	Plasmodium falciparum 3D7	IC50	65.6250	1	2
Macrophage colony-stimulating factor 1 receptor	Homo sapiens (human)	IC50	0.1286	9	15
Macrophage metalloelastase	Homo sapiens (human)	IC50	2.9900	4	4
Macrophage-stimulating protein receptor	Homo sapiens (human)	IC50	10.0000	1	1
MAP kinase-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	IC50	0.1790	1	1
MAP kinase-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.4205	2	2
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	GI50	0.1937	55	55
Mast/stem cell growth factor receptor Kit	Mus musculus (house mouse)	GI50	0.0030	1	1
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	IC50	0.2178	34	46
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	Ki	0.0040	1	1
Matrilysin	Homo sapiens (human)	IC50	3.5012	2	2
Matrix metalloproteinase-14	Homo sapiens (human)	IC50	0.5715	5	5
Matrix metalloproteinase-9	Homo sapiens (human)	IC50	1.3711	6	6
Mcl-1	Homo sapiens (human)	IC50	1.6341	1	1
Melanocortin receptor 3	Homo sapiens (human)	IC50	19.8560	1	1
Melanocortin receptor 3	Homo sapiens (human)	Ki	17.3290	1	1
melanocortin receptor 4	Homo sapiens (human)	IC50	54.8937	3	3
Melanocortin receptor 4	Homo sapiens (human)	Ki	29.3080	1	1
Melanocortin receptor 5	Homo sapiens (human)	IC50	26.5290	1	1
Melanocortin receptor 5	Homo sapiens (human)	Ki	24.8860	1	1
Metabotropic glutamate receptor 5	Rattus norvegicus (Norway rat)	IC50	1.2000	1	1
Methionine aminopeptidase	Escherichia coli K-12	IC50	100.0000	1	1
Methionine aminopeptidase 1	Saccharomyces cerevisiae S288C	IC50	100.0000	1	1
Methionine aminopeptidase 2	Homo sapiens (human)	IC50	0.3006	7	8
Methionine aminopeptidase 2	Homo sapiens (human)	Ki	0.0010	2	2
Mitogen-activated protein kinase 1	Homo sapiens (human)	IC50	9.5548	2	2
Mitogen-activated protein kinase 1	Rattus norvegicus (Norway rat)	IC50	9.0095	1	2
Mitogen-activated protein kinase 10	Homo sapiens (human)	IC50	18.0250	1	4
Mitogen-activated protein kinase 10	Rattus norvegicus (Norway rat)	IC50	6.8000	1	1
Mitogen-activated protein kinase 11	Homo sapiens (human)	IC50	0.0190	1	1
Mitogen-activated protein kinase 12	Homo sapiens (human)	IC50	0.0190	1	1
Mitogen-activated protein kinase 13	Homo sapiens (human)	IC50	0.0190	1	1
Mitogen-activated protein kinase 14	Homo sapiens (human)	IC50	5.0104	15	19
Mitogen-activated protein kinase 3	Homo sapiens (human)	IC50	0.7640	2	2
Monoglyceride lipase	Homo sapiens (human)	IC50	0.8095	2	2
Mu-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	0.0180	1	1
Mu-type opioid receptor	Homo sapiens (human)	IC50	10.5525	1	2
Mu-type opioid receptor	Homo sapiens (human)	Ki	4.2835	1	2
Multidrug resistance-associated protein 1	Homo sapiens (human)	IC50	3.0000	1	1
Multidrug resistance-associated protein 4	Homo sapiens (human)	IC50	110.2250	1	4
Muscarinic acetylcholine receptor M1	Homo sapiens (human)	IC50	2.8290	1	1
Muscarinic acetylcholine receptor M1	Homo sapiens (human)	Ki	0.6810	1	1
Muscarinic acetylcholine receptor M2	Homo sapiens (human)	IC50	7.7930	1	1
Muscarinic acetylcholine receptor M2	Homo sapiens (human)	Ki	2.7710	1	1
Muscarinic acetylcholine receptor M3	Homo sapiens (human)	IC50	2.9740	1	1
Muscarinic acetylcholine receptor M3	Homo sapiens (human)	Ki	0.6300	1	1
Muscarinic acetylcholine receptor M4	Homo sapiens (human)	IC50	4.8170	1	1
Muscarinic acetylcholine receptor M4	Homo sapiens (human)	Ki	0.6720	1	1
Muscarinic acetylcholine receptor M5	Homo sapiens (human)	IC50	2.5850	1	1
Muscarinic acetylcholine receptor M5	Homo sapiens (human)	Ki	1.8570	1	1
NACHT, LRR and PYD domains-containing protein 3	Mus musculus (house mouse)	IC50	1.9050	2	2
NAD-dependent protein deacetylase HST2	Saccharomyces cerevisiae S288C	IC50	240.0000	1	1
NAD-dependent protein deacetylase sirtuin-1	Homo sapiens (human)	IC50	1.3857	7	7
NAD-dependent protein deacetylase sirtuin-2	Homo sapiens (human)	IC50	25.4800	5	5
NAD-dependent protein deacylase sirtuin-5, mitochondrial	Homo sapiens (human)	IC50	20.6000	8	8
NADPH oxidase 4	Homo sapiens (human)	IC50	0.8500	1	1
Neprilysin	Homo sapiens (human)	IC50	100.0000	1	1
Neuraminidase	Influenza A virus (A/Wilson-Smith/1933(H1N1))	IC50	27.9000	4	5
Neuraminidase	Influenza A virus (A/Wilson-Smith/1933(H1N1))	Ki	16.6500	1	2
Neuropilin-1	Homo sapiens (human)	IC50	9.1833	6	6
Neutrophil collagenase	Homo sapiens (human)	IC50	0.7000	1	1
Neutrophil elastase	Homo sapiens (human)	IC50	6.9850	2	2
Neutrophil elastase	Homo sapiens (human)	Ki	10.1000	1	1
NH(3)-dependent NAD(+) synthetase	Bacillus subtilis subsp. subtilis str. 168	IC50	1.0000	1	1
Nitric oxide synthase, brain	Homo sapiens (human)	IC50	4.8900	2	2
Nitric oxide synthase, brain	Homo sapiens (human)	Ki	7.3000	1	1
Nitric oxide synthase, brain	Rattus norvegicus (Norway rat)	IC50	7.5500	2	2
Nitric oxide synthase, endothelial	Bos taurus (cattle)	IC50	611.3333	3	3
Nitric oxide synthase, endothelial	Homo sapiens (human)	IC50	485.0667	3	3
Nitric oxide synthase, inducible	Homo sapiens (human)	IC50	0.1395	3	3
Nitric oxide synthase, inducible	Mus musculus (house mouse)	IC50	2.0828	4	4
NUAK family SNF1-like kinase 1	Homo sapiens (human)	IC50	0.0480	1	1
Nuclear receptor subfamily 3 group C member 3	Bos taurus (cattle)	IC50	0.9670	1	1
Nuclear receptor subfamily 3 group C member 3	Bos taurus (cattle)	Ki	0.7922	1	1
P2X purinoceptor 2	Rattus norvegicus (Norway rat)	IC50	21.9054	1	2
P2Y purinoceptor 11	Homo sapiens (human)	Ki	0.2071	2	2
P2Y purinoceptor 2	Homo sapiens (human)	IC50	75.0000	2	2
P2Y purinoceptor 6	Homo sapiens (human)	IC50	27.0000	1	1
perilipin-1	Homo sapiens (human)	IC50	7.4270	1	2
perilipin-5	Homo sapiens (human)	IC50	5.5450	1	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	IC50	30.5000	1	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	IC50	50.0000	1	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	IC50	37.3333	1	3
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	IC50	31.5000	1	2
Phospholipase A2	Rattus norvegicus (Norway rat)	IC50	100.0000	1	1
Phospholipase A2, membrane associated	Homo sapiens (human)	IC50	23.8000	1	1
Phospholipase D1	Homo sapiens (human)	IC50	20.0000	1	1
Phospholipase D1	Rattus norvegicus (Norway rat)	IC50	20.0000	1	1
Platelet-activating factor acetylhydrolase	Homo sapiens (human)	IC50	0.9040	1	1
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	GI50	0.1939	4	4
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	IC50	0.1144	6	6
Platelet-derived growth factor receptor alpha	Rattus norvegicus (Norway rat)	IC50	50.0000	2	2
Platelet-derived growth factor receptor alpha	Mus musculus (house mouse)	IC50	6.2662	8	8
Platelet-derived growth factor receptor beta	Homo sapiens (human)	GI50	0.1140	1	1
Platelet-derived growth factor receptor beta	Homo sapiens (human)	IC50	8.2102	39	51
Platelet-derived growth factor receptor beta	Mus musculus (house mouse)	IC50	8.3954	12	18
Platelet-derived growth factor receptor beta	Rattus norvegicus (Norway rat)	IC50	50.0000	2	2
Platelet-derived growth factor receptor beta	Homo sapiens (human)	Ki	0.0080	1	1
Poly [ADP-ribose] polymerase 1	Homo sapiens (human)	IC50	0.4834	17	22
Poly [ADP-ribose] polymerase 2	Homo sapiens (human)	IC50	3.0634	5	7
Poly [ADP-ribose] polymerase 2	Mus musculus (house mouse)	IC50	0.0405	1	2
Poly [ADP-ribose] polymerase tankyrase-1	Homo sapiens (human)	IC50	1.4307	5	8
Poly [ADP-ribose] polymerase tankyrase-2	Homo sapiens (human)	IC50	1.2162	4	7
Polyamine deacetylase HDAC10	Homo sapiens (human)	IC50	0.2910	1	1
Polyunsaturated fatty acid 5-lipoxygenase	Homo sapiens (human)	IC50	34.1500	2	3
Polyunsaturated fatty acid 5-lipoxygenase	Rattus norvegicus (Norway rat)	IC50	10.0000	2	2
Polyunsaturated fatty acid 5-lipoxygenase	Homo sapiens (human)	Ki	0.0844	2	2
Polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	IC50	31.5320	2	5
Polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	Ki	1.6000	1	1
Polyunsaturated fatty acid lipoxygenase ALOX15	Homo sapiens (human)	IC50	28.4833	3	6
Polyunsaturated fatty acid lipoxygenase ALOX15	Oryctolagus cuniculus (rabbit)	IC50	9.5075	1	2
Polyunsaturated fatty acid lipoxygenase ALOX15	Homo sapiens (human)	Ki	0.6000	1	1
Polyunsaturated fatty acid lipoxygenase ALOX15B	Homo sapiens (human)	IC50	51.0929	3	7
Polyunsaturated fatty acid lipoxygenase ALOX15B	Rattus norvegicus (Norway rat)	IC50	0.2600	1	1
Potassium voltage-gated channel subfamily D member 3	Homo sapiens (human)	IC50	50.1187	1	1
Potassium voltage-gated channel subfamily E member 1	Homo sapiens (human)	IC50	63.0957	1	1
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	IC50	4.9683	8	8
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	Ki	0.7922	1	1
Potassium voltage-gated channel subfamily KQT member 1	Homo sapiens (human)	IC50	63.0957	1	1
Procathepsin L	Homo sapiens (human)	IC50	8.8250	1	2
Progesterone receptor	Homo sapiens (human)	IC50	38.3763	3	3
Programmed cell death 1 ligand 1	Homo sapiens (human)	IC50	0.0100	1	1
Programmed cell death protein 1	Homo sapiens (human)	IC50	0.0100	1	1
Prolyl endopeptidase	Homo sapiens (human)	IC50	36.0000	1	1
Prostaglandin G/H synthase 1	Homo sapiens (human)	IC50	4.3910	1	1
Prostaglandin G/H synthase 1	Ovis aries (sheep)	IC50	76.6000	2	2
Prostaglandin G/H synthase 1	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	IC50	48.7767	6	6
Prostaglandin G/H synthase 2	Mus musculus (house mouse)	IC50	1.0700	1	1
Prostaglandin G/H synthase 2	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Proteasome subunit beta type-5	Homo sapiens (human)	IC50	1.4000	2	2
Protein arginine N-methyltransferase 1	Homo sapiens (human)	IC50	344.8100	3	3
Protein cereblon	Homo sapiens (human)	IC50	7.2078	6	11
Protein cereblon	Homo sapiens (human)	Ki	9.2633	2	3
Protein delta homolog 1	Homo sapiens (human)	Ki	0.0063	1	1
Protein kinase C alpha type	Homo sapiens (human)	IC50	19.5333	6	6
Protein kinase C alpha type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C beta type	Homo sapiens (human)	IC50	22.5000	4	4
Protein kinase C beta type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C delta type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C delta type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C epsilon type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C epsilon type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C eta type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C eta type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C gamma type	Homo sapiens (human)	IC50	22.5000	4	4
Protein kinase C gamma type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C iota type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C theta type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C theta type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein kinase C zeta type	Homo sapiens (human)	IC50	16.6667	3	3
Protein kinase C zeta type	Rattus norvegicus (Norway rat)	IC50	75.0000	1	1
Protein mono-ADP-ribosyltransferase PARP10	Homo sapiens (human)	IC50	6.3123	2	4
Protein mono-ADP-ribosyltransferase PARP12	Homo sapiens (human)	IC50	0.2269	1	2
Protein mono-ADP-ribosyltransferase PARP14	Homo sapiens (human)	IC50	4.1843	1	2
Protein mono-ADP-ribosyltransferase PARP15	Homo sapiens (human)	IC50	8.9563	1	2
Protein mono-ADP-ribosyltransferase PARP3	Homo sapiens (human)	IC50	1.4377	1	2
Protein mono-ADP-ribosyltransferase PARP4	Homo sapiens (human)	IC50	0.7586	1	1
Protein-glutamine gamma-glutamyltransferase 2	Homo sapiens (human)	IC50	2.2000	1	1
Protein-lysine 6-oxidase	Homo sapiens (human)	IC50	0.3200	1	1
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	GI50	0.1013	3	3
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	IC50	0.3065	12	15
Proto-oncogene tyrosine-protein kinase Src	Gallus gallus (chicken)	IC50	33.5183	3	3
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	IC50	24.6355	8	11
Pyruvate kinase PKM	Homo sapiens (human)	IC50	76.0050	2	2
Pyruvate kinase PKM	Homo sapiens (human)	Ki	3.5300	1	1
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	IC50	30.0000	2	2
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.6814	30	34
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	Ki	0.0060	1	1
Receptor protein-tyrosine kinase	Homo sapiens (human)	IC50	2.2000	1	1
Receptor tyrosine-protein kinase erbB-2	Homo sapiens (human)	IC50	5.6176	5	5
Receptor tyrosine-protein kinase erbB-3	Homo sapiens (human)	IC50	0.0020	1	1
Receptor tyrosine-protein kinase erbB-4	Homo sapiens (human)	IC50	0.0020	1	1
Receptor-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	IC50	1.5000	2	2
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	3.6000	1	1
Receptor-interacting serine/threonine-protein kinase 3	Homo sapiens (human)	IC50	14.5200	1	1
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	GI50	3.1330	3	3
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	IC50	0.2052	51	64
Receptor-type tyrosine-protein phosphatase eta	Homo sapiens (human)	IC50	2.2000	1	1
Receptor-type tyrosine-protein phosphatase S	Homo sapiens (human)	IC50	10.3000	1	1
Replicase polyprotein 1a	Severe acute respiratory syndrome-related coronavirus	IC50	8.8250	1	2
Replicase polyprotein 1ab	Betacoronavirus England 1	IC50	13.6125	2	4
Replicase polyprotein 1ab	Human coronavirus 229E	IC50	8.8250	1	2
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	IC50	6.3339	16	24
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	IC50	10.2778	3	9
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	Ki	8.7550	1	2
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	Ki	10.4367	2	3
Retinal dehydrogenase 1	Homo sapiens (human)	IC50	0.1300	1	1
Reverse transcriptase/RNaseH	Human immunodeficiency virus 1	IC50	47.8000	3	3
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	IC50	0.1313	1	1
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	IC50	0.1839	1	1
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	IC50	10.0000	1	1
Ribosomal protein S6 kinase beta-2	Homo sapiens (human)	IC50	10.0000	1	1
RmtA	Aspergillus nidulans	IC50	5.9000	1	1
RuvB-like 1	Homo sapiens (human)	IC50	66.0000	1	1
RuvB-like 2	Homo sapiens (human)	IC50	66.0000	1	1
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	IC50	8.0500	4	4
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Ki	121.7000	1	1
Serine/threonine-protein kinase A-Raf	Homo sapiens (human)	IC50	0.0087	3	3
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	GI50	1.0000	1	1
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	IC50	0.3699	58	62
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	Ki	0.0327	3	3
Serine/threonine-protein kinase B-raf	Mus musculus (house mouse)	IC50	0.1300	1	1
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	IC50	20.0386	2	2
Serine/threonine-protein kinase Chk2	Homo sapiens (human)	IC50	0.0168	1	1
Serine/threonine-protein kinase D1	Homo sapiens (human)	IC50	16.6667	3	3
Serine/threonine-protein kinase D3	Homo sapiens (human)	IC50	16.6667	3	3
Serine/threonine-protein kinase mTOR	Homo sapiens (human)	IC50	50.0000	1	2
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	IC50	12.0000	1	1
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	IC50	0.5692	2	2
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	Ki	0.5000	1	1
Serine/threonine-protein kinase PAK 5	Homo sapiens (human)	Ki	0.5000	1	1
Serine/threonine-protein kinase PAK 6	Homo sapiens (human)	Ki	0.5000	1	1
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	IC50	5.8000	2	2
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	IC50	9.5000	2	2
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Ki	14.9800	1	8
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	IC50	314.0000	1	1
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	Ki	14.9800	1	8
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	IC50	40.0000	1	1
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	Ki	14.9800	1	8
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Ki	14.9800	1	8
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	IC50	0.2200	1	1
Serine/threonine-protein kinase TNNI3K	Homo sapiens (human)	IC50	0.1750	2	2
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	IC50	0.7900	1	1
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform	Homo sapiens (human)	IC50	30.5730	1	1
Sex hormone-binding globulin	Homo sapiens (human)	IC50	52.0000	1	1
Short transient receptor potential channel 5	Homo sapiens (human)	IC50	10.0000	1	1
Sialidase	Clostridium perfringens	IC50	2.8500	1	2
Sialidase-2	Homo sapiens (human)	IC50	130.0000	1	2
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	IC50	0.0210	1	1
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	Ki	0.0219	2	2
Signal transducer and activator of transcription 1-alpha/beta	Homo sapiens (human)	IC50	9.1000	1	1
Signal transducer and activator of transcription 3	Mus musculus (house mouse)	IC50	100.0000	1	1
Signal transducer and activator of transcription 5A	Homo sapiens (human)	IC50	9.4000	1	1
Signal transducer and activator of transcription 5B	Homo sapiens (human)	IC50	10.4000	1	1
Similar to alpha-tubulin isoform 1	Bos taurus (cattle)	IC50	2.4000	1	2
Similar to alpha-tubulin isoform 1	Bos taurus (cattle)	Ki	3.2000	1	2
Smoothened homolog	Homo sapiens (human)	Ki	0.0876	1	1
Snake venom metalloproteinase BaP1	Bothrops asper (terciopelo)	IC50	1.2000	1	1
Sodium channel protein type 5 subunit alpha	Homo sapiens (human)	IC50	27.8298	2	2
Sodium- and chloride-dependent betaine transporter	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Sodium- and chloride-dependent GABA transporter 1	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Sodium- and chloride-dependent GABA transporter 2	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Sodium- and chloride-dependent GABA transporter 3	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Sodium-dependent dopamine transporter	Homo sapiens (human)	IC50	3.2390	1	2
Sodium-dependent dopamine transporter	Homo sapiens (human)	Ki	2.5730	1	2
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	IC50	35.9210	1	2
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	Ki	35.6355	1	2
Sodium-dependent serotonin transporter	Homo sapiens (human)	IC50	2.3340	1	1
Sodium-dependent serotonin transporter	Rattus norvegicus (Norway rat)	IC50	0.0011	1	1
Sodium-dependent serotonin transporter	Homo sapiens (human)	Ki	1.2400	1	1
Solute carrier family 22 member 1	Homo sapiens (human)	IC50	6.1000	1	1
Solute carrier organic anion transporter family member 1A1	Rattus norvegicus (Norway rat)	Ki	18.2000	1	1
Solute carrier organic anion transporter family member 1A2	Homo sapiens (human)	Ki	51.0000	1	1
Solute carrier organic anion transporter family member 1A4	Rattus norvegicus (Norway rat)	Ki	1.4300	2	2
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	IC50	1.5000	4	4
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	Ki	9.0500	2	2
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	IC50	1.5000	1	1
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	Ki	3.2000	2	2
Solute carrier organic anion transporter family member 2B1	Homo sapiens (human)	IC50	65.0000	1	1
Solute carrier organic anion transporter family member 2B1	Homo sapiens (human)	Ki	63.0000	1	1
Spike glycoprotein	Betacoronavirus England 1	IC50	8.8250	1	2
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	IC50	8.8250	1	2
Steroid hormone receptor ERR1	Homo sapiens (human)	IC50	0.2000	1	1
Stromelysin-1	Homo sapiens (human)	IC50	17.4004	7	7
Substance-K receptor	Cavia porcellus (domestic guinea pig)	IC50	33.7000	1	1
Substance-K receptor	Homo sapiens (human)	IC50	3.6700	1	1
Substance-K receptor	Homo sapiens (human)	Ki	1.2230	1	1
Substance-P receptor	Cavia porcellus (domestic guinea pig)	IC50	33.7000	1	1
Substance-P receptor	Homo sapiens (human)	IC50	15.6560	1	1
Substance-P receptor	Homo sapiens (human)	Ki	8.5400	1	1
Sucrase-isomaltase, intestinal	Homo sapiens (human)	IC50	43.5000	2	2
Sucrase-isomaltase, intestinal	Rattus norvegicus (Norway rat)	IC50	156.0000	2	2
Testosterone 17-beta-dehydrogenase 3	Homo sapiens (human)	IC50	97.6100	2	2
Thiosulfate sulfurtransferase	Homo sapiens (human)	IC50	50.5000	2	2
Thromboxane-A synthase	Homo sapiens (human)	IC50	0.9160	1	1
Transcription factor GATA-4	Mus musculus (house mouse)	IC50	22.0000	1	1
Transcriptional activator protein LuxR	Aliivibrio fischeri	IC50	40.0000	1	1
Transient receptor potential cation channel subfamily M member 8	Mus musculus (house mouse)	IC50	8.0000	2	2
Transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	IC50	34.6667	3	3
Translocator protein	Rattus norvegicus (Norway rat)	IC50	0.0390	1	2
Transmembrane protease serine 2	Homo sapiens (human)	IC50	8.8250	1	2
Transthyretin	Homo sapiens (human)	IC50	6.4000	1	1
Trypanothione reductase	Trypanosoma cruzi	IC50	55.0000	2	2
Trypsin-1	Homo sapiens (human)	IC50	54.3500	1	2
Trypsin-2	Homo sapiens (human)	IC50	54.3500	1	2
Trypsin-3	Homo sapiens (human)	IC50	54.3500	1	2
Tubulin alpha-1A chain	Sus scrofa (pig)	IC50	1.8000	1	1
Tubulin beta chain	Sus scrofa (pig)	IC50	1.8000	1	1
Tubulin beta-2B chain	Bos taurus (cattle)	IC50	2.4000	1	1
Tubulin beta-2B chain	Bos taurus (cattle)	Ki	3.2000	1	1
type-1 angiotensin II receptor	Homo sapiens (human)	IC50	6.6370	1	1
Tyrosinase	Homo sapiens (human)	IC50	60.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	GI50	7.3000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	IC50	8.9610	6	7
Tyrosine-protein kinase ABL1	Mus musculus (house mouse)	IC50	0.2259	1	1
Tyrosine-protein kinase Fgr	Homo sapiens (human)	IC50	500.0000	1	1
Tyrosine-protein kinase Fyn	Homo sapiens (human)	IC50	1.1950	1	1
Tyrosine-protein kinase HCK	Homo sapiens (human)	IC50	12.8125	2	4
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	IC50	40.0000	1	1
Tyrosine-protein kinase JAK3	Homo sapiens (human)	IC50	26.1000	2	2
Tyrosine-protein kinase Lck	Homo sapiens (human)	IC50	91.7670	6	6
Tyrosine-protein kinase Lyn	Homo sapiens (human)	IC50	50.0000	1	1
Tyrosine-protein kinase Lyn	Mus musculus (house mouse)	IC50	11.1000	1	1
Tyrosine-protein kinase Mer	Homo sapiens (human)	IC50	1.3700	1	1
Tyrosine-protein kinase receptor UFO	Homo sapiens (human)	IC50	0.0090	2	2
Tyrosine-protein kinase SYK	Homo sapiens (human)	IC50	12.0000	1	1
Tyrosine-protein kinase Yes	Homo sapiens (human)	IC50	1.1102	3	3
Tyrosine-protein kinase Yes	Homo sapiens (human)	Ki	2.3800	1	1
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	IC50	40.0000	1	1
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	IC50	8.5800	2	2
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	Ki	7.8000	1	1
Ubiquitin carboxyl-terminal hydrolase isozyme L1	Homo sapiens (human)	IC50	290.0000	1	1
Ubiquitin carboxyl-terminal hydrolase isozyme L1	Mus musculus (house mouse)	IC50	180.5000	1	2
Ubiquitin carboxyl-terminal hydrolase isozyme L3	Homo sapiens (human)	IC50	71.0000	2	2
Ubiquitin carboxyl-terminal hydrolase isozyme L3	Mus musculus (house mouse)	IC50	180.5000	1	2
ubiquitin-conjugating enzyme E2 N	Homo sapiens (human)	IC50	20.0000	1	1
UDP-glucuronosyltransferase 1A1	Homo sapiens (human)	IC50	5.7000	2	2
Uracil nucleotide/cysteinyl leukotriene receptor	Homo sapiens (human)	IC50	100.0000	1	1
Urease subunit alpha	Helicobacter pylori 26695	IC50	163.2000	1	2
Urease subunit beta	Helicobacter pylori 26695	IC50	163.2000	1	2
Valosin-containing protein	Homo sapiens (human)	IC50	36.3280	2	3
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	IC50	0.0926	29	40
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	Ki	0.0310	2	2
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	GI50	0.0330	1	1
Vascular endothelial growth factor receptor 2	Danio rerio (zebrafish)	IC50	1.1933	2	3
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	IC50	1.1553	176	214
Vascular endothelial growth factor receptor 2	Mus musculus (house mouse)	IC50	0.1102	3	9
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Ki	0.0098	7	8
Vascular endothelial growth factor receptor 2	Mus musculus (house mouse)	Ki	0.0280	1	1
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	IC50	0.0822	11	12
Vascular endothelial growth factor receptor 3	Mus musculus (house mouse)	IC50	0.1269	1	7
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	Ki	0.0170	1	1
Vitamin K-dependent protein C	Homo sapiens (human)	IC50	0.2640	2	12
Voltage-dependent L-type calcium channel subunit alpha-1C	Homo sapiens (human)	IC50	104.1196	3	3
Voltage-dependent L-type calcium channel subunit alpha-1D	Homo sapiens (human)	IC50	33.4000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1F	Homo sapiens (human)	IC50	33.4000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1S	Homo sapiens (human)	IC50	33.4000	1	1
Voltage-dependent N-type calcium channel subunit alpha-1B	Homo sapiens (human)	IC50	7.0000	2	2
Voltage-dependent T-type calcium channel subunit alpha-1H	Homo sapiens (human)	IC50	2.0000	2	2
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	IC50	59.2800	2	5
Xanthine dehydrogenase/oxidase	Homo sapiens (human)	IC50	5.6700	3	4
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	Ki	1.9000	1	1
Xanthine dehydrogenase/oxidase	Homo sapiens (human)	Ki	2.9000	1	1

Activation Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
26S proteasome regulatory subunit 6B	Homo sapiens (human)	Kd	30.0000	1	9
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase	Homo sapiens (human)	Kd	0.0010	1	1
3-phosphoinositide-dependent protein kinase 1	Homo sapiens (human)	Kd	8.5000	3	13
5'-AMP-activated protein kinase catalytic subunit alpha-1	Homo sapiens (human)	Kd	12.2038	6	23
5'-AMP-activated protein kinase catalytic subunit alpha-2	Homo sapiens (human)	Kd	7.7128	3	13
5'-AMP-activated protein kinase subunit gamma-1	Homo sapiens (human)	Kd	22.8920	1	8
5'-AMP-activated protein kinase subunit gamma-2	Homo sapiens (human)	Kd	22.9382	1	8
7-dehydrocholesterol reductase	Homo sapiens (human)	Kd	0.0010	1	1
AarF domain-containing protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	9
Actin-related protein 2	Homo sapiens (human)	Kd	30.0000	1	8
Actin-related protein 3	Homo sapiens (human)	Kd	30.0000	1	8
Activated CDC42 kinase 1	Homo sapiens (human)	Kd	16.7146	4	21
Activin receptor type-1	Homo sapiens (human)	Kd	17.5510	4	22
Activin receptor type-1B	Homo sapiens (human)	Kd	17.6190	4	21
Activin receptor type-2A	Homo sapiens (human)	Kd	10.0000	3	13
Activin receptor type-2B	Homo sapiens (human)	Kd	18.6957	4	23
Acyl-CoA dehydrogenase family member 10	Homo sapiens (human)	Kd	30.0000	1	6
Acyl-CoA dehydrogenase family member 11	Homo sapiens (human)	Kd	30.0000	1	8
Adenine phosphoribosyltransferase	Homo sapiens (human)	Kd	25.0048	1	6
Adenosine kinase	Homo sapiens (human)	Kd	30.0000	1	8
Adenylate kinase 2, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	9
ADP/ATP translocase 2	Homo sapiens (human)	Kd	30.0000	1	8
ADP/ATP translocase 3	Homo sapiens (human)	Kd	30.0000	1	8
Albumin	Homo sapiens (human)	Kd	12.0000	1	1
ALK tyrosine kinase receptor	Homo sapiens (human)	Kd	9.5807	4	15
Angiopoietin-1 receptor	Homo sapiens (human)	Kd	5.7600	4	14
Angiotensin-converting enzyme 2	Homo sapiens (human)	EC50	37.8633	1	3
Ankyrin repeat and protein kinase domain-containing protein 1	Homo sapiens (human)	Kd	7.7638	3	13
AP2-associated protein kinase 1	Homo sapiens (human)	Kd	12.4233	8	25
ATP-dependent 6-phosphofructokinase, platelet type	Homo sapiens (human)	Kd	30.0000	1	7
ATP-dependent RNA helicase DDX1	Homo sapiens (human)	Kd	30.0000	1	10
ATP-dependent RNA helicase DDX3X	Homo sapiens (human)	Kd	30.0000	1	9
ATP-dependent RNA helicase DDX42	Homo sapiens (human)	Kd	30.0000	1	6
ATP-dependent RNA helicase DHX30	Homo sapiens (human)	Kd	30.0000	1	8
ATP-dependent translocase ABCB1	Homo sapiens (human)	EC50	56.5000	1	1
Atypical kinase COQ8A, mitochondrial	Homo sapiens (human)	Kd	17.6190	4	21
Atypical kinase COQ8B, mitochondrial	Homo sapiens (human)	Kd	9.4538	3	13
Aurora kinase A	Homo sapiens (human)	Kd	14.9864	5	22
Aurora kinase B	Homo sapiens (human)	Kd	11.2790	4	21
Aurora kinase C	Homo sapiens (human)	Kd	3.1368	5	15
BDNF/NT-3 growth factors receptor	Homo sapiens (human)	Kd	4.6362	3	13
Beta-adrenergic receptor kinase 1	Homo sapiens (human)	Kd	30.0000	1	8
BMP-2-inducible protein kinase	Homo sapiens (human)	Kd	12.2339	6	23
Bone morphogenetic protein receptor type-1A	Homo sapiens (human)	Kd	18.1818	4	22
Bone morphogenetic protein receptor type-1B	Homo sapiens (human)	Kd	18.9444	3	16
Bone morphogenetic protein receptor type-2	Homo sapiens (human)	Kd	14.7580	4	21
Breakpoint cluster region protein	Homo sapiens (human)	EC50	1.0000	1	1
Breakpoint cluster region protein	Homo sapiens (human)	Kd	26.3119	1	8
Bromodomain testis-specific protein	Homo sapiens (human)	Kd	0.1786	7	7
Bromodomain-containing protein 2	Homo sapiens (human)	Kd	0.0827	12	12
Bromodomain-containing protein 3	Homo sapiens (human)	Kd	0.0599	10	10
Bromodomain-containing protein 4	Homo sapiens (human)	EC50	0.1203	3	3
Bromodomain-containing protein 4	Homo sapiens (human)	Kd	0.0912	31	57
Bromodomain-containing protein 7	Homo sapiens (human)	Kd	11.0000	1	1
Bromodomain-containing protein 9	Homo sapiens (human)	Kd	17.0000	1	1
Calcium-dependent protein kinase 1	Plasmodium falciparum 3D7	Kd	6.9200	1	6
Calcium/calmodulin-dependent protein kinase kinase 1	Homo sapiens (human)	Kd	7.2971	4	14
Calcium/calmodulin-dependent protein kinase kinase 2	Homo sapiens (human)	Kd	14.5652	5	22
Calcium/calmodulin-dependent protein kinase type 1	Homo sapiens (human)	Kd	7.4936	4	14
Calcium/calmodulin-dependent protein kinase type 1D	Homo sapiens (human)	Kd	7.3307	4	14
Calcium/calmodulin-dependent protein kinase type 1G	Homo sapiens (human)	Kd	9.3746	4	13
Calcium/calmodulin-dependent protein kinase type II subunit alpha	Homo sapiens (human)	Kd	6.7320	5	15
Calcium/calmodulin-dependent protein kinase type II subunit beta	Homo sapiens (human)	Kd	7.6714	4	14
Calcium/calmodulin-dependent protein kinase type II subunit delta	Homo sapiens (human)	Kd	14.2355	5	22
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Homo sapiens (human)	Kd	11.8278	7	25
Calcium/calmodulin-dependent protein kinase type IV	Homo sapiens (human)	Kd	15.0305	4	21
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Kd	19.2286	3	21
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Kd	18.1818	4	22
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	Kd	30.0000	1	8
cAMP-dependent protein kinase catalytic subunit PRKX	Homo sapiens (human)	Kd	11.4286	4	14
cAMP-dependent protein kinase type II-alpha regulatory subunit	Homo sapiens (human)	Kd	30.0000	1	8
Casein kinase I isoform alpha	Homo sapiens (human)	Kd	16.8118	3	16
Casein kinase I isoform alpha-like	Homo sapiens (human)	Kd	8.2818	2	11
Casein kinase I isoform delta	Homo sapiens (human)	Kd	12.7778	4	21
Casein kinase I isoform epsilon	Homo sapiens (human)	Kd	14.6721	4	22
Casein kinase I isoform gamma-1	Homo sapiens (human)	Kd	16.3550	4	23
Casein kinase I isoform gamma-2	Homo sapiens (human)	Kd	16.2062	4	21
Casein kinase I isoform gamma-3	Homo sapiens (human)	Kd	14.9365	4	21
Casein kinase II subunit alpha	Homo sapiens (human)	Kd	7.7740	3	13
Casein kinase II subunit alpha'	Homo sapiens (human)	Kd	14.9572	4	21
Cell division control protein 2 homolog	Plasmodium falciparum 3D7	Kd	10.0000	1	6
Cell division cycle 7-related protein kinase	Homo sapiens (human)	Kd	30.0000	1	5
cGMP-dependent protein kinase 1	Homo sapiens (human)	Kd	17.6190	4	21
cGMP-dependent protein kinase 2	Homo sapiens (human)	Kd	10.0000	3	13
Chain A, Bromodomain testis-specific protein	Homo sapiens (human)	Kd	0.1901	1	1
Chain A, Bromodomain-containing protein 4	Homo sapiens (human)	Kd	0.0490	1	1
Chain A, Mitogen-activated protein kinase 14	Homo sapiens (human)	Kd	0.0914	1	7
Chain A, Transthyretin	Homo sapiens (human)	Kd	0.1000	1	5
Chain B, Transthyretin	Homo sapiens (human)	Kd	0.1000	1	2
Choline-phosphate cytidylyltransferase A	Homo sapiens (human)	Kd	30.0000	1	4
Chromodomain-helicase-DNA-binding protein 4	Homo sapiens (human)	Kd	30.0000	1	7
Citron Rho-interacting kinase	Homo sapiens (human)	Kd	16.4455	4	22
CREB-binding protein	Homo sapiens (human)	Kd	9.6000	1	1
Cyclin-C	Homo sapiens (human)	Kd	0.3100	1	1
Cyclin-dependent kinase 1	Homo sapiens (human)	Kd	22.8258	1	8
Cyclin-dependent kinase 10	Homo sapiens (human)	Kd	30.0000	1	4
Cyclin-dependent kinase 11A	Homo sapiens (human)	Kd	7.1151	3	13
Cyclin-dependent kinase 11B	Homo sapiens (human)	Kd	7.1382	3	13
Cyclin-dependent kinase 12	Homo sapiens (human)	Kd	26.6852	1	9
Cyclin-dependent kinase 13	Homo sapiens (human)	Kd	17.8869	2	14
Cyclin-dependent kinase 14	Homo sapiens (human)	Kd	4.6838	3	13
Cyclin-dependent kinase 15	Homo sapiens (human)	Kd	7.0675	2	8
Cyclin-dependent kinase 16	Homo sapiens (human)	Kd	11.1300	6	23
Cyclin-dependent kinase 17	Homo sapiens (human)	Kd	11.4909	4	21
Cyclin-dependent kinase 18	Homo sapiens (human)	Kd	8.2277	4	14
Cyclin-dependent kinase 19	Homo sapiens (human)	Kd	4.1768	3	13
Cyclin-dependent kinase 2	Homo sapiens (human)	Kd	13.5987	5	22
Cyclin-dependent kinase 3	Homo sapiens (human)	Kd	12.8001	4	20
Cyclin-dependent kinase 4	Homo sapiens (human)	Kd	15.1150	3	20
Cyclin-dependent kinase 6	Homo sapiens (human)	Kd	26.6824	1	9
Cyclin-dependent kinase 7	Homo sapiens (human)	Kd	10.4512	4	21
Cyclin-dependent kinase 8	Homo sapiens (human)	Kd	4.1664	4	14
Cyclin-dependent kinase 9	Homo sapiens (human)	Kd	13.1988	4	21
Cyclin-dependent kinase-like 1	Homo sapiens (human)	Kd	10.0000	1	6
Cyclin-dependent kinase-like 2	Homo sapiens (human)	Kd	4.0626	2	8
Cyclin-dependent kinase-like 3	Homo sapiens (human)	Kd	6.5475	2	8
Cyclin-dependent kinase-like 5	Homo sapiens (human)	Kd	18.6668	3	15
Cyclin-dependent-like kinase 5	Homo sapiens (human)	Kd	13.5080	5	22
Cyclin-G-associated kinase	Homo sapiens (human)	Kd	10.8298	7	24
Cysteine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	30.0000	1	7
Cytochrome c1, heme protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	10
Cytochrome P450 2B6	Homo sapiens (human)	EC50	1.3000	1	1
Cytoplasmic tyrosine-protein kinase BMX	Homo sapiens (human)	Kd	10.0000	3	13
dCTP pyrophosphatase 1	Homo sapiens (human)	Kd	30.0000	1	8
Death-associated protein kinase 1	Homo sapiens (human)	Kd	7.7200	3	13
Death-associated protein kinase 2	Homo sapiens (human)	Kd	6.7593	5	15
Death-associated protein kinase 3	Homo sapiens (human)	Kd	7.0383	6	20
Delta-type opioid receptor	Homo sapiens (human)	EC50	100.0000	1	1
Delta-type opioid receptor	Mus musculus (house mouse)	EC50	0.0030	1	2
Delta(24)-sterol reductase	Homo sapiens (human)	Kd	30.0000	1	9
Deoxycytidine kinase	Homo sapiens (human)	Kd	30.0000	1	8
Discoidin domain-containing receptor 2	Homo sapiens (human)	Kd	12.1245	7	24
DNA damage-binding protein 1	Homo sapiens (human)	EC50	0.0090	1	1
DNA replication licensing factor MCM4	Homo sapiens (human)	Kd	30.0000	1	8
DNA topoisomerase 2-alpha	Homo sapiens (human)	Kd	30.0000	1	6
DNA topoisomerase 2-beta	Homo sapiens (human)	Kd	30.0000	1	8
DNA-binding protein Ikaros	Homo sapiens (human)	EC50	0.0455	1	2
DnaJ homolog subfamily A member 1	Homo sapiens (human)	Kd	30.0000	1	8
Dual serine/threonine and tyrosine protein kinase	Homo sapiens (human)	Kd	8.5500	1	6
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	Kd	14.9033	4	21
Dual specificity mitogen-activated protein kinase kinase 2	Homo sapiens (human)	Kd	15.5458	4	22
Dual specificity mitogen-activated protein kinase kinase 3	Homo sapiens (human)	Kd	17.2238	4	21
Dual specificity mitogen-activated protein kinase kinase 4	Homo sapiens (human)	Kd	13.1688	4	16
Dual specificity mitogen-activated protein kinase kinase 5	Homo sapiens (human)	Kd	13.3951	2	14
Dual specificity mitogen-activated protein kinase kinase 6	Homo sapiens (human)	Kd	17.3905	4	21
Dual specificity mitogen-activated protein kinase kinase 7	Homo sapiens (human)	Kd	10.0000	1	6
Dual specificity protein kinase CLK1	Homo sapiens (human)	Kd	10.7787	7	24
Dual specificity protein kinase CLK2	Homo sapiens (human)	Kd	11.4601	7	23
Dual specificity protein kinase CLK3	Homo sapiens (human)	Kd	17.0000	4	20
Dual specificity protein kinase CLK4	Homo sapiens (human)	Kd	9.2538	7	20
Dual specificity protein kinase TTK	Homo sapiens (human)	Kd	12.4357	6	21
Dual specificity testis-specific protein kinase 1	Homo sapiens (human)	Kd	17.0000	4	20
Dual specificity testis-specific protein kinase 2	Homo sapiens (human)	Kd	30.0000	1	4
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	Kd	13.3015	3	16
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	Kd	11.0812	4	16
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	Kd	6.6325	2	8
Dynamin-like 120 kDa protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	8
eIF-2-alpha kinase GCN2	Homo sapiens (human)	Kd	7.7338	3	13
EKC/KEOPS complex subunit TP53RK	Homo sapiens (human)	Kd	30.0000	1	9
Electron transfer flavoprotein subunit beta	Homo sapiens (human)	Kd	26.2515	1	8
Elongation factor Tu, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	9
Ephrin type-A receptor 1	Homo sapiens (human)	Kd	15.2263	4	19
Ephrin type-A receptor 2	Homo sapiens (human)	Kd	15.9455	5	22
Ephrin type-A receptor 3	Homo sapiens (human)	Kd	5.3857	4	14
Ephrin type-A receptor 4	Homo sapiens (human)	Kd	15.9227	5	22
Ephrin type-A receptor 5	Homo sapiens (human)	Kd	15.3128	6	25
Ephrin type-A receptor 6	Homo sapiens (human)	Kd	2.9575	5	16
Ephrin type-A receptor 7	Homo sapiens (human)	Kd	13.3719	6	26
Ephrin type-A receptor 8	Homo sapiens (human)	Kd	7.2747	5	15
Ephrin type-B receptor 1	Homo sapiens (human)	Kd	4.6838	5	16
Ephrin type-B receptor 2	Homo sapiens (human)	Kd	16.0524	4	21
Ephrin type-B receptor 3	Homo sapiens (human)	Kd	18.4500	4	24
Ephrin type-B receptor 4	Homo sapiens (human)	Kd	14.7416	5	24
Ephrin type-B receptor 6	Homo sapiens (human)	Kd	15.5842	3	15
Epidermal growth factor receptor	Homo sapiens (human)	Kd	9.8653	31	149
Epithelial discoidin domain-containing receptor 1	Homo sapiens (human)	Kd	8.1176	6	23
Estrogen receptor	Homo sapiens (human)	EC50	1.1568	3	5
Estrogen receptor	Rattus norvegicus (Norway rat)	EC50	150.0000	1	4
Estrogen receptor beta	Homo sapiens (human)	EC50	0.9808	3	5
Estrogen receptor beta	Rattus norvegicus (Norway rat)	EC50	150.0000	1	4
Eukaryotic peptide chain release factor GTP-binding subunit ERF3B	Homo sapiens (human)	Kd	30.0000	1	1
Eukaryotic translation initiation factor 2-alpha kinase 1	Homo sapiens (human)	Kd	22.5000	2	16
Eukaryotic translation initiation factor 5B	Homo sapiens (human)	Kd	30.0000	1	5
Exosome RNA helicase MTR4	Homo sapiens (human)	Kd	30.0000	1	8
Ferrochelatase, mitochondrial	Homo sapiens (human)	Kd	24.5727	2	9
Fibroblast growth factor receptor 1	Homo sapiens (human)	Kd	12.5197	5	23
Fibroblast growth factor receptor 2	Homo sapiens (human)	Kd	4.7320	5	15
Fibroblast growth factor receptor 3	Homo sapiens (human)	Kd	6.2067	7	27
Fibroblast growth factor receptor 4	Homo sapiens (human)	Kd	8.6692	3	13
Focal adhesion kinase 1	Homo sapiens (human)	Kd	14.8930	6	23
G protein-coupled receptor kinase 4	Homo sapiens (human)	Kd	7.5350	2	8
G protein-coupled receptor kinase 6	Homo sapiens (human)	Kd	25.2692	1	6
G-protein coupled receptor 35	Homo sapiens (human)	EC50	10.8600	2	4
Gamma-aminobutyric acid receptor subunit alpha-1	Homo sapiens (human)	EC50	3.6000	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Homo sapiens (human)	EC50	3.6000	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Homo sapiens (human)	EC50	3.6000	1	1
General transcription and DNA repair factor IIH helicase subunit XPD	Homo sapiens (human)	Kd	23.5926	1	9
Glycine--tRNA ligase	Homo sapiens (human)	Kd	26.2550	1	8
Glycogen phosphorylase, brain form	Homo sapiens (human)	Kd	30.0000	1	8
Glycogen phosphorylase, liver form	Homo sapiens (human)	Kd	30.0000	1	8
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	Kd	15.2500	4	21
Glycogen synthase kinase-3 beta	Homo sapiens (human)	Kd	15.2559	4	21
glycogen synthase kinase-3 beta isoform 1	Homo sapiens (human)	EC50	3.8120	1	1
GTP-binding nuclear protein Ran	Homo sapiens (human)	Kd	30.0000	1	9
Guanine nucleotide-binding protein G(i) subunit alpha-2	Homo sapiens (human)	Kd	30.0000	1	7
Heat shock protein HSP 90-alpha	Homo sapiens (human)	EC50	0.0070	1	1
Heat shock protein HSP 90-alpha	Homo sapiens (human)	Kd	0.0010	1	1
Heat shock protein HSP 90-beta	Homo sapiens (human)	Kd	0.0017	1	1
Heme oxygenase 2	Homo sapiens (human)	Kd	30.0000	1	8
Hepatocyte growth factor receptor	Homo sapiens (human)	Kd	11.0066	9	37
High affinity nerve growth factor receptor	Homo sapiens (human)	Kd	9.6453	7	24
HLA class I histocompatibility antigen, A alpha chain	Homo sapiens (human)	Kd	21.2000	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	Kd	5.7694	2	8
Homeodomain-interacting protein kinase 2	Homo sapiens (human)	Kd	4.3702	2	8
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	Kd	3.1515	2	8
Homeodomain-interacting protein kinase 4	Homo sapiens (human)	Kd	3.7965	2	8
Hormonally up-regulated neu tumor-associated kinase	Homo sapiens (human)	Kd	7.6250	2	8
Inhibitor of nuclear factor kappa-B kinase subunit alpha	Homo sapiens (human)	Kd	7.6300	2	8
Inhibitor of nuclear factor kappa-B kinase subunit beta	Homo sapiens (human)	Kd	10.0000	2	8
Inhibitor of nuclear factor kappa-B kinase subunit epsilon	Homo sapiens (human)	Kd	14.9329	4	21
Inosine-5'-monophosphate dehydrogenase 2	Homo sapiens (human)	Kd	30.0000	1	8
Insulin receptor	Homo sapiens (human)	Kd	15.4942	6	24
Insulin receptor-related protein	Homo sapiens (human)	Kd	6.8531	3	13
Insulin-like growth factor 1 receptor	Homo sapiens (human)	Kd	17.1727	4	22
Integrin-linked protein kinase	Homo sapiens (human)	Kd	26.4161	1	8
Interferon-induced, double-stranded RNA-activated protein kinase	Homo sapiens (human)	Kd	7.8469	3	13
Interleukin-1 receptor-associated kinase 1	Homo sapiens (human)	Kd	19.4134	3	17
Interleukin-1 receptor-associated kinase 3	Homo sapiens (human)	Kd	14.2917	4	21
Interleukin-1 receptor-associated kinase 4	Homo sapiens (human)	Kd	16.6764	2	14
Isoleucine--tRNA ligase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	6
Kappa-type opioid receptor	Homo sapiens (human)	EC50	100.0000	1	1
LacZ protein (plasmid)	Escherichia coli	EC50	40.0000	1	1
large T antigen	Betapolyomavirus macacae	EC50	47.9300	1	1
Leucine-rich repeat serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	8.3488	2	12
Leukocyte tyrosine kinase receptor	Homo sapiens (human)	Kd	6.6538	3	13
Leukotriene C4 synthase	Cavia porcellus (domestic guinea pig)	Kd	8.4883	1	6
LIM domain kinase 1	Homo sapiens (human)	Kd	15.1144	5	23
LIM domain kinase 2	Homo sapiens (human)	Kd	16.7033	4	21
Long-chain-fatty-acid--CoA ligase 5	Homo sapiens (human)	Kd	30.0000	1	7
Lysosomal acid glucosylceramidase	Homo sapiens (human)	EC50	2.5000	1	1
Macrophage colony-stimulating factor 1 receptor	Homo sapiens (human)	Kd	1.5777	4	14
Macrophage-stimulating protein receptor	Homo sapiens (human)	Kd	19.8500	3	16
MAP kinase-activated protein kinase 2	Homo sapiens (human)	Kd	17.6190	4	21
MAP kinase-activated protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	4
MAP kinase-activated protein kinase 5	Homo sapiens (human)	Kd	17.0000	4	20
MAP kinase-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	5.5377	3	13
MAP kinase-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	5.0843	4	14
MAP/microtubule affinity-regulating kinase 3	Homo sapiens (human)	Kd	12.9390	5	22
MAP/microtubule affinity-regulating kinase 4	Homo sapiens (human)	Kd	15.2774	4	21
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	Kd	2.6495	25	113
Maternal embryonic leucine zipper kinase	Homo sapiens (human)	Kd	13.2300	4	21
Matrix metalloproteinase-9	Homo sapiens (human)	Kd	2.1800	1	1
Megakaryocyte-associated tyrosine-protein kinase	Homo sapiens (human)	Kd	9.7125	2	8
melanocortin receptor 4	Homo sapiens (human)	EC50	50.0000	1	1
Membrane-associated progesterone receptor component 1	Homo sapiens (human)	Kd	30.0000	1	5
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	Kd	18.1818	4	22
Microtubule-associated serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	7.0750	2	8
Midasin	Homo sapiens (human)	Kd	30.0000	1	9
Misshapen-like kinase 1	Homo sapiens (human)	Kd	8.9298	3	9
Mitogen-activated protein kinase 1	Homo sapiens (human)	Kd	17.6190	4	21
Mitogen-activated protein kinase 10	Homo sapiens (human)	Kd	16.8810	4	21
Mitogen-activated protein kinase 11	Homo sapiens (human)	Kd	14.4113	6	23
Mitogen-activated protein kinase 12	Homo sapiens (human)	Kd	8.9071	4	14
Mitogen-activated protein kinase 13	Homo sapiens (human)	Kd	9.1500	2	8
Mitogen-activated protein kinase 14	Homo sapiens (human)	Kd	14.8535	6	23
Mitogen-activated protein kinase 15	Homo sapiens (human)	Kd	14.5704	4	21
Mitogen-activated protein kinase 3	Homo sapiens (human)	Kd	17.6190	4	21
Mitogen-activated protein kinase 4	Homo sapiens (human)	Kd	9.0923	3	13
Mitogen-activated protein kinase 6	Homo sapiens (human)	Kd	8.5385	3	13
Mitogen-activated protein kinase 7	Homo sapiens (human)	Kd	15.5054	4	21
Mitogen-activated protein kinase 8	Homo sapiens (human)	Kd	17.6190	4	21
Mitogen-activated protein kinase 9	Homo sapiens (human)	Kd	15.6309	5	22
Mitogen-activated protein kinase kinase kinase 1	Homo sapiens (human)	Kd	18.3614	3	16
Mitogen-activated protein kinase kinase kinase 10	Homo sapiens (human)	Kd	10.0000	3	13
Mitogen-activated protein kinase kinase kinase 11	Homo sapiens (human)	Kd	13.8125	4	21
Mitogen-activated protein kinase kinase kinase 12	Homo sapiens (human)	Kd	8.3500	1	6
Mitogen-activated protein kinase kinase kinase 13	Homo sapiens (human)	Kd	7.5238	2	8
Mitogen-activated protein kinase kinase kinase 15	Homo sapiens (human)	Kd	7.8250	2	8
Mitogen-activated protein kinase kinase kinase 19	Homo sapiens (human)	Kd	1.6103	2	8
Mitogen-activated protein kinase kinase kinase 2	Homo sapiens (human)	Kd	17.0313	3	16
Mitogen-activated protein kinase kinase kinase 20	Homo sapiens (human)	Kd	13.4850	4	21
Mitogen-activated protein kinase kinase kinase 3	Homo sapiens (human)	Kd	17.1065	3	16
Mitogen-activated protein kinase kinase kinase 4	Homo sapiens (human)	Kd	15.4677	5	22
Mitogen-activated protein kinase kinase kinase 5	Homo sapiens (human)	Kd	17.6190	4	21
Mitogen-activated protein kinase kinase kinase 6	Homo sapiens (human)	Kd	20.0000	3	16
Mitogen-activated protein kinase kinase kinase 7	Homo sapiens (human)	Kd	3.4866	4	10
Mitogen-activated protein kinase kinase kinase 9	Homo sapiens (human)	Kd	8.4769	3	13
Mitogen-activated protein kinase kinase kinase kinase 1	Homo sapiens (human)	Kd	12.8378	4	20
Mitogen-activated protein kinase kinase kinase kinase 2	Homo sapiens (human)	Kd	17.7229	3	16
Mitogen-activated protein kinase kinase kinase kinase 3	Homo sapiens (human)	Kd	14.2554	4	23
Mitogen-activated protein kinase kinase kinase kinase 4	Homo sapiens (human)	Kd	11.6680	4	22
Mitogen-activated protein kinase kinase kinase kinase 5	Homo sapiens (human)	Kd	11.9946	6	26
Mitotic checkpoint serine/threonine-protein kinase BUB1	Homo sapiens (human)	Kd	25.5845	1	6
Mu-type opioid receptor	Homo sapiens (human)	EC50	100.0000	1	1
Multifunctional protein ADE2	Homo sapiens (human)	Kd	30.0000	1	8
Muscle, skeletal receptor tyrosine-protein kinase	Homo sapiens (human)	Kd	3.9908	3	13
Myosin light chain kinase 2, skeletal/cardiac muscle	Homo sapiens (human)	Kd	4.4826	5	16
Myosin light chain kinase 3	Homo sapiens (human)	Kd	19.3325	2	13
Myosin light chain kinase family member 4	Homo sapiens (human)	Kd	7.1112	3	13
Myosin light chain kinase, smooth muscle	Gallus gallus (chicken)	Kd	6.3446	1	5
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Kd	16.4345	5	25
Myosin-10	Homo sapiens (human)	Kd	30.0000	1	7
Myosin-14	Homo sapiens (human)	Kd	30.0000	1	9
Myosin-IIIa	Homo sapiens (human)	Kd	9.4692	3	13
Myosin-IIIb	Homo sapiens (human)	Kd	7.9846	3	13
Myotonin-protein kinase	Homo sapiens (human)	Kd	10.0000	3	13
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13	Homo sapiens (human)	Kd	30.0000	1	9
Non-receptor tyrosine-protein kinase TNK1	Homo sapiens (human)	Kd	15.1876	4	21
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	Kd	14.5173	6	30
NPYLR7B	Aedes aegypti (yellow fever mosquito)	EC50	20.0000	1	1
NT-3 growth factor receptor	Homo sapiens (human)	Kd	5.1938	3	13
NUAK family SNF1-like kinase 1	Homo sapiens (human)	Kd	7.7034	3	13
NUAK family SNF1-like kinase 2	Homo sapiens (human)	Kd	13.8868	4	19
Nuclear receptor subfamily 1 group I member 2	Homo sapiens (human)	EC50	2.0790	9	10
Nucleolar GTP-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	8
Obg-like ATPase 1	Homo sapiens (human)	Kd	25.0012	1	6
P2X purinoceptor 1	Rattus norvegicus (Norway rat)	EC50	1.0000	1	1
P2X purinoceptor 2	Rattus norvegicus (Norway rat)	EC50	10.4000	1	1
P2X purinoceptor 3	Homo sapiens (human)	EC50	8.9500	2	2
P2X purinoceptor 4	Rattus norvegicus (Norway rat)	EC50	100.0000	1	1
P2X purinoceptor 5	Rattus norvegicus (Norway rat)	EC50	4.0000	1	1
P2X purinoceptor 6	Rattus norvegicus (Norway rat)	EC50	100.0000	1	1
P2X purinoceptor 7	Homo sapiens (human)	EC50	92.0000	1	1
P2Y purinoceptor 1	Meleagris gallopavo (turkey)	EC50	10.0000	1	1
P2Y purinoceptor 11	Homo sapiens (human)	EC50	16.0000	1	1
P2Y purinoceptor 12	Rattus norvegicus (Norway rat)	EC50	4.0000	1	1
P2Y purinoceptor 2	Homo sapiens (human)	EC50	48.0000	1	1
P2Y purinoceptor 4	Homo sapiens (human)	EC50	100.0000	1	1
PAS domain-containing serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	7
Peripheral plasma membrane protein CASK	Homo sapiens (human)	Kd	8.4000	1	6
Peroxisomal acyl-coenzyme A oxidase 1	Homo sapiens (human)	Kd	30.0000	1	7
Peroxisomal acyl-coenzyme A oxidase 3	Homo sapiens (human)	Kd	30.0000	1	8
Peroxisome proliferator-activated receptor gamma	Mus musculus (house mouse)	EC50	2.3000	1	1
Phenylalanine--tRNA ligase beta subunit	Homo sapiens (human)	Kd	30.0000	1	8
Phosphatidylethanolamine-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	6
Phosphatidylinositol 4-kinase beta	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha	Homo sapiens (human)	Kd	8.9385	3	13
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma	Homo sapiens (human)	Kd	10.0000	1	6
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	Kd	10.0000	21	88
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	Kd	10.0000	2	8
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha	Homo sapiens (human)	Kd	30.0000	1	8
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta	Homo sapiens (human)	Kd	7.7013	3	13
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma	Homo sapiens (human)	Kd	21.4286	2	14
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform	Homo sapiens (human)	Kd	12.0101	6	23
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform	Homo sapiens (human)	Kd	5.8504	5	15
Placenta growth factor	Homo sapiens (human)	Kd	0.0082	1	1
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	Kd	1.4616	4	14
Platelet-derived growth factor receptor beta	Homo sapiens (human)	Kd	3.7819	6	26
Poly [ADP-ribose] polymerase 1	Homo sapiens (human)	EC50	0.0200	1	1
Poly [ADP-ribose] polymerase 1	Homo sapiens (human)	Kd	0.1100	1	1
Poly [ADP-ribose] polymerase tankyrase-2	Homo sapiens (human)	Kd	9.4500	1	2
POsterior Segregation	Caenorhabditis elegans	EC50	60.3740	1	1
Probable ATP-dependent RNA helicase DDX6	Homo sapiens (human)	Kd	30.0000	1	8
Procathepsin L	Homo sapiens (human)	EC50	37.8633	1	3
Prostaglandin G/H synthase 2	Homo sapiens (human)	Kd	8.3392	1	6
Protein cereblon	Homo sapiens (human)	EC50	0.0418	3	5
Protein delta homolog 1	Homo sapiens (human)	Kd	5.0500	1	2
Protein kinase C alpha type	Homo sapiens (human)	Kd	24.1818	3	11
Protein kinase C beta type	Homo sapiens (human)	Kd	30.0000	1	8
Protein kinase C delta type	Homo sapiens (human)	Kd	16.3328	4	21
Protein kinase C epsilon type	Homo sapiens (human)	Kd	10.0000	3	13
Protein kinase C eta type	Homo sapiens (human)	Kd	10.0000	3	13
Protein kinase C iota type	Homo sapiens (human)	Kd	21.4286	2	14
Protein kinase C theta type	Homo sapiens (human)	Kd	15.5220	4	21
Protein kinase C zeta type	Homo sapiens (human)	Kd	30.0000	1	6
Protein mono-ADP-ribosyltransferase PARP3	Homo sapiens (human)	Kd	0.7000	1	1
Protein polybromo-1	Homo sapiens (human)	Kd	12.9000	1	1
Protein-tyrosine kinase 2-beta	Homo sapiens (human)	Kd	16.8294	4	22
Protein-tyrosine kinase 6	Homo sapiens (human)	Kd	16.0045	5	22
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	Kd	4.5694	12	51
Proto-oncogene tyrosine-protein kinase ROS	Homo sapiens (human)	Kd	10.0000	3	13
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	Kd	15.5000	5	22
Putative heat shock protein HSP 90-beta 2	Homo sapiens (human)	Kd	26.5708	1	8
Pyridoxal kinase	Homo sapiens (human)	Kd	27.0026	1	8
Rab-like protein 3	Homo sapiens (human)	Kd	30.0000	1	8
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	Kd	17.6190	4	21
RAC-beta serine/threonine-protein kinase	Homo sapiens (human)	Kd	16.5762	4	21
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	Kd	17.6190	4	21
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	Kd	7.7454	3	13
Ras-related protein Rab-10	Homo sapiens (human)	Kd	30.0000	1	8
Ras-related protein Rab-27A	Homo sapiens (human)	Kd	30.0000	1	9
Ras-related protein Rab-6A	Homo sapiens (human)	Kd	30.0000	1	8
Receptor tyrosine-protein kinase erbB-2	Homo sapiens (human)	Kd	10.0000	3	13
Receptor tyrosine-protein kinase erbB-3	Homo sapiens (human)	Kd	10.0000	2	8
Receptor tyrosine-protein kinase erbB-4	Homo sapiens (human)	Kd	10.0000	2	8
Receptor-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	6.2200	4	14
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	14.1369	5	22
Receptor-interacting serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	8
Receptor-interacting serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	8.0250	2	8
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	Kd	3.9104	28	106
Replicase polyprotein 1a	Severe acute respiratory syndrome-related coronavirus	EC50	31.0475	2	4
Replicase polyprotein 1ab	Betacoronavirus England 1	EC50	37.8633	1	3
Replicase polyprotein 1ab	Human coronavirus 229E	EC50	31.0475	2	4
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	EC50	23.6440	3	5
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	EC50	25.4260	3	5
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	Kd	18.4000	3	3
Rho-associated protein kinase 1	Homo sapiens (human)	Kd	18.8075	3	16
Rho-associated protein kinase 2	Homo sapiens (human)	Kd	18.1819	3	16
Rhodopsin kinase GRK1	Homo sapiens (human)	Kd	7.5725	2	8
Rhodopsin kinase GRK7	Homo sapiens (human)	Kd	7.5450	2	8
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	Kd	12.4597	7	34
Ribosomal protein S6 kinase alpha-2	Homo sapiens (human)	Kd	7.8099	8	28
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	Kd	13.6942	6	23
Ribosomal protein S6 kinase alpha-4	Homo sapiens (human)	Kd	12.1854	7	34
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	Kd	11.2471	9	36
Ribosomal protein S6 kinase alpha-6	Homo sapiens (human)	Kd	12.9906	7	34
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	Kd	18.3155	3	16
Ribosyldihydronicotinamide dehydrogenase [quinone]	Homo sapiens (human)	Kd	23.0077	1	8
RNA cytidine acetyltransferase	Homo sapiens (human)	Kd	30.0000	1	9
RuvB-like 2	Homo sapiens (human)	Kd	22.0000	1	1
S-adenosylmethionine synthase isoform type-2	Homo sapiens (human)	Kd	30.0000	1	7
Septin-9	Homo sapiens (human)	Kd	30.0000	1	10
Serine/threonine-protein kinase 10	Homo sapiens (human)	Kd	9.2779	6	24
Serine/threonine-protein kinase 16	Homo sapiens (human)	Kd	14.8465	6	23
Serine/threonine-protein kinase 17A	Homo sapiens (human)	Kd	5.3950	5	15
Serine/threonine-protein kinase 17B	Homo sapiens (human)	Kd	6.7180	5	15
Serine/threonine-protein kinase 24	Homo sapiens (human)	Kd	12.7165	4	20
Serine/threonine-protein kinase 25	Homo sapiens (human)	Kd	7.7592	3	13
Serine/threonine-protein kinase 26	Homo sapiens (human)	Kd	13.4080	4	21
Serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	12.6816	4	21
Serine/threonine-protein kinase 3	Mus musculus (house mouse)	Kd	0.1600	1	1
Serine/threonine-protein kinase 32A	Homo sapiens (human)	Kd	8.4400	1	6
Serine/threonine-protein kinase 32B	Homo sapiens (human)	Kd	8.0338	3	13
Serine/threonine-protein kinase 32C	Homo sapiens (human)	Kd	10.0000	3	13
Serine/threonine-protein kinase 33	Homo sapiens (human)	Kd	4.4655	3	13
Serine/threonine-protein kinase 35	Homo sapiens (human)	Kd	6.5782	2	8
Serine/threonine-protein kinase 36	Homo sapiens (human)	Kd	6.9514	4	14
Serine/threonine-protein kinase 38	Homo sapiens (human)	Kd	7.6025	2	8
Serine/threonine-protein kinase 38-like	Homo sapiens (human)	Kd	13.3900	5	19
Serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	12.2953	6	24
Serine/threonine-protein kinase A-Raf	Homo sapiens (human)	Kd	30.0000	1	9
Serine/threonine-protein kinase ATR	Homo sapiens (human)	Kd	30.0000	1	5
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	EC50	0.0030	1	1
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	Kd	12.1595	8	35
Serine/threonine-protein kinase BRSK1	Homo sapiens (human)	Kd	8.5000	3	13
Serine/threonine-protein kinase BRSK2	Homo sapiens (human)	Kd	7.6077	3	13
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Kd	15.6452	4	22
Serine/threonine-protein kinase Chk2	Homo sapiens (human)	Kd	7.5021	2	8
Serine/threonine-protein kinase D1	Homo sapiens (human)	Kd	6.4100	3	13
Serine/threonine-protein kinase D2	Homo sapiens (human)	Kd	14.2888	4	21
Serine/threonine-protein kinase D3	Homo sapiens (human)	Kd	12.8133	4	22
Serine/threonine-protein kinase DCLK1	Homo sapiens (human)	Kd	6.4854	3	13
Serine/threonine-protein kinase DCLK2	Homo sapiens (human)	Kd	6.9308	3	13
Serine/threonine-protein kinase DCLK3	Homo sapiens (human)	Kd	6.4254	3	13
Serine/threonine-protein kinase ICK	Homo sapiens (human)	Kd	17.4060	3	15
Serine/threonine-protein kinase LATS1	Homo sapiens (human)	Kd	13.9773	4	22
Serine/threonine-protein kinase LATS2	Homo sapiens (human)	Kd	6.5215	3	13
Serine/threonine-protein kinase MAK	Homo sapiens (human)	Kd	9.0375	2	8
Serine/threonine-protein kinase MARK1	Homo sapiens (human)	Kd	7.9692	3	13
Serine/threonine-protein kinase MARK2	Homo sapiens (human)	Kd	13.6767	5	23
Serine/threonine-protein kinase MRCK alpha	Homo sapiens (human)	Kd	17.6190	4	21
Serine/threonine-protein kinase MRCK beta	Homo sapiens (human)	Kd	18.1818	4	22
Serine/threonine-protein kinase MRCK gamma	Homo sapiens (human)	Kd	17.5381	4	21
Serine/threonine-protein kinase mTOR	Homo sapiens (human)	Kd	10.0000	1	6
Serine/threonine-protein kinase N1	Homo sapiens (human)	Kd	14.8712	4	21
Serine/threonine-protein kinase N2	Homo sapiens (human)	Kd	15.0055	4	21
Serine/threonine-protein kinase N3	Homo sapiens (human)	Kd	30.0000	1	6
Serine/threonine-protein kinase Nek1	Homo sapiens (human)	Kd	17.6190	4	21
Serine/threonine-protein kinase Nek11	Homo sapiens (human)	Kd	10.0000	1	6
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	Kd	15.0087	6	23
Serine/threonine-protein kinase Nek3	Homo sapiens (human)	Kd	22.0063	2	14
Serine/threonine-protein kinase Nek4	Homo sapiens (human)	Kd	10.0000	1	6
Serine/threonine-protein kinase Nek5	Homo sapiens (human)	Kd	10.0000	3	13
Serine/threonine-protein kinase Nek6	Homo sapiens (human)	Kd	10.0000	3	13
Serine/threonine-protein kinase Nek7	Homo sapiens (human)	Kd	16.1150	4	20
Serine/threonine-protein kinase Nek9	Homo sapiens (human)	Kd	17.6190	4	21
Serine/threonine-protein kinase NIM1	Homo sapiens (human)	Kd	7.7125	2	8
Serine/threonine-protein kinase NLK	Homo sapiens (human)	Kd	16.2819	4	21
Serine/threonine-protein kinase OSR1	Homo sapiens (human)	Kd	7.6325	2	8
Serine/threonine-protein kinase PAK 1	Homo sapiens (human)	Kd	10.0000	3	13
Serine/threonine-protein kinase PAK 2	Homo sapiens (human)	Kd	17.0000	4	20
Serine/threonine-protein kinase PAK 3	Homo sapiens (human)	Kd	6.6960	3	13
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	Kd	15.8140	4	22
Serine/threonine-protein kinase PAK 5	Homo sapiens (human)	Kd	7.8400	3	13
Serine/threonine-protein kinase PAK 6	Homo sapiens (human)	Kd	12.3250	4	16
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	Kd	17.6190	4	21
Serine/threonine-protein kinase pim-2	Homo sapiens (human)	Kd	15.0000	5	19
Serine/threonine-protein kinase pim-3	Homo sapiens (human)	Kd	8.2462	3	13
Serine/threonine-protein kinase PknB	Mycobacterium tuberculosis H37Rv	Kd	8.3478	1	6
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Kd	14.7059	4	17
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	Kd	8.6750	2	8
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	Kd	9.7692	3	13
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Kd	14.0212	6	25
Serine/threonine-protein kinase PRP4 homolog	Homo sapiens (human)	Kd	7.5975	2	8
Serine/threonine-protein kinase receptor R3	Homo sapiens (human)	Kd	11.4286	4	14
Serine/threonine-protein kinase RIO1	Homo sapiens (human)	Kd	7.7004	3	13
Serine/threonine-protein kinase RIO2	Homo sapiens (human)	Kd	5.7553	3	9
Serine/threonine-protein kinase RIO3	Homo sapiens (human)	Kd	8.5692	3	13
Serine/threonine-protein kinase SBK1	Homo sapiens (human)	Kd	8.3667	1	6
Serine/threonine-protein kinase Sgk3	Homo sapiens (human)	Kd	7.0200	1	6
Serine/threonine-protein kinase SIK1	Homo sapiens (human)	Kd	8.4308	3	13
Serine/threonine-protein kinase SIK2	Homo sapiens (human)	Kd	16.0705	4	22
Serine/threonine-protein kinase SIK3	Homo sapiens (human)	Kd	18.8236	3	17
Serine/threonine-protein kinase STK11	Homo sapiens (human)	Kd	16.8234	4	22
Serine/threonine-protein kinase TAO1	Homo sapiens (human)	Kd	14.3488	4	18
Serine/threonine-protein kinase TAO2	Homo sapiens (human)	Kd	20.1671	2	14
Serine/threonine-protein kinase TAO3	Homo sapiens (human)	Kd	16.6688	3	16
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	Kd	18.4301	3	18
Serine/threonine-protein kinase TNNI3K	Homo sapiens (human)	Kd	7.2229	4	14
Serine/threonine-protein kinase tousled-like 1	Homo sapiens (human)	Kd	7.8631	3	13
Serine/threonine-protein kinase tousled-like 2	Homo sapiens (human)	Kd	7.7685	3	13
Serine/threonine-protein kinase ULK1	Homo sapiens (human)	Kd	14.7409	3	16
Serine/threonine-protein kinase ULK2	Homo sapiens (human)	Kd	7.5032	2	8
Serine/threonine-protein kinase ULK3	Homo sapiens (human)	Kd	16.9506	3	16
Serine/threonine-protein kinase ULK3	Mus musculus (house mouse)	Kd	0.1100	1	1
Serine/threonine-protein kinase VRK2	Homo sapiens (human)	Kd	10.0000	1	6
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	Kd	18.8250	3	16
Serine/threonine-protein kinase/endoribonuclease IRE2	Homo sapiens (human)	Kd	30.0000	1	8
Sex hormone-binding globulin	Homo sapiens (human)	Kd	0.3090	1	1
Signal recognition particle receptor subunit alpha	Homo sapiens (human)	Kd	30.0000	1	6
Similar to alpha-tubulin isoform 1	Bos taurus (cattle)	Kd	8.2000	2	4
SNF-related serine/threonine-protein kinase	Homo sapiens (human)	Kd	8.4400	1	6
Sodium-dependent dopamine transporter	Rattus norvegicus (Norway rat)	EC50	1.4500	1	1
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	EC50	31.0000	1	1
Spike glycoprotein	Betacoronavirus England 1	EC50	37.8633	1	3
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	EC50	37.8633	1	3
SRSF protein kinase 1	Homo sapiens (human)	Kd	7.7500	3	13
SRSF protein kinase 2	Homo sapiens (human)	Kd	7.7362	3	13
SRSF protein kinase 3	Homo sapiens (human)	Kd	7.5148	2	8
STE20-like serine/threonine-protein kinase	Homo sapiens (human)	Kd	12.5482	6	24
STE20-related kinase adapter protein alpha	Homo sapiens (human)	Kd	23.7716	1	9
STE20/SPS1-related proline-alanine-rich protein kinase	Homo sapiens (human)	Kd	7.5350	2	8
streptokinase A precursor	Streptococcus pyogenes M1 GAS	EC50	77.1175	2	4
Structural maintenance of chromosomes protein 1A	Homo sapiens (human)	Kd	30.0000	1	9
Structural maintenance of chromosomes protein 2	Homo sapiens (human)	Kd	30.0000	1	9
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial	Homo sapiens (human)	Kd	26.2509	1	8
Testis-specific serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	9.1462	3	13
TGF-beta receptor type-1	Homo sapiens (human)	Kd	18.1818	4	22
TGF-beta receptor type-2	Homo sapiens (human)	Kd	17.3500	4	22
Thyroid hormone receptor-associated protein 3	Homo sapiens (human)	Kd	30.0000	1	8
TRAF2 and NCK-interacting protein kinase	Homo sapiens (human)	Kd	11.3687	6	23
Transient receptor potential cation channel subfamily A member 1	Homo sapiens (human)	EC50	6.3333	3	3
Transient receptor potential cation channel subfamily M member 6	Homo sapiens (human)	Kd	10.0000	1	6
Transient receptor potential cation channel subfamily M member 8	Mus musculus (house mouse)	EC50	8.0000	1	1
Transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	Kd	19.9526	1	1
Transmembrane protease serine 2	Homo sapiens (human)	EC50	37.8633	1	3
Transthyretin	Homo sapiens (human)	Kd	0.0700	1	1
Tubulin alpha-1A chain	Rattus norvegicus (Norway rat)	Kd	10.0000	1	5
Tubulin alpha-1A chain	Sus scrofa (pig)	Kd	1.0450	4	4
Tubulin beta chain	Sus scrofa (pig)	Kd	1.0450	4	4
Tubulin beta-2B chain	Bos taurus (cattle)	Kd	8.2000	2	2
Tyrosine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	26.6645	1	8
Tyrosine-protein kinase ABL1	Homo sapiens (human)	EC50	1.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	Kd	5.8352	41	179
Tyrosine-protein kinase ABL2	Homo sapiens (human)	Kd	13.7885	5	24
Tyrosine-protein kinase Blk	Homo sapiens (human)	Kd	7.0919	3	13
Tyrosine-protein kinase BTK	Homo sapiens (human)	Kd	17.2429	4	21
Tyrosine-protein kinase CSK	Homo sapiens (human)	Kd	17.2810	4	21
Tyrosine-protein kinase Fer	Homo sapiens (human)	Kd	14.3954	5	22
Tyrosine-protein kinase Fes/Fps	Homo sapiens (human)	Kd	16.3276	4	21
Tyrosine-protein kinase Fgr	Homo sapiens (human)	Kd	8.9282	6	18
Tyrosine-protein kinase FRK	Homo sapiens (human)	Kd	11.6183	7	24
Tyrosine-protein kinase Fyn	Homo sapiens (human)	Kd	15.6300	5	22
Tyrosine-protein kinase HCK	Homo sapiens (human)	Kd	14.0492	5	22
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	Kd	7.6953	3	13
Tyrosine-protein kinase JAK1	Homo sapiens (human)	Kd	12.3432	8	31
Tyrosine-protein kinase JAK2	Homo sapiens (human)	Kd	13.2721	5	19
Tyrosine-protein kinase JAK3	Homo sapiens (human)	Kd	7.7615	3	13
Tyrosine-protein kinase Lck	Homo sapiens (human)	Kd	12.3337	5	23
Tyrosine-protein kinase Lyn	Homo sapiens (human)	Kd	12.7090	6	23
Tyrosine-protein kinase Mer	Homo sapiens (human)	Kd	9.5386	4	16
Tyrosine-protein kinase receptor Tie-1	Homo sapiens (human)	Kd	5.0326	3	13
Tyrosine-protein kinase receptor TYRO3	Homo sapiens (human)	Kd	7.7036	3	13
Tyrosine-protein kinase receptor UFO	Homo sapiens (human)	Kd	4.9390	3	13
Tyrosine-protein kinase Srms	Homo sapiens (human)	Kd	9.9538	3	13
Tyrosine-protein kinase SYK	Homo sapiens (human)	EC50	4.5000	1	1
Tyrosine-protein kinase SYK	Homo sapiens (human)	Kd	18.1818	4	22
Tyrosine-protein kinase Tec	Homo sapiens (human)	Kd	17.6190	4	21
Tyrosine-protein kinase TXK	Homo sapiens (human)	Kd	10.0000	3	13
Tyrosine-protein kinase Yes	Homo sapiens (human)	Kd	14.2830	5	23
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	Kd	10.0000	3	13
U5 small nuclear ribonucleoprotein 200 kDa helicase	Homo sapiens (human)	Kd	30.0000	1	8
UMP-CMP kinase	Homo sapiens (human)	Kd	18.0018	1	5
Uncharacterized aarF domain-containing protein kinase 5	Homo sapiens (human)	Kd	30.0000	1	7
Uncharacterized protein FLJ45252	Homo sapiens (human)	Kd	26.7146	1	9
Uncharacterized serine/threonine-protein kinase SBK3	Homo sapiens (human)	Kd	7.9750	2	8
Vascular endothelial growth factor A	Homo sapiens (human)	Kd	0.0165	1	1
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	Kd	1.4338	4	14
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	EC50	0.5000	1	1
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Kd	1.0323	7	20
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	Kd	1.1931	5	18
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	8
Wee1-like protein kinase	Homo sapiens (human)	Kd	18.5663	4	22
Wee1-like protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	8
Zinc finger protein Aiolos	Homo sapiens (human)	EC50	0.0545	1	2
Zinc finger protein mex-5	Caenorhabditis elegans	EC50	31.0000	1	1

Other Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
Androgen receptor	Homo sapiens (human)	EC150	18.4500	1	2
Arylacetamide deacetylase	Homo sapiens (human)	Km	200.0000	1	2
Breakpoint cluster region protein	Homo sapiens (human)	DC50	10.0000	1	2
Bromodomain-containing protein 4	Homo sapiens (human)	DC50	5.0000	1	1
Catechol O-methyltransferase	Rattus norvegicus (Norway rat)	Km	3.2400	2	2
Cholinesterase	Homo sapiens (human)	Activity	0.0400	1	1
Cyclic AMP-responsive element-binding protein 1	Homo sapiens (human)	AC50	13.5000	1	1
cystic fibrosis transmembrane conductance regulator ATP-binding cassette sub-family C member 7	Homo sapiens (human)	AC50	29.2700	1	1
Cytochrome P450 1A2	Homo sapiens (human)	Km	45.0000	1	1
Cytochrome P450 3A4	Homo sapiens (human)	Km	32.7000	1	1
Delta-type opioid receptor	Homo sapiens (human)	Ke	6.0000	1	1
Dihydrolipoyl dehydrogenase, mitochondrial	Sus scrofa (pig)	Km	72.0000	1	1
DNA damage-binding protein 1	Homo sapiens (human)	DC50	5.0000	1	1
DNA-binding protein Ikaros	Homo sapiens (human)	DC50	0.0584	1	2
DNA-binding protein Ikaros	Homo sapiens (human)	fEC50	0.2805	1	2
dual specificity tyrosine-phosphorylation-regulated kinase 1A	Rattus norvegicus (Norway rat)	AC50	14.5280	1	1
E3 ubiquitin-protein ligase ZFP91	Homo sapiens (human)	DC50	0.4200	1	1
Estrogen receptor	Rattus norvegicus (Norway rat)	A50	0.0200	1	1
Estrogen receptor	Homo sapiens (human)	DC50	0.0910	1	1
Estrogen receptor	Homo sapiens (human)	MEC	1.0000	1	1
Estrogen receptor beta	Rattus norvegicus (Norway rat)	A50	0.0200	1	1
Estrogen receptor beta	Homo sapiens (human)	MEC	1.0000	1	1
Fibroblast growth factor receptor 1	Homo sapiens (human)	Activity	0.2760	1	1
Fibroblast growth factor receptor 2	Homo sapiens (human)	Activity	0.2760	1	1
Fibroblast growth factor receptor 3	Homo sapiens (human)	Activity	0.2760	1	1
Fibroblast growth factor receptor 4	Homo sapiens (human)	Activity	0.2760	1	1
Glucocorticoid receptor	Homo sapiens (human)	EC150	18.4500	1	2
Glutathione reductase	Plasmodium falciparum 3D7	Km	82.2000	1	1
Glutathione reductase, mitochondrial	Homo sapiens (human)	Km	31.2000	1	1
H3 histone acetyltransferase	Candida albicans SC5314	AC50	3.2600	1	1
heat shock protein 90, putative	Plasmodium falciparum 3D7	AC50	4.5540	1	1
heat shock protein HSP 90-alpha isoform 2	Homo sapiens (human)	AC50	5.1780	1	1
hypothetical protein CAALFM_CR05890CA	Candida albicans SC5314	AC50	3.2600	1	1
interferon gamma precursor	Homo sapiens (human)	AC50	35.2400	1	1
Kappa-type opioid receptor	Homo sapiens (human)	Ke	0.4900	1	1
Mu-type opioid receptor	Homo sapiens (human)	Ke	10.0000	1	1
NAD	Homo sapiens (human)	Km	1.3000	3	3
NAD	Homo sapiens (human)	Vmax	7,286.0000	1	1
Nuclear receptor subfamily 1 group I member 2	Homo sapiens (human)	MEC	2.0000	1	2
Platelet-activating factor acetylhydrolase	Homo sapiens (human)	Km	72.0000	1	5
Protein cereblon	Homo sapiens (human)	DC50	5.0233	3	5
Protein cereblon	Homo sapiens (human)	fEC50	0.2805	1	2
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	INH	0.0399	2	4
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Km	169.0500	2	2
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Vmax	0.0105	2	2
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	Km	7.2500	2	2
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	Km	2.3000	1	1
Transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	Kb	18.0000	1	1
Trypanothione reductase	Trypanosoma cruzi	Km	21.0000	1	1
Trypanothione reductase	Trypanosoma cruzi	x fold	375.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	DC50	10.0000	1	2
UDP-glucuronosyltransferase 1A4	Homo sapiens (human)	Km	32.0000	1	1
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	Activity	0.0400	1	1
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Activity	0.0400	1	1
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	ED50	0.0340	1	1
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	INH	100.0000	1	1
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	Activity	0.0400	1	1
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	Km	32.3500	4	4

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angiogenesis inhibitor

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Protein Targets (1,248)

Potency Measurements

Inhibition Measurements

Activation Measurements

Other Measurements