Proteins > type-1 angiotensin II receptor
Page last updated: 2024-08-07 15:14:41

type-1 angiotensin II receptor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (19)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
disulfiramHomo sapiens (human)IC506.637010
helenalinHomo sapiens (human)IC5018.639010
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)IC503.673010
n-(6-methoxy-8-quinolyl)-4-toluenesulfonamideHomo sapiens (human)IC503.882010
8-(4-benzenesulfonylamino)quinolineHomo sapiens (human)IC502.747010
miglitolHomo sapiens (human)IC5040.000010
angustibalinHomo sapiens (human)IC5021.974010
4-chloro-1-ethyl-3-nitro-2-quinolinoneHomo sapiens (human)IC502.221010
N-[[3-chloro-2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-methoxy-3-nitrobenzamideHomo sapiens (human)IC5040.000010
7'-hydroxy-4'-(4-methoxyphenyl)-4,4,5'-trimethyl-2-spiro[1,3-diazinane-6,2'-3,4-dihydro-2H-1-benzopyran]thioneHomo sapiens (human)IC5079.000020
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaHomo sapiens (human)IC5018.798010
1,5-dioxo-2,4-dihydropyrrolo[1,2-a]quinazoline-3-carboxylic acid ethyl esterHomo sapiens (human)IC509.246010
4-oxo-6-((pyrimidin-2-ylthio)methyl)-4h-pyran-3-yl 4-nitrobenzoateHomo sapiens (human)IC5079.000020
calcimycinHomo sapiens (human)IC5040.000010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
6-methoxy-3-[[2-oxolanylmethyl-[1-[1-(phenylmethyl)-5-tetrazolyl]propyl]amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)EC50100.000010
N-(4-hydroxy-2-methyl-5-propan-2-ylphenyl)benzenesulfonamideHomo sapiens (human)EC5079.000010
3-[(4-nitrophenyl)methoxy]-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-6-oneHomo sapiens (human)EC50100.000010
N-[(3,5-dimethoxyanilino)-sulfanylidenemethyl]-3-phenylpropanamideHomo sapiens (human)EC50100.000010
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[[3-(phenylmethyl)-2-imidazo[4,5-b]pyridinyl]thio]acetamideHomo sapiens (human)EC5079.000010