An endothelin-1 receptor that is encoded in the genome of rat. [OMA:P26684, PRO:DNx]
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| amlexanox | Rattus norvegicus (Norway rat) | Potency | 7.0795 | 1 | 0 |
| anisindione | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol | Rattus norvegicus (Norway rat) | Potency | 3.1623 | 1 | 0 |
| ebselen | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| indoprofen | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| leflunomide | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| thiabendazole | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| quinophthalone | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| dehydrothio-4-toluidine | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| indirubin | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| hematoxylin | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| 4-(benzoylamino)-2-hydroxybenzoic acid | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 2-phenylbenzimidazole | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 2,5-diphenyloxazole | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| drometrizole | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 2-(alpha-thenoylamino)-2-nitro-5-thiazole | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 1,6-bismaleimidohexane | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| diacerein | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| n-(cyclohexylthio)phthalimide | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| k 308 | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| nitazoxanide | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| xanthyletine | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| pifexole | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 2-(2'-pyridyl)benzimidazole | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| methyl fluorone black | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| 4-(2-thiazolylazo)resorcinol | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3,5-di-tert-butyl-1,2-benzoquinone | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| witisol | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 1,4-di(2'-thienyl)-1,4-butadione | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 2-phenyl-1,2-benzisothiazol-3-(2h)-one | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| N-(4-methoxyphenyl)carbamic acid propan-2-yl ester | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 1-Anilino-9,10-dioxo-2-anthroic acid | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| gossypol acetic acid | Rattus norvegicus (Norway rat) | Potency | 0.7943 | 1 | 0 |
| 2-pyridin-4-yl-1,3-benzothiazole | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2-[(6-butoxy-3-pyridinyl)amino]-4-chlorobenzoic acid | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 2-hydroxyestradiol | Rattus norvegicus (Norway rat) | Potency | 0.5623 | 1 | 0 |
| nsc228155 | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| Dubamine | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 4,5,7-trihydroxy-9,10-dioxo-2-anthracenecarboxylic acid | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| (R)-norlaudanosoline | Rattus norvegicus (Norway rat) | Potency | 0.5012 | 1 | 0 |
| resveratrol | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 3-(3,5-dimethyl-1-pyrazolyl)-1,2-benzothiazole 1,1-dioxide | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| chalcone | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 7-methoxyisoflavone | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2'-hydroxychalcone | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazole | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| N,N-dimethyl-6-phenyl-3-pyridazinamine | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-(3,5-dimethoxyphenyl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 4-cyclohexyl-3-[(3-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| acetic acid (11-oxo-6H-benzo[c][1]benzoxepin-2-yl) ester | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| 4-cyclohexyl-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| 4-cyclohexyl-3-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 4.4668 | 1 | 0 |
| N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-3-furamide | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 2-[(3-methyl-2-thiophenyl)methylidene]indene-1,3-dione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 2-(thiophen-2-ylmethylidene)indene-1,3-dione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| krm iii | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2-(4-hydroxyanilino)-1,4-naphthoquinone | Rattus norvegicus (Norway rat) | Potency | 7.9433 | 1 | 0 |
| 4-[2-(1-methyl-2-benzimidazolyl)ethyl]aniline | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-(2,5-dimethylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| nsc185058 | Rattus norvegicus (Norway rat) | Potency | 13.4270 | 1 | 0 |
| 2-(4-fluorophenyl)-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-[(4-methylphenoxy)methyl]-4-phenyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 1-(4,5-dihydrothiazol-2-yl)-3-phenylurea | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-(2,3-dimethyl-1H-indol-5-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 3-(3-nitrophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| N-(2-fluoro-5-methylphenyl)-3-phenylpropanamide | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 4-[[(4-acetyloxy-3-methoxyphenyl)-oxomethyl]amino]benzoic acid | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| acetic acid [4-[(4-hydroxyanilino)-oxomethyl]-2-methoxyphenyl] ester | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 3-bromo-N-(2-furanylmethyl)benzamide | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| N-(cyclopentylideneamino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 4-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 2-methyl-N-(2-naphthalenyl)-3-furancarboxamide | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 2-(ethylthio)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-one | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 3-(2-furanyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| N-(1,3-benzodioxol-5-yl)-5-methyl-2-furancarboxamide | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 3-(1,3-dimethyl-4-pyrazolyl)-4-(2-methoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 4-(2-methylphenyl)-3-(5-methyl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| 3-(4-ethyl-5-methyl-3-thiophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-(3-methylphenyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 3-(1,3-benzodioxol-5-yl)-4-(2,5-dimethylphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 3.9811 | 1 | 0 |
| 3-(1-benzothiophen-3-yl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 4-(3-methylphenyl)-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| 3-(4,5-dimethyl-3-thiophenyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 7.9433 | 1 | 0 |
| 3-(2-methyl-3-furanyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 4-(phenylmethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-methoxy-2-[3-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]phenol | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 5-(1-methyl-2-benzimidazolyl)-2-thiophenecarboxaldehyde | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| N-(2-fluorophenyl)-3-phenylpropanamide | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| benzoic acid (2-oxo-2-thiophen-2-ylethyl) ester | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 4-sulfanylidene-1,6,7,8,9,10-hexahydropyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrile | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 2-[[anilino(oxo)methyl]amino]-N-(2-furanylmethyl)benzamide | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 4-[methyl(methylsulfonyl)amino]-N-(2-phenylethyl)benzamide | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 4-phenacyloxybenzoic acid methyl ester | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 3-(4-ethoxyphenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| N-(4,5-dihydrothiazol-2-yl)-2-(2-methylphenoxy)acetamide | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 3-[4-(2-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]-1H-pyridazin-6-one | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| 3-[5-(2-furanyl)-1H-pyrazol-3-yl]-4-(2-methoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 3.5481 | 1 | 0 |
| 4-(4-chlorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| N-(4-methoxyphenyl)-2-(methylthio)benzamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 4-phenyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| 4-(2-methylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 3-[[(3-acetylanilino)-oxomethyl]amino]-2-thiophenecarboxylic acid methyl ester | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 6-hydroxy-2-(4-nitrophenyl)-3,1-benzoxazin-4-one | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| umi-77 | Rattus norvegicus (Norway rat) | Potency | 3.5481 | 1 | 0 |
| N-(5-chloro-2-pyridinyl)-2-ethyl-3-pyrazolecarboxamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 1-[4-[3-[5-(2-furanyl)-1H-pyrazol-3-yl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]phenyl]ethanone | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| N-(3-methoxyphenyl)-4-(1-oxopropylamino)benzamide | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 3-[[1-oxo-2-[(4,6,9-trimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)thio]ethyl]amino]benzoic acid | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| N-[5-(4-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-5-methyl-3-isoxazolecarboxamide | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| N-(1,3-benzodioxol-5-yl)-2-[[4-(4-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]thio]acetamide | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| 4-(2-chlorophenyl)-3-(5-methyl-3-phenyl-4-isoxazolyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 3-[(1,3-benzothiazol-2-ylthio)methyl]-4-cyclohexyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 4-methyl-2-(4-nitrophenyl)-5-thiazolecarboxylic acid | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 3-phenyl-2H-1,4-benzoxazine | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| 2-(6-chloro-3-pyridinyl)-1H-benzimidazole | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-butyl-3-(5-ethyl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 4-butyl-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 4-butyl-3-(3-methyl-2-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 1-[[4-[(3,4-dichlorophenyl)thio]-3-pyridinyl]sulfonyl]-3-propylurea | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-(2-bromo-4-methylphenyl)-3-[5-(2-furanyl)-1H-pyrazol-3-yl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 4-(2,5-dimethoxyphenyl)-3-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(3,4-dimethoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| 3-(1,3-benzodioxol-5-yl)-4-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 2-[[4-(2-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]methyl]-1-phthalazinone | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-(phenylmethyl)-3-[2-(4-propoxyphenyl)ethyl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 3.1623 | 1 | 0 |
| 3,4,5-trimethoxy-N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]benzamide | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| 4-(2,5-dimethoxyphenyl)-3-(3-phenyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| 3-(4-bromophenyl)-4-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| N-[(tert-butylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamide | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| N-(3,4-dihydro-2H-pyrrol-5-yl)-5-phenyl-1,3,4-oxadiazol-2-amine | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 5-(3,4-dimethoxyphenyl)-3-(4-methoxyphenyl)-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 7.9433 | 1 | 0 |
| 5-(3,4-dimethoxyphenyl)-3-(4-ethoxyphenyl)-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 2.8184 | 1 | 0 |
| N-[5-(2-methylpropyl)-1,3,4-thiadiazol-2-yl]-4-nitrobenzenesulfonamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 2,5-dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) ester | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 4-butyl-3-(phenylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanone | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 1-(2-chlorophenyl)-2-(3,5-dimethyl-4-nitro-1-pyrazolyl)ethanone | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 2-chloro-3-pyridinecarboxylic acid [2-(4-fluorophenyl)-2-oxoethyl] ester | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-(1,3-benzodioxol-5-yl)-4-phenyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 7.0795 | 1 | 0 |
| 7-methyl-N-[4-(4-morpholinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 3-methoxy-N-(4-methyl-2-thiazolyl)benzamide | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 3-[[(2,4-dichlorophenyl)methylthio]methyl]-4-propan-2-yl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 2-[3-(4-pyridyl)-1H-1,2,4-triazol-5-yl]pyridine | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| N-[(2-hydroxyphenyl)-oxomethyl]-2,3-dihydrobenzofuran-5-carboxamide | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 4-(2-furanylmethyl)-3-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 3-[4-(4-chlorophenyl)-1-piperazinyl]-1-(4-methoxyphenyl)pyrrolidine-2,5-dione | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| 3-(4-methoxyphenyl)-3-(4-methylphenyl)sulfonyl-1-phenyl-1-propanone | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2-(3,4-dimethylphenyl)-5-ethyl-5-phenyl-1,2,4-triazolidine-3-thione | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| 4-(1-phenylethyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 4-[1-(4-fluorophenyl)ethyl]-3-thiophen-2-yl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-(benzenesulfonyl)-3-(4-methoxyphenyl)-1-phenyl-1-propanone | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2-quinolinecarboxylic acid (1-oxo-1-phenylpropan-2-yl) ester | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| yl-109 | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 4-[4-[[1-(2-methylbutan-2-yl)-5-tetrazolyl]-(6-quinolinyl)methyl]-1-piperazinyl]phenol | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-[4-[(1-tert-butyl-5-tetrazolyl)-pyridin-4-ylmethyl]-1-piperazinyl]phenol | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| 3-(4-bromophenyl)-4-(2-furanylmethyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 4-[[(3-methoxyphenyl)-oxomethyl]amino]benzoic acid | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-butyl-3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 4-butyl-3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| N-cycloheptyl-4-(2-oxolanylmethoxy)benzamide | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 2-[(4-amino-7-tert-butyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)thio]acetic acid | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-nitro-N-(2-phenylethyl)-2-pyridinamine | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 4-(2-methylcyclohexyl)-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 0 |
| 2-[2-[5-amino-4-(3-thiophenyl)-1-pyrazolyl]-4-phenyl-5-thiazolyl]acetic acid | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| 4-[[(2-methyl-5-nitro-1H-imidazol-4-yl)thio]methyl]-2-nitrophenol | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 3,5-bis(4-methoxyphenyl)-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 1.4125 | 1 | 0 |
| 4-(1-phenylethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 2-methoxy-N-(5-phenyl-1,2,4-thiadiazol-3-yl)benzamide | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| 2-[[2-(3,4-dimethoxyanilino)-2-oxoethyl]thio]-3-pyridinecarboxylic acid propan-2-yl ester | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| 3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 39.8107 | 1 | 0 |
| 2-(2-fluoroanilino)-3-pyridinecarboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-methylamino]-2-oxoethyl] ester | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| N,N,4-trimethyl-2-[[(5-methyl-2-furanyl)-oxomethyl]amino]-5-thiazolecarboxamide | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| 4-(4-chlorophenyl)-3-[2-(4-methylphenyl)cyclopropyl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 0 |
| 4-(4-chlorophenyl)-3-phenyl-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 2.5119 | 1 | 0 |
| 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[[2-(2-pyridinyl)-1-benzimidazolyl]methyl]-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| 3-(2-methoxyphenyl)-4-phenyl-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 4-(4-methylphenyl)-3-phenyl-1H-imidazole-2-thione | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| 2-cyano-N'-[2,6-dinitro-4-(trifluoromethyl)phenyl]acetohydrazide | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 3-(4-methyl-1,3-dioxan-2-yl)-1-benzopyran-4-one | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| N-[bis(methylthio)methylideneamino]-4-hydroxybenzamide | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 0 |
| chrysoeriol | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 4-hydroxyestradiol | Rattus norvegicus (Norway rat) | Potency | 1.0000 | 1 | 0 |
| 4-hydroxychalcone | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 3-(prop-2-enylthio)-[1,2,4]triazino[5,6-d][3,1]benzoxazepine | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| 5,7-dihydroxy-4',6-dimethoxyflavone | Rattus norvegicus (Norway rat) | Potency | 7.9433 | 1 | 0 |
| erbstatin | Rattus norvegicus (Norway rat) | Potency | 4.4668 | 1 | 0 |
| 2'-hydroxy-4-methoxychalcone | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 0 |
| (2e)-3-phenyl-1-(2,3,4,5-tetrahydro-1,6-benzodioxocin-8-yl)prop-2-en-1-one | Rattus norvegicus (Norway rat) | Potency | 28.1838 | 1 | 0 |
| styrylquinoline | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| 7-hydroxyisoflavone | Rattus norvegicus (Norway rat) | Potency | 12.5893 | 1 | 0 |
| dithiazanine iodide | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| quinaldine red | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| 2',3,4-trihydroxychalcone | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| chloride of pseudoisocyanine | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| alpha-(p-Methoxyphenyl)-2-pyridineacrylonitrile | Rattus norvegicus (Norway rat) | Potency | 8.9125 | 1 | 0 |
| Adenosine 5'-monophosphate monohydrate | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 0 |
| 1-(3-methoxyphenyl)-3-[2-(methylthio)phenyl]urea | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |
| altenusin | Rattus norvegicus (Norway rat) | Potency | 2.8184 | 1 | 0 |
| hydralazine 4-anisaldehyde hydrazone | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 0 |
| lissamine rhodamine b | Rattus norvegicus (Norway rat) | Potency | 15.8489 | 1 | 0 |
| N-[3-[butyl(ethyl)amino]propyl]-2-[6-(4-morpholinylsulfonyl)-3-oxo-1,4-benzothiazin-4-yl]acetamide | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 0 |
| 5-methyl-5-pentyl-2-phenyl-1,2,4-triazolidine-3-thione | Rattus norvegicus (Norway rat) | Potency | 3.9811 | 1 | 0 |
| 1-(1,4-dioxan-2-yl)-N-[[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-N-methylmethanamine | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| acid blue 129 | Rattus norvegicus (Norway rat) | Potency | 14.1254 | 1 | 0 |
| LSM-16789 | Rattus norvegicus (Norway rat) | Potency | 22.3872 | 1 | 0 |