Page last updated: 2024-08-07 10:05:41

Serine/threonine-protein kinase B-raf

A B-Raf proto-oncogene serine/threonine-protein kinase that is encoded in the genome of mouse. [OMA:MOUSE18293, PRO:DNx]

Synonyms

EC 2.7.11.1;
Proto-oncogene B-Raf

Research

Bioassay Publications (4)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (4)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
erlotinibMus musculus (house mouse)IC500.060011
erlotinib hydrochlorideMus musculus (house mouse)IC500.040011
sorafenibMus musculus (house mouse)IC500.130011
plx4032Mus musculus (house mouse)IC500.030011