An agent and endogenous substances that antagonize or inhibit the development of new blood vessels.
| Member | Definition | Class |
|---|
| 2-methyl-1,4-hydroquinone | A member of the class of hydroquinones that is hydroquinone in which one of the benzene hydrogens has been replaced by a methyl group. | toluquinol |
| 3-(3-pyridinyl)-1-(4-pyridinyl)-2-propen-1-one | A member of the class of pyridines that is pyridine substituted by a 3-oxo-3-(pyridin-4-yl)prop-1-en-1-yl group at position 3. An inhibitor of PFKFB3 kinase, an enzyme with a key role in glycolysis. | 3PO |
| abt 869 | A member of the class of phenylureas that is urea in which one of the nitrogens is substituted by a 2-fluoro-5-methylphenyl group, while the other is substituted by a p-(3-amino-1H-indazol-4-yl)phenyl group. It is a potent, selective inhibitor of vascular endothelial growth factor and platelet-derived growth factor receptor tyrosine kinases. | linifanib |
| acetopyrrothine | A dithiolopyrrolone antibiotic that is 4,5-dihydro[1,2]dithiolo[4,3-b]pyrrole in which the hydrogens at positions 4,5 and 6 have been replaced by methyl, oxo and acetamido groups, respectively. It is a potent inhibitor of RNA polymerases, inhibits the angiogenesis of human umbilical vein endothelial cells, and also inhibits JAMM metalloproteases. | thiolutin |
| aee 788 | A 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-N-(1-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine which adopts an R-configuration. It is a potent inhibitor of human EGFR, VEGFR and HER2 receptor tyrosine kinases and exhibits anticancer and antiangiogenic activity. | AEE788 |
| ageladine a | An imidazopyridine that is 1H-imidazo[4,5-c]pyridin-2-amine substituted by a 4,5-dibromo-1H-pyrrol-2-yl group at position 4. It is an alkaloid isolated from a marine sponge Agelas nakamurai and acts as an inhibitor of the matrix metalloproteinases, the key enzymes involved in tumour growth, migration, angiogenesis, invasion and metastasis. | ageladine A |
| amentoflavone | A biflavonoid that is obtained by oxidative coupling of two molecules of apigenin resulting in a bond between positions C-3 of the hydroxyphenyl ring and C-8 of the chromene ring. A natural product found particularly in Ginkgo biloba and Hypericum perforatum. | amentoflavone |
| antofine | An organic heteropentacyclic compound that is (13aR)-9,11,12,13,13a,14-hexahydrodibenzo[f,h]pyrrolo[1,2-b]isoquinoline substituted at positions 2, 3 and 6 by methoxy groups. It is an alkaloid produced by relatives of the milkweed family and exhibits antiviral, anti-inflammatory, antiadipogenic and antitumorigenic activities. | (-)-antofine |
| ascochlorin | A dihydroxybenzaldehyde that is 2,4-dihydroxybenzaldehyde which is substituted by a (1E,3E)-3-methyl-1-[(1R,2R,6R)-1,2,6-trimethyl-3-oxocyclohexyl]penta-1,3-dien-5-yl group at position 3, chlorine at position 5, and a methyl group at position 6. A meroterpenoid produced by several fungi including Ascochyta viciae . It exhibits anticancer, antifungal and antiprotozoal activities. | ascochlorin |
| ascofuranone | A dihydroxybenzaldehyde that is 2,4-dihydroxybenzaldehyde which is substituted by a (2E,6E)-7-[(2S)-5,5-dimethyl-4-oxotetrahydrofuran-2-yl]-3-methylocta-2,6-dien-1-yl group at position 3, chlorine at position 5, and a methyl group at position 6. A meroterpenoid produced by the soil fungus, Acremonium sclerotigenum. It is a promising drug candidate against the tropical disease, African trypanosomiasis. | ascofuranone |
| aureothricin | A dithiolopyrrolone antibiotic that is 4,5-dihydro[1,2]dithiolo[4,3-b]pyrrole in which the hydrogens at positions 4,5 and 6 have been replaced by methyl, oxo and propanoylamino groups, respectively. It is a moderate antimicrobial by-product of the thiolutin fermentation in various Streptomyces species. | aureothricin |
| baicalein | A trihydroxyflavone with the hydroxy groups at positions C-5, -6 and -7. | baicalein |
| batimastat | A secondary carboxamide resulting from the formal condensation of the carboxy group of (2S,3R)-5-methyl-3-{[(2S)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]carbamoyl}-2-[(thiophen-2-ylsulfanyl)methyl]hexanoic acid with the amino group of hydroxylamine. It a broad-spectrum matrix metalloprotease inhibitor. | batimastat |
| bms 387032 | A secondary carboxamide resulting from the formal condensation of the carboxy group of piperidine-4-carboxylic acid with the amino group of 5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-amine. It is an ATP-competitive inhibitor of CDK2, CDK7 and CDK9 kinases and exhibits anti-cancer properties. | N-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide |
| brivanib | A secondary alcohol resulting from the hydrolysis of the carboxylic ester group of brivanib alaninate. It is a dual VEGFR-2/FGFR-1 kinase inhibitor whose alanine prodrug, brivanib alaninate is currently under development as an oral agent for the treatment of cancer. | (2R)-1-[[4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methyl-6-pyrrolo[2,1-f][1,2,4]triazinyl]oxy]-2-propanol; brivanib |
| cafestol | An organic heteropentacyclic compound and furan diterpenoid with formula C20H28O3 obtained from the unsaponifiable fraction of coffee oil (a lipid fraction obtained from coffee beans by organic solvent extraction). | cafestol |
| can 508 | A member of the class of pyrazoles that is 1H-pyrazole substituted by amino, (4-hydroxyphenyl)diazenyl, and amino groups at positions 3, 4 and 5, respectively. It is a CDK9 inhibitor (IC50 = 0.35 muM) with 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. | CAN-508 |
| capsiate | A carboxylic ester obtained by formal condensation of the carboxy group of (6E)-8-methylnon-6-enoic acid with the benzylic hydroxy group of vanillyl alcohol. A non-pungent analogue of capsaicin with a similar biological profile. | capsiate |
| crenolanib | A member of the class of benzimidazoles that is 1H-benzimidazole which is substituted by a 8-(4-aminopiperidin-1-yl)quinolin-2-yl group at position 1 and by a (3-methyloxetan-3-yl)methoxy group at position 5. It is an inhibitor of type III tyrosine kinases, PDGFRalpha/beta and FLT3 (IC50 of 11, 3.2, and 4 nM). Currently under clinical development for the treatment of acute myeloid leukemia. | crenolanib |
| deguelin | A rotenone that is 13,13a-dihydro-3H-chromeno[3,4-b]pyrano[2,3-h]chromen-7(7aH)-one substituted by methoxy groups at positions 9 and 10, and by two methyl groups at position 3 (the 7aS,13aS-stereoisomer). It exists in abundant quantities in the bark, roots, and leaves of the Leguminosae family of plants and reported to exert anti-tumour effects in various cancers. | deguelin |
| diosmetin | A monomethoxyflavone that is the 4'-methyl ether derivative of luteolin. It is a natural product isolated from citrus fruits which exhibits a range of pharmacological activities. | diosmetin |
| disulfiram | An organic disulfide that results from the formal oxidative dimerisation of N,N-diethyldithiocarbamic acid. A multi-enzyme inhibitor that is used in alcohol aversion therapy and also exhibits anticancer properties. | disulfiram |
| EG00229 | A member of the class of thiophenes that is thiophene substituted by a carbonyl-L-arginine and (2,1,3-benzothiadiazole-4-sulfonyl)amino groups at positions 2 and 3. It is an inhibitor of the neuropilin-1 and VEGF-A interaction and a potential anti-cancer agent. | EG00229 |
| fumagillin | A meroterpenoid resulting from the formal condensation of the hydroxy group of fumagillol with the carboxylic acid group of (all-E)-deca-2,4,6,8-tetraenedioic acid. Originally isolated from the fungus Aspergillus fumigatus, it is used for the control of Nosema infection in honey bees. | fumagillin |
| herbacetin | A pentahydroxyflavone that is kaempferol substituted by a hydroxy group at position 8. It is a natural flavonoid from flaxseed which exerts antioxidant, anti-inflammatory and anticancer activities. | herbacetin |
| jq1 compound | A member of the class of thienotriazolodiazepines that is the tert-butyl ester of [(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetic acid. An inhibitor of bromodomain-containing protein 4 that exhibits anti-cancer and cardioprotective properties. | JQ1 |
| kahweol | A diterpenoid with formula C20H26O3, isolated from the beans of Coffea arabica. It exhibits antioxidant, anti-inflammatory, anti-angiogenesis and anti-proliferative properties. | kahweol |
| lenalidomide | A dicarboximide that consists of 1-oxoisoindoline bearing an amino substituent at position 4 and a 2,6-dioxopiperidin-3-yl group at position 2. Inhibits the secretion of TNF-alpha. | lenalidomide |
| lupulon | A beta-bitter acid in which the acyl group is specified as 3-methylbutanoyl. | lupulone |
| luteolin | A tetrahydroxyflavone in which the four hydroxy groups are located at positions 3', 4', 5 and 7. It is thought to play an important role in the human body as an antioxidant, a free radical scavenger, an anti-inflammatory agent and an immune system modulator as well as being active against several cancers. | luteolin |
| matairesinol | A lignan that is gamma-butyrolactone in which the 3 and 4 positions are substituted by 4-hydroxy-3-methoxybenzyl groups (the 3R,4R-diastereomer). | (-)-matairesinol |
| n-(3-(aminomethyl)benzyl)acetamidine | An aralkylamine that is Nbenzylacetamidine substituted at position 3 on the benzene ring by an aminomethyl group. An inhibitor of nitric oxide synthase. | N-[3-(aminomethyl)benzyl]acetamidine |
| nnc 55-0396 | The dihydrochloride salt of NNC 55-0396. It is a stable analogue of mibefradil and a highly selective T-type calcium channel blocker. | NNC 55-0396 dihydrochloride |
| NNC 55-0396 (free base) | | NNC 55-0396 (free base) |
| npi 2358 | A member of the class of 2,5-diketopiperazines that is piperazine-2,5-dione substituted by benzylidene and (5-tert-butyl-1H-imidazol-4-yl)methylidene groups at positions 3 and 6, respectively. It is a vascular disrupting agent and a microtubule destabalising agent which was in clinical trials (now discontinued) for the treatment of non-small cell lung cancer. | plinabulin |
| o-(chloroacetylcarbamoyl)fumagillol | A carbamate ester that is fumagillol in which the hydroxy group has been converted to the corresponding N-(chloroacetyl)carbamate derivative. | O-(chloroacetylcarbamoyl)fumagillol |
| oridonin | An organic heteropentacyclic compound and ent-kaurane diterpenoid with formula C20H28O6 isolated from the leaves of the medicinal herb Rabdosia rubescens. | oridonin |
| pd 166866 | A member of the class of pyridopyrimidines that is pyrido[2,3-d]pyrimidine substituted by an amino group at position 2, 3,5-dimethoxyphenyl group at position 6, and by a (tert-butylcarbamoyl)nitrilo group at position 7. It is a selective ATP competitive inhibitor of the human fibroblast growth factor-1 receptor (FGFR1) tyrosine kinase with an IC50 of 52.4 nM. | PD-166866 |
| pj-34 | A member of the class of phenanthridines that is 5,6-dihydrophenanthridine substituted at positions 2 and 6 by (N,N-dimethylglycyl)amino and oxo groups, respectively. It is a potent inhibitor of poly(ADP-ribose) polymerases PARP1 and PARP2 (IC50 of 110 nM and 86 nM, respectively) and exhibits anti-cancer, cardioprotective and neuroprotective properties. | PJ34 |
| pomalidomide | An aromatic amine that is thalidomide substituted at position 4 on the isoindole ring system by an amino group. Used for the treatment of multiple myeloma in patients who failed to respond to previous therapies. | pomalidomide |
| ptk 787 | A succinate salt obtained by combining vatalanib with one molar equivalent of succinic acid. It is a multi-targeted tyrosine kinase inhibitor for all isoforms of VEGFR, PDGFR and c-Kit. | vatalanib succinate |
| quininib | A styrylquinoline that is trans-2-styrylquinoline in which the the phenyl group has been substituted at position 2 by a hydroxy group. It is an anti-angiogenic compound that exerts a dose-dependent antagonism of the cysteinyl leukotriene pathway, preferentially antagonising cysteinyl leukotriene receptor 1. The major species at pH 7.3 | quininib |
| rhapontin | A rhaponticin in which the double bond adopts a trans-configuration. It possesses a range of pharmacological activities including antitumour, antiinflammatory, antilipemic and neuroprotective activities. | trans-rhaponticin |
| rifampin | A member of the class of rifamycins that is a a semisynthetic antibiotic derived from Amycolatopsis rifamycinica (previously known as Amycolatopsis mediterranei and Streptomyces mediterranei). | rifampicin zwitterion; rifampicin |
| sb 220025 | Am member of the class of imidazoles carrying piperidin-4-yl, 4-fluophenyl and 2-aminopyrimidin-4-yl substituents at posiitons 1, 4 and 5 respectively. | SB220025 |
| sorafenib | A member of the class of phenylureas that is urea in which one of the nitrogens is substituted by a 4-chloro-3-trifluorophenyl group while the other is substituted by a phenyl group which, in turn, is substituted at the para position by a [2-(methylcarbamoyl)pyridin-4-yl]oxy group. | sorafenib |
| su 11248 | | sunitinib |
| suramin | A member of the class of phenylureas that is urea in which each of the amino groups has been substituted by a 3-({2-methyl-5-[(4,6,8-trisulfo-1-naphthyl)carbamoyl]phenyl}carbamoyl)phenyl group. An activator of both the rabbit skeletal muscle RyR1 and sheep cardiac RyR2 isoform ryanodine receptor channels, it has been used for the treatment of human African trypanosomiasis for over 100 years. | suramin |
| suramin sodium | An organic sodium salt that is the hexasodium salt of suramin. It is an FDA approved drug for African sleeping sickness and river blindness. | suramin sodium |
| tamoxifen | | tamoxifen |
| tamoxifen citrate | | tamoxifen citrate |
| vatalanib | A member of the class of phthalazines that is phthalazine in which the hydrogens at positions 1 and 4have been replaced by a p-chlorophenylamino group and a pyridin-4-ylmethyl group, respectively. It is a multi-targeted tyrosine kinase inhibitor for all isoforms of VEGFR, PDGFR and c-Kit. | vatalanib |
| ver 52296 | A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 5-(2,4-dihydroxy-5-isopropylphenyl)-4-[4-(morpholin-4-ylmethyl)phenyl]-1,2-oxazole-3-carboxylic acid with the amino group of ethylamine. | luminespib |
| vitamin k 3 | A member of the class of 1,4-naphthoquinones that is 1,4-naphthoquinone which is substituted at position 2 by a methyl group. It is used as a nutritional supplement and for the treatment of hypoprothrombinemia. | menadione |
| voacamine | A monoterpenoid indole alkaloid with formula C22H28N2O3, isolated from several plant species. | (-)-voacangine |
| wogonin | A dihydroxy- and monomethoxy-flavone in which the hydroxy groups are positioned at C-5 and C-7 and the methoxy group is at C-8. | wogonin |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 10.9165 | 1 | 11 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 5.5253 | 1 | 7 |
| 67.9K protein | Vaccinia virus | Potency | 13.3499 | 2 | 9 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 58.5840 | 4 | 18 |
| acid sphingomyelinase | Homo sapiens (human) | Potency | 89.1251 | 1 | 1 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 32.6305 | 2 | 16 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 14.9990 | 1 | 16 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 16.3696 | 1 | 5 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Potency | 5.1735 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 28.3627 | 1 | 3 |
| AR protein | Homo sapiens (human) | Potency | 26.3833 | 10 | 80 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 30.4024 | 3 | 11 |
| arylsulfatase A | Homo sapiens (human) | Potency | 5.3582 | 1 | 1 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 11.1375 | 4 | 8 |
| Ataxin-2 | Homo sapiens (human) | Potency | 40.6377 | 2 | 12 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 15.3454 | 5 | 11 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 44.9017 | 2 | 15 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 2.3934 | 1 | 1 |
| atrial natriuretic peptide receptor 2 precursor | Homo sapiens (human) | Potency | 5.2119 | 1 | 1 |
| beta-2 adrenergic receptor | Homo sapiens (human) | Potency | 10.6238 | 1 | 2 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 11.6943 | 3 | 10 |
| BRCA1 | Homo sapiens (human) | Potency | 18.7570 | 1 | 4 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 42.3956 | 1 | 4 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 35.0310 | 1 | 9 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| caspase-3 | Cricetulus griseus (Chinese hamster) | Potency | 31.3341 | 1 | 6 |
| caspase-3 | Homo sapiens (human) | Potency | 35.0310 | 1 | 9 |
| Caspase-7 | Cricetulus griseus (Chinese hamster) | Potency | 31.3341 | 1 | 6 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 43.1928 | 3 | 26 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 15.3659 | 2 | 17 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 12.0057 | 1 | 8 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 17.5505 | 4 | 14 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 32.7114 | 2 | 6 |
| Chain A, Breast cancer type 1 susceptibility protein | Homo sapiens (human) | Potency | 14.2191 | 1 | 2 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 16.9329 | 2 | 13 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 27.7928 | 2 | 4 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 12.7718 | 2 | 14 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 54.3177 | 1 | 6 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 7.2337 | 3 | 18 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 10.4465 | 2 | 10 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 15.1259 | 2 | 12 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 12.7718 | 2 | 14 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 24.4517 | 2 | 5 |
| core-binding factor subunit beta isoform 2 | Homo sapiens (human) | Potency | 17.6943 | 3 | 5 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 7.9113 | 1 | 8 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 12.9128 | 1 | 6 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 16.4462 | 1 | 11 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 14.4115 | 1 | 7 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 21.0124 | 1 | 7 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 17.5388 | 2 | 28 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 13.9527 | 2 | 11 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 13.2008 | 1 | 12 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 5.1014 | 2 | 3 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 14.6892 | 1 | 1 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | Potency | 3.4703 | 1 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 27.9428 | 2 | 2 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 3.9854 | 1 | 2 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 23.1951 | 2 | 7 |
| DNA polymerase III, partial | Bacillus subtilis | Potency | 29.9349 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 36.6778 | 2 | 9 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 13.2029 | 1 | 16 |
| endonuclease IV | Escherichia coli | Potency | 17.8010 | 2 | 4 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 20.5990 | 11 | 104 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 36.7051 | 3 | 23 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 23.5576 | 10 | 86 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 13.0388 | 1 | 21 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 11.9376 | 4 | 56 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 36.0896 | 5 | 24 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 43.9639 | 2 | 9 |
| fructose-bisphosphate aldolase A | Oryctolagus cuniculus (rabbit) | Potency | 6.3096 | 1 | 1 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 26.0872 | 1 | 16 |
| G | Vesicular stomatitis virus | Potency | 16.4462 | 1 | 11 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| galactokinase | Homo sapiens (human) | Potency | 32.5259 | 2 | 2 |
| GALC protein | Homo sapiens (human) | Potency | 0.6310 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 17.5388 | 1 | 14 |
| geminin | Homo sapiens (human) | Potency | 12.2316 | 4 | 24 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 15.6191 | 3 | 27 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 16.6351 | 1 | 3 |
| GLS protein | Homo sapiens (human) | Potency | 24.3396 | 2 | 10 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 26.1355 | 1 | 11 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 34.7278 | 4 | 23 |
| Glutamate receptor 1 | Rattus norvegicus (Norway rat) | Potency | 4.7718 | 1 | 2 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 12.7124 | 2 | 15 |
| Glutamate receptor 3 | Rattus norvegicus (Norway rat) | Potency | 4.7718 | 1 | 2 |
| Glutamate receptor 4 | Rattus norvegicus (Norway rat) | Potency | 4.7718 | 1 | 2 |
| glyceraldehyde-3-phosphate dehydrogenase isoform 1 | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| GTP-binding nuclear protein Ran isoform 1 | Homo sapiens (human) | Potency | 27.6461 | 1 | 2 |
| Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 4.4668 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 26.2698 | 2 | 20 |
| hemoglobin subunit beta | Homo sapiens (human) | Potency | 22.1060 | 2 | 2 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 11.1962 | 2 | 48 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 31.3838 | 1 | 3 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 17.7310 | 1 | 2 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 39.5267 | 2 | 21 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 39.1539 | 1 | 5 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 16.4462 | 1 | 11 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 23.9190 | 1 | 3 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 15.0506 | 2 | 5 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 27.8007 | 2 | 20 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 16.2246 | 3 | 9 |
| IDH1 | Homo sapiens (human) | Potency | 10.9111 | 1 | 3 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 33.3202 | 2 | 3 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 16.4462 | 1 | 22 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 7.0348 | 1 | 4 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 16.7946 | 1 | 9 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 16.7946 | 1 | 9 |
| Interferon beta | Homo sapiens (human) | Potency | 14.4472 | 3 | 55 |
| interleukin 8 | Homo sapiens (human) | Potency | 66.8242 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 11.2702 | 3 | 14 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 18.4528 | 1 | 11 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 27.8298 | 1 | 2 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 18.3626 | 4 | 11 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 45.8624 | 3 | 3 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 14.4719 | 1 | 4 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 17.4592 | 2 | 35 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 13.4067 | 1 | 3 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 5.5620 | 1 | 3 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 23.9063 | 1 | 3 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 56.2341 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 56.2341 | 1 | 1 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 19.7830 | 1 | 2 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 4.7427 | 2 | 8 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 10.4356 | 1 | 4 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 58.0479 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 26.6298 | 4 | 31 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 20.5962 | 1 | 1 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 47.3936 | 1 | 2 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 27.7047 | 2 | 17 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 29.8493 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 42.2402 | 2 | 39 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 29.6917 | 3 | 32 |
| Ornithine decarboxylase | Rattus norvegicus (Norway rat) | Potency | 28.3708 | 1 | 2 |
| P53 | Homo sapiens (human) | Potency | 39.1512 | 1 | 2 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 125.8920 | 1 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 54.1162 | 1 | 4 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 20.9168 | 2 | 9 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 21.0634 | 1 | 2 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 34.2171 | 5 | 29 |
| Peroxisome proliferator-activated receptor alpha | Homo sapiens (human) | Potency | 50.1187 | 1 | 2 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 33.3517 | 5 | 24 |
| phosphoglycerate kinase | Trypanosoma brucei brucei TREU927 | Potency | 28.1838 | 1 | 1 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 34.8307 | 2 | 19 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 10.1775 | 1 | 3 |
| Platelet-activating factor receptor | Homo sapiens (human) | Potency | 14.2191 | 1 | 2 |
| polyprotein | Zika virus | Potency | 26.0872 | 1 | 16 |
| polypyrimidine tract-binding protein 1 isoform a | Homo sapiens (human) | Potency | 14.5500 | 2 | 2 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 8.5438 | 1 | 8 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 10.1662 | 1 | 15 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 9.5352 | 1 | 6 |
| PPM1D protein | Homo sapiens (human) | Potency | 13.1893 | 1 | 28 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 18.4450 | 3 | 20 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 79.4328 | 1 | 1 |
| progesterone receptor | Homo sapiens (human) | Potency | 44.6219 | 3 | 22 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 8.3216 | 2 | 4 |
| pyruvate kinase PKM isoform a | Homo sapiens (human) | Potency | 15.8489 | 2 | 2 |
| pyruvate kinase PKM isoform b | Homo sapiens (human) | Potency | 28.3708 | 2 | 4 |
| Rap guanine nucleotide exchange factor 3 | Homo sapiens (human) | Potency | 59.6193 | 2 | 5 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 20.6003 | 2 | 26 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 91.9997 | 1 | 1 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 5.7764 | 1 | 4 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 32.6123 | 3 | 34 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 20.8661 | 4 | 25 |
| runt-related transcription factor 1 isoform AML1b | Homo sapiens (human) | Potency | 17.6943 | 3 | 5 |
| serine-protein kinase ATM isoform a | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 11.8094 | 5 | 8 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 11.0180 | 1 | 2 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 47.1852 | 3 | 13 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 47.1852 | 3 | 13 |
| Smad3 | Homo sapiens (human) | Potency | 17.2863 | 1 | 8 |
| snurportin-1 | Homo sapiens (human) | Potency | 33.3202 | 2 | 3 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 29.0691 | 1 | 5 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 14.2728 | 1 | 6 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 3.3998 | 1 | 2 |
| TDP1 protein | Homo sapiens (human) | Potency | 15.1954 | 2 | 48 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 26.6514 | 1 | 2 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 21.6856 | 2 | 5 |
| Thrombopoietin | Homo sapiens (human) | Potency | 4.7931 | 2 | 6 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 13.9030 | 3 | 33 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 40.9168 | 4 | 7 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 39.0962 | 6 | 34 |
| thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 27.1740 | 2 | 10 |
| transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 14.4834 | 2 | 11 |
| ubiquitin carboxyl-terminal hydrolase 2 isoform a | Homo sapiens (human) | Potency | 3.4703 | 1 | 2 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 10.1775 | 1 | 3 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 10.1775 | 1 | 3 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 38.6476 | 2 | 16 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 16.4073 | 2 | 24 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 26.2985 | 5 | 28 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 26.2830 | 1 | 13 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 13.9340 | 1 | 13 |
| Vpr | Human immunodeficiency virus 1 | Potency | 26.2000 | 1 | 2 |
| WRN | Homo sapiens (human) | Potency | 17.1205 | 2 | 4 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a | Homo sapiens (human) | IC50 | 6.4860 | 2 | 4 |
| 1-deoxy-D-xylulose 5-phosphate reductoisomerase | Escherichia coli K-12 | IC50 | 2.8000 | 1 | 2 |
| 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 | Bos taurus (cattle) | IC50 | 29.0000 | 1 | 1 |
| 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 | Homo sapiens (human) | IC50 | 29.0000 | 1 | 1 |
| 10 kDa chaperonin | Escherichia coli | IC50 | 52.8750 | 4 | 4 |
| 10 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 57.5000 | 2 | 2 |
| 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | Homo sapiens (human) | IC50 | 0.0120 | 1 | 1 |
| 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | Homo sapiens (human) | Ki | 0.0050 | 1 | 1 |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 4.0000 | 1 | 1 |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 1.3000 | 2 | 2 |
| 4-aminobutyrate aminotransferase, mitochondrial | Homo sapiens (human) | IC50 | 12,800.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 26.0800 | 2 | 2 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 1.1810 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | Ki | 6.9490 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | IC50 | 26.0800 | 2 | 2 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | Ki | 6.9490 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Rattus norvegicus (Norway rat) | IC50 | 40.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Sus scrofa (pig) | Ki | 4.0940 | 1 | 1 |
| 5-hydroxytryptamine receptor 1F | Rattus norvegicus (Norway rat) | IC50 | 40.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | IC50 | 4.8010 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | Ki | 1.6655 | 2 | 2 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | IC50 | 18.3155 | 1 | 2 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | Ki | 7.7887 | 2 | 3 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | IC50 | 0.4600 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 1.0710 | 3 | 3 |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| 5-hydroxytryptamine receptor 3B | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| 5-hydroxytryptamine receptor 3C | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| 5-hydroxytryptamine receptor 3D | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| 5-hydroxytryptamine receptor 3E | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | IC50 | 0.4600 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | Ki | 0.2410 | 1 | 1 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 3.2960 | 1 | 1 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | IC50 | 9.3400 | 1 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 3.9818 | 3 | 4 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | IC50 | 350.0000 | 1 | 2 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 7.0710 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | IC50 | 0.1580 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | IC50 | 0.0617 | 1 | 1 |
| 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 | Homo sapiens (human) | IC50 | 49.3000 | 3 | 3 |
| 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 | Homo sapiens (human) | Ki | 25.1000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli K-12 | IC50 | 250.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli | IC50 | 52.8750 | 4 | 4 |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 57.5000 | 2 | 2 |
| 7-dehydrocholesterol reductase | Homo sapiens (human) | IC50 | 0.0120 | 1 | 1 |
| 72 kDa type IV collagenase | Homo sapiens (human) | IC50 | 4.1597 | 9 | 9 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | IC50 | 4.4000 | 1 | 1 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 66.2850 | 2 | 2 |
| Acetylcholinesterase | Homo sapiens (human) | Ki | 65.8000 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | IC50 | 23.7670 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | Ki | 13.8640 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | IC50 | 7.0990 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | Ki | 3.9850 | 1 | 1 |
| Adenosine receptor A3 | Homo sapiens (human) | IC50 | 2.0285 | 1 | 2 |
| Adenosine receptor A3 | Homo sapiens (human) | Ki | 1.1465 | 1 | 2 |
| ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 | Homo sapiens (human) | IC50 | 8.2000 | 1 | 1 |
| Aldehyde dehydrogenase, mitochondrial | Homo sapiens (human) | IC50 | 3.4000 | 1 | 1 |
| Aldehyde oxidase | Homo sapiens (human) | IC50 | 0.2000 | 1 | 1 |
| Aldehyde oxidase 1 | Macaca fascicularis (crab-eating macaque) | IC50 | 0.1100 | 1 | 1 |
| Aldehyde oxidase 1 | Mus musculus (house mouse) | IC50 | 0.1500 | 1 | 1 |
| Aldehyde oxidase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 2.0000 | 1 | 1 |
| Aldehyde oxidase 1 | Cavia porcellus (domestic guinea pig) | Ki | 7.2300 | 1 | 1 |
| Aldehyde oxidase 1 | Rattus norvegicus (Norway rat) | IC50 | 0.1900 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Bos taurus (cattle) | IC50 | 5.1620 | 2 | 2 |
| Aldo-keto reductase family 1 member B1 | Homo sapiens (human) | IC50 | 1.9000 | 2 | 2 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 24.4607 | 2 | 3 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 35.6355 | 1 | 2 |
| Aldo-keto reductase family 1 member B10 | Homo sapiens (human) | IC50 | 58.5000 | 2 | 2 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | IC50 | 1.1773 | 2 | 2 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 2.0285 | 1 | 2 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 1.1465 | 1 | 2 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 2.0285 | 1 | 2 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 1.1465 | 1 | 2 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | IC50 | 4.9820 | 1 | 1 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | Ki | 2.4490 | 1 | 1 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | IC50 | 3.4195 | 1 | 2 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 1.2825 | 1 | 2 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | IC50 | 3.3680 | 1 | 2 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 1.5375 | 1 | 2 |
| Alpha-amylase 1A | Homo sapiens (human) | IC50 | 18.4000 | 2 | 2 |
| Alpha-synuclein | Homo sapiens (human) | IC50 | 20.9000 | 3 | 5 |
| Alternative oxidase, mitochondrial | Trypanosoma brucei brucei | IC50 | 0.0020 | 1 | 1 |
| Alternative oxidase, mitochondrial | Trypanosoma brucei brucei | Ki | 0.0001 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 7.9635 | 3 | 4 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | Ki | 26.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | IC50 | 59.7000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | Ki | 0.4000 | 1 | 1 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 5.6000 | 2 | 2 |
| Androgen receptor | Rattus norvegicus (Norway rat) | IC50 | 17.3423 | 2 | 2 |
| Androgen receptor | Rattus norvegicus (Norway rat) | Ki | 15.1080 | 1 | 1 |
| Angiopoietin-1 receptor | Homo sapiens (human) | IC50 | 0.7468 | 9 | 14 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | IC50 | 193.6557 | 3 | 3 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | Ki | 0.7922 | 1 | 1 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | IC50 | 8.8250 | 1 | 2 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | IC50 | 0.0462 | 2 | 2 |
| apelin receptor | Homo sapiens (human) | IC50 | 2.6300 | 1 | 1 |
| Aromatase | Homo sapiens (human) | IC50 | 0.0826 | 3 | 14 |
| Arylacetamide deacetylase | Homo sapiens (human) | Ki | 300.0000 | 1 | 1 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 117.0000 | 1 | 4 |
| ATP-dependent 6-phosphofructokinase | Trypanosoma brucei brucei | IC50 | 3.0000 | 1 | 1 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 23.2500 | 6 | 6 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | Ki | 0.1000 | 1 | 1 |
| Aurora kinase A | Homo sapiens (human) | IC50 | 2.4146 | 5 | 8 |
| Aurora kinase B | Homo sapiens (human) | IC50 | 3.3250 | 2 | 4 |
| B2 bradykinin receptor | Homo sapiens (human) | IC50 | 20.3560 | 1 | 1 |
| B2 bradykinin receptor | Homo sapiens (human) | Ki | 12.0480 | 1 | 1 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | IC50 | 17.2890 | 1 | 1 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | Ki | 9.9840 | 1 | 1 |
| Beta-3 adrenergic receptor | Homo sapiens (human) | IC50 | 7.7030 | 1 | 1 |
| Beta-3 adrenergic receptor | Homo sapiens (human) | Ki | 5.7780 | 1 | 1 |
| Beta-adrenergic receptor kinase 1 | Bos taurus (cattle) | IC50 | 130.0000 | 1 | 1 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 5.0000 | 1 | 1 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 11.5000 | 1 | 1 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 1.5400 | 1 | 1 |
| Bifunctional epoxide hydrolase 2 | Homo sapiens (human) | IC50 | 5.0060 | 1 | 2 |
| bifunctional UDP-N-acetylglucosamine pyrophosphorylase/glucosamine-1-phosphate N-acetyltransferase | Mycobacterium tuberculosis H37Rv | IC50 | 85.0300 | 1 | 1 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 44.4182 | 8 | 17 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | IC50 | 34.7000 | 1 | 1 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | Ki | 11.9000 | 1 | 1 |
| Breakpoint cluster region protein | Homo sapiens (human) | GI50 | 7.3000 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 17.7500 | 3 | 4 |
| Bromodomain testis-specific protein | Homo sapiens (human) | IC50 | 0.1902 | 13 | 13 |
| Bromodomain-containing protein 1 | Homo sapiens (human) | IC50 | 44.5000 | 1 | 1 |
| Bromodomain-containing protein 2 | Homo sapiens (human) | IC50 | 0.0959 | 22 | 22 |
| Bromodomain-containing protein 2 | Homo sapiens (human) | Ki | 0.0128 | 4 | 4 |
| Bromodomain-containing protein 3 | Homo sapiens (human) | IC50 | 0.0573 | 18 | 18 |
| Bromodomain-containing protein 3 | Homo sapiens (human) | Ki | 0.0078 | 4 | 4 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | IC50 | 0.8621 | 120 | 120 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | Ki | 0.0193 | 8 | 8 |
| C-8 sterol isomerase | Saccharomyces cerevisiae S288C | Ki | 1.5000 | 1 | 1 |
| C-C chemokine receptor type 2 | Homo sapiens (human) | IC50 | 2.4680 | 1 | 1 |
| C-C chemokine receptor type 2 | Homo sapiens (human) | Ki | 0.9540 | 1 | 1 |
| C-C chemokine receptor type 4 | Homo sapiens (human) | IC50 | 8.3950 | 1 | 1 |
| C-C chemokine receptor type 4 | Homo sapiens (human) | Ki | 4.3970 | 1 | 1 |
| C-C chemokine receptor type 5 | Homo sapiens (human) | IC50 | 23.6610 | 1 | 1 |
| C-C chemokine receptor type 5 | Homo sapiens (human) | Ki | 18.2840 | 1 | 1 |
| C-X-C chemokine receptor type 2 | Homo sapiens (human) | IC50 | 6.0130 | 1 | 1 |
| C-X-C chemokine receptor type 2 | Homo sapiens (human) | Ki | 4.2090 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 100.4000 | 2 | 5 |
| Cannabinoid receptor 2 | Mus musculus (house mouse) | IC50 | 50.0310 | 2 | 2 |
| Carbamate kinase | Giardia intestinalis | IC50 | 0.6000 | 1 | 1 |
| Carbonic anhydrase 1 | Homo sapiens (human) | Ki | 5.4567 | 3 | 6 |
| Carbonic anhydrase 12 | Homo sapiens (human) | Ki | 0.0603 | 1 | 1 |
| Carbonic anhydrase 2 | Homo sapiens (human) | Ki | 4.4053 | 3 | 6 |
| Carbonic anhydrase 3 | Bos taurus (cattle) | Ki | 3.1850 | 1 | 4 |
| Carbonic anhydrase 4 | Homo sapiens (human) | Ki | 2.6066 | 2 | 5 |
| Carbonic anhydrase 7 | Homo sapiens (human) | Ki | 4.0706 | 2 | 2 |
| Carbonic anhydrase 9 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Casein kinase I isoform alpha | Homo sapiens (human) | IC50 | 0.1255 | 1 | 2 |
| Casein kinase I isoform alpha | Sus scrofa (pig) | IC50 | 50.0000 | 1 | 1 |
| Casein kinase II subunit alpha | Homo sapiens (human) | IC50 | 3.8333 | 2 | 3 |
| Casein kinase II subunit alpha 3 | Homo sapiens (human) | IC50 | 5.2500 | 1 | 2 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | IC50 | 3.1250 | 3 | 4 |
| Casein kinase II subunit beta | Homo sapiens (human) | IC50 | 3.1250 | 3 | 4 |
| Caspase-1 | Homo sapiens (human) | IC50 | 5.0595 | 2 | 2 |
| Cathepsin B | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| Cationic trypsin | Bos taurus (cattle) | IC50 | 35.3000 | 1 | 1 |
| CDK-activating kinase assembly factor MAT1 | Homo sapiens (human) | IC50 | 3.1520 | 4 | 4 |
| Cereblon isoform 4 | Magnetospirillum gryphiswaldense | Ki | 1.9500 | 1 | 2 |
| Chain A, Casein kinase II subunit alpha | Zea mays | IC50 | 0.3500 | 1 | 3 |
| Chain A, CES1 protein | Homo sapiens (human) | Ki | 15.2000 | 1 | 1 |
| Chain A, Cyclin-dependent kinase 9 | Homo sapiens (human) | IC50 | 0.7400 | 1 | 1 |
| Chain A, Exotoxin A | Pseudomonas aeruginosa | Ki | 0.1400 | 1 | 1 |
| Chain A, Extracellular Regulated Kinase 2 | Rattus norvegicus (Norway rat) | IC50 | 9.0095 | 1 | 4 |
| Chain A, MAP KINASE P38 | Homo sapiens (human) | IC50 | 9.0095 | 1 | 2 |
| Chain A, PROTEIN (MAP KINASE P38) | Homo sapiens (human) | IC50 | 9.0095 | 1 | 6 |
| Chain A, RNA-directed RNA polymerase NS5 | Dengue virus 2 16681-PDK53 | IC50 | 35.0600 | 1 | 1 |
| Chain A, VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 | Homo sapiens (human) | Ki | 0.0005 | 1 | 5 |
| Chemotaxis protein CheA | Escherichia coli K-12 | IC50 | 111.0000 | 1 | 1 |
| Collagenase 3 | Homo sapiens (human) | IC50 | 5.0275 | 2 | 2 |
| CREB-binding protein | Homo sapiens (human) | IC50 | 9.7153 | 3 | 3 |
| Cruzipain | Trypanosoma cruzi | IC50 | 91.5000 | 2 | 2 |
| Cyclin homolog | Herpesvirus saimiri (strain 11) | IC50 | 77.7000 | 1 | 4 |
| Cyclin-A1 | Homo sapiens (human) | IC50 | 34.5105 | 2 | 2 |
| Cyclin-A1 | Homo sapiens (human) | Ki | 69.0000 | 1 | 1 |
| Cyclin-A2 | Homo sapiens (human) | IC50 | 21.3782 | 7 | 12 |
| Cyclin-A2 | Homo sapiens (human) | Ki | 69.0000 | 1 | 1 |
| Cyclin-C | Homo sapiens (human) | IC50 | 2.0108 | 3 | 3 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 16.1804 | 17 | 26 |
| Cyclin-dependent kinase 1 | Oryzias latipes (Japanese medaka) | IC50 | 77.7000 | 1 | 4 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Ki | 0.4800 | 1 | 1 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | IC50 | 0.1150 | 1 | 2 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 20.9140 | 27 | 37 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Ki | 27.4460 | 3 | 3 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | IC50 | 15.6734 | 11 | 20 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Ki | 0.9250 | 1 | 1 |
| Cyclin-dependent kinase 5 activator 1 | Homo sapiens (human) | IC50 | 45.0400 | 4 | 7 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | IC50 | 101.8217 | 3 | 6 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | IC50 | 15.5281 | 13 | 22 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | IC50 | 2.3242 | 11 | 14 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | IC50 | 9.3365 | 21 | 30 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Ki | 0.1770 | 2 | 2 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | IC50 | 45.0400 | 4 | 7 |
| Cyclin-H | Homo sapiens (human) | IC50 | 15.8429 | 10 | 15 |
| Cyclin-T1 | Homo sapiens (human) | IC50 | 9.1942 | 14 | 19 |
| Cyclin-T1 | Homo sapiens (human) | Ki | 0.3500 | 1 | 1 |
| Cytochrome P450 11B1, mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Cytochrome P450 1A1 | Homo sapiens (human) | IC50 | 0.6945 | 1 | 2 |
| Cytochrome P450 1A1 | Homo sapiens (human) | Ki | 1.3998 | 2 | 5 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 10.1254 | 4 | 5 |
| Cytochrome P450 1B1 | Homo sapiens (human) | IC50 | 0.1560 | 2 | 3 |
| Cytochrome P450 1B1 | Homo sapiens (human) | Ki | 0.5496 | 3 | 5 |
| Cytochrome P450 2B6 | Homo sapiens (human) | Ki | 0.9000 | 1 | 1 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 20.0040 | 2 | 2 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 19.4270 | 3 | 4 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 11.9167 | 8 | 8 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Ki | 0.2000 | 1 | 1 |
| Cytosol aminopeptidase | Sus scrofa (pig) | IC50 | 49.6000 | 1 | 1 |
| Cytosolic phospholipase A2 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| D(1A) dopamine receptor | Homo sapiens (human) | IC50 | 5.3300 | 1 | 2 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 2.6650 | 1 | 2 |
| D(2) dopamine receptor | Homo sapiens (human) | IC50 | 18.4515 | 1 | 2 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 6.1505 | 1 | 2 |
| D(3) dopamine receptor | Homo sapiens (human) | IC50 | 1.0780 | 1 | 2 |
| D(3) dopamine receptor | Rattus norvegicus (Norway rat) | IC50 | 18.1000 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 0.6577 | 2 | 3 |
| D(4) dopamine receptor | Homo sapiens (human) | IC50 | 7.1555 | 1 | 2 |
| D(4) dopamine receptor | Homo sapiens (human) | Ki | 2.5090 | 1 | 2 |
| Death-associated protein kinase 1 | Homo sapiens (human) | IC50 | 70.5000 | 1 | 2 |
| Delta-type opioid receptor | Homo sapiens (human) | IC50 | 13.3390 | 1 | 1 |
| Delta-type opioid receptor | Homo sapiens (human) | Ki | 1.5915 | 3 | 3 |
| Delta-type opioid receptor | Sus scrofa (pig) | Ki | 0.0365 | 1 | 1 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | IC50 | 3.3500 | 1 | 2 |
| Dipeptidyl peptidase 3 | Homo sapiens (human) | IC50 | 22.0000 | 1 | 1 |
| Dipeptidyl peptidase 4 | Homo sapiens (human) | IC50 | 100.0600 | 2 | 2 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | IC50 | 0.0215 | 2 | 2 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | IC50 | 0.0149 | 1 | 1 |
| DNA damage-binding protein 1 | Homo sapiens (human) | IC50 | 1.7972 | 3 | 5 |
| DNA gyrase subunit A | Mycobacterium tuberculosis H37Rv | IC50 | 150.0000 | 3 | 3 |
| DNA gyrase subunit B | Mycobacterium tuberculosis H37Rv | IC50 | 125.0000 | 2 | 2 |
| DNA primase | Mycobacterium tuberculosis CDC1551 | IC50 | 8.2000 | 1 | 1 |
| DNA topoisomerase 1 | Rattus norvegicus (Norway rat) | IC50 | 2.8300 | 2 | 2 |
| DNA-dependent protein kinase catalytic subunit | Homo sapiens (human) | IC50 | 33.9000 | 2 | 3 |
| DNA-directed RNA polymerase subunit beta | Escherichia coli O127:H6 str. E2348/69 | IC50 | 511.3333 | 3 | 3 |
| DNA-directed RNA polymerase subunit beta | Mycobacterium tuberculosis H37Rv | IC50 | 0.0100 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | IC50 | 3.3000 | 1 | 1 |
| Dual specificity protein phosphatase 1 | Mus musculus (house mouse) | IC50 | 24.0000 | 1 | 1 |
| Dual specificity protein phosphatase 5 | Homo sapiens (human) | Ki | 0.0250 | 1 | 1 |
| Dual specificity protein phosphatase 6 | Rattus norvegicus (Norway rat) | IC50 | 20.5000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| Ectonucleoside triphosphate diphosphohydrolase 1 | Rattus norvegicus (Norway rat) | Ki | 300.0000 | 2 | 2 |
| Ectonucleoside triphosphate diphosphohydrolase 2 | Rattus norvegicus (Norway rat) | Ki | 65.4000 | 2 | 2 |
| Ectonucleoside triphosphate diphosphohydrolase 3 | Rattus norvegicus (Norway rat) | Ki | 12.7000 | 1 | 1 |
| Ectonucleoside triphosphate diphosphohydrolase 8 | Homo sapiens (human) | Ki | 100.0000 | 1 | 1 |
| Emopamil-binding protein-like | Homo sapiens (human) | Ki | 0.0028 | 1 | 1 |
| Endoplasmin | Canis lupus familiaris (dog) | IC50 | 0.0120 | 1 | 1 |
| Endoplasmin | Homo sapiens (human) | IC50 | 0.0850 | 1 | 1 |
| Endoplasmin | Homo sapiens (human) | Ki | 0.0040 | 1 | 1 |
| Endothelin-converting enzyme 2 | Homo sapiens (human) | IC50 | 6.4200 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] | Mycobacterium tuberculosis H37Rv | IC50 | 0.0300 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli K-12 | Ki | 7.0500 | 1 | 1 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 2.0000 | 2 | 2 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 2.1000 | 1 | 1 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | IC50 | 6.7262 | 6 | 8 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 35.3205 | 33 | 37 |
| Estrogen receptor | Homo sapiens (human) | IC50 | 1.1920 | 42 | 42 |
| Estrogen receptor | Homo sapiens (human) | Ki | 0.0586 | 4 | 4 |
| Estrogen receptor beta | Homo sapiens (human) | IC50 | 1.2236 | 23 | 23 |
| Estrogen receptor beta | Homo sapiens (human) | Ki | 0.0510 | 4 | 4 |
| Estrogen-related receptor gamma | Homo sapiens (human) | IC50 | 0.0622 | 1 | 1 |
| Fatty acid synthase | Gallus gallus (chicken) | IC50 | 62.5000 | 1 | 1 |
| Fatty acid synthase | Homo sapiens (human) | IC50 | 62.5000 | 1 | 1 |
| Fatty-acid amide hydrolase 1 | Homo sapiens (human) | IC50 | 363.0780 | 1 | 1 |
| Fatty-acid amide hydrolase 1 | Rattus norvegicus (Norway rat) | IC50 | 6.1000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | IC50 | 4.9864 | 22 | 32 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | IC50 | 3.1700 | 4 | 4 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | IC50 | 3.1700 | 4 | 4 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | IC50 | 3.1700 | 4 | 4 |
| Focal adhesion kinase 1 | Homo sapiens (human) | IC50 | 20.8000 | 2 | 2 |
| Fructose-1,6-bisphosphatase 1 | Homo sapiens (human) | IC50 | 87.5067 | 11 | 12 |
| G protein-coupled receptor kinase 5 | Homo sapiens (human) | IC50 | 0.8300 | 1 | 1 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | IC50 | 8.7000 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | IC50 | 23.4000 | 1 | 2 |
| G1/S-specific cyclin-D1 | Homo sapiens (human) | IC50 | 17.1354 | 7 | 12 |
| G1/S-specific cyclin-D2 | Homo sapiens (human) | IC50 | 0.9250 | 1 | 1 |
| G1/S-specific cyclin-D3 | Homo sapiens (human) | IC50 | 0.9250 | 1 | 1 |
| G1/S-specific cyclin-E1 | Homo sapiens (human) | IC50 | 17.7863 | 11 | 16 |
| G1/S-specific cyclin-E1 | Homo sapiens (human) | Ki | 13.3000 | 1 | 1 |
| G1/S-specific cyclin-E2 | Homo sapiens (human) | IC50 | 17.8870 | 4 | 4 |
| G1/S-specific cyclin-E2 | Homo sapiens (human) | Ki | 13.3000 | 1 | 1 |
| G2/mitotic-specific cyclin-B | Marthasterias glacialis (spiny starfish) | IC50 | 77.7000 | 1 | 4 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 16.8565 | 12 | 17 |
| G2/mitotic-specific cyclin-B2 | Homo sapiens (human) | IC50 | 16.8933 | 3 | 3 |
| G2/mitotic-specific cyclin-B3 | Homo sapiens (human) | IC50 | 16.8933 | 3 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit delta | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | IC50 | 281,838.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | IC50 | 0.0149 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit pi | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gamma-aminobutyric acid receptor subunit theta | Homo sapiens (human) | Ki | 1.9193 | 3 | 4 |
| Gasdermin-D | Homo sapiens (human) | IC50 | 0.4000 | 1 | 1 |
| Gasdermin-D | Mus musculus (house mouse) | IC50 | 0.4000 | 1 | 1 |
| Gastrin/cholecystokinin type B receptor | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 2 | 2 |
| Genome polyprotein | Zika virus | IC50 | 53.0000 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | IC50 | 19.0000 | 1 | 1 |
| glucose-6-phosphate 1-dehydrogenase isoform b | Homo sapiens (human) | IC50 | 80.0000 | 1 | 1 |
| glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase | Plasmodium berghei | IC50 | 56.7000 | 3 | 3 |
| Glutathione reductase, mitochondrial | Homo sapiens (human) | Ki | 14.1000 | 2 | 2 |
| Glutathione S-transferase omega-1 | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | IC50 | 0.8000 | 1 | 1 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 10.1500 | 4 | 5 |
| Glycogen synthase kinase-3 beta | Rattus norvegicus (Norway rat) | IC50 | 77.7000 | 1 | 4 |
| Group 10 secretory phospholipase A2 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Heat shock protein 75 kDa, mitochondrial | Homo sapiens (human) | IC50 | 0.3577 | 3 | 3 |
| Heat shock protein 75 kDa, mitochondrial | Homo sapiens (human) | Ki | 0.0160 | 1 | 1 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | IC50 | 2.8407 | 16 | 16 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Ki | 0.0055 | 2 | 2 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | IC50 | 0.0657 | 12 | 12 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Ki | 0.0026 | 4 | 4 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 7.2188 | 8 | 8 |
| Histamine H2 receptor | Homo sapiens (human) | IC50 | 9.3960 | 1 | 1 |
| Histamine H2 receptor | Homo sapiens (human) | Ki | 9.2400 | 1 | 1 |
| Histidine kinase | Caulobacter vibrioides | IC50 | 7.3000 | 1 | 1 |
| histidine kinase | Streptococcus pneumoniae TIGR4 | IC50 | 216.0000 | 1 | 1 |
| Histone acetyltransferase p300 | Homo sapiens (human) | IC50 | 19.4000 | 1 | 1 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Histone-lysine N-methyltransferase EHMT1 | Homo sapiens (human) | IC50 | 1.6000 | 1 | 1 |
| Histone-lysine N-methyltransferase EHMT2 | Homo sapiens (human) | IC50 | 0.6000 | 1 | 1 |
| Histone-lysine N-methyltransferase SETD7 | Homo sapiens (human) | IC50 | 6.0800 | 1 | 1 |
| Homeobox protein Nkx-2.5 | Mus musculus (house mouse) | IC50 | 22.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | IC50 | 0.0515 | 2 | 2 |
| hypothetical protein SA1422 | Staphylococcus aureus subsp. aureus N315 | IC50 | 19.3900 | 2 | 2 |
| Indoleamine 2,3-dioxygenase 1 | Homo sapiens (human) | IC50 | 0.8925 | 4 | 4 |
| Inositol hexakisphosphate kinase 2 | Homo sapiens (human) | IC50 | 1.1000 | 1 | 2 |
| Inositol polyphosphate multikinase | Homo sapiens (human) | IC50 | 6.3500 | 1 | 2 |
| Insulin receptor | Homo sapiens (human) | IC50 | 19.5000 | 2 | 3 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 15.0000 | 3 | 3 |
| Integrase | Human immunodeficiency virus 1 | IC50 | 10.3730 | 5 | 10 |
| integrase, partial | Human immunodeficiency virus 1 | IC50 | 7.8945 | 2 | 2 |
| Interstitial collagenase | Homo sapiens (human) | IC50 | 0.6551 | 8 | 8 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 0.6600 | 1 | 1 |
| Kappa-type opioid receptor | Homo sapiens (human) | IC50 | 10.8660 | 1 | 2 |
| Kappa-type opioid receptor | Homo sapiens (human) | Ki | 4.3465 | 1 | 2 |
| Lactoylglutathione lyase | Homo sapiens (human) | IC50 | 9.3500 | 1 | 2 |
| Lanosterol 14-alpha demethylase | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| large T antigen | Betapolyomavirus macacae | IC50 | 11.3150 | 1 | 2 |
| lens epithelium-derived growth factor p75 | Homo sapiens (human) | IC50 | 7.8945 | 2 | 2 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.0215 | 2 | 2 |
| Linoleate 9S-lipoxygenase-4 | Glycine max (soybean) | IC50 | 22.0000 | 1 | 1 |
| Low affinity immunoglobulin epsilon Fc receptor | Homo sapiens (human) | IC50 | 0.1000 | 2 | 2 |
| Lysine-specific demethylase 4E | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Lysine-specific demethylase 4E | Homo sapiens (human) | Ki | 4.3300 | 1 | 1 |
| Lysine-specific demethylase 5A | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Lysine-specific histone demethylase 1A | Homo sapiens (human) | IC50 | 16.4233 | 2 | 3 |
| Lysosomal alpha-glucosidase | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Lysyl oxidase homolog 2 | Homo sapiens (human) | IC50 | 0.1500 | 1 | 1 |
| Lysyl oxidase homolog 3 | Homo sapiens (human) | IC50 | 0.0930 | 1 | 1 |
| Lysyl oxidase homolog 4 | Homo sapiens (human) | IC50 | 0.0590 | 1 | 1 |
| M-phase inducer phosphatase 1 | Homo sapiens (human) | IC50 | 4.5500 | 2 | 2 |
| M-phase inducer phosphatase 2 | Homo sapiens (human) | IC50 | 3.1600 | 3 | 3 |
| M-phase inducer phosphatase 3 | Homo sapiens (human) | IC50 | 18.9000 | 2 | 2 |
| M1-family alanyl aminopeptidase | Plasmodium falciparum 3D7 | IC50 | 65.6250 | 1 | 2 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | IC50 | 0.1286 | 9 | 15 |
| Macrophage metalloelastase | Homo sapiens (human) | IC50 | 2.9900 | 4 | 4 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | IC50 | 0.1790 | 1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.4205 | 2 | 2 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | GI50 | 0.1937 | 55 | 55 |
| Mast/stem cell growth factor receptor Kit | Mus musculus (house mouse) | GI50 | 0.0030 | 1 | 1 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | IC50 | 0.2178 | 34 | 46 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Ki | 0.0040 | 1 | 1 |
| Matrilysin | Homo sapiens (human) | IC50 | 3.5012 | 2 | 2 |
| Matrix metalloproteinase-14 | Homo sapiens (human) | IC50 | 0.5715 | 5 | 5 |
| Matrix metalloproteinase-9 | Homo sapiens (human) | IC50 | 1.3711 | 6 | 6 |
| Mcl-1 | Homo sapiens (human) | IC50 | 1.6341 | 1 | 1 |
| Melanocortin receptor 3 | Homo sapiens (human) | IC50 | 19.8560 | 1 | 1 |
| Melanocortin receptor 3 | Homo sapiens (human) | Ki | 17.3290 | 1 | 1 |
| melanocortin receptor 4 | Homo sapiens (human) | IC50 | 54.8937 | 3 | 3 |
| Melanocortin receptor 4 | Homo sapiens (human) | Ki | 29.3080 | 1 | 1 |
| Melanocortin receptor 5 | Homo sapiens (human) | IC50 | 26.5290 | 1 | 1 |
| Melanocortin receptor 5 | Homo sapiens (human) | Ki | 24.8860 | 1 | 1 |
| Metabotropic glutamate receptor 5 | Rattus norvegicus (Norway rat) | IC50 | 1.2000 | 1 | 1 |
| Methionine aminopeptidase | Escherichia coli K-12 | IC50 | 100.0000 | 1 | 1 |
| Methionine aminopeptidase 1 | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 1 |
| Methionine aminopeptidase 2 | Homo sapiens (human) | IC50 | 0.3006 | 7 | 8 |
| Methionine aminopeptidase 2 | Homo sapiens (human) | Ki | 0.0010 | 2 | 2 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | IC50 | 9.5548 | 2 | 2 |
| Mitogen-activated protein kinase 1 | Rattus norvegicus (Norway rat) | IC50 | 9.0095 | 1 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 18.0250 | 1 | 4 |
| Mitogen-activated protein kinase 10 | Rattus norvegicus (Norway rat) | IC50 | 6.8000 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | IC50 | 0.0190 | 1 | 1 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | IC50 | 0.0190 | 1 | 1 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | IC50 | 0.0190 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 5.0104 | 15 | 19 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | IC50 | 0.7640 | 2 | 2 |
| Monoglyceride lipase | Homo sapiens (human) | IC50 | 0.8095 | 2 | 2 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 0.0180 | 1 | 1 |
| Mu-type opioid receptor | Homo sapiens (human) | IC50 | 10.5525 | 1 | 2 |
| Mu-type opioid receptor | Homo sapiens (human) | Ki | 4.2835 | 1 | 2 |
| Multidrug resistance-associated protein 1 | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 110.2250 | 1 | 4 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | IC50 | 2.8290 | 1 | 1 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 0.6810 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | IC50 | 7.7930 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 2.7710 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | IC50 | 2.9740 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 0.6300 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | IC50 | 4.8170 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | Ki | 0.6720 | 1 | 1 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | IC50 | 2.5850 | 1 | 1 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | Ki | 1.8570 | 1 | 1 |
| NACHT, LRR and PYD domains-containing protein 3 | Mus musculus (house mouse) | IC50 | 1.9050 | 2 | 2 |
| NAD-dependent protein deacetylase HST2 | Saccharomyces cerevisiae S288C | IC50 | 240.0000 | 1 | 1 |
| NAD-dependent protein deacetylase sirtuin-1 | Homo sapiens (human) | IC50 | 1.3857 | 7 | 7 |
| NAD-dependent protein deacetylase sirtuin-2 | Homo sapiens (human) | IC50 | 25.4800 | 5 | 5 |
| NAD-dependent protein deacylase sirtuin-5, mitochondrial | Homo sapiens (human) | IC50 | 20.6000 | 8 | 8 |
| NADPH oxidase 4 | Homo sapiens (human) | IC50 | 0.8500 | 1 | 1 |
| Neprilysin | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Neuraminidase | Influenza A virus (A/Wilson-Smith/1933(H1N1)) | IC50 | 27.9000 | 4 | 5 |
| Neuraminidase | Influenza A virus (A/Wilson-Smith/1933(H1N1)) | Ki | 16.6500 | 1 | 2 |
| Neuropilin-1 | Homo sapiens (human) | IC50 | 9.1833 | 6 | 6 |
| Neutrophil collagenase | Homo sapiens (human) | IC50 | 0.7000 | 1 | 1 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 6.9850 | 2 | 2 |
| Neutrophil elastase | Homo sapiens (human) | Ki | 10.1000 | 1 | 1 |
| NH(3)-dependent NAD(+) synthetase | Bacillus subtilis subsp. subtilis str. 168 | IC50 | 1.0000 | 1 | 1 |
| Nitric oxide synthase, brain | Homo sapiens (human) | IC50 | 4.8900 | 2 | 2 |
| Nitric oxide synthase, brain | Homo sapiens (human) | Ki | 7.3000 | 1 | 1 |
| Nitric oxide synthase, brain | Rattus norvegicus (Norway rat) | IC50 | 7.5500 | 2 | 2 |
| Nitric oxide synthase, endothelial | Bos taurus (cattle) | IC50 | 611.3333 | 3 | 3 |
| Nitric oxide synthase, endothelial | Homo sapiens (human) | IC50 | 485.0667 | 3 | 3 |
| Nitric oxide synthase, inducible | Homo sapiens (human) | IC50 | 0.1395 | 3 | 3 |
| Nitric oxide synthase, inducible | Mus musculus (house mouse) | IC50 | 2.0828 | 4 | 4 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | IC50 | 0.0480 | 1 | 1 |
| Nuclear receptor subfamily 3 group C member 3 | Bos taurus (cattle) | IC50 | 0.9670 | 1 | 1 |
| Nuclear receptor subfamily 3 group C member 3 | Bos taurus (cattle) | Ki | 0.7922 | 1 | 1 |
| P2X purinoceptor 2 | Rattus norvegicus (Norway rat) | IC50 | 21.9054 | 1 | 2 |
| P2Y purinoceptor 11 | Homo sapiens (human) | Ki | 0.2071 | 2 | 2 |
| P2Y purinoceptor 2 | Homo sapiens (human) | IC50 | 75.0000 | 2 | 2 |
| P2Y purinoceptor 6 | Homo sapiens (human) | IC50 | 27.0000 | 1 | 1 |
| perilipin-1 | Homo sapiens (human) | IC50 | 7.4270 | 1 | 2 |
| perilipin-5 | Homo sapiens (human) | IC50 | 5.5450 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 30.5000 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | IC50 | 50.0000 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | IC50 | 37.3333 | 1 | 3 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | IC50 | 31.5000 | 1 | 2 |
| Phospholipase A2 | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Phospholipase A2, membrane associated | Homo sapiens (human) | IC50 | 23.8000 | 1 | 1 |
| Phospholipase D1 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| Phospholipase D1 | Rattus norvegicus (Norway rat) | IC50 | 20.0000 | 1 | 1 |
| Platelet-activating factor acetylhydrolase | Homo sapiens (human) | IC50 | 0.9040 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | GI50 | 0.1939 | 4 | 4 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | IC50 | 0.1144 | 6 | 6 |
| Platelet-derived growth factor receptor alpha | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 2 | 2 |
| Platelet-derived growth factor receptor alpha | Mus musculus (house mouse) | IC50 | 6.2662 | 8 | 8 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | GI50 | 0.1140 | 1 | 1 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | IC50 | 8.2102 | 39 | 51 |
| Platelet-derived growth factor receptor beta | Mus musculus (house mouse) | IC50 | 8.3954 | 12 | 18 |
| Platelet-derived growth factor receptor beta | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 2 | 2 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Ki | 0.0080 | 1 | 1 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | IC50 | 0.4834 | 17 | 22 |
| Poly [ADP-ribose] polymerase 2 | Homo sapiens (human) | IC50 | 3.0634 | 5 | 7 |
| Poly [ADP-ribose] polymerase 2 | Mus musculus (house mouse) | IC50 | 0.0405 | 1 | 2 |
| Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens (human) | IC50 | 1.4307 | 5 | 8 |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | IC50 | 1.2162 | 4 | 7 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 0.2910 | 1 | 1 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | IC50 | 34.1500 | 2 | 3 |
| Polyunsaturated fatty acid 5-lipoxygenase | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | Ki | 0.0844 | 2 | 2 |
| Polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | IC50 | 31.5320 | 2 | 5 |
| Polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Ki | 1.6000 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens (human) | IC50 | 28.4833 | 3 | 6 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | IC50 | 9.5075 | 1 | 2 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens (human) | Ki | 0.6000 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | IC50 | 51.0929 | 3 | 7 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Rattus norvegicus (Norway rat) | IC50 | 0.2600 | 1 | 1 |
| Potassium voltage-gated channel subfamily D member 3 | Homo sapiens (human) | IC50 | 50.1187 | 1 | 1 |
| Potassium voltage-gated channel subfamily E member 1 | Homo sapiens (human) | IC50 | 63.0957 | 1 | 1 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 4.9683 | 8 | 8 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | Ki | 0.7922 | 1 | 1 |
| Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens (human) | IC50 | 63.0957 | 1 | 1 |
| Procathepsin L | Homo sapiens (human) | IC50 | 8.8250 | 1 | 2 |
| Progesterone receptor | Homo sapiens (human) | IC50 | 38.3763 | 3 | 3 |
| Programmed cell death 1 ligand 1 | Homo sapiens (human) | IC50 | 0.0100 | 1 | 1 |
| Programmed cell death protein 1 | Homo sapiens (human) | IC50 | 0.0100 | 1 | 1 |
| Prolyl endopeptidase | Homo sapiens (human) | IC50 | 36.0000 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Homo sapiens (human) | IC50 | 4.3910 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Ovis aries (sheep) | IC50 | 76.6000 | 2 | 2 |
| Prostaglandin G/H synthase 1 | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | IC50 | 48.7767 | 6 | 6 |
| Prostaglandin G/H synthase 2 | Mus musculus (house mouse) | IC50 | 1.0700 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 1.4000 | 2 | 2 |
| Protein arginine N-methyltransferase 1 | Homo sapiens (human) | IC50 | 344.8100 | 3 | 3 |
| Protein cereblon | Homo sapiens (human) | IC50 | 7.2078 | 6 | 11 |
| Protein cereblon | Homo sapiens (human) | Ki | 9.2633 | 2 | 3 |
| Protein delta homolog 1 | Homo sapiens (human) | Ki | 0.0063 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 19.5333 | 6 | 6 |
| Protein kinase C alpha type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 22.5000 | 4 | 4 |
| Protein kinase C beta type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C delta type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C epsilon type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C eta type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 22.5000 | 4 | 4 |
| Protein kinase C gamma type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C theta type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Protein kinase C zeta type | Rattus norvegicus (Norway rat) | IC50 | 75.0000 | 1 | 1 |
| Protein mono-ADP-ribosyltransferase PARP10 | Homo sapiens (human) | IC50 | 6.3123 | 2 | 4 |
| Protein mono-ADP-ribosyltransferase PARP12 | Homo sapiens (human) | IC50 | 0.2269 | 1 | 2 |
| Protein mono-ADP-ribosyltransferase PARP14 | Homo sapiens (human) | IC50 | 4.1843 | 1 | 2 |
| Protein mono-ADP-ribosyltransferase PARP15 | Homo sapiens (human) | IC50 | 8.9563 | 1 | 2 |
| Protein mono-ADP-ribosyltransferase PARP3 | Homo sapiens (human) | IC50 | 1.4377 | 1 | 2 |
| Protein mono-ADP-ribosyltransferase PARP4 | Homo sapiens (human) | IC50 | 0.7586 | 1 | 1 |
| Protein-glutamine gamma-glutamyltransferase 2 | Homo sapiens (human) | IC50 | 2.2000 | 1 | 1 |
| Protein-lysine 6-oxidase | Homo sapiens (human) | IC50 | 0.3200 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | GI50 | 0.1013 | 3 | 3 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 0.3065 | 12 | 15 |
| Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | IC50 | 33.5183 | 3 | 3 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 24.6355 | 8 | 11 |
| Pyruvate kinase PKM | Homo sapiens (human) | IC50 | 76.0050 | 2 | 2 |
| Pyruvate kinase PKM | Homo sapiens (human) | Ki | 3.5300 | 1 | 1 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 30.0000 | 2 | 2 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 0.6814 | 30 | 34 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Ki | 0.0060 | 1 | 1 |
| Receptor protein-tyrosine kinase | Homo sapiens (human) | IC50 | 2.2000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 5.6176 | 5 | 5 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | IC50 | 0.0020 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | IC50 | 0.0020 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | IC50 | 1.5000 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 3.6000 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | IC50 | 14.5200 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | GI50 | 3.1330 | 3 | 3 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 0.2052 | 51 | 64 |
| Receptor-type tyrosine-protein phosphatase eta | Homo sapiens (human) | IC50 | 2.2000 | 1 | 1 |
| Receptor-type tyrosine-protein phosphatase S | Homo sapiens (human) | IC50 | 10.3000 | 1 | 1 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | IC50 | 8.8250 | 1 | 2 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 13.6125 | 2 | 4 |
| Replicase polyprotein 1ab | Human coronavirus 229E | IC50 | 8.8250 | 1 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 6.3339 | 16 | 24 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 10.2778 | 3 | 9 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Ki | 8.7550 | 1 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | Ki | 10.4367 | 2 | 3 |
| Retinal dehydrogenase 1 | Homo sapiens (human) | IC50 | 0.1300 | 1 | 1 |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | IC50 | 47.8000 | 3 | 3 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | IC50 | 0.1313 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | IC50 | 0.1839 | 1 | 1 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase beta-2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| RmtA | Aspergillus nidulans | IC50 | 5.9000 | 1 | 1 |
| RuvB-like 1 | Homo sapiens (human) | IC50 | 66.0000 | 1 | 1 |
| RuvB-like 2 | Homo sapiens (human) | IC50 | 66.0000 | 1 | 1 |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max (soybean) | IC50 | 8.0500 | 4 | 4 |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max (soybean) | Ki | 121.7000 | 1 | 1 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | IC50 | 0.0087 | 3 | 3 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | GI50 | 1.0000 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | IC50 | 0.3699 | 58 | 62 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Ki | 0.0327 | 3 | 3 |
| Serine/threonine-protein kinase B-raf | Mus musculus (house mouse) | IC50 | 0.1300 | 1 | 1 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | IC50 | 20.0386 | 2 | 2 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | IC50 | 0.0168 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 16.6667 | 3 | 3 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | IC50 | 50.0000 | 1 | 2 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | IC50 | 12.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | IC50 | 0.5692 | 2 | 2 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 5.8000 | 2 | 2 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | IC50 | 9.5000 | 2 | 2 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Ki | 14.9800 | 1 | 8 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | IC50 | 314.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Ki | 14.9800 | 1 | 8 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Ki | 14.9800 | 1 | 8 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Ki | 14.9800 | 1 | 8 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | IC50 | 0.2200 | 1 | 1 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | IC50 | 0.1750 | 2 | 2 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | IC50 | 0.7900 | 1 | 1 |
| Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 30.5730 | 1 | 1 |
| Sex hormone-binding globulin | Homo sapiens (human) | IC50 | 52.0000 | 1 | 1 |
| Short transient receptor potential channel 5 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Sialidase | Clostridium perfringens | IC50 | 2.8500 | 1 | 2 |
| Sialidase-2 | Homo sapiens (human) | IC50 | 130.0000 | 1 | 2 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | IC50 | 0.0210 | 1 | 1 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | Ki | 0.0219 | 2 | 2 |
| Signal transducer and activator of transcription 1-alpha/beta | Homo sapiens (human) | IC50 | 9.1000 | 1 | 1 |
| Signal transducer and activator of transcription 3 | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| Signal transducer and activator of transcription 5A | Homo sapiens (human) | IC50 | 9.4000 | 1 | 1 |
| Signal transducer and activator of transcription 5B | Homo sapiens (human) | IC50 | 10.4000 | 1 | 1 |
| Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | IC50 | 2.4000 | 1 | 2 |
| Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | Ki | 3.2000 | 1 | 2 |
| Smoothened homolog | Homo sapiens (human) | Ki | 0.0876 | 1 | 1 |
| Snake venom metalloproteinase BaP1 | Bothrops asper (terciopelo) | IC50 | 1.2000 | 1 | 1 |
| Sodium channel protein type 5 subunit alpha | Homo sapiens (human) | IC50 | 27.8298 | 2 | 2 |
| Sodium- and chloride-dependent betaine transporter | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Sodium- and chloride-dependent GABA transporter 1 | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Sodium- and chloride-dependent GABA transporter 2 | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Sodium- and chloride-dependent GABA transporter 3 | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | IC50 | 3.2390 | 1 | 2 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | Ki | 2.5730 | 1 | 2 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 35.9210 | 1 | 2 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 35.6355 | 1 | 2 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | IC50 | 2.3340 | 1 | 1 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | IC50 | 0.0011 | 1 | 1 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 1.2400 | 1 | 1 |
| Solute carrier family 22 member 1 | Homo sapiens (human) | IC50 | 6.1000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1A1 | Rattus norvegicus (Norway rat) | Ki | 18.2000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1A2 | Homo sapiens (human) | Ki | 51.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1A4 | Rattus norvegicus (Norway rat) | Ki | 1.4300 | 2 | 2 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | IC50 | 1.5000 | 4 | 4 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | Ki | 9.0500 | 2 | 2 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | IC50 | 1.5000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | Ki | 3.2000 | 2 | 2 |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens (human) | IC50 | 65.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens (human) | Ki | 63.0000 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | IC50 | 8.8250 | 1 | 2 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | IC50 | 8.8250 | 1 | 2 |
| Steroid hormone receptor ERR1 | Homo sapiens (human) | IC50 | 0.2000 | 1 | 1 |
| Stromelysin-1 | Homo sapiens (human) | IC50 | 17.4004 | 7 | 7 |
| Substance-K receptor | Cavia porcellus (domestic guinea pig) | IC50 | 33.7000 | 1 | 1 |
| Substance-K receptor | Homo sapiens (human) | IC50 | 3.6700 | 1 | 1 |
| Substance-K receptor | Homo sapiens (human) | Ki | 1.2230 | 1 | 1 |
| Substance-P receptor | Cavia porcellus (domestic guinea pig) | IC50 | 33.7000 | 1 | 1 |
| Substance-P receptor | Homo sapiens (human) | IC50 | 15.6560 | 1 | 1 |
| Substance-P receptor | Homo sapiens (human) | Ki | 8.5400 | 1 | 1 |
| Sucrase-isomaltase, intestinal | Homo sapiens (human) | IC50 | 43.5000 | 2 | 2 |
| Sucrase-isomaltase, intestinal | Rattus norvegicus (Norway rat) | IC50 | 156.0000 | 2 | 2 |
| Testosterone 17-beta-dehydrogenase 3 | Homo sapiens (human) | IC50 | 97.6100 | 2 | 2 |
| Thiosulfate sulfurtransferase | Homo sapiens (human) | IC50 | 50.5000 | 2 | 2 |
| Thromboxane-A synthase | Homo sapiens (human) | IC50 | 0.9160 | 1 | 1 |
| Transcription factor GATA-4 | Mus musculus (house mouse) | IC50 | 22.0000 | 1 | 1 |
| Transcriptional activator protein LuxR | Aliivibrio fischeri | IC50 | 40.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily M member 8 | Mus musculus (house mouse) | IC50 | 8.0000 | 2 | 2 |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | IC50 | 34.6667 | 3 | 3 |
| Translocator protein | Rattus norvegicus (Norway rat) | IC50 | 0.0390 | 1 | 2 |
| Transmembrane protease serine 2 | Homo sapiens (human) | IC50 | 8.8250 | 1 | 2 |
| Transthyretin | Homo sapiens (human) | IC50 | 6.4000 | 1 | 1 |
| Trypanothione reductase | Trypanosoma cruzi | IC50 | 55.0000 | 2 | 2 |
| Trypsin-1 | Homo sapiens (human) | IC50 | 54.3500 | 1 | 2 |
| Trypsin-2 | Homo sapiens (human) | IC50 | 54.3500 | 1 | 2 |
| Trypsin-3 | Homo sapiens (human) | IC50 | 54.3500 | 1 | 2 |
| Tubulin alpha-1A chain | Sus scrofa (pig) | IC50 | 1.8000 | 1 | 1 |
| Tubulin beta chain | Sus scrofa (pig) | IC50 | 1.8000 | 1 | 1 |
| Tubulin beta-2B chain | Bos taurus (cattle) | IC50 | 2.4000 | 1 | 1 |
| Tubulin beta-2B chain | Bos taurus (cattle) | Ki | 3.2000 | 1 | 1 |
| type-1 angiotensin II receptor | Homo sapiens (human) | IC50 | 6.6370 | 1 | 1 |
| Tyrosinase | Homo sapiens (human) | IC50 | 60.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | GI50 | 7.3000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 8.9610 | 6 | 7 |
| Tyrosine-protein kinase ABL1 | Mus musculus (house mouse) | IC50 | 0.2259 | 1 | 1 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 1.1950 | 1 | 1 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | IC50 | 12.8125 | 2 | 4 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | IC50 | 26.1000 | 2 | 2 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 91.7670 | 6 | 6 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Mus musculus (house mouse) | IC50 | 11.1000 | 1 | 1 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | IC50 | 1.3700 | 1 | 1 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | IC50 | 0.0090 | 2 | 2 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | IC50 | 12.0000 | 1 | 1 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | IC50 | 1.1102 | 3 | 3 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Ki | 2.3800 | 1 | 1 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 8.5800 | 2 | 2 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | Ki | 7.8000 | 1 | 1 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L1 | Homo sapiens (human) | IC50 | 290.0000 | 1 | 1 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L1 | Mus musculus (house mouse) | IC50 | 180.5000 | 1 | 2 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L3 | Homo sapiens (human) | IC50 | 71.0000 | 2 | 2 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L3 | Mus musculus (house mouse) | IC50 | 180.5000 | 1 | 2 |
| ubiquitin-conjugating enzyme E2 N | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| UDP-glucuronosyltransferase 1A1 | Homo sapiens (human) | IC50 | 5.7000 | 2 | 2 |
| Uracil nucleotide/cysteinyl leukotriene receptor | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Urease subunit alpha | Helicobacter pylori 26695 | IC50 | 163.2000 | 1 | 2 |
| Urease subunit beta | Helicobacter pylori 26695 | IC50 | 163.2000 | 1 | 2 |
| Valosin-containing protein | Homo sapiens (human) | IC50 | 36.3280 | 2 | 3 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | IC50 | 0.0926 | 29 | 40 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Ki | 0.0310 | 2 | 2 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | GI50 | 0.0330 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Danio rerio (zebrafish) | IC50 | 1.1933 | 2 | 3 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 1.1553 | 176 | 214 |
| Vascular endothelial growth factor receptor 2 | Mus musculus (house mouse) | IC50 | 0.1102 | 3 | 9 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Ki | 0.0098 | 7 | 8 |
| Vascular endothelial growth factor receptor 2 | Mus musculus (house mouse) | Ki | 0.0280 | 1 | 1 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | IC50 | 0.0822 | 11 | 12 |
| Vascular endothelial growth factor receptor 3 | Mus musculus (house mouse) | IC50 | 0.1269 | 1 | 7 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Ki | 0.0170 | 1 | 1 |
| Vitamin K-dependent protein C | Homo sapiens (human) | IC50 | 0.2640 | 2 | 12 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | IC50 | 104.1196 | 3 | 3 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | IC50 | 33.4000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | IC50 | 33.4000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | IC50 | 33.4000 | 1 | 1 |
| Voltage-dependent N-type calcium channel subunit alpha-1B | Homo sapiens (human) | IC50 | 7.0000 | 2 | 2 |
| Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens (human) | IC50 | 2.0000 | 2 | 2 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | IC50 | 59.2800 | 2 | 5 |
| Xanthine dehydrogenase/oxidase | Homo sapiens (human) | IC50 | 5.6700 | 3 | 4 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | Ki | 1.9000 | 1 | 1 |
| Xanthine dehydrogenase/oxidase | Homo sapiens (human) | Ki | 2.9000 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | Homo sapiens (human) | Kd | 0.0010 | 1 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | Kd | 8.5000 | 3 | 13 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 12.2038 | 6 | 23 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | Kd | 7.7128 | 3 | 13 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 22.8920 | 1 | 8 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 22.9382 | 1 | 8 |
| 7-dehydrocholesterol reductase | Homo sapiens (human) | Kd | 0.0010 | 1 | 1 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 16.7146 | 4 | 21 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 17.5510 | 4 | 22 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Activin receptor type-2A | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 18.6957 | 4 | 23 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 25.0048 | 1 | 6 |
| Adenosine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Albumin | Homo sapiens (human) | Kd | 12.0000 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 9.5807 | 4 | 15 |
| Angiopoietin-1 receptor | Homo sapiens (human) | Kd | 5.7600 | 4 | 14 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | EC50 | 37.8633 | 1 | 3 |
| Ankyrin repeat and protein kinase domain-containing protein 1 | Homo sapiens (human) | Kd | 7.7638 | 3 | 13 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 12.4233 | 8 | 25 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 10 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | EC50 | 56.5000 | 1 | 1 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Atypical kinase COQ8B, mitochondrial | Homo sapiens (human) | Kd | 9.4538 | 3 | 13 |
| Aurora kinase A | Homo sapiens (human) | Kd | 14.9864 | 5 | 22 |
| Aurora kinase B | Homo sapiens (human) | Kd | 11.2790 | 4 | 21 |
| Aurora kinase C | Homo sapiens (human) | Kd | 3.1368 | 5 | 15 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | Kd | 4.6362 | 3 | 13 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 12.2339 | 6 | 23 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 18.9444 | 3 | 16 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 14.7580 | 4 | 21 |
| Breakpoint cluster region protein | Homo sapiens (human) | EC50 | 1.0000 | 1 | 1 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 26.3119 | 1 | 8 |
| Bromodomain testis-specific protein | Homo sapiens (human) | Kd | 0.1786 | 7 | 7 |
| Bromodomain-containing protein 2 | Homo sapiens (human) | Kd | 0.0827 | 12 | 12 |
| Bromodomain-containing protein 3 | Homo sapiens (human) | Kd | 0.0599 | 10 | 10 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | EC50 | 0.1203 | 3 | 3 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | Kd | 0.0912 | 31 | 57 |
| Bromodomain-containing protein 7 | Homo sapiens (human) | Kd | 11.0000 | 1 | 1 |
| Bromodomain-containing protein 9 | Homo sapiens (human) | Kd | 17.0000 | 1 | 1 |
| Calcium-dependent protein kinase 1 | Plasmodium falciparum 3D7 | Kd | 6.9200 | 1 | 6 |
| Calcium/calmodulin-dependent protein kinase kinase 1 | Homo sapiens (human) | Kd | 7.2971 | 4 | 14 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 14.5652 | 5 | 22 |
| Calcium/calmodulin-dependent protein kinase type 1 | Homo sapiens (human) | Kd | 7.4936 | 4 | 14 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | Kd | 7.3307 | 4 | 14 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 9.3746 | 4 | 13 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | Kd | 6.7320 | 5 | 15 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | Kd | 7.6714 | 4 | 14 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 14.2355 | 5 | 22 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 11.8278 | 7 | 25 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 15.0305 | 4 | 21 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 19.2286 | 3 | 21 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| cAMP-dependent protein kinase catalytic subunit PRKX | Homo sapiens (human) | Kd | 11.4286 | 4 | 14 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 16.8118 | 3 | 16 |
| Casein kinase I isoform alpha-like | Homo sapiens (human) | Kd | 8.2818 | 2 | 11 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 12.7778 | 4 | 21 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 14.6721 | 4 | 22 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 16.3550 | 4 | 23 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 16.2062 | 4 | 21 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 14.9365 | 4 | 21 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Kd | 7.7740 | 3 | 13 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 14.9572 | 4 | 21 |
| Cell division control protein 2 homolog | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 6 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| cGMP-dependent protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Chain A, Bromodomain testis-specific protein | Homo sapiens (human) | Kd | 0.1901 | 1 | 1 |
| Chain A, Bromodomain-containing protein 4 | Homo sapiens (human) | Kd | 0.0490 | 1 | 1 |
| Chain A, Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 0.0914 | 1 | 7 |
| Chain A, Transthyretin | Homo sapiens (human) | Kd | 0.1000 | 1 | 5 |
| Chain B, Transthyretin | Homo sapiens (human) | Kd | 0.1000 | 1 | 2 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 16.4455 | 4 | 22 |
| CREB-binding protein | Homo sapiens (human) | Kd | 9.6000 | 1 | 1 |
| Cyclin-C | Homo sapiens (human) | Kd | 0.3100 | 1 | 1 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 22.8258 | 1 | 8 |
| Cyclin-dependent kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 11A | Homo sapiens (human) | Kd | 7.1151 | 3 | 13 |
| Cyclin-dependent kinase 11B | Homo sapiens (human) | Kd | 7.1382 | 3 | 13 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 26.6852 | 1 | 9 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 17.8869 | 2 | 14 |
| Cyclin-dependent kinase 14 | Homo sapiens (human) | Kd | 4.6838 | 3 | 13 |
| Cyclin-dependent kinase 15 | Homo sapiens (human) | Kd | 7.0675 | 2 | 8 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 11.1300 | 6 | 23 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 11.4909 | 4 | 21 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 8.2277 | 4 | 14 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | Kd | 4.1768 | 3 | 13 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 13.5987 | 5 | 22 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 12.8001 | 4 | 20 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 15.1150 | 3 | 20 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 26.6824 | 1 | 9 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 10.4512 | 4 | 21 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | Kd | 4.1664 | 4 | 14 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 13.1988 | 4 | 21 |
| Cyclin-dependent kinase-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Cyclin-dependent kinase-like 2 | Homo sapiens (human) | Kd | 4.0626 | 2 | 8 |
| Cyclin-dependent kinase-like 3 | Homo sapiens (human) | Kd | 6.5475 | 2 | 8 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 18.6668 | 3 | 15 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 13.5080 | 5 | 22 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 10.8298 | 7 | 24 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 10 |
| Cytochrome P450 2B6 | Homo sapiens (human) | EC50 | 1.3000 | 1 | 1 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Death-associated protein kinase 1 | Homo sapiens (human) | Kd | 7.7200 | 3 | 13 |
| Death-associated protein kinase 2 | Homo sapiens (human) | Kd | 6.7593 | 5 | 15 |
| Death-associated protein kinase 3 | Homo sapiens (human) | Kd | 7.0383 | 6 | 20 |
| Delta-type opioid receptor | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Delta-type opioid receptor | Mus musculus (house mouse) | EC50 | 0.0030 | 1 | 2 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 12.1245 | 7 | 24 |
| DNA damage-binding protein 1 | Homo sapiens (human) | EC50 | 0.0090 | 1 | 1 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| DNA-binding protein Ikaros | Homo sapiens (human) | EC50 | 0.0455 | 1 | 2 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Dual serine/threonine and tyrosine protein kinase | Homo sapiens (human) | Kd | 8.5500 | 1 | 6 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 14.9033 | 4 | 21 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 15.5458 | 4 | 22 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 17.2238 | 4 | 21 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | Kd | 13.1688 | 4 | 16 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 13.3951 | 2 | 14 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 17.3905 | 4 | 21 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 10.7787 | 7 | 24 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 11.4601 | 7 | 23 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 17.0000 | 4 | 20 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 9.2538 | 7 | 20 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 12.4357 | 6 | 21 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 17.0000 | 4 | 20 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 13.3015 | 3 | 16 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 11.0812 | 4 | 16 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | Kd | 6.6325 | 2 | 8 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| eIF-2-alpha kinase GCN2 | Homo sapiens (human) | Kd | 7.7338 | 3 | 13 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 26.2515 | 1 | 8 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 15.2263 | 4 | 19 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 15.9455 | 5 | 22 |
| Ephrin type-A receptor 3 | Homo sapiens (human) | Kd | 5.3857 | 4 | 14 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 15.9227 | 5 | 22 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 15.3128 | 6 | 25 |
| Ephrin type-A receptor 6 | Homo sapiens (human) | Kd | 2.9575 | 5 | 16 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 13.3719 | 6 | 26 |
| Ephrin type-A receptor 8 | Homo sapiens (human) | Kd | 7.2747 | 5 | 15 |
| Ephrin type-B receptor 1 | Homo sapiens (human) | Kd | 4.6838 | 5 | 16 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 16.0524 | 4 | 21 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 18.4500 | 4 | 24 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 14.7416 | 5 | 24 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 15.5842 | 3 | 15 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 9.8653 | 31 | 149 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 8.1176 | 6 | 23 |
| Estrogen receptor | Homo sapiens (human) | EC50 | 1.1568 | 3 | 5 |
| Estrogen receptor | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 4 |
| Estrogen receptor beta | Homo sapiens (human) | EC50 | 0.9808 | 3 | 5 |
| Estrogen receptor beta | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 4 |
| Eukaryotic peptide chain release factor GTP-binding subunit ERF3B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 22.5000 | 2 | 16 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 24.5727 | 2 | 9 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 12.5197 | 5 | 23 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | Kd | 4.7320 | 5 | 15 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | Kd | 6.2067 | 7 | 27 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | Kd | 8.6692 | 3 | 13 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 14.8930 | 6 | 23 |
| G protein-coupled receptor kinase 4 | Homo sapiens (human) | Kd | 7.5350 | 2 | 8 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 25.2692 | 1 | 6 |
| G-protein coupled receptor 35 | Homo sapiens (human) | EC50 | 10.8600 | 2 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | EC50 | 3.6000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | EC50 | 3.6000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | EC50 | 3.6000 | 1 | 1 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 23.5926 | 1 | 9 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 26.2550 | 1 | 8 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 15.2500 | 4 | 21 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 15.2559 | 4 | 21 |
| glycogen synthase kinase-3 beta isoform 1 | Homo sapiens (human) | EC50 | 3.8120 | 1 | 1 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | EC50 | 0.0070 | 1 | 1 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Kd | 0.0010 | 1 | 1 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Kd | 0.0017 | 1 | 1 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 11.0066 | 9 | 37 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 9.6453 | 7 | 24 |
| HLA class I histocompatibility antigen, A alpha chain | Homo sapiens (human) | Kd | 21.2000 | 1 | 1 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | Kd | 5.7694 | 2 | 8 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | Kd | 4.3702 | 2 | 8 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | Kd | 3.1515 | 2 | 8 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | Kd | 3.7965 | 2 | 8 |
| Hormonally up-regulated neu tumor-associated kinase | Homo sapiens (human) | Kd | 7.6250 | 2 | 8 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | Kd | 7.6300 | 2 | 8 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 14.9329 | 4 | 21 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Insulin receptor | Homo sapiens (human) | Kd | 15.4942 | 6 | 24 |
| Insulin receptor-related protein | Homo sapiens (human) | Kd | 6.8531 | 3 | 13 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 17.1727 | 4 | 22 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 26.4161 | 1 | 8 |
| Interferon-induced, double-stranded RNA-activated protein kinase | Homo sapiens (human) | Kd | 7.8469 | 3 | 13 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 19.4134 | 3 | 17 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 14.2917 | 4 | 21 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 16.6764 | 2 | 14 |
| Isoleucine--tRNA ligase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Kappa-type opioid receptor | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| LacZ protein (plasmid) | Escherichia coli | EC50 | 40.0000 | 1 | 1 |
| large T antigen | Betapolyomavirus macacae | EC50 | 47.9300 | 1 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 8.3488 | 2 | 12 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | Kd | 6.6538 | 3 | 13 |
| Leukotriene C4 synthase | Cavia porcellus (domestic guinea pig) | Kd | 8.4883 | 1 | 6 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 15.1144 | 5 | 23 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 16.7033 | 4 | 21 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Lysosomal acid glucosylceramidase | Homo sapiens (human) | EC50 | 2.5000 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Kd | 1.5777 | 4 | 14 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 19.8500 | 3 | 16 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| MAP kinase-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 17.0000 | 4 | 20 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 5.5377 | 3 | 13 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 5.0843 | 4 | 14 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 12.9390 | 5 | 22 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 15.2774 | 4 | 21 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Kd | 2.6495 | 25 | 113 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 13.2300 | 4 | 21 |
| Matrix metalloproteinase-9 | Homo sapiens (human) | Kd | 2.1800 | 1 | 1 |
| Megakaryocyte-associated tyrosine-protein kinase | Homo sapiens (human) | Kd | 9.7125 | 2 | 8 |
| melanocortin receptor 4 | Homo sapiens (human) | EC50 | 50.0000 | 1 | 1 |
| Membrane-associated progesterone receptor component 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| Microtubule-associated serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 7.0750 | 2 | 8 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 8.9298 | 3 | 9 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 16.8810 | 4 | 21 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 14.4113 | 6 | 23 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | Kd | 8.9071 | 4 | 14 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | Kd | 9.1500 | 2 | 8 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 14.8535 | 6 | 23 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 14.5704 | 4 | 21 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Mitogen-activated protein kinase 4 | Homo sapiens (human) | Kd | 9.0923 | 3 | 13 |
| Mitogen-activated protein kinase 6 | Homo sapiens (human) | Kd | 8.5385 | 3 | 13 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 15.5054 | 4 | 21 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 15.6309 | 5 | 22 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 18.3614 | 3 | 16 |
| Mitogen-activated protein kinase kinase kinase 10 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 13.8125 | 4 | 21 |
| Mitogen-activated protein kinase kinase kinase 12 | Homo sapiens (human) | Kd | 8.3500 | 1 | 6 |
| Mitogen-activated protein kinase kinase kinase 13 | Homo sapiens (human) | Kd | 7.5238 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 15 | Homo sapiens (human) | Kd | 7.8250 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 19 | Homo sapiens (human) | Kd | 1.6103 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 17.0313 | 3 | 16 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 13.4850 | 4 | 21 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 17.1065 | 3 | 16 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 15.4677 | 5 | 22 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 20.0000 | 3 | 16 |
| Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens (human) | Kd | 3.4866 | 4 | 10 |
| Mitogen-activated protein kinase kinase kinase 9 | Homo sapiens (human) | Kd | 8.4769 | 3 | 13 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 12.8378 | 4 | 20 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 17.7229 | 3 | 16 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 14.2554 | 4 | 23 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 11.6680 | 4 | 22 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 11.9946 | 6 | 26 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 25.5845 | 1 | 6 |
| Mu-type opioid receptor | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Muscle, skeletal receptor tyrosine-protein kinase | Homo sapiens (human) | Kd | 3.9908 | 3 | 13 |
| Myosin light chain kinase 2, skeletal/cardiac muscle | Homo sapiens (human) | Kd | 4.4826 | 5 | 16 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 19.3325 | 2 | 13 |
| Myosin light chain kinase family member 4 | Homo sapiens (human) | Kd | 7.1112 | 3 | 13 |
| Myosin light chain kinase, smooth muscle | Gallus gallus (chicken) | Kd | 6.3446 | 1 | 5 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 16.4345 | 5 | 25 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Myosin-IIIa | Homo sapiens (human) | Kd | 9.4692 | 3 | 13 |
| Myosin-IIIb | Homo sapiens (human) | Kd | 7.9846 | 3 | 13 |
| Myotonin-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 15.1876 | 4 | 21 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 14.5173 | 6 | 30 |
| NPYLR7B | Aedes aegypti (yellow fever mosquito) | EC50 | 20.0000 | 1 | 1 |
| NT-3 growth factor receptor | Homo sapiens (human) | Kd | 5.1938 | 3 | 13 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | Kd | 7.7034 | 3 | 13 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 13.8868 | 4 | 19 |
| Nuclear receptor subfamily 1 group I member 2 | Homo sapiens (human) | EC50 | 2.0790 | 9 | 10 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 25.0012 | 1 | 6 |
| P2X purinoceptor 1 | Rattus norvegicus (Norway rat) | EC50 | 1.0000 | 1 | 1 |
| P2X purinoceptor 2 | Rattus norvegicus (Norway rat) | EC50 | 10.4000 | 1 | 1 |
| P2X purinoceptor 3 | Homo sapiens (human) | EC50 | 8.9500 | 2 | 2 |
| P2X purinoceptor 4 | Rattus norvegicus (Norway rat) | EC50 | 100.0000 | 1 | 1 |
| P2X purinoceptor 5 | Rattus norvegicus (Norway rat) | EC50 | 4.0000 | 1 | 1 |
| P2X purinoceptor 6 | Rattus norvegicus (Norway rat) | EC50 | 100.0000 | 1 | 1 |
| P2X purinoceptor 7 | Homo sapiens (human) | EC50 | 92.0000 | 1 | 1 |
| P2Y purinoceptor 1 | Meleagris gallopavo (turkey) | EC50 | 10.0000 | 1 | 1 |
| P2Y purinoceptor 11 | Homo sapiens (human) | EC50 | 16.0000 | 1 | 1 |
| P2Y purinoceptor 12 | Rattus norvegicus (Norway rat) | EC50 | 4.0000 | 1 | 1 |
| P2Y purinoceptor 2 | Homo sapiens (human) | EC50 | 48.0000 | 1 | 1 |
| P2Y purinoceptor 4 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Peripheral plasma membrane protein CASK | Homo sapiens (human) | Kd | 8.4000 | 1 | 6 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Peroxisome proliferator-activated receptor gamma | Mus musculus (house mouse) | EC50 | 2.3000 | 1 | 1 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha | Homo sapiens (human) | Kd | 8.9385 | 3 | 13 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | Kd | 10.0000 | 21 | 88 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | Homo sapiens (human) | Kd | 7.7013 | 3 | 13 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 21.4286 | 2 | 14 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 12.0101 | 6 | 23 |
| Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | Homo sapiens (human) | Kd | 5.8504 | 5 | 15 |
| Placenta growth factor | Homo sapiens (human) | Kd | 0.0082 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Kd | 1.4616 | 4 | 14 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 3.7819 | 6 | 26 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | EC50 | 0.0200 | 1 | 1 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | Kd | 0.1100 | 1 | 1 |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | Kd | 9.4500 | 1 | 2 |
| POsterior Segregation | Caenorhabditis elegans | EC50 | 60.3740 | 1 | 1 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Procathepsin L | Homo sapiens (human) | EC50 | 37.8633 | 1 | 3 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Kd | 8.3392 | 1 | 6 |
| Protein cereblon | Homo sapiens (human) | EC50 | 0.0418 | 3 | 5 |
| Protein delta homolog 1 | Homo sapiens (human) | Kd | 5.0500 | 1 | 2 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 24.1818 | 3 | 11 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 16.3328 | 4 | 21 |
| Protein kinase C epsilon type | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Protein kinase C eta type | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 21.4286 | 2 | 14 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 15.5220 | 4 | 21 |
| Protein kinase C zeta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Protein mono-ADP-ribosyltransferase PARP3 | Homo sapiens (human) | Kd | 0.7000 | 1 | 1 |
| Protein polybromo-1 | Homo sapiens (human) | Kd | 12.9000 | 1 | 1 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 16.8294 | 4 | 22 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 16.0045 | 5 | 22 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 4.5694 | 12 | 51 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 15.5000 | 5 | 22 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 26.5708 | 1 | 8 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 27.0026 | 1 | 8 |
| Rab-like protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 16.5762 | 4 | 21 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Kd | 7.7454 | 3 | 13 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 6.2200 | 4 | 14 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 14.1369 | 5 | 22 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Receptor-interacting serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 8.0250 | 2 | 8 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 3.9104 | 28 | 106 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | EC50 | 31.0475 | 2 | 4 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | EC50 | 37.8633 | 1 | 3 |
| Replicase polyprotein 1ab | Human coronavirus 229E | EC50 | 31.0475 | 2 | 4 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | EC50 | 23.6440 | 3 | 5 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | EC50 | 25.4260 | 3 | 5 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Kd | 18.4000 | 3 | 3 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 18.8075 | 3 | 16 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 18.1819 | 3 | 16 |
| Rhodopsin kinase GRK1 | Homo sapiens (human) | Kd | 7.5725 | 2 | 8 |
| Rhodopsin kinase GRK7 | Homo sapiens (human) | Kd | 7.5450 | 2 | 8 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 12.4597 | 7 | 34 |
| Ribosomal protein S6 kinase alpha-2 | Homo sapiens (human) | Kd | 7.8099 | 8 | 28 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 13.6942 | 6 | 23 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 12.1854 | 7 | 34 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 11.2471 | 9 | 36 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 12.9906 | 7 | 34 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 18.3155 | 3 | 16 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 23.0077 | 1 | 8 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| RuvB-like 2 | Homo sapiens (human) | Kd | 22.0000 | 1 | 1 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Septin-9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 10 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 9.2779 | 6 | 24 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 14.8465 | 6 | 23 |
| Serine/threonine-protein kinase 17A | Homo sapiens (human) | Kd | 5.3950 | 5 | 15 |
| Serine/threonine-protein kinase 17B | Homo sapiens (human) | Kd | 6.7180 | 5 | 15 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 12.7165 | 4 | 20 |
| Serine/threonine-protein kinase 25 | Homo sapiens (human) | Kd | 7.7592 | 3 | 13 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 13.4080 | 4 | 21 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 12.6816 | 4 | 21 |
| Serine/threonine-protein kinase 3 | Mus musculus (house mouse) | Kd | 0.1600 | 1 | 1 |
| Serine/threonine-protein kinase 32A | Homo sapiens (human) | Kd | 8.4400 | 1 | 6 |
| Serine/threonine-protein kinase 32B | Homo sapiens (human) | Kd | 8.0338 | 3 | 13 |
| Serine/threonine-protein kinase 32C | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Serine/threonine-protein kinase 33 | Homo sapiens (human) | Kd | 4.4655 | 3 | 13 |
| Serine/threonine-protein kinase 35 | Homo sapiens (human) | Kd | 6.5782 | 2 | 8 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | Kd | 6.9514 | 4 | 14 |
| Serine/threonine-protein kinase 38 | Homo sapiens (human) | Kd | 7.6025 | 2 | 8 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 13.3900 | 5 | 19 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 12.2953 | 6 | 24 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Serine/threonine-protein kinase ATR | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | EC50 | 0.0030 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 12.1595 | 8 | 35 |
| Serine/threonine-protein kinase BRSK1 | Homo sapiens (human) | Kd | 8.5000 | 3 | 13 |
| Serine/threonine-protein kinase BRSK2 | Homo sapiens (human) | Kd | 7.6077 | 3 | 13 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 15.6452 | 4 | 22 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | Kd | 7.5021 | 2 | 8 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | Kd | 6.4100 | 3 | 13 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 14.2888 | 4 | 21 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 12.8133 | 4 | 22 |
| Serine/threonine-protein kinase DCLK1 | Homo sapiens (human) | Kd | 6.4854 | 3 | 13 |
| Serine/threonine-protein kinase DCLK2 | Homo sapiens (human) | Kd | 6.9308 | 3 | 13 |
| Serine/threonine-protein kinase DCLK3 | Homo sapiens (human) | Kd | 6.4254 | 3 | 13 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 17.4060 | 3 | 15 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 13.9773 | 4 | 22 |
| Serine/threonine-protein kinase LATS2 | Homo sapiens (human) | Kd | 6.5215 | 3 | 13 |
| Serine/threonine-protein kinase MAK | Homo sapiens (human) | Kd | 9.0375 | 2 | 8 |
| Serine/threonine-protein kinase MARK1 | Homo sapiens (human) | Kd | 7.9692 | 3 | 13 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 13.6767 | 5 | 23 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 17.5381 | 4 | 21 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 14.8712 | 4 | 21 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 15.0055 | 4 | 21 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Serine/threonine-protein kinase Nek11 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 15.0087 | 6 | 23 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 22.0063 | 2 | 14 |
| Serine/threonine-protein kinase Nek4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Serine/threonine-protein kinase Nek5 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 16.1150 | 4 | 20 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Serine/threonine-protein kinase NIM1 | Homo sapiens (human) | Kd | 7.7125 | 2 | 8 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 16.2819 | 4 | 21 |
| Serine/threonine-protein kinase OSR1 | Homo sapiens (human) | Kd | 7.6325 | 2 | 8 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 17.0000 | 4 | 20 |
| Serine/threonine-protein kinase PAK 3 | Homo sapiens (human) | Kd | 6.6960 | 3 | 13 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 15.8140 | 4 | 22 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Kd | 7.8400 | 3 | 13 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 12.3250 | 4 | 16 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 15.0000 | 5 | 19 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | Kd | 8.2462 | 3 | 13 |
| Serine/threonine-protein kinase PknB | Mycobacterium tuberculosis H37Rv | Kd | 8.3478 | 1 | 6 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 14.7059 | 4 | 17 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Kd | 8.6750 | 2 | 8 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Kd | 9.7692 | 3 | 13 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 14.0212 | 6 | 25 |
| Serine/threonine-protein kinase PRP4 homolog | Homo sapiens (human) | Kd | 7.5975 | 2 | 8 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 11.4286 | 4 | 14 |
| Serine/threonine-protein kinase RIO1 | Homo sapiens (human) | Kd | 7.7004 | 3 | 13 |
| Serine/threonine-protein kinase RIO2 | Homo sapiens (human) | Kd | 5.7553 | 3 | 9 |
| Serine/threonine-protein kinase RIO3 | Homo sapiens (human) | Kd | 8.5692 | 3 | 13 |
| Serine/threonine-protein kinase SBK1 | Homo sapiens (human) | Kd | 8.3667 | 1 | 6 |
| Serine/threonine-protein kinase Sgk3 | Homo sapiens (human) | Kd | 7.0200 | 1 | 6 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Kd | 8.4308 | 3 | 13 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 16.0705 | 4 | 22 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 18.8236 | 3 | 17 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 16.8234 | 4 | 22 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 14.3488 | 4 | 18 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 20.1671 | 2 | 14 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 16.6688 | 3 | 16 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 18.4301 | 3 | 18 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | Kd | 7.2229 | 4 | 14 |
| Serine/threonine-protein kinase tousled-like 1 | Homo sapiens (human) | Kd | 7.8631 | 3 | 13 |
| Serine/threonine-protein kinase tousled-like 2 | Homo sapiens (human) | Kd | 7.7685 | 3 | 13 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 14.7409 | 3 | 16 |
| Serine/threonine-protein kinase ULK2 | Homo sapiens (human) | Kd | 7.5032 | 2 | 8 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 16.9506 | 3 | 16 |
| Serine/threonine-protein kinase ULK3 | Mus musculus (house mouse) | Kd | 0.1100 | 1 | 1 |
| Serine/threonine-protein kinase VRK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 18.8250 | 3 | 16 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Sex hormone-binding globulin | Homo sapiens (human) | Kd | 0.3090 | 1 | 1 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | Kd | 8.2000 | 2 | 4 |
| SNF-related serine/threonine-protein kinase | Homo sapiens (human) | Kd | 8.4400 | 1 | 6 |
| Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | EC50 | 1.4500 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | EC50 | 31.0000 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | EC50 | 37.8633 | 1 | 3 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | EC50 | 37.8633 | 1 | 3 |
| SRSF protein kinase 1 | Homo sapiens (human) | Kd | 7.7500 | 3 | 13 |
| SRSF protein kinase 2 | Homo sapiens (human) | Kd | 7.7362 | 3 | 13 |
| SRSF protein kinase 3 | Homo sapiens (human) | Kd | 7.5148 | 2 | 8 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 12.5482 | 6 | 24 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 23.7716 | 1 | 9 |
| STE20/SPS1-related proline-alanine-rich protein kinase | Homo sapiens (human) | Kd | 7.5350 | 2 | 8 |
| streptokinase A precursor | Streptococcus pyogenes M1 GAS | EC50 | 77.1175 | 2 | 4 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 9 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 26.2509 | 1 | 8 |
| Testis-specific serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 9.1462 | 3 | 13 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 17.3500 | 4 | 22 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 11.3687 | 6 | 23 |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens (human) | EC50 | 6.3333 | 3 | 3 |
| Transient receptor potential cation channel subfamily M member 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 6 |
| Transient receptor potential cation channel subfamily M member 8 | Mus musculus (house mouse) | EC50 | 8.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | Kd | 19.9526 | 1 | 1 |
| Transmembrane protease serine 2 | Homo sapiens (human) | EC50 | 37.8633 | 1 | 3 |
| Transthyretin | Homo sapiens (human) | Kd | 0.0700 | 1 | 1 |
| Tubulin alpha-1A chain | Rattus norvegicus (Norway rat) | Kd | 10.0000 | 1 | 5 |
| Tubulin alpha-1A chain | Sus scrofa (pig) | Kd | 1.0450 | 4 | 4 |
| Tubulin beta chain | Sus scrofa (pig) | Kd | 1.0450 | 4 | 4 |
| Tubulin beta-2B chain | Bos taurus (cattle) | Kd | 8.2000 | 2 | 2 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 26.6645 | 1 | 8 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | EC50 | 1.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 5.8352 | 41 | 179 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 13.7885 | 5 | 24 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | Kd | 7.0919 | 3 | 13 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 17.2429 | 4 | 21 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 17.2810 | 4 | 21 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 14.3954 | 5 | 22 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 16.3276 | 4 | 21 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 8.9282 | 6 | 18 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 11.6183 | 7 | 24 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 15.6300 | 5 | 22 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 14.0492 | 5 | 22 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | Kd | 7.6953 | 3 | 13 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 12.3432 | 8 | 31 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 13.2721 | 5 | 19 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Kd | 7.7615 | 3 | 13 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 12.3337 | 5 | 23 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 12.7090 | 6 | 23 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 9.5386 | 4 | 16 |
| Tyrosine-protein kinase receptor Tie-1 | Homo sapiens (human) | Kd | 5.0326 | 3 | 13 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | Kd | 7.7036 | 3 | 13 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | Kd | 4.9390 | 3 | 13 |
| Tyrosine-protein kinase Srms | Homo sapiens (human) | Kd | 9.9538 | 3 | 13 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | EC50 | 4.5000 | 1 | 1 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 18.1818 | 4 | 22 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 17.6190 | 4 | 21 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 14.2830 | 5 | 23 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | Kd | 10.0000 | 3 | 13 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 18.0018 | 1 | 5 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 26.7146 | 1 | 9 |
| Uncharacterized serine/threonine-protein kinase SBK3 | Homo sapiens (human) | Kd | 7.9750 | 2 | 8 |
| Vascular endothelial growth factor A | Homo sapiens (human) | Kd | 0.0165 | 1 | 1 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Kd | 1.4338 | 4 | 14 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | EC50 | 0.5000 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Kd | 1.0323 | 7 | 20 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Kd | 1.1931 | 5 | 18 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 18.5663 | 4 | 22 |
| Wee1-like protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 8 |
| Zinc finger protein Aiolos | Homo sapiens (human) | EC50 | 0.0545 | 1 | 2 |
| Zinc finger protein mex-5 | Caenorhabditis elegans | EC50 | 31.0000 | 1 | 1 |