An estrogen receptor that is encoded in the genome of rat. [OMA:P06211, PRO:DNx]
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| benzbromarone | Rattus norvegicus (Norway rat) | EC50 | 17.1820 | 1 | 0 |
| eucalyptol | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| clofazimine | Rattus norvegicus (Norway rat) | EC50 | 2.2810 | 1 | 0 |
| clotrimazole | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| safingol | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| ellipticine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| hexachlorophene | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| pyrimethamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| ici 204,219 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 0 |
| norethindrone | Rattus norvegicus (Norway rat) | Kd | 0.0006 | 1 | 1 |
| azoviolet | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 0 |
| dehydrothio-4-toluidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| naphthyl red | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| metformin hydrochloride | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| nsc-145,668 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| thiamphenicol | Rattus norvegicus (Norway rat) | EC50 | 4.0180 | 1 | 0 |
| cetyldimethylethylammonium bromide | Rattus norvegicus (Norway rat) | EC50 | 23.2480 | 1 | 0 |
| thymolphthalein | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| triclabendazole | Rattus norvegicus (Norway rat) | EC50 | 4.6950 | 1 | 0 |
| cefaclor anhydrous | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| chaetochromin | Rattus norvegicus (Norway rat) | EC50 | 1.7390 | 1 | 0 |
| 4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol | Rattus norvegicus (Norway rat) | EC50 | 0.0060 | 1 | 1 |
| physodic acid | Rattus norvegicus (Norway rat) | EC50 | 15.8990 | 1 | 0 |
| dimidium bromide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 9-methoxyellipticine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| pyridaben | Rattus norvegicus (Norway rat) | EC50 | 20.7650 | 1 | 0 |
| 9,10-phenanthrenequinone monoxime | Rattus norvegicus (Norway rat) | EC50 | 7.1120 | 1 | 0 |
| tanshinone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| pefloxacin mesylate | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| n-(6-methoxy-8-quinolyl)-4-toluenesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| sch 45752 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| cryptotanshinone | Rattus norvegicus (Norway rat) | EC50 | 14.8160 | 1 | 0 |
| 8-(4-benzenesulfonylamino)quinoline | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-phenyl-1,2-benzisothiazol-3-(2h)-one | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| nbi 27914 | Rattus norvegicus (Norway rat) | EC50 | 1.3070 | 1 | 0 |
| estradiol 3-benzoate | Rattus norvegicus (Norway rat) | EC50 | 2.4310 | 1 | 0 |
| 6,7-bis(4-aminophenyl)pteridine-2,4-diamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| nsc-260594 | Rattus norvegicus (Norway rat) | EC50 | 27.9550 | 1 | 0 |
| linezolid | Rattus norvegicus (Norway rat) | EC50 | 5.9980 | 1 | 0 |
| mupirocin | Rattus norvegicus (Norway rat) | EC50 | 0.4230 | 1 | 0 |
| 6-bromoindirubin-3'-oxime | Rattus norvegicus (Norway rat) | EC50 | 44.9450 | 1 | 0 |
| 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 9-carbazolyl-(4-methylphenyl)methanone | Rattus norvegicus (Norway rat) | EC50 | 6.4540 | 1 | 0 |
| idarubicin hydrochloride | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| LSM-28231 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(1-ethyl-6-methyl-3-pyrazolo[3,4-b]quinolinyl)-4-pyridinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanol | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(3,4-dihydro-2H-quinolin-1-yl)-6-[(4-phenyl-1-piperazinyl)methyl]-1,3,5-triazin-2-amine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-(4-chlorophenyl)-3H-thieno[2,3-d]pyrimidine-4-thione | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-(3,5-dichlorophenyl)-3-phenylurea | Rattus norvegicus (Norway rat) | EC50 | 16.8190 | 1 | 0 |
| 3-[2-(4-methyl-2-propan-2-ylphenoxy)ethyl]-1H-benzimidazole-2-thione | Rattus norvegicus (Norway rat) | EC50 | 15.2370 | 1 | 0 |
| N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-5-nitro-2-furancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 111.4710 | 1 | 0 |
| 2-(2-methylphenoxy)-N-[2-(4-methyl-1-piperidinyl)phenyl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 45.0230 | 1 | 0 |
| 3-phenyl-5-(2-phenylphenyl)-1,2,4-oxadiazole | Rattus norvegicus (Norway rat) | EC50 | 21.5130 | 1 | 0 |
| 1-[[[2-(2,4-dichlorophenyl)-4-quinolinyl]-oxomethyl]amino]-3-phenylurea | Rattus norvegicus (Norway rat) | EC50 | 20.3880 | 1 | 0 |
| N-[[3-chloro-4-(4-morpholinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[[3-cyano-4-(2-methoxyphenyl)-6-phenyl-2-pyridinyl]thio]acetic acid | Rattus norvegicus (Norway rat) | EC50 | 1.7240 | 1 | 0 |
| LSM-16285 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[5-(2-fluorophenyl)-2-tetrazolyl]-N-[2-oxo-2-[(phenylmethyl)amino]ethyl]-N-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-[(3,5-dichloro-2-hydroxyphenyl)methylamino]-1,5-dimethyl-2-phenyl-3-pyrazolone | Rattus norvegicus (Norway rat) | EC50 | 21.0910 | 1 | 0 |
| 4-(4-methylphenyl)-2-[[3-(4-morpholinyl)-1-oxopropyl]amino]-3-thiophenecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 65.4060 | 1 | 0 |
| 4-(4-anilinoanilino)-2-quinazolinecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(3-bromophenyl)-2-(4-bromophenyl)-7-methylpyrazolo[3,4-d]pyridazine | Rattus norvegicus (Norway rat) | EC50 | 19.1850 | 1 | 0 |
| 4-(3-bromophenyl)-7-methyl-2-(4-methylphenyl)pyrazolo[3,4-d]pyridazine | Rattus norvegicus (Norway rat) | EC50 | 94.1220 | 1 | 0 |
| LSM-27108 | Rattus norvegicus (Norway rat) | EC50 | 27.7820 | 1 | 0 |
| 5-bromo-N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-2-furancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-bromo-N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[(4-chlorophenyl)thio]-N-(5-oxo-1-phenyl-4H-pyrazol-3-yl)acetamide | Rattus norvegicus (Norway rat) | EC50 | 9.3320 | 1 | 0 |
| [4-[(2-chlorophenyl)methyl]-1-piperazinyl]-(6,8-dimethyl-2-pyridin-4-yl-4-quinolinyl)methanone | Rattus norvegicus (Norway rat) | EC50 | 10.3150 | 1 | 0 |
| 4,6-bis(1-pyrrolidinyl)-N-[3-(trifluoromethyl)phenyl]-1,3,5-triazin-2-amine | Rattus norvegicus (Norway rat) | EC50 | 17.4810 | 1 | 0 |
| 3-[[[[[5-(4-chlorophenyl)-2-furanyl]-oxomethyl]amino]-sulfanylidenemethyl]amino]-4-methoxybenzoic acid | Rattus norvegicus (Norway rat) | EC50 | 23.7880 | 1 | 0 |
| N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 96.9890 | 1 | 0 |
| 2-[1-(4-tert-butylphenyl)sulfonyl-4-piperidinyl]-6-chloro-1H-benzimidazole | Rattus norvegicus (Norway rat) | EC50 | 4.1290 | 1 | 0 |
| N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-[4-[5-(trifluoromethyl)-1-benzotriazolyl]-1-piperidinyl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-[4-(2-fluorophenyl)-2-thiazolyl]-5-(trifluoromethyl)-4-pyrazolecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 34.3350 | 1 | 0 |
| 4-[(4-chloro-1-naphthalenyl)oxy]-5-methoxy-2-(2-pyridinyl)pyrimidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(methylthio)-7-(4-phenylphenyl)-[1,2,4]triazolo[1,5-a]pyrimidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1,1-bis(4-chlorophenyl)-2-[(3-methoxyphenyl)methylamino]ethanol | Rattus norvegicus (Norway rat) | EC50 | 18.9470 | 1 | 0 |
| 5-[(4-methyl-1-piperidinyl)methyl]-1-[4-(1-pyrrolyl)-1,2,5-oxadiazol-3-yl]-4-triazolecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 14.9060 | 1 | 0 |
| 1,4-benzoquinone guanylhydrazone thiosemicarbazone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-methoxy-2-(4-propoxyphenyl)quinazoline | Rattus norvegicus (Norway rat) | EC50 | 6.0180 | 1 | 0 |
| N-[(2-adamantylamino)-sulfanylidenemethyl]hexanamide | Rattus norvegicus (Norway rat) | EC50 | 11.5250 | 1 | 0 |
| N-[[[2-(2-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-methyl-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-tert-butyl-3-(4-chlorophenyl)-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-[2-[(3-chloro-4-methoxyphenyl)methylthio]ethyl]-3-phenylthiourea | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| amn082 | Rattus norvegicus (Norway rat) | EC50 | 12.0430 | 1 | 0 |
| 6-chloro-4-phenyl-2-(prop-2-enylthio)quinazoline | Rattus norvegicus (Norway rat) | EC50 | 29.4320 | 1 | 0 |
| 2-[[[2-amino-1-(3-methoxypropyl)-3-pyrrolo[3,2-b]quinoxalinyl]-oxomethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-[[(4-ethoxyanilino)-sulfanylidenemethyl]amino]-3-[3-(trifluoromethyl)phenyl]thiourea | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[[[(4-methoxyphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 5.1780 | 1 | 0 |
| 3-cyclohexyl-10-methyl-2-thiophen-2-ylpyrimido[4,5-b]quinoline-4,5-dione | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(4,5-diphenyl-2-oxazolyl)-2-[(1-methyl-5-tetrazolyl)thio]acetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2,2-diphenylacetic acid (2,6-dimethylphenyl) ester | Rattus norvegicus (Norway rat) | EC50 | 17.0390 | 1 | 0 |
| 5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| benzoic acid [2-oxo-2-[2-(phenylthio)anilino]ethyl] ester | Rattus norvegicus (Norway rat) | EC50 | 28.8160 | 1 | 0 |
| 3-[[4-(2-benzofuranyl)-2-thiazolyl]methyl]-2-[(dimethylamino)methyl]-4-quinazolinone | Rattus norvegicus (Norway rat) | EC50 | 103.9270 | 1 | 0 |
| N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2,5-diphenyl-3-pyrazolecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 8.3220 | 1 | 0 |
| 4-(4-tert-butylphenoxy)-N-(4,5-dihydrothiazol-2-yl)butanamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(1H-benzimidazol-2-yl)-3-[methyl-(4-methylphenyl)sulfamoyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[methyl(phenyl)sulfamoyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[[[[4-[(2-methyl-1-oxopropyl)amino]phenyl]-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-thiophenecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (3-anilino-5-methyl-1-pyrazolyl)-(4-bromophenyl)methanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-(4-propylphenyl)-1H-pyrazol-3-amine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(3-chloro-2-quinoxalinyl)-2-naphthalenesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 15.0930 | 1 | 0 |
| 2-[[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]thio]-N-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[4-bromo-3-(trifluoromethyl)phenyl]-2,4,6-trimethylbenzamide | Rattus norvegicus (Norway rat) | EC50 | 3.2900 | 1 | 0 |
| N-[4-(difluoromethylthio)phenyl]-5-[(2-hydroxy-5-methoxyphenyl)-oxomethyl]-2-imino-3-pyrancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 6-[[(2-chlorophenyl)methyl-methylamino]methyl]-N2-(2-methylphenyl)-1,3,5-triazine-2,4-diamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 6-amino-1-(2-methoxyethyl)-N-(4-methylphenyl)sulfonyl-2,4-dioxo-5-pyrimidinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (2S)-3-methyl-2-[[(3-methylphenyl)-oxomethyl]amino]butanoic acid (4-oxo-2-pyrimido[2,1-b][1,3]benzothiazolyl)methyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-[[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]methyl]-2-furancarboxylic acid methyl ester | Rattus norvegicus (Norway rat) | EC50 | 5.6120 | 1 | 0 |
| 4-chloro-N-[3-[(3,5-dimethyl-4-isoxazolyl)methylthio]-2-quinoxalinyl]benzenesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 5.5080 | 1 | 0 |
| tamoxifen | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 3-(2,4-dichlorophenyl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-chloro-N-[3-cyano-4-[(4-methoxyphenyl)thio]phenyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 4.9840 | 1 | 0 |
| 5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 2.8520 | 1 | 0 |
| 2-[[2-[[5-(4-tert-butylphenyl)-2-methoxycarbonyl-3-thiophenyl]amino]-2-oxoethyl]thio]acetic acid | Rattus norvegicus (Norway rat) | EC50 | 6.6890 | 1 | 0 |
| 2-amino-4-(2-chlorophenyl)-6-[(4-chlorophenyl)thio]pyridine-3,5-dicarbonitrile | Rattus norvegicus (Norway rat) | EC50 | 13.1540 | 1 | 0 |
| 2-[4-[[4-[bis(2-hydroxyethyl)amino]-2-chlorophenyl]-(2-chlorophenyl)methyl]-3-chloro-N-(2-hydroxyethyl)anilino]ethanol | Rattus norvegicus (Norway rat) | EC50 | 4.8400 | 1 | 0 |
| 2,4-dichloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 20.8570 | 1 | 0 |
| 1-hexadecyl-3-methylimidazolium bromide | Rattus norvegicus (Norway rat) | EC50 | 77.9860 | 1 | 0 |
| 2,4-dichloro-6-[1-(4-morpholinyl)-3-phenylprop-2-ynyl]phenol | Rattus norvegicus (Norway rat) | EC50 | 26.7640 | 1 | 0 |
| 4-[3-[[(2,5-dichloroanilino)-methyliminomethyl]thio]-2,5-dioxo-1-pyrrolidinyl]benzoic acid methyl ester | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 0 |
| N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-2-phenyl-4-quinolinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-[[3-[2-(1-cyclohexenyl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazolin-7-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 29.7590 | 1 | 0 |
| 4-[[1-[(3,4-dichlorophenyl)methyl]-3-indolyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-one | Rattus norvegicus (Norway rat) | EC50 | 10.0720 | 1 | 0 |
| 2-methyl-3-[(2-methyl-1H-indol-3-yl)-(2-pyridinyl)methyl]-1H-indole | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| LSM-19894 | Rattus norvegicus (Norway rat) | EC50 | 4.0390 | 1 | 0 |
| 1-[1-(1-adamantyl)butyl]-3-(2-oxolanylmethyl)thiourea | Rattus norvegicus (Norway rat) | EC50 | 18.0260 | 1 | 0 |
| 5-chloro-7-[3-pyridinyl-(2-pyridinylamino)methyl]-8-quinolinol | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-[[2-(dimethylamino)-2-thiophen-2-ylethyl]amino]-5-methyl-6-thieno[2,3-d]pyrimidinecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(6-imidazo[2,1-b]thiazolyl)acetic acid [2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl] ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| fusidic acid | Rattus norvegicus (Norway rat) | EC50 | 0.3620 | 1 | 0 |
| toremifene citrate | Rattus norvegicus (Norway rat) | EC50 | 25.9470 | 1 | 0 |
| N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) ester | Rattus norvegicus (Norway rat) | EC50 | 3.0140 | 1 | 0 |
| 2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl ester | Rattus norvegicus (Norway rat) | EC50 | 2.7960 | 1 | 0 |
| 1-(4-bromophenyl)-N-(3,4-dichlorophenyl)-5-oxo-3-pyrrolidinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 20.1340 | 1 | 0 |
| 2-[[2-(2,4-dichlorophenoxy)-1-oxopropyl]hydrazo]-N-(4-methoxyphenyl)-2-oxoacetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[(3-cyano-4,6-diphenyl-2-pyridinyl)thio]-3-methylbutanoic acid | Rattus norvegicus (Norway rat) | EC50 | 10.0580 | 1 | 0 |
| 2-(2-bromophenyl)-2,3-dihydro-1H-perimidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 9-(1H-indol-3-yl)acridine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(6-bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline | Rattus norvegicus (Norway rat) | EC50 | 2.5520 | 1 | 0 |
| 4-(6-bromo-1,3-benzodioxol-5-yl)-7,9-dimethyl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 7-(2-ethyl-1-piperidinyl)-5-methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidine | Rattus norvegicus (Norway rat) | EC50 | 15.2560 | 1 | 0 |
| 5-(4-bromophenyl)-N,N-diethyl-3-isoxazolecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 3,5-dimethyl-N-(2-phenylethyl)-N-(phenylmethyl)-4-isoxazolesulfonamide | Rattus norvegicus (Norway rat) | EC50 | 21.6590 | 1 | 0 |
| 6-[(2-chlorophenyl)methyl]-3-(3-methoxyphenyl)-7-triazolo[4,5-d]pyrimidinone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamine | Rattus norvegicus (Norway rat) | EC50 | 9.3190 | 1 | 0 |
| N-[[3-[(3-chlorophenyl)sulfamoyl]-4-methylanilino]-sulfanylidenemethyl]-4-fluorobenzamide | Rattus norvegicus (Norway rat) | EC50 | 11.5100 | 1 | 0 |
| 5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinol | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)-N-(5-ethyl-1,3,4-oxadiazol-2-yl)benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (S)-4',5,7-Trihydroxy-6-prenylflavanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(4-chlorophenyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]phenyl]-4-oxobutanamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]-5-nitro-2-thiophenecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| l 663536 | Rattus norvegicus (Norway rat) | EC50 | 1.2370 | 1 | 0 |
| N-[2-[[2-(4-chlorophenyl)-2-oxoethyl]thio]-4-oxo-3-quinazolinyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 105.6150 | 1 | 0 |
| 4-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitrobenzoic acid methyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitropyridine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-(benzenesulfonyl)-4-(2,6-dimethylphenoxy)-2-phenylpyrimidine | Rattus norvegicus (Norway rat) | EC50 | 3.9870 | 1 | 0 |
| 2-[4-(3-chlorophenyl)-1-piperazinyl]-3-pyridinecarboxylic acid propan-2-yl ester | Rattus norvegicus (Norway rat) | EC50 | 19.3340 | 1 | 0 |
| 4-fluoro-N-[[2-(3-pyridinyl)-1-piperidinyl]-sulfanylidenemethyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(2-chlorophenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(1H-benzimidazol-2-yl)-5-methyl-4-(phenylmethyl)-4H-pyrazol-3-one | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-(carbamoylamino)benzoic acid [2-(3-chloro-4-methylanilino)-2-oxo-1-phenylethyl] ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-benzoyl-2-heptyl-5-methyl-4H-pyrazol-3-one | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 6-(4-morpholinyl)-3-(2-phenylethyl)-2-sulfanylidene-1H-quinazolin-4-one | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (6-bromo-5-methoxy-2-methyl-3-benzofuranyl)-[4-(2-methylphenyl)-1-piperazinyl]methanone | Rattus norvegicus (Norway rat) | EC50 | 79.7540 | 1 | 0 |
| [3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methyl-1-piperidinyl)sulfonyl]benzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(4-chlorophenyl)-3-methyl-N-(2-thiazolyl)butanamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| LSM-16826 | Rattus norvegicus (Norway rat) | EC50 | 1.5300 | 1 | 0 |
| N-(1,3-benzodioxol-5-yl)-6-chloro-2-(2-pyridinyl)-3-imidazo[1,2-a]pyridinamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(1H-benzimidazol-2-yl)-3-phenylbutanamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[[(3,4-dimethoxyphenyl)-oxomethyl]amino]acetic acid [2-[5-(4-chlorophenyl)-3-(2-furanyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-bromo-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-2-thiophenecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-[3-(dimethylamino)propyl]thiourea | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[3-[(4-chlorophenyl)methylthio]-1H-1,2,4-triazol-5-yl]-4-cyanobenzamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 3-(1-methyl-2-benzimidazolyl)-1-(3-methylphenyl)-2-pyrrolo[3,2-b]quinoxalinamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(4-Nitro-1,2,5-oxadiazol-3-yl)-2-pyridin-2-ylsulfanylacetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (4-chloro-1-ethyl-3-pyrazolyl)-[3-(2-hydroxyphenyl)-5-(2-naphthalenyl)-3,4-dihydropyrazol-2-yl]methanone | Rattus norvegicus (Norway rat) | EC50 | 13.0080 | 1 | 0 |
| 2-[[4-amino-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]thio]-1-(1H-indol-3-yl)-2-phenylethanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| sphingosine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| amentoflavone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| morusin | Rattus norvegicus (Norway rat) | EC50 | 1.1490 | 1 | 0 |
| bornyl ferulate | Rattus norvegicus (Norway rat) | EC50 | 7.3170 | 1 | 0 |
| cycloheterophyllin | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| muromonab-cd3 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| chloride of pseudoisocyanine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5233705 compound | Rattus norvegicus (Norway rat) | EC50 | 13.2710 | 1 | 0 |
| nifuratrone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-(3-methylphenyl)-4-[4-(4-morpholinyl)-3-nitrophenyl]-1-phthalazinamine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| nitrofurantoin | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| am 404 | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-3-methyl-2-thiophenecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 3-(2,4-dimethoxyphenyl)-N-(3-fluoro-4-methylphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[(4-fluorophenyl)methyl]-2-[3-oxo-6-(1-piperidinylsulfonyl)-1,4-benzoxazin-4-yl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| N-[2-(3,4-dimethoxyphenyl)ethyl]-N'-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)oxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1,2-dihydroacenaphthylen-5-yl-[1-[(6-methyl-2-pyridinyl)methyl]-3-piperidinyl]methanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 1-cyclohexyl-2-[(1-ethyl-2-imidazolyl)methyl]-1,3,4,9-tetrahydropyrido[3,4-b]indole | Rattus norvegicus (Norway rat) | EC50 | 42.1440 | 1 | 0 |
| 4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidine | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid (phenylmethyl) ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-(3-methyl-1-piperidinyl)-3-oxopropyl]-4-phenyl-1-benzopyran-2-one | Rattus norvegicus (Norway rat) | EC50 | 41.2420 | 1 | 0 |
| 4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl ester | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| montelukast sodium | Rattus norvegicus (Norway rat) | EC50 | 3.4080 | 1 | 0 |
| cefoxitin sodium | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| (5R)-5-tert-butyl-1-[(3S)-3-phenyl-3-(phenylthio)propyl]-2-azepanone | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-[1-[(4-chlorophenyl)-oxomethyl]-5-methoxy-2-methyl-3-indolyl]-N-[(2-hydroxy-5-nitrophenyl)methyl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 20.1910 | 1 | 0 |
| 1-(3-methoxyphenyl)-3-(4-phenylbutyl)urea | Rattus norvegicus (Norway rat) | EC50 | 106.4670 | 1 | 0 |
| 2-(2,6-dimethylphenoxy)-N-[2-(1-piperidinyl)phenyl]acetamide | Rattus norvegicus (Norway rat) | EC50 | 4.1510 | 1 | 0 |
| N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-5-bromo-2-furancarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-hydroxy-1-methyl-N'-[(3-methylphenyl)-oxomethyl]-2-oxo-3-quinolinecarbohydrazide | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 4-hydroxy-6-propan-2-ylpyrano[3,2-c]quinoline-2,5-dione | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 6,8-dibromo-2-[[[4-(difluoromethoxy)phenyl]methyl-methylamino]methyl]-1H-quinazolin-4-one | Rattus norvegicus (Norway rat) | EC50 | 29.3720 | 1 | 0 |
| 7-methyl-2-[(4-methyl-6-phenyl-2-pyrimidinyl)amino]-1H-quinazolin-4-one | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| carbadox | Rattus norvegicus (Norway rat) | EC50 | 150.0000 | 1 | 0 |
| 2-(4-chloroanilino)-5-[(2,3-dichlorophenyl)methyl]-4-thiazolone | Rattus norvegicus (Norway rat) | EC50 | 130.5170 | 1 | 0 |