Page last updated: 2024-08-07 16:48:08

P2X purinoceptor 4

A P2X purinoceptor 4 that is encoded in the genome of rat. [OMA:P51577, PRO:DNx]

Synonyms

P2X4;
ATP receptor;
Purinergic receptor

Research

Bioassay Publications (5)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Compounds (12)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acidRattus norvegicus (Norway rat)IC50251.300022
paroxetineRattus norvegicus (Norway rat)IC502.450022
mrs 2219Rattus norvegicus (Norway rat)IC50100.000011
acid blue 40Rattus norvegicus (Norway rat)IC5010.000011
acid blue 25Rattus norvegicus (Norway rat)IC5010.000011
acid blue 129Rattus norvegicus (Norway rat)IC5010.000011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pyridoxal phosphateRattus norvegicus (Norway rat)EC50219.000011
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acidRattus norvegicus (Norway rat)EC5010.000011
suraminRattus norvegicus (Norway rat)EC50100.000011
adenosine diphosphateRattus norvegicus (Norway rat)EC5028.000011
alpha,beta-methyleneadenosine 5'-triphosphateRattus norvegicus (Norway rat)EC5033.000011
adenosine 5'-o-(3-thiotriphosphate)Rattus norvegicus (Norway rat)EC502.300011
2-methylthio-atpRattus norvegicus (Norway rat)EC508.700022