Page last updated: 2024-08-07 12:33:50

M18 aspartyl aminopeptidase

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (22)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
protocatechuic acidPlasmodium falciparum 3D7IC500.479410
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolPlasmodium falciparum 3D7IC503.669010
bufexamacPlasmodium falciparum 3D7IC5010.020010
n,n-naphthaloylhydroxylaminePlasmodium falciparum 3D7IC50100.000010
dopamine hydrochloridePlasmodium falciparum 3D7IC501.979010
epicatechinPlasmodium falciparum 3D7IC501.376010
rg 6866Plasmodium falciparum 3D7IC5029.240010
resveratrolPlasmodium falciparum 3D7IC502.242010
1-(4-ethoxyphenyl)-3-(6-quinoxalinyl)ureaPlasmodium falciparum 3D7IC5073.456010
2-[[2-[(3,7-dimethyl-2-quinolinyl)thio]-1-oxoethyl]amino]-4,5-dimethoxybenzoic acidPlasmodium falciparum 3D7IC5073.456010
4,5-dimethoxy-2-[[1-oxo-2-[(3,5,8-trimethyl-2-quinolinyl)thio]ethyl]amino]benzoic acidPlasmodium falciparum 3D7IC5073.456010
N-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamidePlasmodium falciparum 3D7IC502.784010
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-onePlasmodium falciparum 3D7IC500.648110
7-[[[5-(2,4-dimethylanilino)-1,3,4-thiadiazol-2-yl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinonePlasmodium falciparum 3D7IC5073.456010
2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-onePlasmodium falciparum 3D7IC504.284010
N-(2,3-dihydro-1H-inden-5-yl)-2-[(4-hydroxy-6-oxo-1H-pyrimidin-2-yl)thio]acetamidePlasmodium falciparum 3D7IC5073.456010
esculetinPlasmodium falciparum 3D7IC5044.190010
4-hydroxyestradiolPlasmodium falciparum 3D7IC501.220010
erbstatinPlasmodium falciparum 3D7IC503.719010
epinephrine bitartratePlasmodium falciparum 3D7IC503.015010
3-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-2-oxolanonePlasmodium falciparum 3D7IC5073.456010
quercetinPlasmodium falciparum 3D7IC500.385110