Page last updated: 2024-08-07 18:05:31
Endoplasmin
An endoplasmin that is encoded in the genome of dog. [OMA:P41148, PRO:DAN]
Synonyms
94 kDa glucose-regulated protein;
GRP-94;
Heat shock protein 90 kDa beta member 1
Research
Bioassay Publications (5)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 1 (20.00) | 24.3611 |
| 2020's | 3 (60.00) | 2.80 |
Compounds (13)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| adenosine diphosphate | Canis lupus familiaris (dog) | IC50 | 11.4470 | 1 | 1 |
| geldanamycin | Canis lupus familiaris (dog) | IC50 | 0.0100 | 1 | 1 |
| tanespimycin | Canis lupus familiaris (dog) | IC50 | 0.0310 | 1 | 1 |
| 9h-purine-9-propanamine, 6-amino-8-((6-iodo-1,3-benzodioxol-5-yl)thio)-n-(1-methylethyl)- | Canis lupus familiaris (dog) | IC50 | 0.0300 | 1 | 1 |
| at 13387 | Canis lupus familiaris (dog) | IC50 | 0.0130 | 1 | 1 |
| cnf 2024 | Canis lupus familiaris (dog) | IC50 | 0.1240 | 1 | 1 |
| snx 2112 | Canis lupus familiaris (dog) | IC50 | 0.5310 | 2 | 2 |
| debio 0932 | Canis lupus familiaris (dog) | IC50 | 0.1900 | 1 | 1 |
| ver 52296 | Canis lupus familiaris (dog) | IC50 | 0.0120 | 1 | 1 |
| sta 9090 | Canis lupus familiaris (dog) | IC50 | 0.0100 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| adenosine diphosphate | Canis lupus familiaris (dog) | EC50 | 21.0000 | 1 | 1 |
| adenosine-5'-(n-ethylcarboxamide) | Canis lupus familiaris (dog) | Kd | 2.8000 | 1 | 1 |
| 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin | Canis lupus familiaris (dog) | EC50 | 0.0650 | 1 | 1 |
| tanespimycin | Canis lupus familiaris (dog) | EC50 | 0.1240 | 1 | 1 |
| ipi 493 | Canis lupus familiaris (dog) | EC50 | 0.0480 | 1 | 1 |