Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
astemizole | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
safingol | Homo sapiens (human) | IC50 | 14.4325 | 2 | 0 |
nafamostat | Homo sapiens (human) | IC50 | 14.0000 | 1 | 0 |
oxethazaine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
perphenazine | Homo sapiens (human) | IC50 | 14.7900 | 2 | 0 |
ritanserin | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
terfenadine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
benzethonium chloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
wr 171,699 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
butoconazole nitrate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
cerm-1978 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
amlodipine besylate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
fluoxetine hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
sertraline hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
mefloquine hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
nsc 38280 | Homo sapiens (human) | IC50 | 2.5125 | 2 | 0 |
econazole nitrate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
methixene hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
prochlorperazine edisylate salt | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
imidocarb | Homo sapiens (human) | IC50 | 11.8920 | 2 | 0 |
amiodarone hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
mefloquine hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
naringin | Homo sapiens (human) | IC50 | 7.6785 | 2 | 0 |
afimoxifene | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
trimethylcolchicinic acid | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-methyl-2-[(5-methyl-2-thiophenyl)methylideneamino]phenol | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazoline | Homo sapiens (human) | IC50 | 1.1845 | 2 | 0 |
calmidazolium | Homo sapiens (human) | IC50 | 8.2315 | 2 | 0 |
N-butyl-N-[5-(3,4,5-trimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-furancarboxamide | Homo sapiens (human) | IC50 | 10.0845 | 2 | 0 |
(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-(butylamino)-N-[4-[5-[[2-(butylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
LSM-28489 | Homo sapiens (human) | IC50 | 3.0260 | 2 | 0 |
isatin beta-thiosemicarbazone | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
6-bromo-3-phenyl-2-sulfanylidene-1H-quinazolin-4-one | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
thiothixene | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acid | Homo sapiens (human) | IC50 | 78.4000 | 1 | 0 |
LSM-16526 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-(dimethylsulfamoyl)-N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
6-(4-methyl-1-piperazinyl)-2-(3,4,5-trimethoxyphenyl)-1H-benzimidazole | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
1-[[[1-(6-methyl-2-pyridinyl)-4-imidazolyl]-oxomethyl]amino]-3-phenylthiourea | Homo sapiens (human) | IC50 | 10.8905 | 2 | 0 |
enclomiphene | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
CID 2131972 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
3-[[2-(6-methoxy-3-benzofuranyl)-1-oxoethyl]amino]benzoic acid methyl ester | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
tamoxifen | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
jnj-1661010 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
1-hexadecyl-3-methylimidazolium bromide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
cid 2858522 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
eskazine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-[2-[4-[2-hydroxy-3-(2-methylphenoxy)propyl]-1-piperazinyl]ethyl]benzo[de]isoquinoline-1,3-dione | Homo sapiens (human) | IC50 | 16.4000 | 2 | 0 |
zuclomifene citrate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
3-[5-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl ester | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
1-(4-chlorophenyl)sulfonyl-N'-[oxo-[4-(1-piperidinylsulfonyl)phenyl]methyl]-4-piperidinecarbohydrazide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
6-bromo-3-[4-oxo-4-[4-(2-pyridinyl)-1-piperazinyl]butyl]-2-sulfanylidene-1H-quinazolin-4-one | Homo sapiens (human) | IC50 | 19.8730 | 2 | 0 |
N-[2-(2,3-dimethylphenyl)-5,5-dioxo-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-2-methoxybenzamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-[(1-acetyl-2-benzimidazolyl)thio]-N-(2-methoxyphenyl)acetamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
1-pyrenebutylamine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
5-(4-ethoxyphenyl)-1,3-diphenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dione | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
5,5,7,7-tetramethyl-2-[[oxo-(4-propan-2-yloxyphenyl)methyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid methyl ester | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
1-[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-[3-(dimethylamino)propyl]thiourea | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-tert-butyl-N-[3-[4-[3-[[(4-tert-butylphenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]benzamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
sphingosine | Homo sapiens (human) | IC50 | 6.3125 | 2 | 0 |
perhexiline maleate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
N-[3-[butyl(ethyl)amino]propyl]-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-amino-5-chloro-N-[(3R,4S)-1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
baohuoside ii | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
methylbenzethonium chloride | Homo sapiens (human) | IC50 | 9.2060 | 2 | 0 |
5233705 compound | Homo sapiens (human) | IC50 | 8.6275 | 2 | 0 |
fluphenazine | Homo sapiens (human) | IC50 | 17.4345 | 2 | 0 |
dibenzheptropine citrate | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-(2-phenylethyl)benzo[de]isoquinoline-1,3-dione | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
chlorhexidine | Homo sapiens (human) | IC50 | 2.6045 | 2 | 0 |
a 77636 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
emergil | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
GR 127935 hydrochloride | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 15.3705 | 2 | 0 |
1-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)-3-[3-[4-(phenylmethyl)-1-piperidinyl]propyl]thiourea | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
N-[2-(dipropylamino)ethyl]-5-ethyl-4-oxo-2-thieno[3,2-c]quinolinecarboxamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-[[(4S)-2-amino-3-[2-(1-naphthalenyl)ethyl]-4,5-dihydroimidazol-4-yl]methyl]phenol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-[[(4S)-3-[2-(1-adamantyl)ethyl]-2-amino-4,5-dihydroimidazol-4-yl]methyl]phenol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
(5S)-1-(4-cyclohexylbutyl)-5-phenyl-4,5-dihydroimidazol-2-amine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
(5S)-1-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]-5-phenyl-4,5-dihydroimidazol-2-amine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
(5R)-1-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]-5-butyl-4,5-dihydroimidazol-2-amine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
3-bromo-N-[2-[(3R,6S)-6-[(4-methoxyphenyl)methyl]-3-(phenylmethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]imidazol-7-yl]ethyl]-4-methylbenzamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
3-(4-bromophenyl)-N-[5-[[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-oxomethyl]-2-methylphenyl]-1H-pyrazole-5-carboxamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-one | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-[[4-(5-chloro-2-methoxyanilino)-6-(1-piperidinyl)-1,3,5-triazin-2-yl]amino]ethanol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-[[4-(5-chloro-2-propan-2-yloxyanilino)-6-(1-pyrrolidinyl)-1,3,5-triazin-2-yl]amino]ethanol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 4.4013 | 3 | 0 |
N-[5-Fluoro-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chloride | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
(2R)-N2-[2-(4-bicyclo[2.2.1]heptanyl)ethyl]-N1-[(2R,3R)-3-methyl-1-(methylamino)pentan-2-yl]hexane-1,2-diamine | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
3-(4-Amino-3,5-dichlorobenzoyl)-2-(3-amino-3-oxopropyl)-2H-indazole 1-oxide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
pd 120697 | Homo sapiens (human) | IC50 | 16.1595 | 2 | 0 |
5-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]methyl]-8-quinolinol | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamide | Homo sapiens (human) | IC50 | 20.0000 | 1 | 0 |
tegaserod maleate | Homo sapiens (human) | IC50 | 10.3500 | 2 | 0 |