Page last updated: 2024-08-07 13:19:40
P2Y purinoceptor 1
A P2Y purinoceptor 1 that is encoded in the genome of turkey. [OMA:P49652, PRO:DNx]
Synonyms
P2Y1;
6H1 orphan receptor;
ADP receptor;
Purinergic receptor
Research
Bioassay Publications (10)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (20.00) | 18.2507 |
| 2000's | 5 (50.00) | 29.6817 |
| 2010's | 3 (30.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (17)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acid | Meleagris gallopavo (turkey) | IC50 | 16.6000 | 1 | 1 |
| adenosine 3'-phosphate-5'-phosphate | Meleagris gallopavo (turkey) | IC50 | 9.5450 | 2 | 2 |
| adenosine 2',5'-diphosphate | Meleagris gallopavo (turkey) | IC50 | 8.4600 | 1 | 1 |
| mrs2159 | Meleagris gallopavo (turkey) | IC50 | 100.0000 | 1 | 1 |
| 2'-deoxyadenosine-3',5'-diphosphate | Meleagris gallopavo (turkey) | IC50 | 5.7600 | 2 | 2 |
| 2'-deoxyguanosine 3',5'-diphosphate | Meleagris gallopavo (turkey) | IC50 | 14.9000 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| suramin | Meleagris gallopavo (turkey) | EC50 | 10.0000 | 1 | 1 |
| adenosine diphosphate | Meleagris gallopavo (turkey) | EC50 | 4.0500 | 2 | 2 |
| adenosine monophosphate | Meleagris gallopavo (turkey) | EC50 | 3.1500 | 1 | 2 |
| 2'-deoxyadenosine triphosphate | Meleagris gallopavo (turkey) | EC50 | 19.0000 | 1 | 1 |
| 5'-adenylyl (beta,gamma-methylene)diphosphonate | Meleagris gallopavo (turkey) | EC50 | 100.0000 | 1 | 1 |
| alpha,beta-methyleneadenosine 5'-triphosphate | Meleagris gallopavo (turkey) | EC50 | 100.0000 | 1 | 1 |
| methylthio-adp | Meleagris gallopavo (turkey) | EC50 | 0.0042 | 6 | 6 |
| adenosine 3'-phosphate-5'-phosphate | Meleagris gallopavo (turkey) | EC50 | 1.8100 | 2 | 2 |
| 2-chloro-atp | Meleagris gallopavo (turkey) | EC50 | 0.7200 | 1 | 1 |
| adenosine 2',5'-diphosphate | Meleagris gallopavo (turkey) | EC50 | 1.3700 | 1 | 1 |
| adenosine 5'-o-(3-thiotriphosphate) | Meleagris gallopavo (turkey) | EC50 | 1.3000 | 1 | 1 |
| 2-methylthio-atp | Meleagris gallopavo (turkey) | EC50 | 0.0080 | 2 | 2 |
| adp beta s | Meleagris gallopavo (turkey) | EC50 | 0.0960 | 1 | 1 |
| 2'-deoxyadenosine-3',5'-diphosphate | Meleagris gallopavo (turkey) | EC50 | 6.2750 | 2 | 2 |