Proteins > melanocortin receptor 4
Page last updated: 2024-08-07 18:24:35

melanocortin receptor 4

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (28)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
n-(cyclohexylthio)phthalimideHomo sapiens (human)IC5062.013010
thymolphthaleinHomo sapiens (human)IC5064.584010
sorafenibHomo sapiens (human)IC5067.100020
nexavarHomo sapiens (human)IC504.480010
6-bromoindirubin-3'-oximeHomo sapiens (human)IC506.370010
2-[[(2,3-dimethoxyphenyl)-oxomethyl]amino]-5-propan-2-yl-3-thiophenecarboxamideHomo sapiens (human)IC5064.573010
4-bromo-3-nitrobenzoic acid [2-[anilino(oxo)methyl]phenyl] esterHomo sapiens (human)IC5064.574010
2-[(2-propyl-4-quinazolinyl)thio]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)IC5064.583010
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideHomo sapiens (human)IC5064.575010
2-chloro-N-[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]acetamideHomo sapiens (human)IC507.177010
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterHomo sapiens (human)IC5064.578010
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)IC5064.564010
nsc 105827Homo sapiens (human)IC5064.577010
ML162Homo sapiens (human)IC5064.585010
chlorhexidineHomo sapiens (human)IC501.997010
chlorhexidine hydrochlorideHomo sapiens (human)IC501.547010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
benzethonium chlorideHomo sapiens (human)EC5089.188010
cetylpyridinium chlorideHomo sapiens (human)EC5089.211010
9-methoxyellipticineHomo sapiens (human)EC5089.313010
sorafenibHomo sapiens (human)EC5050.000010
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)EC5089.167010
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)EC5089.177010
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideHomo sapiens (human)EC5089.186010
N-[(3-benzamidoanilino)-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)EC5089.200010
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideHomo sapiens (human)EC5089.179010
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)EC5089.198010
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideHomo sapiens (human)EC5089.224010
dihydroxanthohumolHomo sapiens (human)EC5089.202010
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)EC5089.208010