Page last updated: 2024-08-07 19:30:34
P2X purinoceptor 6
A P2X purinoceptor 6 that is encoded in the genome of rat. [OMA:P51579, PRO:DNx]
Synonyms
P2X6;
ATP receptor;
P2XM;
Purinergic receptor;
Purinergic receptor P2X-like 1
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (6)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acid | Rattus norvegicus (Norway rat) | IC50 | 251.0000 | 2 | 2 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acid | Rattus norvegicus (Norway rat) | EC50 | 100.0000 | 1 | 1 |
suramin | Rattus norvegicus (Norway rat) | EC50 | 100.0000 | 1 | 1 |
adenosine diphosphate | Rattus norvegicus (Norway rat) | EC50 | 11.0000 | 1 | 1 |
alpha,beta-methyleneadenosine 5'-triphosphate | Rattus norvegicus (Norway rat) | EC50 | 8.0000 | 1 | 1 |
adenosine 5'-o-(3-thiotriphosphate) | Rattus norvegicus (Norway rat) | EC50 | 1.3000 | 1 | 1 |
2-methylthio-atp | Rattus norvegicus (Norway rat) | EC50 | 0.6000 | 1 | 1 |