A role played by a substance that can react readily with, and thereby eliminate, radicals.
| Member | Definition | Class |
|---|
| (E)-5-hydroxy-6-(3-methylbut-2-enyl)-2-(pent-1-enyl)benzofuran-4-carbaldehyde | A member of the class of 1-benzofurans that is 1-benzofuran substituted by a hydroxy group at position 5, a prenyl group at position 6 and a pent-1-en-1-yl group at position 2. Isolated from Chaetomium globosum, it exhibits radical scavenging activity. | (E)-5-hydroxy-6-(3-methylbut-2-enyl)-2-(pent-1-enyl)benzofuran-4-carbaldehyde |
| 1,2,3,4,6-pentakis-O-galloyl-beta-D-glucose | A galloyl-beta-D-glucose compound having five galloyl groups in the 1-, 2-, 3-, 4- and 6-positions. | 1,2,3,4,6-pentakis-O-galloyl-beta-D-glucose |
| 1,3-dihydroxy-4,4,5,5-tetramethyl-2-(4-carboxyphenyl)tetrahydroimidazole | A mmeber of the class of imidazolines and organic radical that is 4,4,5,5-tetramethyl-3-oxo-4,5-dihydro-1H-3lambda(5)-imidazol-1-yl]oxidanyl substituted at position 2 by a 4-carboxyphenyl group. | carboxy-PTIO |
| 2-naphthol | A naphthol carrying a hydroxy group at position 2. | 2-naphthol |
| 2',6'-dihydroxy-4'-methoxydihydrochalcone | A member of the class of dihydrochalcones that is dihydrochalcone substituted by hydroxy groups at positions 2' and 6' and a methoxy group at position 4' respectively. | 2',6'-dihydroxy-4'-methoxydihydrochalcone |
| 4-maleimido-2,2,6,6-tetramethylpiperidinooxyl | A member of the class of piperidines that is TEMPO carrying a maleimido group at position 4. | 4-maleimido-TEMPO |
| 6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid | A chromanol that is 6-hydroxychromane which is substituted by a carboxy group at position 2 and by methyl groups at positions 2, 5, 7, and 8. A cell-permeable, water-soluble analogue of vitamin E, it is used as a standard for measuring the antioxidant capacity of complex mixtures. | Trolox |
| 6,6'-bieckol | A phlorotanin that is 1,1'-bioxanthrene substituted by 3,5-dihydroxyphenoxy groups at position 6 and 6' and hydroxy groups at positions 2, 2', 4, 4', 7, 7', 9 and 9' respectively. It is isolated from an edible marine brown alga Ecklonia cava and exhibits antioxidant activity. | 6,6'-bieckol |
| acetylcysteine | An N-acetyl-L-amino acid that is the N-acetylated derivative of the natural amino acid L-cysteine. | N-acetyl-L-cysteine |
| allopurinol | A bicyclic structure comprising a pyrazole ring fused to a hydroxy-substituted pyrimidine ring. | allopurinol |
| anthrone | A member of the class of anthracenes that is 9,10-dihydroanthracene carrying an oxo group at C-9. | anthrone |
| astilbin | A flavanone glycoside that is (+)-taxifolin substituted by a alpha-L-rhamnosyl moiety at position 3 via a glycosidic linkage. | astilbin |
| baicalein | A trihydroxyflavone with the hydroxy groups at positions C-5, -6 and -7. | baicalein |
| bendazac | A monocarboxylic acid that is glycolic acid in which the hydrogen attached to the 2-hydroxy group is replaced by a 1-benzyl-1H-indazol-3-yl group. Although it has anti-inflammatory, antinecrotic, choleretic and antilipidaemic properties and has been used for the treatment of various inflammatory skin disorders, its principal effect is to inhibit the denaturation of proteins. Its lysine salt is used in the management of cataracts. | bendazac |
| cupressuflavone | A biflavonoid that is obtained by oxidative coupling of two molecules of apigenin resulting in a bond between positions C-8 of the two chromene rings respectively. Isolated from Cupressus sempervirens and Juniperus occidentalis, it exhibits free radical scavenging and antielastase activities. | cupressuflavone |
| curcumin | A beta-diketone that is methane in which two of the hydrogens are substituted by feruloyl groups. A natural dyestuff found in the root of Curcuma longa. | curcumin |
| deanol | A tertiary amine that is ethanolamine having two N-methyl substituents. | N,N-dimethylethanolamine |
| demethylbellidifolin | A member of the class of xanthones that is xanthone which is substituted by hydroxy groups at positions 1, 3, 5, and 8. A natural product found particularly in Iris nigricans and Gentiana campestris. | bellidin |
| dieckol | A phlorotannin isolated from a brown alga Ecklonia cava which exhibits antioxidant, hepatoprotective and anticoagulant activities. | dieckol |
| dimethyl sulfoxide | A 2-carbon sulfoxide in which the sulfur atom has two methyl substituents. | dimethyl sulfoxide |
| diphenylamine | An aromatic amine containing two phenyl substituents. It has been used as a fungicide for the treatment of superficial scald in apples and pears, but is no longer approved for this purpose within the European Union. | diphenylamine |
| ebselen | A benzoselenazole that is 1,2-benzoselenazol-3-one carrying an additional phenyl substituent at position 2. Acts as a mimic of glutathione peroxidase. | ebselen |
| eckstolonol | A phlorotannin that is [1,4]benzodioxino[2,3-a]oxanthrene substituted by hydroxy groups at positions 1, 3, 6, 9 and 11. Isolated from the brown alga Ecklonia stolonifera, it exhibits radical scavenging activity. | eckstolonol |
| edaravone | A pyrazolone that is 2,4-dihydro-3H-pyrazol-3-one which is substituted at positions 2 and 5 by phenyl and methyl groups, respectively. | edaravone |
| eriodictyol 7-O-beta-D-glucopyranoside | A flavanone glycoside that is eriodictyol attached to a beta-D-glucopyranosyl residue at position 7 via a glycosidic linkage. It is an Nrf2 activator and provides protection against cisplatin-induced toxicity. | eriodictyol 7-O-beta-D-glucopyranoside |
| ferrostatin-1 | An ethyl ester resulting from the formal condensation of the carboxy group of 3-amino-4-(cyclohexylamino)benzoic acid with ethanol. It is a potent inhibitor of ferroptosis, a distinct non-apoptotic form of cell death caused by lipid peroxidation. It is also a radical-trapping antioxidant and has the ability to reduce the accumulation of lipid peroxides and chain-carrying peroxyl radicals. | ferrostatin-1 |
| gallocatechol | A gallocatechin that has (2R,3S)-configuration. It is found in green tea and bananas. | (+)-gallocatechin |
| ginsenoside rb1 | A ginsenoside found in Panax ginseng and Panax japonicus var. major that is ginsenoside Rd in which the beta-D-glucopyranoside group at position 20 is replaced by a beta-D-glucopyranosyl-beta-D-glucopyranoside group. | ginsenoside Rb1 |
| gliclazide | | gliclazide |
| homoorientin | A flavone C-glycoside consisting of luteolin having a beta-D-glucosyl residue at the 6-position. | isoorientin |
| hydroxyurea | A member of the class of ureas that is urea in which one of the hydrogens is replaced by a hydroxy group. An antineoplastic used in the treatment of chronic myeloid leukaemia as well as for sickle-cell disease. | hydroxyurea |
| ibuprofen | A monocarboxylic acid that is propionic acid in which one of the hydrogens at position 2 is substituted by a 4-(2-methylpropyl)phenyl group. | ibuprofen |
| kaempferol 7-o-glucoside | A kaempferol O-glucoside that is kaempferol attached to a beta-D-glucopyranosyl moiety at position 7 via a glycosidic linkage. | kaempferol 7-O-beta-D-glucopyranoside |
| kaempferol-3-o-rutinoside | A kaempferol O-glucoside that is kaempferol attached to a rutinosyl [6-deoxy-alpha-L-mannosyl-(1->6)-beta-D-glucosyl] residue at position 3 via a glycosidic linkage. It has been isolated from the leaves of Solanum campaniforme. | kaempferol-3-rutinoside |
| ladanein | A dimethoxyflavone that is scutellarein in which the hydroxy groups at positions 4' and 7 are replaced by methoxy groups. It is an effective anti-HCV agent. | ladanein |
| liproxstatin-1 | An azaspiro compound that is 1'H-spiro[piperidine-4,2'-quinoxaline] in which the hydrogen at position 3' is replaced by a (3-chlorobenzyl)amino group. It is a potent inhibitor of ferroptosis. | liproxstatin-1 |
| luteolin | A tetrahydroxyflavone in which the four hydroxy groups are located at positions 3', 4', 5 and 7. It is thought to play an important role in the human body as an antioxidant, a free radical scavenger, an anti-inflammatory agent and an immune system modulator as well as being active against several cancers. | luteolin |
| matteucinol | A dihydroxyflavanone that is (2S)-flavanone with hydroxy groups at positions 5 and 7, methyl groups at positions 6 and 8 and a methoxy group at position 4'. | matteucinol |
| melatonin | A member of the class of acetamides that is acetamide in which one of the hydrogens attached to the nitrogen atom is replaced by a 2-(5-methoxy-1H-indol-3-yl)ethyl group. It is a hormone secreted by the pineal gland in humans. | melatonin |
| methyl brevifolincarboxylate | An organic heterotricyclic compound that is 1,2,3,5-tetrahydrocyclopenta[c]isochromene substituted by hydroxy groups at positions 7, 8 and 9, oxo groups at positions 3 and 5 and a methoxycarbonyl group at position 1. Isolated from Phyllanthus urinaria and Phyllanthus niruri, it exhibits vasorelaxant activity. | methyl brevifolincarboxylate |
| n-(1-oxyl-2,2,6,6-tetramethyl-4-piperidinyl)iodoacetamide | A piperidinecarboxamide that is TEMPO carrying an 2-iodoacetamido group at position 4. | 4-(2-iodacetamido)-TEMPO |
| nigerloxin | A member of the class of benzoic acids that is benzoic acid which is substituted at positions 2, 3, 4, 5, and 6 by carbamoyl, hydroxy, E)-prop-1-en-1-yl, methyl, and methoxy groups, respectively. Obtained from solid-state fermentation of Aspergillus niger CFR-W-105, it inhibits soy bean lipoxygenase-1 (LOX-1) and rat lens aldose reductase (RLAR). It also shows free radical scavenging activity. | nigerloxin |
| nymphaeol c | A tetrahydroxyflavanone that is (2S)-flavanone substituted by hydroxy group at positions 5, 7, 3' and 4', a geranyl group at position 2' and a prenyl group at position 6. Isolated from Macaranga tanarius and propolis collected in Okinawa, it exhibits radical scavenging activity. | nymphaeol C |
| oleuropein | A secoiridoid glycoside that is the methyl ester of 3,4-dihydro-2H-pyran-5-carboxylic acid which is substituted at positions 2, 3, and 4 by hydroxy, ethylidene, and carboxymethyl groups, respectively and in which the anomeric hydroxy group at position 2 has been converted into its beta-D-glucoside and the carboxylic acid moiety of the carboxymethyl substituent has been converted to the corresponding 3,4-dihydroxyphenethyl ester (the 2S,3E,4S stereoisomer). The most important phenolic compound present in olive cultivars. | oleuropein |
| orobol | A member of the class of 7-hydroxyisoflavones which consists of isoflavone substituted by hydroxy groups at positions 5, 7, 3' and 4'. It has been isolated from the mycelia of Cordyceps sinensis. | orobol |
| ovothiol a | A L-histidine derivative that is L-histidine substituted at positions N3 and C5 on the imidazole ring by methyl and mercapto groups respectively. | ovothiol A zwitterion; ovothiol A |
| ovothiol c | A L-histidine derivative that is N,N-dimethyl-L-histidine substituted at positions N3 and C5 on the imidazole ring by methyl and mercapto groups respectively. | ovothiol C zwitterion; ovothiol C |
| phenothiazine | The 10H-tautomer of phenothiazine. | 10H-phenothiazine |
| phenoxazine | A member of the class of phenoxazines that is morpholine which is ortho-fused to two benzene rings at positions 2-3 and 5-6. | 10H-phenoxazine |
| potassium iodide | A metal iodide salt with a K(+) counterion. It is a scavenger of hydroxyl radicals. | potassium iodide |
| pramipexole | A member of the class of benzothiazoles that is 4,5,6,7-tetrahydro-1,3-benzothiazole in which the hydrogens at the 2 and 6-pro-S-positions are substituted by amino and propylamino groups, respectively. | pramipexole |
| propofol | A phenol resulting from the formal substitution of the hydrogen at the 2 position of 1,3-diisopropylbenzene by a hydroxy group. | propofol |
| propolin c | A tetrahydroxyflavanone that is (2S)-flavanone substituted by hydroxy group at positions 5, 7, 3' and 4' and a geranyl group at position 6. Isolated from Macaranga tanarius and propolis collected in Okinawa, it exhibits radical scavenging activity. | nymphaeol A |
| proxyl nitroxide | | PROXYL |
| pterostilbene | A stilbenol that consists of trans-stilbene bearing a hydroxy group at position 4 as well as two methoxy substituents at positions 3' and 5'. | pterostilbene |
| pyrrolidine dithiocarbamate | A member of the class of dithiocarbamic acids that is the N-dithiocarboxy derivative of pyrrolidine. | pyrrolidine dithiocarbamate |
| quercetin | A pentahydroxyflavone having the five hydroxy groups placed at the 3-, 3'-, 4'-, 5- and 7-positions. It is one of the most abundant flavonoids in edible vegetables, fruit and wine. | quercetin |
| resveratrol | A resveratrol in which the double bond has E configuration. | trans-resveratrol |
| rosiglitazone | A coumarin substituted by a methyl group at position 4 and by acetyloxy groups at positions 7 and 8. It exhibits strong antioxidant and radical scavenging properties. | 7,8-diacetoxy-4-methylcoumarin |
| sigmoidin a | A tetrahydroxyflavanone that is (2S)-flavanone substituted by hydroxy groups at positions 5, 7, 3' and 4' and prenyl groups at positions 2' and 5'. Isolated from Erythrina sigmoidea, it exhibits anti-inflammatory and antioxidant activities. | sigmoidin A |
| silychristin | A flavonolignan isolated from Silybum marianum and has been shown to exhibit inhibitory activities against lipoxygenase and prostaglandin synthetase. | silychristin |
| sugiol | An abietane diterpenoid that is ferruginol in which the methylene group para to the phenolic hydroxy group has been substituted by an oxo group. | sugiol |
| taurine | An amino sulfonic acid that is the 2-amino derivative of ethanesulfonic acid. It is a naturally occurring amino acid derived from methionine and cysteine metabolism. An abundant component of fish- and meat-based foods, it has been used as an oral supplement in the treatment of disorders such as cystic fibrosis and hypertension. | taurine zwitterion; taurine |
| tempace | A piperidinecarboxamide that is TEMPO carrying an acetamido group at position 4. | 4-acetamido-TEMPO |
| tempo | A member of the class of aminoxyls that is piperidine that carries an oxidanediyl group at position 1 and methyl groups at positions 2, 2, 6, and 6, respectively. | TEMPO |
| tempo carboxylic acid | A member of the class of aminoxyls that is TEMPO carrying a carboxy group at position 4. | 4-carboxy-TEMPO |
| tempol | A member of the class of aminoxyls that is TEMPO carrying a hydroxy substituent at position 4. It is a radical scavenger which exhibits anti-inflammatory and analgesic properties. | 4-hydroxy-TEMPO |
| triacetoneamine-n-oxyl | A member of the class of aminoxyls that is TEMPO carrying an oxo group at position 4. | 4-oxo-TEMPO |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 16.0888 | 1 | 19 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 4.2120 | 1 | 10 |
| 2,3-bisphosphoglycerate-independent phosphoglycerate mutase | Leishmania major strain Friedlin | Potency | 7.5686 | 1 | 1 |
| 67.9K protein | Vaccinia virus | Potency | 17.3932 | 2 | 6 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 51.6351 | 4 | 11 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 20.5940 | 2 | 6 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 21.3376 | 1 | 28 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 38.3494 | 3 | 3 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 10.2284 | 1 | 5 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Potency | 16.3601 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 21.2804 | 1 | 2 |
| AR protein | Homo sapiens (human) | Potency | 20.7265 | 12 | 88 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 31.2570 | 3 | 36 |
| arylsulfatase A | Homo sapiens (human) | Potency | 16.1246 | 1 | 5 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 12.7265 | 4 | 13 |
| Ataxin-2 | Homo sapiens (human) | Potency | 16.2713 | 2 | 7 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 10.2171 | 5 | 13 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 21.1329 | 2 | 10 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 6.7456 | 1 | 1 |
| atrial natriuretic peptide receptor 2 precursor | Homo sapiens (human) | Potency | 23.4354 | 1 | 2 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 30.7324 | 3 | 24 |
| BRCA1 | Homo sapiens (human) | Potency | 17.5235 | 1 | 5 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 42.5356 | 1 | 5 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 44.2412 | 1 | 7 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 23.7358 | 1 | 2 |
| caspase-3 | Homo sapiens (human) | Potency | 44.2412 | 1 | 7 |
| Caspase-7 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 40.8275 | 3 | 24 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 10.9817 | 2 | 13 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 15.3370 | 1 | 24 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 8.2654 | 4 | 17 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 33.4836 | 2 | 5 |
| Chain A, Breast cancer type 1 susceptibility protein | Homo sapiens (human) | Potency | 5.0119 | 1 | 3 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 26.0843 | 2 | 8 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 16.5203 | 3 | 5 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 11.9424 | 2 | 23 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 54.8787 | 1 | 9 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 7.0433 | 3 | 26 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 16.3695 | 3 | 12 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 21.5381 | 1 | 18 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 11.9424 | 2 | 23 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 32.2288 | 2 | 7 |
| ClpP | Bacillus subtilis | Potency | 28.3085 | 1 | 3 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 13.4400 | 1 | 7 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 10.5076 | 1 | 7 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 14.8924 | 1 | 4 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 18.5250 | 1 | 4 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 22.2399 | 1 | 7 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 18.7851 | 2 | 32 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 11.8160 | 2 | 10 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 35.2905 | 1 | 17 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 10.1786 | 3 | 5 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 3.6898 | 1 | 1 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | Potency | 16.1269 | 1 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3F isoform a | Homo sapiens (human) | Potency | 28.9342 | 1 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 27.2454 | 2 | 3 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 31.4839 | 1 | 6 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 11.6211 | 2 | 6 |
| DNA polymerase III, partial | Bacillus subtilis | Potency | 7.6828 | 1 | 2 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 37.2992 | 2 | 16 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 13.3188 | 1 | 24 |
| dopamine D1 receptor | Homo sapiens (human) | Potency | 0.0206 | 1 | 1 |
| endonuclease IV | Escherichia coli | Potency | 7.9433 | 1 | 1 |
| Endothelin receptor type B | Rattus norvegicus (Norway rat) | Potency | 20.0850 | 1 | 2 |
| Endothelin-1 receptor | Rattus norvegicus (Norway rat) | Potency | 20.0850 | 1 | 2 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 29.7695 | 12 | 104 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 25.8927 | 3 | 17 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 25.1106 | 10 | 85 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 11.9998 | 1 | 23 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 15.3085 | 4 | 23 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 29.8564 | 4 | 12 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 35.1983 | 2 | 16 |
| fructose-bisphosphate aldolase A | Oryctolagus cuniculus (rabbit) | Potency | 22.3872 | 1 | 1 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 31.7859 | 1 | 2 |
| G | Vesicular stomatitis virus | Potency | 14.8924 | 1 | 4 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| galactokinase | Homo sapiens (human) | Potency | 44.6988 | 1 | 2 |
| GALC protein | Homo sapiens (human) | Potency | 0.5623 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 18.7851 | 1 | 16 |
| geminin | Homo sapiens (human) | Potency | 11.0739 | 5 | 27 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 25.4807 | 3 | 28 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 14.9776 | 2 | 4 |
| GLS protein | Homo sapiens (human) | Potency | 15.3849 | 2 | 13 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 29.0621 | 1 | 14 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 21.1406 | 4 | 19 |
| glucokinase regulatory protein | Homo sapiens (human) | Potency | 18.2563 | 1 | 2 |
| Glutamate receptor 1 | Rattus norvegicus (Norway rat) | Potency | 0.6310 | 1 | 1 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 40.6088 | 2 | 8 |
| Glutamate receptor 3 | Rattus norvegicus (Norway rat) | Potency | 0.6310 | 1 | 1 |
| Glutamate receptor 4 | Rattus norvegicus (Norway rat) | Potency | 0.6310 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2D | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3A | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3B | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Glycoprotein hormones alpha chain | Homo sapiens (human) | Potency | 5.0119 | 1 | 1 |
| GTP-binding nuclear protein Ran isoform 1 | Homo sapiens (human) | Potency | 42.8000 | 1 | 2 |
| Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 42.8000 | 1 | 2 |
| guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 16.3577 | 2 | 5 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 34.8731 | 2 | 5 |
| hemoglobin subunit beta | Homo sapiens (human) | Potency | 35.7168 | 2 | 2 |
| hexokinase-4 isoform 1 | Homo sapiens (human) | Potency | 18.2563 | 1 | 2 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 9.9788 | 2 | 43 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 0.4496 | 1 | 4 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 10.3265 | 2 | 12 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 57.1732 | 2 | 22 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 42.5765 | 1 | 4 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 14.8924 | 1 | 4 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 13.7560 | 2 | 3 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 15.2028 | 4 | 6 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 35.8690 | 2 | 4 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 12.4208 | 2 | 14 |
| IDH1 | Homo sapiens (human) | Potency | 25.7676 | 1 | 7 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 51.9700 | 2 | 6 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 14.8923 | 1 | 8 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 12.8342 | 1 | 6 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 12.3175 | 1 | 6 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 12.3175 | 1 | 6 |
| Interferon beta | Homo sapiens (human) | Potency | 17.0911 | 2 | 10 |
| interleukin 8 | Homo sapiens (human) | Potency | 77.2652 | 1 | 4 |
| isocitrate dehydrogenase 1, partial | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 9.7663 | 2 | 16 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 6.2481 | 1 | 9 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 23.7358 | 1 | 2 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 29.5493 | 4 | 25 |
| luciferase | Photuris pensylvanica (Pennsylania firefly) | Potency | 18.0789 | 3 | 5 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 28.7737 | 1 | 6 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 9.6305 | 1 | 5 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 10.9403 | 2 | 38 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 36.5355 | 2 | 5 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 10.7100 | 2 | 5 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 26.2185 | 1 | 6 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 3.4916 | 1 | 3 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 5.2131 | 2 | 10 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 6.1188 | 1 | 3 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 8.8306 | 1 | 3 |
| Nrf2 | Homo sapiens (human) | Potency | 25.3935 | 2 | 4 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 31.2307 | 4 | 30 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 20.5962 | 1 | 1 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 35.1177 | 1 | 5 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 38.2509 | 1 | 4 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 19.0289 | 4 | 40 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 31.5965 | 3 | 42 |
| Ornithine decarboxylase | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 1 |
| P53 | Homo sapiens (human) | Potency | 39.1512 | 1 | 2 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 76.4710 | 1 | 4 |
| Parkin | Homo sapiens (human) | Potency | 9.2296 | 3 | 4 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 28.9055 | 2 | 5 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 22.9558 | 1 | 4 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 51.3601 | 1 | 5 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 30.5475 | 5 | 19 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 36.1777 | 5 | 14 |
| phosphoglycerate kinase | Trypanosoma brucei brucei TREU927 | Potency | 17.8762 | 2 | 2 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 36.9545 | 1 | 18 |
| PINK1 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 10.0693 | 2 | 7 |
| polyprotein | Zika virus | Potency | 31.7859 | 1 | 2 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 9.9264 | 1 | 10 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 9.4740 | 1 | 11 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 12.5558 | 1 | 5 |
| PPM1D protein | Homo sapiens (human) | Potency | 18.5569 | 1 | 4 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 44.0007 | 3 | 27 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 45.3915 | 1 | 3 |
| progesterone receptor | Homo sapiens (human) | Potency | 24.6995 | 2 | 16 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 16.1889 | 5 | 7 |
| pyruvate kinase PKM isoform a | Homo sapiens (human) | Potency | 12.8072 | 4 | 6 |
| pyruvate kinase PKM isoform b | Homo sapiens (human) | Potency | 10.0000 | 2 | 2 |
| Rap guanine nucleotide exchange factor 3 | Homo sapiens (human) | Potency | 38.1456 | 1 | 2 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 20.5668 | 2 | 22 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 10.2723 | 1 | 5 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 7.3130 | 1 | 8 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 32.9808 | 3 | 45 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 1,129.4180 | 4 | 18 |
| RGS12 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 15.7483 | 3 | 4 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 2.9935 | 1 | 1 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | Potency | 5.7988 | 1 | 1 |
| signal transducer and activator of transcription 6, interleukin-4 induced | Homo sapiens (human) | Potency | 2.5119 | 2 | 2 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 31.1085 | 2 | 7 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 31.1085 | 2 | 7 |
| Smad3 | Homo sapiens (human) | Potency | 25.3460 | 1 | 6 |
| snurportin-1 | Homo sapiens (human) | Potency | 51.9700 | 2 | 6 |
| Sodium channel protein type 1 subunit alpha | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Sodium channel protein type 2 subunit alpha | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Sodium channel protein type 3 subunit alpha | Rattus norvegicus (Norway rat) | Potency | 5.7988 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 25.1189 | 1 | 1 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 13.1384 | 1 | 10 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 23.3352 | 1 | 5 |
| TDP1 protein | Homo sapiens (human) | Potency | 16.7125 | 2 | 58 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 42.2395 | 1 | 2 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 23.3035 | 4 | 15 |
| Thrombopoietin | Homo sapiens (human) | Potency | 17.3926 | 2 | 4 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 37.8758 | 3 | 27 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 49.7592 | 4 | 9 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 28.5762 | 5 | 31 |
| thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 27.7247 | 1 | 1 |
| transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 9.2878 | 1 | 3 |
| transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| tumor susceptibility gene 101 protein | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 15.4103 | 1 | 1 |
| ubiquitin carboxyl-terminal hydrolase 2 isoform a | Homo sapiens (human) | Potency | 16.9155 | 2 | 3 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 10.0693 | 2 | 7 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 10.0693 | 2 | 7 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 25.0514 | 2 | 11 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 39.0320 | 2 | 19 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 19.3056 | 5 | 11 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 20.0725 | 1 | 7 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 46.3199 | 1 | 7 |
| WRN | Homo sapiens (human) | Potency | 6.1212 | 2 | 3 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a | Homo sapiens (human) | IC50 | 5.9775 | 2 | 4 |
| 1-deoxy-D-xylulose 5-phosphate reductoisomerase | Escherichia coli K-12 | IC50 | 2.5000 | 1 | 3 |
| 10 kDa chaperonin | Escherichia coli | IC50 | 3.0000 | 2 | 2 |
| 10 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| 17-beta-hydroxysteroid dehydrogenase type 2 | Homo sapiens (human) | IC50 | 1.6033 | 2 | 3 |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 4.7000 | 1 | 2 |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 1.3000 | 2 | 2 |
| 4-aminobutyrate aminotransferase, mitochondrial | Homo sapiens (human) | IC50 | 12,800.0000 | 1 | 1 |
| 4-aminobutyrate aminotransferase, mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 1.1000 | 1 | 2 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 4.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 6.5140 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Homo sapiens (human) | Ki | 3.5080 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1E | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | Ki | 3.9000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | IC50 | 5.4990 | 1 | 1 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | Ki | 3.4990 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | IC50 | 6.8945 | 1 | 2 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 3.6110 | 1 | 2 |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | IC50 | 6.8945 | 1 | 2 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | Ki | 3.6110 | 1 | 2 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | IC50 | 350.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 1.1880 | 1 | 1 |
| 5-lipoxygenase | Bos taurus (cattle) | IC50 | 2.0000 | 1 | 1 |
| 5'-nucleotidase | Homo sapiens (human) | IC50 | 10.5400 | 1 | 1 |
| 5'-nucleotidase | Mus musculus (house mouse) | IC50 | 100.0000 | 1 | 1 |
| 5'-nucleotidase | Rattus norvegicus (Norway rat) | Ki | 0.0453 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli K-12 | IC50 | 250.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli | IC50 | 3.0000 | 2 | 2 |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| 72 kDa type IV collagenase | Homo sapiens (human) | IC50 | 5.1450 | 1 | 2 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | IC50 | 264.0540 | 5 | 5 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 494.3233 | 7 | 9 |
| Acetylcholinesterase | Homo sapiens (human) | Ki | 37.5000 | 2 | 3 |
| Acetylcholinesterase | Bos taurus (cattle) | IC50 | 0.1000 | 2 | 3 |
| Acid-sensing ion channel 1 | Rattus norvegicus (Norway rat) | IC50 | 288.0192 | 5 | 9 |
| Acid-sensing ion channel 3 | Rattus norvegicus (Norway rat) | IC50 | 512.8610 | 1 | 1 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | IC50 | 1,030.0000 | 1 | 1 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | Ki | 8.9000 | 3 | 3 |
| Adenosine receptor A2a | Rattus norvegicus (Norway rat) | IC50 | 1,030.0000 | 1 | 1 |
| Adenosine receptor A2a | Rattus norvegicus (Norway rat) | Ki | 5.1250 | 2 | 2 |
| Adenosine receptor A3 | Homo sapiens (human) | IC50 | 25.6400 | 1 | 1 |
| Adenosine receptor A3 | Homo sapiens (human) | Ki | 22.2460 | 2 | 2 |
| ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 | Homo sapiens (human) | IC50 | 48.7000 | 1 | 3 |
| Albumin | Bos taurus (cattle) | IC50 | 3.0000 | 1 | 1 |
| Albumin | Homo sapiens (human) | Ki | 165,959,000,000.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member A1 | Rattus norvegicus (Norway rat) | IC50 | 2.3200 | 1 | 1 |
| Aldo-keto reductase family 1 member A1 | Sus scrofa (pig) | IC50 | 38.4000 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Bos taurus (cattle) | IC50 | 14.1563 | 5 | 7 |
| Aldo-keto reductase family 1 member B1 | Homo sapiens (human) | IC50 | 2.1356 | 8 | 8 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 7.4880 | 8 | 12 |
| Aldo-keto reductase family 1 member B1 | Sus scrofa (pig) | IC50 | 50.1000 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 4.0220 | 1 | 3 |
| Aldo-keto reductase family 1 member B10 | Homo sapiens (human) | IC50 | 58.5000 | 2 | 2 |
| Aldo-keto reductase family 1 member C1 | Homo sapiens (human) | IC50 | 300.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member C2 | Homo sapiens (human) | IC50 | 1,000.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member C21 | Mus musculus (house mouse) | IC50 | 6.9000 | 1 | 1 |
| Aldo-keto reductase family 1 member C21 | Mus musculus (house mouse) | Ki | 11.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member C3 | Homo sapiens (human) | IC50 | 20.8733 | 3 | 3 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | IC50 | 3.3200 | 1 | 1 |
| alkaline phosphatase, germ cell type preproprotein | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| alkaline phosphatase, intestinal | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| alkaline phosphatase, tissue-nonspecific isozyme isoform 1 preproprotein | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 10.3468 | 3 | 3 |
| Alpha-1A adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 14.4920 | 1 | 1 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 27.7100 | 3 | 4 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 14.4920 | 1 | 1 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 5.4000 | 1 | 1 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 0.0757 | 1 | 1 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 0.0677 | 1 | 1 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | Ki | 0.0522 | 1 | 1 |
| Alpha-amylase 1A | Homo sapiens (human) | IC50 | 16.3900 | 3 | 5 |
| Alpha-amylase 1A | Homo sapiens (human) | Ki | 2.6000 | 1 | 1 |
| Alpha-glucosidase MAL12 | Saccharomyces cerevisiae S288C | Ki | 21.5000 | 1 | 1 |
| Alpha-synuclein | Homo sapiens (human) | IC50 | 36.1600 | 4 | 7 |
| Alpha-synuclein | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 5.8032 | 11 | 13 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | Ki | 0.7100 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Bos taurus (cattle) | IC50 | 0.0100 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Bos taurus (cattle) | IC50 | 20.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | IC50 | 29.1989 | 8 | 9 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | Ki | 21.5000 | 1 | 1 |
| Aminopeptidase N | Homo sapiens (human) | IC50 | 15.5000 | 1 | 1 |
| Aminopeptidase N | Sus scrofa (pig) | IC50 | 15.5000 | 1 | 1 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 13.6169 | 40 | 48 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | IC50 | 290.0000 | 2 | 2 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | IC50 | 0.6700 | 1 | 1 |
| Anthrax toxin receptor 2 | Homo sapiens (human) | IC50 | 100.3023 | 2 | 3 |
| Arginase | Leishmania amazonensis | IC50 | 4.0000 | 1 | 1 |
| Aromatase | Homo sapiens (human) | IC50 | 22.7413 | 8 | 9 |
| Aromatase | Homo sapiens (human) | Ki | 41.6700 | 1 | 1 |
| Arrestin, beta 1 | Homo sapiens (human) | IC50 | 1.5240 | 1 | 1 |
| Aryl hydrocarbon receptor | Oryctolagus cuniculus (rabbit) | Ki | 0.3743 | 2 | 3 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 6 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 43.0200 | 3 | 5 |
| Aurora kinase B | Homo sapiens (human) | IC50 | 3.2025 | 2 | 4 |
| B2 bradykinin receptor | Cavia porcellus (domestic guinea pig) | IC50 | 4.0000 | 2 | 2 |
| Bcl-2-like protein 1 | Homo sapiens (human) | IC50 | 190.0000 | 1 | 1 |
| Beta lactamase (plasmid) | Pseudomonas aeruginosa | IC50 | 7.7510 | 1 | 1 |
| Beta-2 adrenergic receptor | Homo sapiens (human) | Ki | 55.0000 | 2 | 2 |
| Beta-3 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 3.2500 | 1 | 2 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 11.5000 | 1 | 1 |
| Beta-lactamase | Enterobacter cloacae | IC50 | 269.6667 | 3 | 3 |
| Beta-lactamase | Escherichia coli K-12 | IC50 | 58.0000 | 4 | 4 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 43.3044 | 7 | 9 |
| Beta-secretase 1 | Homo sapiens (human) | Ki | 7.1575 | 2 | 4 |
| Bifunctional epoxide hydrolase 2 | Homo sapiens (human) | IC50 | 7.2617 | 6 | 6 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 343.7600 | 5 | 15 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | IC50 | 645.4500 | 1 | 2 |
| Breakpoint cluster region protein | Homo sapiens (human) | IC50 | 19.0000 | 1 | 2 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 6.2575 | 4 | 4 |
| C-C chemokine receptor type 4 | Homo sapiens (human) | IC50 | 47.2409 | 3 | 6 |
| C-X-C chemokine receptor type 1 | Homo sapiens (human) | IC50 | 35.3780 | 2 | 4 |
| Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B | Rattus norvegicus (Norway rat) | IC50 | 275.0000 | 1 | 1 |
| Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C | Rattus norvegicus (Norway rat) | IC50 | 275.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Calmodulin-1 | Homo sapiens (human) | IC50 | 12.9700 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 6 |
| Cannabinoid receptor 1 | Homo sapiens (human) | IC50 | 24.8570 | 1 | 1 |
| Cannabinoid receptor 1 | Mus musculus (house mouse) | IC50 | 1,000.0000 | 1 | 2 |
| Cannabinoid receptor 1 | Homo sapiens (human) | Ki | 19.6240 | 1 | 1 |
| Carbonic anhydrase 1 | Homo sapiens (human) | Ki | 41.4475 | 8 | 16 |
| Carbonic anhydrase 12 | Homo sapiens (human) | Ki | 3.4668 | 3 | 3 |
| Carbonic anhydrase 13 | Homo sapiens (human) | Ki | 4.0900 | 1 | 1 |
| Carbonic anhydrase 13 | Mus musculus (house mouse) | Ki | 9.0300 | 1 | 1 |
| Carbonic anhydrase 14 | Homo sapiens (human) | Ki | 3.1200 | 2 | 2 |
| Carbonic anhydrase 15 | Mus musculus (house mouse) | Ki | 9.3600 | 1 | 1 |
| Carbonic anhydrase 2 | Homo sapiens (human) | Ki | 1,547.4042 | 9 | 17 |
| Carbonic anhydrase 3 | Bos taurus (cattle) | Ki | 5.0411 | 2 | 9 |
| Carbonic anhydrase 3 | Homo sapiens (human) | Ki | 8.5950 | 2 | 2 |
| Carbonic anhydrase 4 | Homo sapiens (human) | Ki | 17.9302 | 7 | 14 |
| Carbonic anhydrase 5A, mitochondrial | Homo sapiens (human) | Ki | 6,260.6400 | 4 | 4 |
| Carbonic anhydrase 5B, mitochondrial | Homo sapiens (human) | Ki | 8.2700 | 2 | 2 |
| Carbonic anhydrase 6 | Homo sapiens (human) | Ki | 5.9900 | 3 | 3 |
| Carbonic anhydrase 7 | Homo sapiens (human) | Ki | 3.0649 | 3 | 3 |
| Carbonic anhydrase 9 | Homo sapiens (human) | Ki | 1,757.7025 | 4 | 4 |
| Carboxylic ester hydrolase | Equus caballus (horse) | IC50 | 0.7500 | 2 | 2 |
| Carboxylic ester hydrolase | Equus caballus (horse) | Ki | 1.2000 | 1 | 1 |
| Casein kinase II subunit alpha | Homo sapiens (human) | IC50 | 2.4688 | 5 | 8 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Ki | 1.1800 | 4 | 4 |
| Casein kinase II subunit alpha 3 | Homo sapiens (human) | IC50 | 3.6833 | 1 | 3 |
| Casein kinase II subunit alpha 3 | Homo sapiens (human) | Ki | 1.1800 | 1 | 1 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | IC50 | 2.3056 | 6 | 9 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Ki | 1.1800 | 1 | 1 |
| Casein kinase II subunit beta | Homo sapiens (human) | IC50 | 2.3056 | 6 | 9 |
| Casein kinase II subunit beta | Homo sapiens (human) | Ki | 1.1800 | 1 | 1 |
| Caspase-1 | Homo sapiens (human) | IC50 | 18.3680 | 2 | 5 |
| Caspase-3 | Homo sapiens (human) | IC50 | 21.9500 | 1 | 4 |
| Caspase-4 | Homo sapiens (human) | IC50 | 21.9500 | 1 | 4 |
| Caspase-5 | Homo sapiens (human) | IC50 | 21.9500 | 1 | 4 |
| Caspase-9 | Homo sapiens (human) | IC50 | 21.9500 | 1 | 4 |
| Cathepsin D | Homo sapiens (human) | IC50 | 138.0000 | 1 | 1 |
| cathepsin L1 | Homo sapiens (human) | IC50 | 59.6420 | 1 | 1 |
| Cationic trypsin | Bos taurus (cattle) | IC50 | 26.2333 | 2 | 6 |
| CDGSH iron-sulfur domain-containing protein 1 | Homo sapiens (human) | IC50 | 2.3600 | 1 | 1 |
| CDGSH iron-sulfur domain-containing protein 1 | Homo sapiens (human) | Ki | 0.1010 | 1 | 1 |
| Cereblon isoform 4 | Magnetospirillum gryphiswaldense | IC50 | 20.8000 | 1 | 1 |
| Cereblon isoform 4 | Magnetospirillum gryphiswaldense | Ki | 5,570.2333 | 3 | 3 |
| cGMP-dependent 3',5'-cyclic phosphodiesterase | Rattus norvegicus (Norway rat) | IC50 | 81.3000 | 1 | 1 |
| Chain A, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase | Helicobacter pylori | Ki | 12.7000 | 1 | 3 |
| Chain A, APH(2')-Id | Enterococcus casseliflavus | Ki | 25.1000 | 1 | 1 |
| Chain A, Casein kinase II subunit alpha | Zea mays | IC50 | 0.3500 | 1 | 3 |
| Chain A, Leukotriene A-4 hydrolase | Homo sapiens (human) | IC50 | 212.0000 | 1 | 17 |
| Chain A, RNA-directed RNA polymerase NS5 | Dengue virus 2 16681-PDK53 | IC50 | 35.0600 | 1 | 1 |
| Chain B, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase | Helicobacter pylori | Ki | 12.7000 | 1 | 3 |
| Chemotaxis protein CheA | Escherichia coli K-12 | IC50 | 111.0000 | 1 | 1 |
| Choline O-acetyltransferase | Rattus norvegicus (Norway rat) | IC50 | 200.0000 | 1 | 1 |
| Choline O-acetyltransferase | Rattus norvegicus (Norway rat) | Ki | 25,000.0000 | 1 | 1 |
| Cholinesterase | Equus caballus (horse) | IC50 | 180.2370 | 4 | 4 |
| Cholinesterase | Homo sapiens (human) | IC50 | 122.0400 | 3 | 5 |
| Chymotrypsin-C | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Chymotrypsin-like elastase family member 1 | Sus scrofa (pig) | IC50 | 28.7500 | 1 | 4 |
| Chymotrypsinogen A | Bos taurus (cattle) | IC50 | 292.5000 | 2 | 2 |
| Chymotrypsinogen B | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Coagulation factor X | Homo sapiens (human) | IC50 | 0.1700 | 1 | 1 |
| Coagulation factor X | Homo sapiens (human) | Ki | 0.5700 | 1 | 1 |
| Collagenase 3 | Homo sapiens (human) | IC50 | 9.2550 | 1 | 2 |
| CREB-binding protein | Homo sapiens (human) | IC50 | 25.0000 | 4 | 4 |
| Cruzipain | Trypanosoma cruzi | IC50 | 91.5000 | 2 | 2 |
| Cyclin homolog | Herpesvirus saimiri (strain 11) | IC50 | 54.4875 | 1 | 8 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 21.3633 | 4 | 6 |
| Cyclin-dependent kinase 1 | Oryzias latipes (Japanese medaka) | IC50 | 54.4875 | 1 | 8 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 30.0000 | 1 | 2 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | IC50 | 61.0000 | 1 | 1 |
| Cyclin-dependent kinase 5 activator 1 | Homo sapiens (human) | IC50 | 39.3492 | 4 | 12 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | IC50 | 76.0900 | 2 | 10 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | IC50 | 39.3492 | 4 | 12 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Ki | 0.1700 | 1 | 2 |
| Cystathionine beta-synthase | Homo sapiens (human) | IC50 | 11.5000 | 1 | 1 |
| Cystathionine gamma-lyase | Homo sapiens (human) | IC50 | 400.0000 | 1 | 1 |
| Cysteine protease | Trypanosoma brucei rhodesiense | IC50 | 7.7500 | 1 | 1 |
| Cytochrome P450 11B1, mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 2 |
| Cytochrome P450 1A1 | Homo sapiens (human) | IC50 | 12.3812 | 8 | 9 |
| Cytochrome P450 1A1 | Homo sapiens (human) | Ki | 8.4638 | 4 | 8 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 9.6404 | 5 | 7 |
| Cytochrome P450 1A2 | Homo sapiens (human) | Ki | 12.0000 | 1 | 1 |
| Cytochrome P450 1A2 | Rattus norvegicus (Norway rat) | Ki | 0.0003 | 1 | 1 |
| Cytochrome P450 1B1 | Homo sapiens (human) | IC50 | 6.9326 | 8 | 9 |
| Cytochrome P450 1B1 | Homo sapiens (human) | Ki | 2.7817 | 8 | 11 |
| Cytochrome P450 2A5 | Mus musculus (house mouse) | IC50 | 77.9915 | 2 | 2 |
| Cytochrome P450 2A6 | Homo sapiens (human) | IC50 | 139.9795 | 2 | 2 |
| Cytochrome P450 2C11 | Rattus norvegicus (Norway rat) | Ki | 0.0003 | 1 | 1 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Cytochrome P450 2C8 | Homo sapiens (human) | IC50 | 13.5000 | 2 | 2 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 28.6667 | 3 | 3 |
| Cytochrome P450 2C9 | Homo sapiens (human) | Ki | 38.5000 | 2 | 2 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 20.0000 | 2 | 2 |
| Cytochrome P450 2D6 | Homo sapiens (human) | Ki | 0.0003 | 1 | 1 |
| Cytochrome P450 2J2 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 12.0833 | 6 | 6 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Ki | 20.0000 | 1 | 1 |
| Cytosol aminopeptidase | Sus scrofa (pig) | IC50 | 41.9500 | 1 | 2 |
| D | Bos taurus (cattle) | Ki | 20.0000 | 1 | 1 |
| D | Rattus norvegicus (Norway rat) | Ki | 50.0135 | 2 | 2 |
| D-amino-acid oxidase | Sus scrofa (pig) | IC50 | 1.0700 | 2 | 2 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(1B) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 1.0903 | 17 | 17 |
| D(2) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0390 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 0.0082 | 17 | 17 |
| D(3) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0006 | 2 | 2 |
| D(4) dopamine receptor | Homo sapiens (human) | Ki | 0.7548 | 9 | 11 |
| Death-associated protein kinase 1 | Homo sapiens (human) | IC50 | 49.9667 | 1 | 3 |
| Dehydrogenase/reductase SDR family member 9 | Homo sapiens (human) | IC50 | 1,000.0000 | 1 | 1 |
| Dehydrogenase/reductase SDR family member 9 | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Delta-type opioid receptor | Mus musculus (house mouse) | IC50 | 14.4000 | 1 | 1 |
| Delta-type opioid receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Dihydrofolate reductase | Homo sapiens (human) | Ki | 560.0000 | 1 | 1 |
| Dipeptidyl peptidase 3 | Homo sapiens (human) | IC50 | 48.0500 | 1 | 2 |
| Dipeptidyl peptidase 4 | Homo sapiens (human) | IC50 | 66.6081 | 2 | 5 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | IC50 | 25.3100 | 1 | 1 |
| DNA polymerase alpha catalytic subunit | Homo sapiens (human) | IC50 | 3.3000 | 1 | 1 |
| DNA topoisomerase 1 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| DNA topoisomerase 1 | Rattus norvegicus (Norway rat) | IC50 | 2.8300 | 2 | 2 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ectonucleoside triphosphate diphosphohydrolase 1 | Mus musculus (house mouse) | IC50 | 1.5600 | 1 | 1 |
| ELAV-like protein 1 | Homo sapiens (human) | IC50 | 1.4000 | 1 | 1 |
| ELAV-like protein 3 | Homo sapiens (human) | IC50 | 1.8000 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli K-12 | IC50 | 20.0000 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli K-12 | Ki | 7.0500 | 1 | 1 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 1.9000 | 3 | 5 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 0.9212 | 4 | 4 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 53.9500 | 4 | 4 |
| Epoxide hydrolase 1 | Homo sapiens (human) | IC50 | 7.0000 | 1 | 1 |
| Estrogen receptor | Homo sapiens (human) | Ki | 0.5797 | 2 | 3 |
| eukaryotic translation initiation factor 4 gamma 1 isoform 4 | Homo sapiens (human) | IC50 | 1.1500 | 1 | 1 |
| eukaryotic translation initiation factor 4E isoform 1 | Mus musculus (house mouse) | IC50 | 1.1500 | 1 | 1 |
| Fatty acid synthase | Gallus gallus (chicken) | IC50 | 62.5000 | 1 | 1 |
| Fatty acid synthase | Homo sapiens (human) | IC50 | 62.5000 | 1 | 1 |
| Fatty acid-binding protein, intestinal | Homo sapiens (human) | Ki | 263.5000 | 1 | 1 |
| Fatty acid-binding protein, liver | Rattus norvegicus (Norway rat) | Ki | 247.8000 | 2 | 2 |
| Fatty-acid amide hydrolase 1 | Homo sapiens (human) | IC50 | 52.0000 | 1 | 1 |
| Fatty-acid amide hydrolase 1 | Rattus norvegicus (Norway rat) | IC50 | 79.0000 | 3 | 4 |
| Focal adhesion kinase 1 | Homo sapiens (human) | IC50 | 1.2000 | 1 | 1 |
| Fructose-1,6-bisphosphatase 1 | Homo sapiens (human) | IC50 | 29.0000 | 1 | 1 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | IC50 | 8.7000 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | IC50 | 20.7333 | 1 | 3 |
| G1/S-specific cyclin-D1 | Homo sapiens (human) | IC50 | 61.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B | Marthasterias glacialis (spiny starfish) | IC50 | 54.4875 | 1 | 8 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 25.5460 | 3 | 5 |
| G2/mitotic-specific cyclin-B2 | Homo sapiens (human) | IC50 | 40.6000 | 1 | 2 |
| G2/mitotic-specific cyclin-B3 | Homo sapiens (human) | IC50 | 40.6000 | 1 | 2 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | IC50 | 28.0000 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | IC50 | 28.0000 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit delta | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | IC50 | 28.0000 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | IC50 | 13.7857 | 4 | 7 |
| Gamma-aminobutyric acid receptor subunit pi | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit theta | Homo sapiens (human) | Ki | 77.2078 | 2 | 3 |
| Gamma-butyrobetaine dioxygenase | Homo sapiens (human) | IC50 | 0.7420 | 5 | 5 |
| Genome polyprotein | Coxsackievirus B3 (strain Nancy) | IC50 | 1.1000 | 1 | 1 |
| Genome polyprotein | | IC50 | 1.6000 | 1 | 1 |
| Genome polyprotein | Zika virus | IC50 | 53.0000 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | IC50 | 19.0000 | 1 | 1 |
| glucose-6-phosphate 1-dehydrogenase isoform b | Homo sapiens (human) | IC50 | 13.2000 | 1 | 1 |
| glucose-6-phosphate dehydrogenase | Leuconostoc mesenteroides | IC50 | 25.0000 | 1 | 1 |
| glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase | Plasmodium berghei | IC50 | 15.0867 | 3 | 3 |
| Glutathione reductase | Saccharomyces cerevisiae S288C | IC50 | 48.8000 | 1 | 1 |
| Glutathione reductase, mitochondrial | Homo sapiens (human) | IC50 | 218.0000 | 1 | 1 |
| Glutathione S-transferase P | Homo sapiens (human) | IC50 | 69.0000 | 1 | 1 |
| Glyceraldehyde-3-phosphate dehydrogenase, glycosomal | Trypanosoma cruzi | IC50 | 142.0000 | 1 | 1 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | IC50 | 4.8000 | 1 | 1 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | IC50 | 1.4500 | 1 | 2 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 51.4625 | 3 | 4 |
| Glycogen synthase kinase-3 beta | Rattus norvegicus (Norway rat) | IC50 | 48.4407 | 2 | 9 |
| Heat shock factor protein 1 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Heme oxygenase 1 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| Heme oxygenase 2 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 0.5800 | 1 | 1 |
| hexokinase | Trypanosoma brucei brucei TREU927 | IC50 | 11.6394 | 2 | 2 |
| Histamine H2 receptor | Homo sapiens (human) | Ki | 8.2434 | 2 | 2 |
| Histamine H3 receptor | Cavia porcellus (domestic guinea pig) | IC50 | 8.6900 | 1 | 1 |
| Histamine H3 receptor | Homo sapiens (human) | Ki | 0.0005 | 1 | 1 |
| Histamine H4 receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| histidine kinase | Streptococcus pneumoniae TIGR4 | IC50 | 216.0000 | 1 | 1 |
| Histone acetyltransferase p300 | Homo sapiens (human) | IC50 | 21.9167 | 6 | 6 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 1 | Homo sapiens (human) | Ki | 50.7900 | 1 | 1 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 2 | Homo sapiens (human) | Ki | 97.6700 | 1 | 1 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 1,116.8000 | 3 | 3 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 673.3200 | 5 | 5 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Histone deacetylase 8 | Homo sapiens (human) | Ki | 64.9800 | 1 | 1 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 1,116.9000 | 3 | 3 |
| Histone-lysine N-methyltransferase EHMT1 | Homo sapiens (human) | IC50 | 0.7300 | 1 | 1 |
| Histone-lysine N-methyltransferase EHMT2 | Homo sapiens (human) | IC50 | 0.4000 | 1 | 1 |
| Histone-lysine N-methyltransferase SETD7 | Homo sapiens (human) | IC50 | 6.0800 | 1 | 1 |
| Homeobox protein Nkx-2.5 | Mus musculus (house mouse) | IC50 | 22.0000 | 1 | 1 |
| hypothetical protein SA1422 | Staphylococcus aureus subsp. aureus N315 | IC50 | 42.9000 | 2 | 2 |
| Hypoxia-inducible factor 1-alpha inhibitor | Homo sapiens (human) | IC50 | 10.2000 | 1 | 1 |
| Indoleamine 2,3-dioxygenase 1 | Homo sapiens (human) | Ki | 0.0940 | 3 | 3 |
| Inositol hexakisphosphate kinase 2 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 2 |
| Inositol polyphosphate multikinase | Homo sapiens (human) | IC50 | 3.9000 | 1 | 2 |
| Insulin-degrading enzyme | Homo sapiens (human) | IC50 | 33.3520 | 3 | 3 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 0.3000 | 1 | 1 |
| Integrase | Human immunodeficiency virus 1 | IC50 | 11.3020 | 5 | 15 |
| integrase, partial | Human immunodeficiency virus 1 | IC50 | 7.8945 | 2 | 2 |
| Interstitial collagenase | Homo sapiens (human) | IC50 | 2.2600 | 1 | 2 |
| intestinal alkaline phosphatase precursor | Mus musculus (house mouse) | IC50 | 18.7000 | 1 | 1 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 83.8867 | 3 | 3 |
| Lactoperoxidase | Bos taurus (cattle) | IC50 | 6.1000 | 1 | 1 |
| Lactoylglutathione lyase | Homo sapiens (human) | IC50 | 7.3000 | 1 | 3 |
| Lactoylglutathione lyase | Homo sapiens (human) | Ki | 7.5703 | 2 | 2 |
| large T antigen | Betapolyomavirus macacae | IC50 | 17.3367 | 1 | 3 |
| lens epithelium-derived growth factor p75 | Homo sapiens (human) | IC50 | 7.8945 | 2 | 2 |
| Leukotriene A-4 hydrolase | Homo sapiens (human) | IC50 | 289.0000 | 2 | 2 |
| Linoleate 9S-lipoxygenase-4 | Glycine max (soybean) | IC50 | 22.0000 | 1 | 1 |
| Luciferin 4-monooxygenase | Photinus pyralis (common eastern firefly) | IC50 | 0.0589 | 1 | 1 |
| Lysine-specific demethylase 4E | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Lysine-specific demethylase 4E | Homo sapiens (human) | Ki | 4.3300 | 1 | 1 |
| Lysine-specific histone demethylase 1A | Homo sapiens (human) | IC50 | 9.7120 | 5 | 5 |
| Lysosomal alpha-glucosidase | Homo sapiens (human) | IC50 | 253.9000 | 2 | 2 |
| Lysosomal alpha-glucosidase | Rattus norvegicus (Norway rat) | IC50 | 400.0000 | 1 | 1 |
| M1-family alanyl aminopeptidase | Plasmodium falciparum 3D7 | IC50 | 22.8600 | 1 | 1 |
| M18 aspartyl aminopeptidase | Plasmodium falciparum 3D7 | IC50 | 2.2420 | 1 | 1 |
| Macrophage metalloelastase | Homo sapiens (human) | IC50 | 5.6050 | 1 | 2 |
| Macrophage migration inhibitory factor | Homo sapiens (human) | IC50 | 2.4000 | 1 | 1 |
| Macrophage migration inhibitory factor | Homo sapiens (human) | Ki | 0.5700 | 2 | 2 |
| Malate dehydrogenase | Thermus thermophilus | IC50 | 6.0000 | 1 | 1 |
| Maltase-glucoamylase, intestinal | Homo sapiens (human) | IC50 | 9.3000 | 2 | 2 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | IC50 | 0.1790 | 1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.5790 | 1 | 1 |
| Matrix metalloproteinase-9 | Homo sapiens (human) | IC50 | 2.4679 | 2 | 3 |
| Melatonin receptor type 1A | Homo sapiens (human) | IC50 | 0.0025 | 18 | 18 |
| Melatonin receptor type 1A | Gallus gallus (chicken) | Ki | 0.0007 | 7 | 8 |
| Melatonin receptor type 1A | Homo sapiens (human) | Ki | 0.0003 | 67 | 69 |
| Melatonin receptor type 1B | Homo sapiens (human) | IC50 | 0.0035 | 12 | 12 |
| Melatonin receptor type 1B | Gallus gallus (chicken) | Ki | 0.0007 | 8 | 9 |
| Melatonin receptor type 1B | Homo sapiens (human) | Ki | 0.0004 | 62 | 64 |
| Melatonin receptor type 1C | Gallus gallus (chicken) | Ki | 0.0007 | 7 | 8 |
| Metabotropic glutamate receptor 1 | Rattus norvegicus (Norway rat) | IC50 | 0.0004 | 2 | 2 |
| Methionine aminopeptidase 2 | Homo sapiens (human) | IC50 | 2.4300 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | IC50 | 54.8750 | 4 | 4 |
| Microtubule-associated protein tau | Rattus norvegicus (Norway rat) | IC50 | 0.2000 | 1 | 1 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 5.8150 | 1 | 6 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 5.8150 | 1 | 6 |
| Monocarboxylate transporter 1 | Rattus norvegicus (Norway rat) | IC50 | 14.0000 | 1 | 1 |
| Monocarboxylate transporter 2 | Rattus norvegicus (Norway rat) | IC50 | 5.0000 | 1 | 1 |
| MPI protein | Homo sapiens (human) | IC50 | 0.2905 | 2 | 2 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 2.9000 | 1 | 1 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 0.0003 | 1 | 1 |
| Multidrug resistance-associated protein 1 | Homo sapiens (human) | Ki | 5.2500 | 2 | 2 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 114.3000 | 1 | 6 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Myc proto-oncogene protein | Homo sapiens (human) | IC50 | 60.0000 | 1 | 1 |
| Myeloperoxidase | Homo sapiens (human) | IC50 | 1.9580 | 5 | 5 |
| N1L | Vaccinia virus | IC50 | 21.9000 | 2 | 2 |
| NACHT, LRR and PYD domains-containing protein 3 | Homo sapiens (human) | IC50 | 24.2000 | 1 | 1 |
| NACHT, LRR and PYD domains-containing protein 3 | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| NADPH oxidase 1 | Homo sapiens (human) | IC50 | 0.3588 | 2 | 2 |
| NADPH oxidase 4 | Homo sapiens (human) | IC50 | 0.7650 | 1 | 2 |
| Neuraminidase | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | IC50 | 16.4750 | 2 | 2 |
| Neuraminidase | Influenza A virus (A/RI/5+/1957(H2N2)) | IC50 | 11.9000 | 1 | 1 |
| Neuraminidase | Influenza A virus (A/Wilson-Smith/1933(H1N1)) | IC50 | 42.0000 | 4 | 9 |
| Neuraminidase | Influenza A virus (A/Wilson-Smith/1933(H1N1)) | Ki | 18.7000 | 1 | 3 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 0.7300 | 2 | 3 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 0.7300 | 2 | 3 |
| Neuronal proto-oncogene tyrosine-protein kinase Src | Mus musculus (house mouse) | IC50 | 2.2000 | 1 | 1 |
| neutrophil cytosol factor 1 | Homo sapiens (human) | IC50 | 0.3900 | 1 | 1 |
| Neutrophil cytosol factor 1 | Homo sapiens (human) | Ki | 125.0000 | 3 | 3 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 18.0445 | 2 | 4 |
| Neutrophil elastase | Homo sapiens (human) | Ki | 12.5667 | 1 | 3 |
| Nitric oxide synthase, inducible | Mus musculus (house mouse) | IC50 | 19.4500 | 4 | 4 |
| Nociceptin receptor | Mus musculus (house mouse) | Ki | 0.0003 | 1 | 1 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | IC50 | 5.0900 | 1 | 1 |
| Nuclear factor NF-kappa-B p100 subunit | Homo sapiens (human) | IC50 | 24.7333 | 3 | 3 |
| Nuclear factor NF-kappa-B p105 subunit | Homo sapiens (human) | IC50 | 24.7333 | 3 | 3 |
| Nuclear receptor ROR-gamma | Mus musculus (house mouse) | IC50 | 11.1000 | 1 | 1 |
| Oligo-1,6-glucosidase IMA1 | Saccharomyces cerevisiae S288C | IC50 | 530.0000 | 1 | 1 |
| Ornithine decarboxylase | Homo sapiens (human) | IC50 | 19.0000 | 1 | 1 |
| Palmitoleoyl-protein carboxylesterase NOTUM | Homo sapiens (human) | IC50 | 75.4000 | 1 | 1 |
| Pancreatic triacylglycerol lipase | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
| perilipin-1 | Homo sapiens (human) | IC50 | 6.2885 | 1 | 2 |
| perilipin-5 | Homo sapiens (human) | IC50 | 5.6665 | 1 | 2 |
| Phosphatidylinositol 3-kinase regulatory subunit alpha | Homo sapiens (human) | IC50 | 3.8000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | IC50 | 8.7950 | 2 | 2 |
| Phosphodiesterase | Rattus norvegicus (Norway rat) | IC50 | 275.0000 | 1 | 1 |
| phosphoethanolamine/phosphocholine phosphatase isoform 1 | Homo sapiens (human) | IC50 | 0.1110 | 1 | 1 |
| Phospholipase A2 | Homo sapiens (human) | IC50 | 6.5500 | 2 | 2 |
| phosphomannomutase 2 | Homo sapiens (human) | IC50 | 0.6720 | 1 | 1 |
| Pleiotropic ABC efflux transporter of multiple drugs | Saccharomyces cerevisiae S288C | IC50 | 400.0000 | 1 | 1 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | IC50 | 4.2329 | 1 | 2 |
| Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens (human) | IC50 | 2.3994 | 1 | 2 |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | IC50 | 1.0858 | 1 | 2 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 1,673.5000 | 2 | 2 |
| Polyphenol oxidase 2 | Agaricus bisporus | IC50 | 166.0850 | 10 | 10 |
| Polyphenol oxidase 2 | Agaricus bisporus | Ki | 8.7000 | 4 | 4 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | IC50 | 13.2821 | 10 | 14 |
| Polyunsaturated fatty acid 5-lipoxygenase | Rattus norvegicus (Norway rat) | IC50 | 12.2850 | 10 | 12 |
| Polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | IC50 | 26.3500 | 2 | 6 |
| Polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Ki | 1.6000 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens (human) | IC50 | 24.7286 | 3 | 7 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | IC50 | 12.4173 | 3 | 4 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens (human) | Ki | 0.6000 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | IC50 | 57.2062 | 3 | 8 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Rattus norvegicus (Norway rat) | IC50 | 0.2600 | 1 | 1 |
| Probable maltase-glucoamylase 2 | Homo sapiens (human) | IC50 | 7.8000 | 1 | 1 |
| Procathepsin L | Homo sapiens (human) | IC50 | 0.6700 | 1 | 1 |
| Progesterone receptor | Homo sapiens (human) | IC50 | 15.0000 | 1 | 1 |
| Prolyl endopeptidase | Homo sapiens (human) | IC50 | 24.5000 | 1 | 2 |
| Prostaglandin E synthase | Homo sapiens (human) | IC50 | 1.8000 | 3 | 3 |
| Prostaglandin G/H synthase 1 | Homo sapiens (human) | IC50 | 18.2118 | 16 | 22 |
| Prostaglandin G/H synthase 1 | Mus musculus (house mouse) | IC50 | 0.2200 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Ovis aries (sheep) | IC50 | 13.2471 | 43 | 49 |
| Prostaglandin G/H synthase 1 | Ovis aries (sheep) | Ki | 9.0000 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Bos taurus (cattle) | IC50 | 178.1500 | 6 | 6 |
| Prostaglandin G/H synthase 1 | Rattus norvegicus (Norway rat) | IC50 | 21.9843 | 5 | 7 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | IC50 | 34.0591 | 47 | 54 |
| Prostaglandin G/H synthase 2 | Mus musculus (house mouse) | IC50 | 0.5400 | 2 | 2 |
| Prostaglandin G/H synthase 2 | Ovis aries (sheep) | IC50 | 139.8408 | 12 | 12 |
| Prostaglandin G/H synthase 2 | Ovis aries (sheep) | Ki | 9.0000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Bos taurus (cattle) | IC50 | 1.1000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Rattus norvegicus (Norway rat) | IC50 | 21.9843 | 5 | 7 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 4.7167 | 4 | 6 |
| Protein cereblon | Homo sapiens (human) | IC50 | 264.0000 | 1 | 1 |
| Protein cereblon | Homo sapiens (human) | Ki | 68,568.5000 | 2 | 2 |
| Protein E6 | Human papillomavirus 16 | IC50 | 20.0000 | 1 | 1 |
| Prothrombin | Homo sapiens (human) | IC50 | 15.7500 | 2 | 2 |
| Prothrombin | Bos taurus (cattle) | IC50 | 19.1933 | 3 | 6 |
| Prothrombin | Bos taurus (cattle) | Ki | 3.9000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 78.1000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 7.5600 | 2 | 2 |
| Proton-coupled amino acid transporter 1 | Homo sapiens (human) | Ki | 7,800.0000 | 1 | 1 |
| rac GTPase-activating protein 1 isoform a | Homo sapiens (human) | IC50 | 29.7100 | 1 | 2 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 5.3900 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 3.8067 | 1 | 3 |
| Receptor-type tyrosine-protein phosphatase S | Homo sapiens (human) | IC50 | 10.3000 | 1 | 1 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | IC50 | 0.6700 | 1 | 1 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 6.8900 | 2 | 3 |
| Replicase polyprotein 1ab | Human coronavirus 229E | IC50 | 0.6700 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 5.4610 | 19 | 29 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 36.1982 | 7 | 17 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Ki | 7.4000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | Ki | 4.9000 | 2 | 2 |
| Ribonucleoside-diphosphate reductase large subunit | Homo sapiens (human) | IC50 | 997.0000 | 1 | 1 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | IC50 | 3.8283 | 17 | 21 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Ki | 0.0575 | 3 | 3 |
| RNA polymerase beta subunit (EC 2.7.7.6), partial | Escherichia coli | IC50 | 11.6872 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 6.0000 | 2 | 2 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | Ki | 5.8000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Homo sapiens (human) | IC50 | 7.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Homo sapiens (human) | Ki | 53.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Rattus norvegicus (Norway rat) | Ki | 5.8000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 | Homo sapiens (human) | IC50 | 7.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 | Homo sapiens (human) | Ki | 8.6000 | 1 | 1 |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max (soybean) | IC50 | 8.0500 | 4 | 4 |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max (soybean) | Ki | 114.2000 | 1 | 2 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | IC50 | 7.5890 | 1 | 1 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | IC50 | 5.8000 | 1 | 1 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | IC50 | 5.7300 | 1 | 1 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | IC50 | 4.2300 | 1 | 1 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | IC50 | 15.5000 | 1 | 2 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 0.9072 | 5 | 6 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | IC50 | 26.2500 | 3 | 3 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | IC50 | 314.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Shiga toxin subunit A | Shigella dysenteriae | IC50 | 23.9000 | 1 | 1 |
| Short transient receptor potential channel 5 | Homo sapiens (human) | IC50 | 8.2500 | 1 | 2 |
| Sialidase | Clostridium perfringens | IC50 | 15.6286 | 5 | 7 |
| Sialidase-2 | Homo sapiens (human) | IC50 | 140.0000 | 1 | 3 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | Ki | 4.4460 | 1 | 1 |
| Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | IC50 | 40.0000 | 1 | 2 |
| Sodium- and chloride-dependent betaine transporter | Rattus norvegicus (Norway rat) | IC50 | 36.1000 | 2 | 3 |
| Sodium- and chloride-dependent GABA transporter 1 | Rattus norvegicus (Norway rat) | IC50 | 36.1000 | 2 | 3 |
| Sodium- and chloride-dependent GABA transporter 2 | Rattus norvegicus (Norway rat) | IC50 | 36.1000 | 2 | 3 |
| Sodium- and chloride-dependent GABA transporter 3 | Rattus norvegicus (Norway rat) | IC50 | 36.1000 | 2 | 3 |
| Sodium- and chloride-dependent taurine transporter | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | IC50 | 510.0000 | 2 | 2 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | IC50 | 18.6360 | 1 | 1 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | Ki | 14.8070 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 4.0553 | 1 | 3 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 4.0220 | 1 | 3 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | IC50 | 1.0000 | 1 | 1 |
| Solute carrier family 2, facilitated glucose transporter member 2 | Homo sapiens (human) | IC50 | 12.0000 | 2 | 2 |
| Solute carrier family 2, facilitated glucose transporter member 4 | Rattus norvegicus (Norway rat) | Ki | 16.0000 | 1 | 1 |
| Solute carrier family 22 member 20 | Mus musculus (house mouse) | Ki | 1.1110 | 1 | 2 |
| Solute carrier family 22 member 6 | Homo sapiens (human) | IC50 | 8.0000 | 1 | 1 |
| Solute carrier family 22 member 6 | Mus musculus (house mouse) | Ki | 4.6887 | 1 | 2 |
| Solute carrier family 22 member 6 | Rattus norvegicus (Norway rat) | Ki | 1,001.7500 | 2 | 2 |
| Solute carrier family 22 member 8 | Homo sapiens (human) | Ki | 1,170.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1A1 | Rattus norvegicus (Norway rat) | Ki | 126.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1A4 | Rattus norvegicus (Norway rat) | Ki | 2,430.0000 | 1 | 1 |
| Sorbitol dehydrogenase | Homo sapiens (human) | IC50 | 106.3000 | 2 | 2 |
| Sortase A | Streptococcus mutans | IC50 | 10.2000 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | IC50 | 0.6700 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | IC50 | 0.6700 | 1 | 1 |
| Squalene monooxygenase | Rattus norvegicus (Norway rat) | IC50 | 0.4700 | 1 | 1 |
| Squalene synthase | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Stromelysin-1 | Homo sapiens (human) | IC50 | 10.8850 | 1 | 2 |
| Structural capsid protein | Human immunodeficiency virus 1 | IC50 | 0.0467 | 1 | 1 |
| Substance-K receptor | Cavia porcellus (domestic guinea pig) | IC50 | 46.0500 | 1 | 2 |
| Substance-P receptor | Cavia porcellus (domestic guinea pig) | IC50 | 31.0667 | 2 | 3 |
| Sucrase-isomaltase, intestinal | Homo sapiens (human) | IC50 | 31.6000 | 3 | 3 |
| Sucrase-isomaltase, intestinal | Rattus norvegicus (Norway rat) | IC50 | 237.3333 | 3 | 3 |
| Sulfhydryl oxidase 1 | Homo sapiens (human) | IC50 | 5.4000 | 1 | 1 |
| Synaptojanin-1 | Homo sapiens (human) | IC50 | 15.9000 | 2 | 2 |
| Synaptojanin-2 | Homo sapiens (human) | IC50 | 0.8740 | 3 | 3 |
| Testosterone 17-beta-dehydrogenase 3 | Homo sapiens (human) | IC50 | 97.6100 | 2 | 2 |
| Thioredoxin reductase 1, cytoplasmic | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thioredoxin reductase 1, cytoplasmic | Rattus norvegicus (Norway rat) | IC50 | 200.0000 | 1 | 1 |
| Thioredoxin reductase 2, mitochondrial | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thioredoxin reductase 2, mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 200.0000 | 1 | 1 |
| Thioredoxin reductase 3 | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thiosulfate sulfurtransferase | Homo sapiens (human) | IC50 | 56.0000 | 1 | 1 |
| Tissue factor | Homo sapiens (human) | IC50 | 0.0132 | 1 | 1 |
| toll-like receptor 9 | Homo sapiens (human) | IC50 | 8.3620 | 1 | 1 |
| Toxin B | Clostridioides difficile | IC50 | 0.0172 | 1 | 1 |
| TPA: protein transporter TIM10 | Saccharomyces cerevisiae S288C | IC50 | 10.0933 | 2 | 3 |
| TPA: protein transporter TIM23 | Saccharomyces cerevisiae S288C | IC50 | 0.8800 | 1 | 1 |
| Transcription factor GATA-4 | Mus musculus (house mouse) | IC50 | 22.0000 | 1 | 1 |
| Transcription factor p65 | Homo sapiens (human) | IC50 | 24.7333 | 3 | 3 |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens (human) | IC50 | 15.3750 | 2 | 2 |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus (Norway rat) | IC50 | 6.4580 | 4 | 5 |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Transmembrane protease serine 2 | Homo sapiens (human) | IC50 | 0.6700 | 1 | 1 |
| Transthyretin | Homo sapiens (human) | IC50 | 6.4000 | 1 | 1 |
| Triosephosphate isomerase | Homo sapiens (human) | IC50 | 1,000.0000 | 1 | 1 |
| Triosephosphate isomerase, glycosomal | Trypanosoma cruzi | IC50 | 6.5000 | 1 | 1 |
| Trypsin-1 | Homo sapiens (human) | IC50 | 9.5500 | 2 | 2 |
| Trypsin-2 | Homo sapiens (human) | IC50 | 9.5500 | 2 | 2 |
| Trypsin-3 | Homo sapiens (human) | IC50 | 9.5500 | 2 | 2 |
| Tubulin alpha-1A chain | Sus scrofa (pig) | IC50 | 10.0000 | 1 | 1 |
| Tubulin beta chain | Sus scrofa (pig) | IC50 | 10.0000 | 1 | 1 |
| Tubulin beta-2B chain | Bos taurus (cattle) | IC50 | 40.0000 | 1 | 1 |
| Tyrosinase | Homo sapiens (human) | IC50 | 578.5829 | 7 | 7 |
| Tyrosinase | Mus musculus (house mouse) | IC50 | 10.7800 | 1 | 1 |
| Tyrosinase | Mus musculus (house mouse) | Ki | 2,900.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 19.0000 | 1 | 2 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 46.0000 | 3 | 3 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | IC50 | 0.9600 | 1 | 1 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | IC50 | 16.0000 | 1 | 2 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | IC50 | 3.3000 | 1 | 1 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Ki | 1.4260 | 1 | 2 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 186.7667 | 6 | 6 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | Ki | 10.7000 | 1 | 1 |
| UDP-glucose 4-epimerase | Homo sapiens (human) | IC50 | 0.0140 | 1 | 1 |
| UDP-glucuronosyltransferase 1A1 | Homo sapiens (human) | IC50 | 5.7000 | 2 | 2 |
| Urease subunit alpha | Helicobacter pylori 26695 | IC50 | 141.7900 | 8 | 11 |
| Urease subunit alpha | Helicobacter pylori 26695 | Ki | 4.7830 | 2 | 2 |
| Urease subunit beta | Helicobacter pylori 26695 | IC50 | 141.7900 | 8 | 11 |
| Urease subunit beta | Helicobacter pylori 26695 | Ki | 4.7830 | 2 | 2 |
| Urokinase-type plasminogen activator | Homo sapiens (human) | IC50 | 25.4200 | 2 | 5 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 0.9700 | 2 | 2 |
| Vasopressin V2 receptor | Homo sapiens (human) | IC50 | 20.3282 | 3 | 6 |
| Vif | Human immunodeficiency virus 1 | IC50 | 25.3100 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | IC50 | 14.8443 | 43 | 47 |
| Xanthine dehydrogenase/oxidase | Homo sapiens (human) | IC50 | 30.3362 | 42 | 49 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | Ki | 1.6750 | 3 | 4 |
| Xanthine dehydrogenase/oxidase | Homo sapiens (human) | Ki | 2.5662 | 7 | 8 |
| Xanthine dehydrogenase/oxidase [Includes: Xanthine dehydrogenase | Rattus norvegicus (Norway rat) | IC50 | 9.3177 | 3 | 3 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | EC50 | 1.1749 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Homo sapiens (human) | EC50 | 10.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit beta-1 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | Kd | 77.0000 | 1 | 1 |
| Albumin | Homo sapiens (human) | Kd | 73.0000 | 1 | 1 |
| Albumin | Rattus norvegicus (Norway rat) | Kd | 1.4700 | 1 | 1 |
| Alpha-synuclein | Homo sapiens (human) | Kd | 3.5000 | 4 | 4 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Kd | 38.5000 | 1 | 1 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | EC50 | 32.8900 | 1 | 3 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | Kd | 7.0795 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | EC50 | 0.1953 | 3 | 3 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Kd | 460.0000 | 1 | 7 |
| Chain A, Transthyretin | Homo sapiens (human) | Kd | 0.1000 | 1 | 5 |
| Chain A, Troponin C, slow skeletal and cardiac muscles | Homo sapiens (human) | Kd | 243.0000 | 1 | 1 |
| Chain B, Transthyretin | Homo sapiens (human) | Kd | 0.1000 | 1 | 2 |
| Cystic fibrosis transmembrane conductance regulator | Homo sapiens (human) | Kd | 25.6000 | 1 | 1 |
| Cytochrome P450 1A1 | Homo sapiens (human) | EC50 | 8.8000 | 1 | 1 |
| Cytochrome P450 1B1 | Homo sapiens (human) | EC50 | 1.1000 | 1 | 1 |
| D(1A) dopamine receptor | Homo sapiens (human) | EC50 | 10.0000 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | EC50 | 0.0260 | 7 | 7 |
| D(2) dopamine receptor | Rattus norvegicus (Norway rat) | EC50 | 0.0088 | 5 | 5 |
| D(2) dopamine receptor | Homo sapiens (human) | Kd | 0.0000 | 2 | 2 |
| D(3) dopamine receptor | Homo sapiens (human) | EC50 | 0.0020 | 6 | 6 |
| D(3) dopamine receptor | Rattus norvegicus (Norway rat) | EC50 | 0.0002 | 1 | 2 |
| D(3) dopamine receptor | Homo sapiens (human) | Kd | 0.0000 | 1 | 1 |
| D(4) dopamine receptor | Homo sapiens (human) | EC50 | 0.0150 | 2 | 2 |
| DNA repair and recombination protein RadA | Pyrococcus furiosus DSM 3638 | Kd | 460.0000 | 1 | 1 |
| Estrogen receptor | Mus musculus (house mouse) | EC50 | 5.2030 | 1 | 2 |
| Estrogen receptor beta | Mus musculus (house mouse) | EC50 | 5.2030 | 1 | 2 |
| G-protein coupled receptor 35 | Homo sapiens (human) | EC50 | 9.5650 | 2 | 6 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | EC50 | 19.8550 | 9 | 9 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | EC50 | 22.1333 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | EC50 | 27.6000 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | EC50 | 27.6000 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | EC50 | 27.6000 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | EC50 | 27.6000 | 2 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | EC50 | 26.8000 | 4 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | EC50 | 15.6791 | 5 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | EC50 | 22.9400 | 5 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | EC50 | 16.8369 | 8 | 8 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | EC50 | 50.0000 | 1 | 2 |
| Gamma-butyrobetaine dioxygenase | Homo sapiens (human) | Kd | 4.1000 | 2 | 2 |
| glycogen synthase kinase-3 beta isoform 1 | Homo sapiens (human) | EC50 | 3.8120 | 1 | 1 |
| Heterogeneous nuclear ribonucleoprotein A1 | Homo sapiens (human) | Kd | 5.3000 | 1 | 2 |
| hexokinase HKDC1 | Homo sapiens (human) | EC50 | 38.8000 | 1 | 1 |
| hexokinase-1 isoform HKI | Homo sapiens (human) | EC50 | 41.9000 | 1 | 1 |
| Histamine H1 receptor | Homo sapiens (human) | Kd | 0.0045 | 1 | 1 |
| Histamine H2 receptor | Homo sapiens (human) | EC50 | 0.1660 | 1 | 1 |
| Histamine H2 receptor | Homo sapiens (human) | Kd | 0.0122 | 1 | 1 |
| Histamine H4 receptor | Homo sapiens (human) | Kd | 0.0160 | 1 | 1 |
| Insulin-like growth factor-binding protein 5 | Homo sapiens (human) | Kd | 696,000.0000 | 7 | 7 |
| Interstitial collagenase | Homo sapiens (human) | Kd | 51.8000 | 1 | 1 |
| large T antigen | Betapolyomavirus macacae | EC50 | 47.9300 | 1 | 1 |
| Lymphocyte antigen 96 | Homo sapiens (human) | Kd | 379.0000 | 1 | 1 |
| Melatonin receptor type 1A | Gallus gallus (chicken) | EC50 | 0.0226 | 1 | 1 |
| Melatonin receptor type 1A | Homo sapiens (human) | EC50 | 0.0008 | 11 | 11 |
| Melatonin receptor type 1B | Gallus gallus (chicken) | EC50 | 0.0226 | 1 | 1 |
| Melatonin receptor type 1B | Homo sapiens (human) | EC50 | 0.0025 | 12 | 12 |
| Melatonin receptor type 1C | Gallus gallus (chicken) | EC50 | 0.0226 | 1 | 1 |
| Melatonin receptor type 1C | Xenopus laevis (African clawed frog) | EC50 | 0.0001 | 3 | 3 |
| NAD-dependent protein deacetylase sirtuin-1 | Homo sapiens (human) | EC50 | 52.3333 | 3 | 3 |
| NAD-dependent protein deacetylase sirtuin-2 | Homo sapiens (human) | EC50 | 300.0000 | 1 | 1 |
| NAD-dependent protein deacetylase sirtuin-3, mitochondrial | Homo sapiens (human) | EC50 | 177.5950 | 2 | 2 |
| Nuclear factor erythroid 2-related factor 2 | Homo sapiens (human) | EC50 | 13.2000 | 2 | 2 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | EC50 | 5.2030 | 1 | 1 |
| Peroxisome proliferator-activated receptor gamma | Mus musculus (house mouse) | EC50 | 2.3000 | 1 | 1 |
| POsterior Segregation | Caenorhabditis elegans | EC50 | 220.1247 | 1 | 3 |
| Procathepsin L | Homo sapiens (human) | EC50 | 32.8900 | 1 | 3 |
| Prostaglandin G/H synthase 1 | Ovis aries (sheep) | Kd | 11.7000 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | EC50 | 5,780.0000 | 1 | 1 |
| Protein polybromo-1 | Homo sapiens (human) | Kd | 12.9000 | 1 | 1 |
| Prothrombin | Homo sapiens (human) | Kd | 0.0387 | 1 | 1 |
| Purine nucleoside phosphorylase | Mycobacterium tuberculosis H37Rv | Kd | 1,000.0000 | 1 | 1 |
| recombinase A | Mycobacterium tuberculosis H37Rv | EC50 | 3.0245 | 2 | 2 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | EC50 | 38.5340 | 2 | 5 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | EC50 | 32.8900 | 1 | 3 |
| Replicase polyprotein 1ab | Human coronavirus 229E | EC50 | 38.5340 | 2 | 5 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | EC50 | 16.8529 | 3 | 7 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | EC50 | 26.2850 | 3 | 8 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Kd | 18.4000 | 3 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | Kd | 10.3000 | 1 | 1 |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | EC50 | 1.0700 | 1 | 1 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 0.0540 | 1 | 1 |
| serine/threonine-protein kinase 33 isoform a | Homo sapiens (human) | EC50 | 12.3300 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 0.0250 | 1 | 1 |
| Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | EC50 | 1.4500 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | EC50 | 97.0655 | 1 | 2 |
| Sodium/bile acid cotransporter | Homo sapiens (human) | Kd | 64.3000 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | EC50 | 32.8900 | 1 | 3 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | EC50 | 32.8900 | 1 | 3 |
| streptokinase A precursor | Streptococcus pyogenes M1 GAS | EC50 | 1.5190 | 1 | 1 |
| Stromelysin-1 | Homo sapiens (human) | Kd | 25,000.0000 | 1 | 1 |
| transcription factor p65 isoform 1 | Homo sapiens (human) | EC50 | 5.2030 | 1 | 1 |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens (human) | EC50 | 30.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus (Norway rat) | EC50 | 3.6000 | 1 | 1 |
| Transmembrane protease serine 2 | Homo sapiens (human) | EC50 | 32.8900 | 1 | 3 |
| Transthyretin | Homo sapiens (human) | Kd | 0.2700 | 2 | 2 |
| Triosephosphate isomerase, glycosomal | Trypanosoma cruzi | Kd | 10.4000 | 1 | 1 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | EC50 | 19.7500 | 1 | 2 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | Kd | 0.0005 | 1 | 1 |
| Zinc finger protein mex-5 | Caenorhabditis elegans | EC50 | 97.0655 | 1 | 2 |