Any protein kinase inhibitor that interferes with the action of tyrosine kinase.
| Member | Definition | Class |
|---|
| 1-NA-PP1 | | 1-NA-PP1 |
| 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine | | 1-NM-PP1 |
| 3,3',4,5'-tetrahydroxystilbene | A stilbenol that is trans-stilbene in which one of the phenyl groups is substituted by hydroxy groups at positions 3 and 4, while the other phenyl group is substituted by hydroxy groups at positions 3 and 5. | piceatannol |
| axitinib | An indazole substituted at position 3 by a 2-(pyridin-2-yl)vinyl group and at position 6 by a 2-(N-methylaminocarboxy)phenylsulfanyl group. Used for the treatment of advanced renal cell carcinoma after failure of a first line systemic treatment. | axitinib |
| bibw 2992 | A quinazoline compound having a 3-chloro-4-fluoroanilino group at the 4-position, a 4-dimethylamino-trans-but-2-enamido group at the 6-position, and an (S)-tetrahydrofuran-3-yloxy group at the 7-position. Used (as its dimaleate salt) for the first-line treatment of patients with metastatic non-small cell lung cancer. | afatinib |
| biochanin a | A member of the class of 7-hydroxyisoflavones that is 7-hydroxyisoflavone which is substituted by an additional hydroxy group at position 5 and a methoxy group at position 4'. A phytoestrogen, it has putative benefits in dietary cancer prophylaxis. | biochanin A |
| bosutinib | An aminoquinoline that is 4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline bearing additional cyano and methoxy substituents at positions 3 and 6 respectively. | bosutinib |
| butein | A chalcone that is (E)-chalcone bearing four additional hydroxy substituents at positions 2', 3, 4 and 4'. | butein |
| cabozantinib | A dicarboxylic acid diamide that is N-phenyl-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide in which the hydrogen at position 4 on the phenyl ring is substituted by a (6,7-dimethoxyquinolin-4-yl)oxy group. A multi-tyrosine kinase inhibitor, used (as its malate salt) for the treatment of progressive, metastatic, medullary thyroid cancer. | cabozantinib |
| canertinib | A quinazoline compound having a 3-chloro-4-fluoroanilino group at the 4-position, a propenamido group at the 6-position, and a 3-morpholinopropoxy group at the 7-position. | canertinib |
| cgp 52411 | Phthalimide substituted at the 4- and 5-positions by anilino groups. | 4,5-dianilinophthalimide |
| dasatinib | An aminopyrimidine that is 2-methylpyrimidine which is substituted at position 4 by the primary amino group of 2-amino-1,3-thiazole-5-carboxylic acid and at position 6 by a 4-(2-hydroxyethyl)piperazin-1-yl group, and in which the carboxylic acid group has been formally condensed with 2-chloro-6-methylaniline to afford the corresponding amide. A multi-targeted kinase inhibitor, it is used, particularly as the monohydrate, for the treatment of chronic, accelerated, or myeloid or lymphoid blast phase chronic myeloid leukemia. Note that the name 'dasatinib' is used to refer to the monohydrate (USAN) as well as to anhydrous dasatinib (INN). | dasatinib (anhydrous) |
| dcc-2036 | A member of the class of ureas that is urea in which one of the nitrogens bears a 3-tert-butyl-1-(quinolin-6-yl)-1H-pyrazol-5-yl substituent, while the other bears a 2-fluoro-4-{[2-(methylcarbamoyl)pyridin-4-yl]oxy}phenyl substituent. | DCC-2036 |
| emodin | A trihydroxyanthraquinone that is 9,10-anthraquinone which is substituted by hydroxy groups at positions 1, 3, and 8 and by a methyl group at position 6. It is present in the roots and barks of numerous plants (particularly rhubarb and buckthorn), moulds, and lichens. It is an active ingredient of various Chinese herbs. | emodin |
| genistein | A 7-hydroxyisoflavone with additional hydroxy groups at positions 5 and 4'. It is a phytoestrogenic isoflavone with antioxidant properties. | genistein |
| herbimycin | A 19-membered macrocyle incorporating a benzoquinone ring and a lactam functionality. It is an ansamycin antibiotic that induces apoptosis and displays antitumour effects. | herbimycin |
| hki 272 | A quinoline compound having a cyano group at the 3-position, a 3-chloro-4-(2-pyridylmethoxy)anilino group at the 4-position, a 4-dimethylamino-trans-but-2-enoylamido group at the 6-position, and an ethoxy group at the 7-position. | neratinib |
| hydroxy-2-naphthalenyl-methyl phosphonic acid trisacetoxymethylester | An organic phosphonate that is the trisacetoxymethylester derivative of naphthalene substituted hydroxymethylphosphonic acid. It has been found to inhibit insulin receptor tyrosine kinase activity and insulin stimulated glucose oxidation. | hydroxy-2-naphthalenyl-methyl phosphonic acid trisacetoxymethylester |
| imatinib | A benzamide obtained by formal condensation of the carboxy group of 4-[(4-methylpiperazin-1-yl)methyl]benzoic acid with the primary aromatic amino group of 4-methyl-N(3)-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine. Used (as its mesylate salt) for treatment of chronic myelogenous leukemia and gastrointestinal stromal tumours. | imatinib |
| imatinib mesylate | A methanesulfonate (mesylate) salt that is the monomesylate salt of imatinib. Used for treatment of chronic myelogenous leukemia and gastrointestinal stromal tumours. | imatinib methanesulfonate |
| lapatinib | | lapatinib |
| leflunomide | A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 5-methyl-1,2-oxazole-4-carboxylic acid with the anilino group of 4-(trifluoromethyl)aniline. The prodrug of teriflunomide. | leflunomide |
| masitinib | A member of the class of benzamides that is the carboxamide resulting from the formal condensation of the carboxy group of 4-[(4-methylpiperazin-1-yl)methyl]benzoic acid with the primary amino group of 4-methyl-N(3)-[4-(pyridin-3-yl)-1,3-thiazol-2-yl]benzene-1,3-diamine. It is a highly selective oral tyrosine kinase inhibitor. | masitinib |
| monorden | An antifungal macrolactone antibiotic, obtained from Diheterospora chlamydosporia and Chaetomium chiversii that inhibits protein tyrosine kinase and heat shock protein 90 (Hsp90). | radicicol |
| pazopanib | A pyrimidine that is 5-(pyrimidin-2-yl}amino-2-methylbenzenesulfonamide substituted at position 4 by a (2,3-dimethylindazol-6-yl)(methyl)amino group. Used as its hydrochloride salt for treatment of kidney cancer. | pazopanib |
| pd 173955 | | PD173955 |
| picropodophyllin | An organic heterotetracyclic compound that has a furonaphthodioxole skeleton bearing 3,4,5-trimethoxyphenyl and hydroxy substituents. | picropodophyllotoxin |
| ponatinib | A benzamide obtained by the formal condensation of the carboxy group of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methylbenzoic acid with the anilino group of 4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)aniline. It is a multi-target tyrosine kinase inhibitor that targets ABL, SRC, FGFR, and others and was designed to overcome the resistance of BCR-ABL mutation to imatinib, in particular the gatekeeper mutation ABL(T315I). | ponatinib |
| PP121 | A pyrazolopyrimidine that is 1H-pyrazolo[3,4-d]pyrimidine which is substituted by a cyclopentyl, 1H-pyrrolo[2,3-b]pyridin-5-yl, and amino groups at positions 1, 3 and 4, respectively. It is a dual inhibitor of tyrosine and phosphoinositide kinases and exhibits anti-cancer properties. | PP121 |
| regorafenib | A pyridinecarboxamide obtained by condensation of 4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)-3-fluorophenoxy]pyridine-2-carboxylic acid with methylamine. Used for for the treatment of metastatic colorectal cancer in patients who have previously received chemotherapy, anti-EGFR or anti-VEGF therapy. | regorafenib |
| s 1033 | | nilotinib |
| sorafenib | A member of the class of phenylureas that is urea in which one of the nitrogens is substituted by a 4-chloro-3-trifluorophenyl group while the other is substituted by a phenyl group which, in turn, is substituted at the para position by a [2-(methylcarbamoyl)pyridin-4-yl]oxy group. | sorafenib |
| teriflunomide | An enamide obtained by formal condensation of the carboxy group of (2Z)-2-cyano-3-hydroxybut-2-enoic acid with the anilino group of 4-(trifluoromethyl)aniline. Used for the treatment of relapsing forms of multiple sclerosis and rheumatoid arthritis. | teriflunomide |
| thiopental sodium | A pyrimidine compound having a 2-methoxy-4-(4-methylpiperazin-1-yl)anilino group at the 2-position, a 3-(acryloylamino)phenoxy group at the 4-position, and a chloro substituent at the 5-position. | WZ4002 |
| zd 6474 | A quinazoline that is 7-[(1-methylpiperidin-4-yl)methoxy]quinazoline bearing additional methoxy and 4-bromo-2-fluorophenylamino substituents at positions 6 and 4 respectively. Used for the treatment of symptomatic or progressive medullary thyroid cancer in patients with unresectable locally advanced or metastatic disease. | vandetanib |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 22.5372 | 1 | 9 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 20.5251 | 1 | 3 |
| 2,3-bisphosphoglycerate-independent phosphoglycerate mutase | Leishmania major strain Friedlin | Potency | 37.9330 | 1 | 1 |
| 67.9K protein | Vaccinia virus | Potency | 14.8873 | 2 | 11 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 23.9645 | 3 | 11 |
| acid sphingomyelinase | Homo sapiens (human) | Potency | 293.7300 | 1 | 2 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 51.0926 | 2 | 5 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 24.1669 | 1 | 11 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 10.7509 | 1 | 2 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 8.9125 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 7.0795 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 15.2408 | 12 | 106 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 12.4266 | 3 | 26 |
| arylsulfatase A | Homo sapiens (human) | Potency | 16.3776 | 1 | 4 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 10.6323 | 6 | 18 |
| Ataxin-2 | Homo sapiens (human) | Potency | 8.4313 | 2 | 15 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 20.3664 | 3 | 5 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 6.9479 | 2 | 22 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 22.6327 | 1 | 2 |
| atrial natriuretic peptide receptor 2 precursor | Homo sapiens (human) | Potency | 21.3016 | 1 | 2 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 14.9268 | 2 | 10 |
| BRCA1 | Homo sapiens (human) | Potency | 10.0982 | 1 | 3 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| C-terminal-binding protein 1 | Homo sapiens (human) | Potency | 7.5699 | 1 | 1 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 14.1953 | 1 | 7 |
| caspase-3 | Homo sapiens (human) | Potency | 14.1953 | 1 | 7 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 25.5418 | 3 | 21 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 14.3778 | 2 | 10 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 30.2785 | 1 | 4 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 1.2589 | 1 | 1 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 11.5574 | 1 | 2 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 37.7637 | 2 | 4 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 16.0105 | 2 | 2 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 44.6684 | 1 | 2 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 22.0966 | 2 | 11 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 15.8114 | 1 | 1 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 27.1694 | 1 | 6 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 16.0105 | 2 | 2 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 47.4541 | 2 | 6 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 14.4678 | 1 | 6 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 8.9145 | 1 | 5 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 8.2736 | 1 | 13 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 21.4596 | 1 | 9 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 25.2783 | 1 | 3 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 8.2447 | 2 | 14 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 9.7221 | 1 | 15 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 9.6787 | 1 | 14 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 0.5804 | 1 | 1 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 23.2809 | 1 | 1 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 29.5981 | 2 | 2 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 36.0962 | 1 | 3 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 16.8158 | 1 | 2 |
| DNA polymerase III, partial | Bacillus subtilis | Potency | 28.6828 | 1 | 2 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 46.9355 | 1 | 8 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 35.5313 | 1 | 9 |
| endonuclease IV | Escherichia coli | Potency | 7.9433 | 1 | 1 |
| Endothelin receptor type B | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 1 |
| Endothelin-1 receptor | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 15.2780 | 12 | 131 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 13.6622 | 3 | 27 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 9.7804 | 10 | 104 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 8.4500 | 2 | 12 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 12.3284 | 4 | 75 |
| eyes absent homolog 2 isoform a | Homo sapiens (human) | Potency | 9.5300 | 1 | 1 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 25.6563 | 3 | 19 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 22.9300 | 2 | 8 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 24.6067 | 1 | 19 |
| G | Vesicular stomatitis virus | Potency | 8.2736 | 1 | 13 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| GALC protein | Homo sapiens (human) | Potency | 0.7079 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 8.2447 | 1 | 7 |
| geminin | Homo sapiens (human) | Potency | 16.0480 | 3 | 21 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 10.6564 | 3 | 31 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 13.9028 | 2 | 5 |
| GLS protein | Homo sapiens (human) | Potency | 11.8742 | 2 | 6 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 14.6878 | 1 | 7 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 19.2682 | 4 | 19 |
| glucokinase regulatory protein | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 10.3384 | 1 | 15 |
| guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1 | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 11.1302 | 2 | 6 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 23.6110 | 2 | 7 |
| hexokinase-4 isoform 1 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 8.3912 | 2 | 17 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 34.9134 | 1 | 3 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 7.1907 | 2 | 20 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 69.6220 | 2 | 12 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 8.2736 | 1 | 13 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 13.5026 | 3 | 4 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 9.4096 | 4 | 5 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 33.9588 | 2 | 8 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 8.3373 | 2 | 6 |
| IDH1 | Homo sapiens (human) | Potency | 19.4288 | 1 | 3 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 8.2736 | 1 | 26 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 31.6228 | 1 | 1 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 16.0530 | 1 | 4 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 16.0530 | 1 | 4 |
| Interferon beta | Homo sapiens (human) | Potency | 12.8502 | 3 | 91 |
| interleukin 8 | Homo sapiens (human) | Potency | 66.8242 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 11.2025 | 2 | 11 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 12.4716 | 2 | 4 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 15.2828 | 3 | 20 |
| luciferase | Photuris pensylvanica (Pennsylania firefly) | Potency | 12.5893 | 1 | 1 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 33.8540 | 1 | 7 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 11.5176 | 2 | 17 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 15.4374 | 2 | 7 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 11.3735 | 2 | 3 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 16.8158 | 1 | 2 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 6.3344 | 1 | 2 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 10.0000 | 2 | 2 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 17.7082 | 1 | 3 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 6.0025 | 1 | 7 |
| Nrf2 | Homo sapiens (human) | Potency | 32.6427 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 13.1405 | 4 | 36 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 18.2488 | 1 | 4 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 37.1211 | 1 | 5 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 42.1632 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 25.2607 | 2 | 9 |
| nuclear receptor subfamily 1, group I, member 2 | Rattus norvegicus (Norway rat) | Potency | 11.8930 | 1 | 3 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 14.3486 | 3 | 43 |
| Ornithine decarboxylase | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 1 |
| P53 | Homo sapiens (human) | Potency | 31.2450 | 1 | 4 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 23.6858 | 1 | 6 |
| Parkin | Homo sapiens (human) | Potency | 9.4506 | 2 | 5 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 37.0264 | 2 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 8.6038 | 2 | 10 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 30.7354 | 1 | 4 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 24.8227 | 4 | 21 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 24.2079 | 5 | 21 |
| phosphoglycerate kinase | Trypanosoma brucei brucei TREU927 | Potency | 23.1606 | 2 | 2 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 45.7743 | 1 | 6 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 7.5787 | 1 | 4 |
| polyprotein | Zika virus | Potency | 24.6067 | 1 | 19 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 10.1578 | 1 | 2 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 4.4668 | 1 | 1 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 22.1751 | 1 | 3 |
| PPM1D protein | Homo sapiens (human) | Potency | 13.4567 | 1 | 48 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 19.1723 | 3 | 23 |
| progesterone receptor | Homo sapiens (human) | Potency | 20.6634 | 2 | 14 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 15.1861 | 4 | 4 |
| pyruvate kinase PKM isoform b | Homo sapiens (human) | Potency | 25.1189 | 2 | 2 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 8.8065 | 2 | 27 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 13.2633 | 1 | 6 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 10.3240 | 1 | 5 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 6.5617 | 3 | 40 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 17.8953 | 4 | 26 |
| RGS12 | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 11.6910 | 5 | 10 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 26.6795 | 1 | 1 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 17.7786 | 2 | 11 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 17.7786 | 2 | 11 |
| Smad3 | Homo sapiens (human) | Potency | 11.0011 | 1 | 5 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 15.6290 | 2 | 15 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 18.2195 | 2 | 15 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 3.1623 | 1 | 1 |
| TDP1 protein | Homo sapiens (human) | Potency | 12.4867 | 2 | 51 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 22.3872 | 1 | 1 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 10.3121 | 3 | 10 |
| Thrombopoietin | Homo sapiens (human) | Potency | 11.8091 | 2 | 8 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 19.8430 | 3 | 31 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 55.5574 | 3 | 5 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 16.5584 | 4 | 14 |
| transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 7.2025 | 2 | 19 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 7.5787 | 1 | 4 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 7.5787 | 1 | 4 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 35.1338 | 1 | 4 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 52.8773 | 2 | 5 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 16.2746 | 5 | 19 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 57.8681 | 1 | 3 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 10.3384 | 1 | 15 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial | Homo sapiens (human) | IC50 | 235.9333 | 3 | 3 |
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial | Homo sapiens (human) | IC50 | 77.8000 | 1 | 1 |
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial | Homo sapiens (human) | IC50 | 153.9000 | 2 | 2 |
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial | Homo sapiens (human) | IC50 | 77.8000 | 1 | 1 |
| 17-beta-hydroxysteroid dehydrogenase type 1 | Homo sapiens (human) | IC50 | 2.2100 | 1 | 1 |
| 17-beta-hydroxysteroid dehydrogenase type 2 | Homo sapiens (human) | IC50 | 12.0200 | 2 | 5 |
| 3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ | Yersinia pseudotuberculosis YPIII | IC50 | 36.4000 | 1 | 2 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 1.1810 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | IC50 | 6.1800 | 1 | 2 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | IC50 | 36.4000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | Ki | 1.8300 | 2 | 3 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | Ki | 0.0560 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | IC50 | 14.9100 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 4.1115 | 2 | 2 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | IC50 | 14.9100 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | Ki | 7.8060 | 1 | 1 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 3.2960 | 1 | 1 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 6.2130 | 1 | 1 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 7.0710 | 1 | 1 |
| Accessory gene regulator protein A | Staphylococcus aureus | IC50 | 17.1000 | 1 | 1 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 0.9300 | 1 | 1 |
| Acetylcholinesterase | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | IC50 | 0.0027 | 2 | 2 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Acyl-CoA desaturase 1 | Rattus norvegicus (Norway rat) | IC50 | 0.0013 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | IC50 | 19.9040 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | Ki | 11.6110 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | IC50 | 17.4420 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | Ki | 9.7920 | 1 | 1 |
| Adenosine receptor A2a | Rattus norvegicus (Norway rat) | Ki | 36.0000 | 1 | 1 |
| ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Aldehyde oxidase | Homo sapiens (human) | IC50 | 0.3400 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Homo sapiens (human) | IC50 | 49.8967 | 3 | 3 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 4.6300 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Homo sapiens (human) | Ki | 2.1130 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 4.5910 | 1 | 1 |
| Aldo-keto reductase family 1 member B10 | Homo sapiens (human) | IC50 | 36.1000 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | IC50 | 22.0646 | 5 | 13 |
| Alpha-1A adrenergic receptor | Sus scrofa (pig) | IC50 | 0.0600 | 1 | 1 |
| Alpha-glucosidase MAL32 | Saccharomyces cerevisiae S288C | IC50 | 61.0000 | 1 | 2 |
| Alpha-mannosidase | Canavalia ensiformis (jack bean) | IC50 | 49.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 5.7920 | 6 | 8 |
| Amine oxidase [flavin-containing] A | Bos taurus (cattle) | IC50 | 95.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Rattus norvegicus (Norway rat) | IC50 | 40.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Bos taurus (cattle) | IC50 | 95.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | IC50 | 3.0880 | 4 | 5 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Ki | 1.0000 | 1 | 1 |
| Androgen receptor | Homo sapiens (human) | IC50 | 1,450.0000 | 1 | 2 |
| Androgen receptor | Rattus norvegicus (Norway rat) | IC50 | 85.1138 | 1 | 1 |
| Angiopoietin-1 receptor | Homo sapiens (human) | IC50 | 0.3105 | 15 | 15 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | IC50 | 243,576.9100 | 3 | 3 |
| Angiotensin-converting enzyme | Homo sapiens (human) | Ki | 715.0000 | 1 | 1 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Arginase-1 | Bos taurus (cattle) | IC50 | 47.0000 | 1 | 1 |
| Arginase-1 | Homo sapiens (human) | IC50 | 622.5000 | 2 | 2 |
| Arginase-1 | Bos taurus (cattle) | Ki | 136.0000 | 3 | 3 |
| Aromatase | Homo sapiens (human) | IC50 | 2,606,492,330.3768 | 7 | 13 |
| Aromatase | Homo sapiens (human) | Ki | 45.1667 | 5 | 6 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 5 |
| ATP-citrate synthase | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 4 | 4 |
| ATP-dependent molecular chaperone HSC82 | Saccharomyces cerevisiae S288C | IC50 | 0.2000 | 1 | 1 |
| ATP-dependent molecular chaperone HSP82 | Saccharomyces cerevisiae S288C | IC50 | 0.1192 | 3 | 4 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 6.9145 | 4 | 4 |
| Aurora kinase A | Homo sapiens (human) | IC50 | 24.6718 | 6 | 13 |
| Aurora kinase B | Homo sapiens (human) | IC50 | 34.3761 | 2 | 9 |
| Aurora kinase C | Homo sapiens (human) | IC50 | 37.8625 | 1 | 8 |
| BCR/ABL p210 fusion protein | Homo sapiens (human) | GI50 | 0.2700 | 1 | 1 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | IC50 | 0.0270 | 1 | 1 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 7.5000 | 1 | 2 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 2.3700 | 1 | 1 |
| Bifunctional epoxide hydrolase 2 | Homo sapiens (human) | IC50 | 12.1375 | 2 | 3 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 34.4222 | 6 | 18 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | IC50 | 111.6000 | 1 | 1 |
| Breakpoint cluster region protein | Homo sapiens (human) | GI50 | 1.0636 | 28 | 89 |
| Breakpoint cluster region protein | Mus musculus (house mouse) | GI50 | 0.0010 | 1 | 1 |
| Breakpoint cluster region protein | Homo sapiens (human) | IC50 | 1.7575 | 49 | 72 |
| Breakpoint cluster region protein | Homo sapiens (human) | Ki | 0.0140 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 3.0749 | 15 | 16 |
| Calcium dependent protein kinase | Triticum aestivum (bread wheat) | IC50 | 19.0000 | 1 | 1 |
| Calcium release-activated calcium channel protein 1 | Homo sapiens (human) | IC50 | 4.3000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | IC50 | 0.0920 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | IC50 | 0.0525 | 1 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | IC50 | 0.1840 | 1 | 1 |
| cAMP-dependent protein kinase | Oryctolagus cuniculus (rabbit) | IC50 | 500.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | IC50 | 39.5681 | 3 | 9 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 5 |
| Carbonic anhydrase 1 | Homo sapiens (human) | Ki | 5.0153 | 3 | 4 |
| Carbonic anhydrase 12 | Homo sapiens (human) | Ki | 0.4448 | 2 | 3 |
| Carbonic anhydrase 13 | Mus musculus (house mouse) | Ki | 6.0575 | 1 | 2 |
| Carbonic anhydrase 14 | Homo sapiens (human) | Ki | 0.3455 | 1 | 2 |
| Carbonic anhydrase 15 | Mus musculus (house mouse) | Ki | 0.0785 | 1 | 2 |
| Carbonic anhydrase 2 | Homo sapiens (human) | IC50 | 0.2000 | 1 | 2 |
| Carbonic anhydrase 2 | Homo sapiens (human) | Ki | 5.0086 | 3 | 4 |
| Carbonic anhydrase 3 | Homo sapiens (human) | Ki | 0.4855 | 1 | 2 |
| Carbonic anhydrase 4 | Homo sapiens (human) | Ki | 4.0258 | 2 | 3 |
| Carbonic anhydrase 5A, mitochondrial | Homo sapiens (human) | Ki | 12.8425 | 1 | 2 |
| Carbonic anhydrase 5B, mitochondrial | Homo sapiens (human) | Ki | 15.9625 | 1 | 2 |
| Carbonic anhydrase 6 | Homo sapiens (human) | Ki | 0.4265 | 1 | 2 |
| Carbonic anhydrase 7 | Homo sapiens (human) | Ki | 2.1790 | 3 | 4 |
| Carbonic anhydrase 9 | Homo sapiens (human) | Ki | 2.5317 | 3 | 4 |
| Carbonyl reductase [NADPH] 1 | Homo sapiens (human) | IC50 | 7.9900 | 1 | 2 |
| Carbonyl reductase [NADPH] 1 | Homo sapiens (human) | Ki | 1.2750 | 1 | 2 |
| Carboxylic ester hydrolase | Rattus norvegicus (Norway rat) | IC50 | 50.0000 | 1 | 1 |
| Casein kinase I isoform alpha | Homo sapiens (human) | IC50 | 0.1255 | 1 | 2 |
| Casein kinase I isoform delta | Homo sapiens (human) | IC50 | 0.1500 | 1 | 1 |
| Casein kinase II subunit alpha | Homo sapiens (human) | IC50 | 1.0112 | 8 | 8 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Ki | 9.4200 | 5 | 5 |
| Casein kinase II subunit alpha | Zea mays | Ki | 1.8500 | 1 | 1 |
| Casein kinase II subunit alpha 3 | Homo sapiens (human) | Ki | 1.9000 | 1 | 1 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | IC50 | 1.0400 | 4 | 4 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Ki | 1.9000 | 1 | 1 |
| Casein kinase II subunit beta | Homo sapiens (human) | IC50 | 0.8667 | 6 | 6 |
| Casein kinase II subunit beta | Homo sapiens (human) | Ki | 1.9000 | 1 | 1 |
| Chain A [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 1 | Homo sapiens (human) | IC50 | 400.0000 | 1 | 1 |
| Chain A [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 3 | Homo sapiens (human) | IC50 | 400.0000 | 1 | 1 |
| Chain A, Casein kinase II, alpha chain | Zea mays | Ki | 1.8500 | 1 | 1 |
| Chain A, Epidermal growth factor receptor | Homo sapiens (human) | Ki | 0.0030 | 1 | 1 |
| Chain A, Estrogen receptor 1 (alpha) | Homo sapiens (human) | IC50 | 0.0090 | 1 | 1 |
| Chain A, PROTEIN KINASE CK2, ALPHA SUBUNIT | Zea mays | IC50 | 1.0000 | 1 | 1 |
| Chain A, PROTO-ONCOGENE TYROSINE-PROTEIN KINASE ABL | Mus musculus (house mouse) | IC50 | 0.1000 | 1 | 1 |
| Chain A, Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 0.0024 | 1 | 6 |
| Chain A, Tyrosine-protein kinase SYK | Homo sapiens (human) | Ki | 5.0000 | 1 | 1 |
| Chain A, VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2 | Homo sapiens (human) | Ki | 0.0005 | 1 | 15 |
| Coiled-coil domain-containing protein 6 | Homo sapiens (human) | GI50 | 0.0290 | 1 | 1 |
| Coiled-coil domain-containing protein 6 | Homo sapiens (human) | IC50 | 0.2808 | 3 | 4 |
| Cruzipain | Trypanosoma cruzi | IC50 | 246.6750 | 4 | 4 |
| Cyclin-C | Homo sapiens (human) | IC50 | 0.0662 | 2 | 2 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 62.9909 | 4 | 11 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | IC50 | 0.2060 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 39.6383 | 14 | 24 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | IC50 | 85.3333 | 3 | 3 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | IC50 | 0.1300 | 1 | 1 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | IC50 | 2.0165 | 10 | 10 |
| Cytochrome P450 1A1 | Homo sapiens (human) | IC50 | 12.2500 | 1 | 1 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 13.3034 | 5 | 5 |
| Cytochrome P450 2A6 | Homo sapiens (human) | IC50 | 35.0000 | 1 | 1 |
| Cytochrome P450 2B6 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 25.0185 | 2 | 2 |
| Cytochrome P450 2C8 | Homo sapiens (human) | IC50 | 0.0370 | 1 | 1 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 25.0150 | 2 | 2 |
| Cytochrome P450 2E1 | Homo sapiens (human) | IC50 | 0.0140 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 3.2366 | 5 | 7 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Ki | 14.3000 | 1 | 1 |
| Cytochrome P450 3A5 | Homo sapiens (human) | IC50 | 0.3000 | 1 | 2 |
| Cytochrome P450 3A5 | Homo sapiens (human) | Ki | 37.6000 | 1 | 1 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | IC50 | 13.7294 | 5 | 5 |
| D(1A) dopamine receptor | Sus scrofa (pig) | IC50 | 0.0600 | 1 | 1 |
| Death-associated protein kinase 1 | Homo sapiens (human) | IC50 | 98.0000 | 1 | 1 |
| Dihydrofolate reductase | Escherichia coli K-12 | IC50 | 0.2000 | 1 | 2 |
| Dihydrofolate reductase | Homo sapiens (human) | IC50 | 0.3880 | 1 | 1 |
| Dihydroorotate dehydrogenase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 98.8725 | 4 | 4 |
| Dihydroorotate dehydrogenase | Schistosoma mansoni | IC50 | 50.0000 | 2 | 2 |
| Dihydroorotate dehydrogenase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 22.6750 | 2 | 2 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | IC50 | 1.5822 | 23 | 23 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Mus musculus (house mouse) | IC50 | 0.1030 | 4 | 5 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 0.0160 | 6 | 7 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | Ki | 0.9207 | 3 | 3 |
| Dipeptidyl peptidase 1 | Homo sapiens (human) | IC50 | 4.2250 | 2 | 4 |
| Dipeptidyl peptidase 3 | Homo sapiens (human) | IC50 | 36.6000 | 1 | 1 |
| Dipeptidyl peptidase 4 | Homo sapiens (human) | IC50 | 0.4800 | 1 | 1 |
| Dipeptidyl peptidase 4 | Rattus norvegicus (Norway rat) | IC50 | 27.3333 | 1 | 3 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | GI50 | 5.5250 | 2 | 4 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | IC50 | 0.1294 | 10 | 24 |
| DNA (cytosine-5)-methyltransferase 1 | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| DNA (cytosine-5)-methyltransferase 3-like | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| DNA (cytosine-5)-methyltransferase 3A | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| DNA-dependent protein kinase catalytic subunit | Homo sapiens (human) | IC50 | 33.3533 | 1 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | IC50 | 1.6670 | 3 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | IC50 | 1.7000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | IC50 | 0.4000 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli K-12 | IC50 | 30.0000 | 1 | 1 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 12.5000 | 1 | 1 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 2.8280 | 3 | 3 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | IC50 | 0.1430 | 1 | 1 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | IC50 | 1.4546 | 3 | 7 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | IC50 | 0.0065 | 1 | 2 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | IC50 | 0.4006 | 7 | 10 |
| Epidermal growth factor receptor | Homo sapiens (human) | GI50 | 0.6276 | 7 | 7 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 3.3065 | 252 | 307 |
| Epidermal growth factor receptor | Homo sapiens (human) | Ki | 0.0544 | 3 | 3 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | GI50 | 4.2750 | 2 | 4 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | IC50 | 1.9277 | 8 | 17 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Estrogen receptor | Homo sapiens (human) | IC50 | 1.3997 | 23 | 26 |
| Estrogen receptor | Homo sapiens (human) | Ki | 0.3930 | 2 | 3 |
| Estrogen receptor beta | Homo sapiens (human) | IC50 | 2.1691 | 24 | 28 |
| Estrogen receptor beta | Homo sapiens (human) | Ki | 0.5082 | 2 | 3 |
| Fatty-acid amide hydrolase 1 | Rattus norvegicus (Norway rat) | IC50 | 6.1000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | IC50 | 1.1384 | 32 | 46 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Ki | 0.0560 | 1 | 1 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | IC50 | 0.0364 | 4 | 4 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | IC50 | 0.0099 | 3 | 3 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | IC50 | 0.0058 | 3 | 3 |
| Fibronectin | Homo sapiens (human) | IC50 | 1.9400 | 1 | 3 |
| Focal adhesion kinase 1 | Homo sapiens (human) | IC50 | 25.2690 | 2 | 2 |
| G1/S-specific cyclin-D1 | Homo sapiens (human) | IC50 | 126.5000 | 2 | 2 |
| G1/S-specific cyclin-E1 | Homo sapiens (human) | IC50 | 66.0000 | 5 | 5 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 190.0000 | 2 | 2 |
| Genome polyprotein | Dengue virus 2 Puerto Rico/PR159-S1/1969 | IC50 | 48.3350 | 2 | 2 |
| Genome polyprotein | Human rhinovirus sp. | IC50 | 150.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | IC50 | 0.0016 | 1 | 1 |
| Glycogen phosphorylase, muscle form | Homo sapiens (human) | IC50 | 0.0012 | 1 | 1 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 16.4357 | 3 | 7 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | IC50 | 0.2092 | 5 | 5 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Ki | 20.0000 | 1 | 1 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | IC50 | 0.1148 | 6 | 6 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Ki | 20.0000 | 1 | 1 |
| Heme oxygenase 1 | Rattus norvegicus (Norway rat) | IC50 | 1.2200 | 1 | 2 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 0.2577 | 29 | 31 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | IC50 | 0.0278 | 3 | 4 |
| Histamine H2 receptor | Homo sapiens (human) | IC50 | 1.9630 | 1 | 1 |
| Histamine H2 receptor | Homo sapiens (human) | Ki | 1.9300 | 1 | 1 |
| Histidine kinase | Caulobacter vibrioides | IC50 | 184.0000 | 1 | 1 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 40.0000 | 6 | 6 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 28.0000 | 5 | 5 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 40.0000 | 6 | 6 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 28.0000 | 5 | 5 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | IC50 | 0.0515 | 2 | 2 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Insulin receptor | Homo sapiens (human) | GI50 | 0.7450 | 1 | 2 |
| Insulin receptor | Homo sapiens (human) | IC50 | 30.5750 | 3 | 4 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | GI50 | 0.7450 | 1 | 2 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 17.2857 | 7 | 7 |
| Integrase | Human immunodeficiency virus 1 | IC50 | 16.2105 | 5 | 5 |
| Integrin alpha-IIb | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| Integrin beta-3 | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | IC50 | 0.5740 | 1 | 1 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 4.5000 | 1 | 1 |
| Kinesin-1 heavy chain | Homo sapiens (human) | GI50 | 0.0870 | 1 | 1 |
| Kinesin-1 heavy chain | Homo sapiens (human) | IC50 | 0.2950 | 1 | 2 |
| L-lactate dehydrogenase A chain | Rattus norvegicus (Norway rat) | Ki | 14.3000 | 1 | 1 |
| Lactoylglutathione lyase | Homo sapiens (human) | IC50 | 0.7600 | 1 | 1 |
| large T antigen | Betapolyomavirus macacae | IC50 | 16.3500 | 1 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 24.8150 | 1 | 4 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| LIM domain kinase 1 | Homo sapiens (human) | IC50 | 0.6097 | 5 | 5 |
| LIM domain kinase 2 | Homo sapiens (human) | IC50 | 0.5186 | 4 | 4 |
| Low-density lipoprotein receptor | Homo sapiens (human) | IC50 | 9.8000 | 1 | 1 |
| Lysine-specific histone demethylase 1A | Homo sapiens (human) | IC50 | 2.9500 | 3 | 3 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | GI50 | 0.1100 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | IC50 | 0.3813 | 12 | 14 |
| Macrophage colony-stimulating factor 1 receptor | Mus musculus (house mouse) | IC50 | 0.5340 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | IC50 | 1.7195 | 2 | 2 |
| Maltase-glucoamylase, intestinal | Homo sapiens (human) | IC50 | 6.5050 | 2 | 2 |
| Maltase-glucoamylase, intestinal | Homo sapiens (human) | Ki | 10.4000 | 1 | 1 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.2620 | 1 | 1 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | GI50 | 2.4701 | 91 | 125 |
| Mast/stem cell growth factor receptor Kit | Mus musculus (house mouse) | GI50 | 0.3500 | 1 | 1 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | IC50 | 4.1466 | 75 | 98 |
| melanocortin receptor 4 | Homo sapiens (human) | IC50 | 67.1000 | 2 | 2 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | IC50 | 0.3137 | 4 | 6 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Ki | 0.1218 | 4 | 9 |
| Misshapen-like kinase 1 | Homo sapiens (human) | IC50 | 0.0220 | 1 | 1 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | IC50 | 0.1095 | 1 | 1 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 61.4000 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | IC50 | 17.5750 | 3 | 4 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | IC50 | 17.5750 | 3 | 4 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | IC50 | 17.5750 | 3 | 4 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 15.6495 | 14 | 16 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | IC50 | 0.0181 | 1 | 1 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | IC50 | 0.3200 | 2 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | IC50 | 0.0099 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | IC50 | 0.0003 | 1 | 1 |
| MO15-related protein kinase Pfmrk | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 93.0000 | 1 | 1 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 16.0000 | 1 | 1 |
| Multidrug and toxin extrusion protein 1 | Homo sapiens (human) | IC50 | 0.1467 | 3 | 3 |
| Multidrug and toxin extrusion protein 2 | Homo sapiens (human) | IC50 | 1.6250 | 2 | 2 |
| Multidrug resistance-associated protein 1 | Rattus norvegicus (Norway rat) | Ki | 0.0597 | 3 | 8 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 64.8800 | 1 | 5 |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | IC50 | 0.4000 | 1 | 1 |
| Myelin transcription factor 1 | Homo sapiens (human) | IC50 | 0.0630 | 1 | 1 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | IC50 | 12.0000 | 2 | 2 |
| Neuraminidase | Influenza A virus (A/Wilson-Smith/1933(H1N1)) | IC50 | 98.2667 | 3 | 3 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 52.0000 | 1 | 1 |
| NF-kappa-B essential modulator | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | IC50 | 0.0250 | 1 | 1 |
| Nuclear factor NF-kappa-B p100 subunit | Homo sapiens (human) | IC50 | 38.0000 | 1 | 1 |
| Nuclear factor NF-kappa-B p105 subunit | Homo sapiens (human) | IC50 | 38.0000 | 1 | 1 |
| Nucleophosmin | Homo sapiens (human) | IC50 | 23.8208 | 4 | 12 |
| Ornithine decarboxylase | Homo sapiens (human) | IC50 | 26.0000 | 1 | 1 |
| Oxysterols receptor LXR-alpha | Homo sapiens (human) | IC50 | 46.0000 | 3 | 4 |
| Oxysterols receptor LXR-beta | Homo sapiens (human) | IC50 | 48.0000 | 2 | 3 |
| P2Y purinoceptor 12 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Pancreatic triacylglycerol lipase | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 2 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | IC50 | 0.0600 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 18.9008 | 3 | 5 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | IC50 | 33.8000 | 1 | 3 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | IC50 | 32.5375 | 1 | 4 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | IC50 | 33.7000 | 1 | 3 |
| Phospholipase D | Streptomyces chromofuscus | IC50 | 0.0650 | 1 | 1 |
| Phospholipase D1 | Homo sapiens (human) | IC50 | 0.3870 | 1 | 3 |
| Phospholipase D2 | Homo sapiens (human) | IC50 | 0.3870 | 1 | 3 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | GI50 | 1.4081 | 6 | 8 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | IC50 | 3.5130 | 24 | 25 |
| Platelet-derived growth factor receptor alpha | Rattus norvegicus (Norway rat) | IC50 | 4.0000 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Mus musculus (house mouse) | IC50 | 50.1500 | 2 | 2 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | GI50 | 0.0422 | 3 | 4 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | IC50 | 6.3377 | 29 | 36 |
| Platelet-derived growth factor receptor beta | Mus musculus (house mouse) | IC50 | 10.1288 | 4 | 10 |
| Platelet-derived growth factor receptor beta | Rattus norvegicus (Norway rat) | IC50 | 2.0810 | 2 | 2 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 32.5000 | 4 | 4 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | IC50 | 0.6700 | 2 | 2 |
| Polyunsaturated fatty acid 5-lipoxygenase | Rattus norvegicus (Norway rat) | IC50 | 0.0046 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | IC50 | 9.0330 | 1 | 1 |
| Potassium voltage-gated channel subfamily D member 3 | Homo sapiens (human) | IC50 | 1,739.2540 | 2 | 2 |
| Potassium voltage-gated channel subfamily E member 1 | Homo sapiens (human) | IC50 | 300.1617 | 3 | 3 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 7,758.8296 | 12 | 13 |
| Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens (human) | IC50 | 300.1617 | 3 | 3 |
| Potassium-transporting ATPase alpha chain 1 | Rattus norvegicus (Norway rat) | IC50 | 4.5000 | 1 | 1 |
| Potassium-transporting ATPase subunit beta | Rattus norvegicus (Norway rat) | IC50 | 4.5000 | 1 | 1 |
| Procathepsin L | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Proprotein convertase subtilisin/kexin type 9 | Homo sapiens (human) | IC50 | 9.8000 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Homo sapiens (human) | IC50 | 80.0000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | IC50 | 0.0270 | 1 | 1 |
| Proteasome subunit beta type-1 | Homo sapiens (human) | IC50 | 0.2400 | 1 | 1 |
| Proteasome subunit beta type-2 | Homo sapiens (human) | IC50 | 20.8500 | 1 | 1 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 25.1600 | 3 | 3 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 62.2727 | 5 | 11 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 80.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 76.6667 | 3 | 3 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 60.0070 | 3 | 3 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 80.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 90.0000 | 2 | 2 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 90.0000 | 2 | 2 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 80.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 65.0000 | 2 | 2 |
| Protein tyrosine phosphatase type IVA 3 | Homo sapiens (human) | IC50 | 22.1667 | 3 | 3 |
| Protein-arginine deiminase type-4 | Homo sapiens (human) | IC50 | 2,400.0000 | 1 | 1 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | IC50 | 0.1340 | 1 | 1 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | IC50 | 0.0072 | 2 | 2 |
| Proto-oncogene tyrosine-protein kinase LCK | Mus musculus (house mouse) | IC50 | 0.3735 | 2 | 3 |
| Proto-oncogene tyrosine-protein kinase LCK | Mus musculus (house mouse) | Ki | 0.0001 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | GI50 | 0.2669 | 13 | 13 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 0.4992 | 48 | 70 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | GI50 | 0.8568 | 1 | 3 |
| Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | IC50 | 0.5229 | 6 | 9 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 5.2017 | 73 | 92 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Ki | 18.6001 | 5 | 5 |
| Proto-oncogene tyrosine-protein kinase Src | Rattus norvegicus (Norway rat) | IC50 | 0.1800 | 1 | 1 |
| Quinolone resistance protein NorA | Staphylococcus aureus | IC50 | 11.5000 | 1 | 1 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 60.0000 | 2 | 2 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 0.1537 | 32 | 36 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Ki | 0.0060 | 1 | 1 |
| Receptor protein-tyrosine kinase | Homo sapiens (human) | IC50 | 2.2043 | 1 | 3 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 0.0923 | 69 | 84 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | IC50 | 0.0151 | 2 | 3 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | IC50 | 0.1419 | 11 | 17 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | IC50 | 0.7794 | 5 | 5 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.6611 | 4 | 6 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | IC50 | 4.8411 | 3 | 3 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | GI50 | 3.1330 | 3 | 3 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 1.9028 | 35 | 39 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | IC50 | 10.0000 | 1 | 1 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 10.0000 | 2 | 2 |
| Replicase polyprotein 1ab | Human coronavirus 229E | IC50 | 10.0000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 6.2500 | 2 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | IC50 | 0.5412 | 3 | 5 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Ki | 0.0390 | 1 | 1 |
| RuvB-like 1 | Homo sapiens (human) | IC50 | 66.0000 | 1 | 1 |
| RuvB-like 2 | Homo sapiens (human) | IC50 | 66.0000 | 1 | 1 |
| SAFB-like transcription modulator | Homo sapiens (human) | IC50 | 0.0013 | 1 | 1 |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max (soybean) | IC50 | 100.0000 | 1 | 1 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | IC50 | 0.0520 | 1 | 1 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | IC50 | 0.0039 | 1 | 1 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | IC50 | 0.1910 | 1 | 1 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | IC50 | 0.0087 | 3 | 3 |
| Serine/threonine-protein kinase ATR | Homo sapiens (human) | IC50 | 1.4200 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | GI50 | 1.0000 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | IC50 | 1.7836 | 63 | 69 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Ki | 0.0327 | 3 | 3 |
| Serine/threonine-protein kinase B-raf | Mus musculus (house mouse) | IC50 | 0.1300 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 20.5408 | 3 | 4 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | IC50 | 0.7860 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 40.3080 | 2 | 2 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | IC50 | 15.8383 | 4 | 6 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | IC50 | 0.2740 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 2.5000 | 1 | 1 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | IC50 | 41.2900 | 3 | 10 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Ki | 15.8704 | 1 | 12 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Ki | 15.8704 | 1 | 12 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Ki | 15.8704 | 1 | 12 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | IC50 | 0.0450 | 3 | 3 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Ki | 12.6971 | 4 | 15 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | IC50 | 0.0010 | 1 | 1 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | IC50 | 0.0030 | 1 | 1 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | IC50 | 0.0050 | 1 | 1 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | IC50 | 0.5370 | 2 | 3 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | IC50 | 0.1750 | 2 | 2 |
| Sialidase | Clostridium perfringens | IC50 | 12.0500 | 1 | 1 |
| Sialidase-2 | Homo sapiens (human) | IC50 | 570.0000 | 1 | 2 |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus (Norway rat) | Ki | 14.3000 | 1 | 1 |
| Signal transducer and activator of transcription 3 | Homo sapiens (human) | IC50 | 24.8000 | 1 | 1 |
| Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | IC50 | 15.0000 | 2 | 4 |
| Smoothened homolog | Homo sapiens (human) | Ki | 0.0462 | 1 | 1 |
| Sodium channel protein type 5 subunit alpha | Homo sapiens (human) | IC50 | 1,934.4514 | 5 | 5 |
| Sodium- and chloride-dependent GABA transporter 1 | Rattus norvegicus (Norway rat) | IC50 | 0.0013 | 1 | 1 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | IC50 | 9.9010 | 1 | 2 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | Ki | 7.8665 | 1 | 2 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 4.6300 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 4.5910 | 1 | 1 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | IC50 | 1.4020 | 1 | 1 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | IC50 | 0.1980 | 2 | 2 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 0.7450 | 1 | 1 |
| Solute carrier family 2, facilitated glucose transporter member 1 | Homo sapiens (human) | Ki | 7.0000 | 3 | 3 |
| Solute carrier family 2, facilitated glucose transporter member 4 | Mus musculus (house mouse) | IC50 | 6.8383 | 2 | 3 |
| Solute carrier family 22 member 1 | Homo sapiens (human) | IC50 | 107.0000 | 1 | 1 |
| Solute carrier family 22 member 2 | Homo sapiens (human) | IC50 | 4.2000 | 1 | 1 |
| Solute carrier family 22 member 3 | Homo sapiens (human) | IC50 | 13.0000 | 2 | 2 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | IC50 | 9.1201 | 1 | 1 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | Ki | 5.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | IC50 | 3.8904 | 1 | 1 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | Ki | 2.9600 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | IC50 | 10.0000 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome coronavirus 2 | IC50 | 200.0000 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | IC50 | 10.0000 | 1 | 1 |
| Steroid hormone receptor ERR1 | Homo sapiens (human) | IC50 | 0.0100 | 1 | 1 |
| Steroid hormone receptor ERR2 | Homo sapiens (human) | IC50 | 0.3950 | 1 | 1 |
| Stromal interaction molecule 1 | Homo sapiens (human) | IC50 | 4.3000 | 1 | 1 |
| Substance-K receptor | Cavia porcellus (domestic guinea pig) | IC50 | 77.1000 | 1 | 1 |
| Substance-P receptor | Cavia porcellus (domestic guinea pig) | IC50 | 77.1000 | 1 | 1 |
| Synaptic vesicular amine transporter | Rattus norvegicus (Norway rat) | IC50 | 0.1000 | 1 | 1 |
| Testosterone 17-beta-dehydrogenase 3 | Homo sapiens (human) | IC50 | 20.5500 | 1 | 2 |
| Thromboxane-A synthase | Homo sapiens (human) | IC50 | 3.9590 | 1 | 2 |
| Tissue alpha-L-fucosidase | Bos taurus (cattle) | IC50 | 43.0000 | 1 | 2 |
| Transcription factor p65 | Homo sapiens (human) | IC50 | 38.0000 | 1 | 1 |
| Transmembrane protease serine 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Transthyretin | Homo sapiens (human) | IC50 | 53.9000 | 2 | 2 |
| Triosephosphate isomerase | Oryctolagus cuniculus (rabbit) | Ki | 67.5000 | 1 | 2 |
| Tubulin beta-2B chain | Bos taurus (cattle) | IC50 | 15.0000 | 2 | 2 |
| Tyrosinase | Mus musculus (house mouse) | IC50 | 500.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | GI50 | 1.1306 | 30 | 93 |
| Tyrosine-protein kinase ABL1 | Mus musculus (house mouse) | GI50 | 0.0010 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 24.3882 | 170 | 265 |
| Tyrosine-protein kinase ABL1 | Mus musculus (house mouse) | IC50 | 7.8278 | 3 | 6 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Ki | 0.8863 | 8 | 8 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | IC50 | 8.6164 | 7 | 7 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | GI50 | 3.8512 | 2 | 4 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | IC50 | 0.0395 | 2 | 2 |
| Tyrosine-protein kinase Blk | Mus musculus (house mouse) | IC50 | 0.0076 | 1 | 2 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | IC50 | 0.0431 | 7 | 7 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | IC50 | 29.7964 | 5 | 12 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | IC50 | 0.4900 | 1 | 1 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | IC50 | 0.3580 | 1 | 1 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | IC50 | 0.0011 | 1 | 1 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | IC50 | 0.0018 | 2 | 2 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 5.1006 | 11 | 12 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | GI50 | 4.6130 | 1 | 3 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | IC50 | 0.1787 | 3 | 6 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | IC50 | 2.9390 | 2 | 2 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | IC50 | 0.0322 | 1 | 1 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | IC50 | 0.1690 | 1 | 1 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | IC50 | 2.9400 | 2 | 2 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | GI50 | 2.8428 | 2 | 4 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 6.5387 | 21 | 24 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | IC50 | 0.1901 | 8 | 8 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | IC50 | 1.3700 | 1 | 1 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | IC50 | 0.5145 | 13 | 13 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | IC50 | 15.2674 | 5 | 7 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Ki | 5.0000 | 2 | 2 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | IC50 | 0.2895 | 2 | 2 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | IC50 | 0.0202 | 1 | 2 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | IC50 | 0.0009 | 7 | 9 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | IC50 | 0.5641 | 28 | 35 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | GI50 | 6.0234 | 4 | 5 |
| Vascular endothelial growth factor receptor 2 | Danio rerio (zebrafish) | IC50 | 2.6000 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 2.0971 | 173 | 210 |
| Vascular endothelial growth factor receptor 2 | Mus musculus (house mouse) | IC50 | 0.1005 | 3 | 9 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Ki | 0.0065 | 4 | 4 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | IC50 | 0.0638 | 14 | 19 |
| Vascular endothelial growth factor receptor 3 | Mus musculus (house mouse) | IC50 | 0.1112 | 2 | 8 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | IC50 | 2,742.6327 | 8 | 8 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | IC50 | 42.9000 | 2 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | IC50 | 42.9000 | 2 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | IC50 | 42.9000 | 2 | 2 |
| Xanthine dehydrogenase/oxidase | Bos taurus (cattle) | IC50 | 1.5150 | 2 | 2 |
| Xanthine dehydrogenase/oxidase | Homo sapiens (human) | IC50 | 616.2500 | 2 | 2 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial | Homo sapiens (human) | Kd | 12.4154 | 1 | 3 |
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 18.4610 | 5 | 41 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 29.2343 | 1 | 18 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 15.9230 | 4 | 40 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 17.9786 | 4 | 42 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 18.1408 | 4 | 42 |
| Activin receptor type-2A | Homo sapiens (human) | Kd | 8.6559 | 3 | 22 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 17.4057 | 4 | 41 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 14 |
| Adenosine kinase | Homo sapiens (human) | Kd | 28.5274 | 1 | 18 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 28.3337 | 1 | 18 |
| Albumin | Homo sapiens (human) | Kd | 78.6400 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | EC50 | 6.2580 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 10.6796 | 4 | 25 |
| Angiopoietin-1 receptor | Homo sapiens (human) | Kd | 5.6954 | 4 | 24 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | EC50 | 62.5093 | 1 | 7 |
| Ankyrin repeat and protein kinase domain-containing protein 1 | Homo sapiens (human) | Kd | 9.3500 | 3 | 22 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 17.1147 | 5 | 43 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| ATP-dependent molecular chaperone HSP82 | Saccharomyces cerevisiae S288C | Kd | 0.0190 | 1 | 1 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 28.4256 | 1 | 19 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 28.3575 | 1 | 18 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 14 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 13 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | EC50 | 2.7900 | 1 | 1 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | Kd | 26.3027 | 1 | 1 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 17.8851 | 4 | 41 |
| Atypical kinase COQ8B, mitochondrial | Homo sapiens (human) | Kd | 8.1921 | 3 | 22 |
| Aurora kinase A | Homo sapiens (human) | Kd | 17.1017 | 5 | 42 |
| Aurora kinase B | Homo sapiens (human) | Kd | 17.3163 | 4 | 41 |
| Aurora kinase C | Homo sapiens (human) | Kd | 5.6231 | 4 | 23 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | Kd | 8.0905 | 3 | 22 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 16.3718 | 5 | 41 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 18.9554 | 4 | 41 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 19.2969 | 3 | 33 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 18.7645 | 4 | 40 |
| Breakpoint cluster region protein | Homo sapiens (human) | EC50 | 1.3483 | 4 | 9 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 11.2637 | 1 | 19 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | EC50 | 3.2000 | 1 | 1 |
| Calcium-dependent protein kinase 1 | Plasmodium falciparum 3D7 | Kd | 6.8086 | 1 | 14 |
| Calcium/calmodulin-dependent protein kinase kinase 1 | Homo sapiens (human) | Kd | 9.6091 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 18.4297 | 4 | 42 |
| Calcium/calmodulin-dependent protein kinase type 1 | Homo sapiens (human) | Kd | 9.2818 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | Kd | 9.3705 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 10.3364 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | Kd | 9.7500 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 18.6244 | 5 | 41 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 19.2683 | 4 | 41 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 19.5000 | 3 | 40 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 19.0980 | 4 | 43 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| cAMP-dependent protein kinase catalytic subunit PRKX | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 21.1509 | 3 | 35 |
| Casein kinase I isoform alpha-like | Homo sapiens (human) | Kd | 9.6476 | 2 | 21 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 18.5304 | 4 | 42 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 16.2223 | 5 | 41 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 17.9093 | 4 | 39 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 19.7163 | 4 | 43 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 18.1661 | 4 | 40 |
| Cell division control protein 2 homolog | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 14 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 10 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| cGMP-dependent protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Chain A, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase | Helicobacter pylori | Kd | 0.4500 | 1 | 1 |
| Chain A, Atp-dependent Molecular Chaperone Hsp82 | Saccharomyces cerevisiae (brewer's yeast) | Kd | 0.0900 | 1 | 2 |
| Chain A, HEAT SHOCK PROTEIN 90 | Saccharomyces cerevisiae (brewer's yeast) | Kd | 0.0027 | 1 | 1 |
| Chain A, Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 0.0914 | 1 | 7 |
| Chain A, Transthyretin | Homo sapiens (human) | Kd | 2.1500 | 1 | 4 |
| Chain A, Virulence sensor histidine kinase phoQ | Salmonella enterica subsp. enterica serovar Typhimurium | Kd | 715.0000 | 1 | 1 |
| Chain B, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase | Helicobacter pylori | Kd | 0.4500 | 1 | 1 |
| Chain B, Type 2 DNA topoisomerase 6 subunit B | Saccharolobus shibatae | Kd | 2.0000 | 1 | 1 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 10 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 17.5025 | 4 | 40 |
| Cyclin-C | Homo sapiens (human) | Kd | 0.3100 | 1 | 1 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 28.4774 | 1 | 19 |
| Cyclin-dependent kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Cyclin-dependent kinase 11A | Homo sapiens (human) | Kd | 9.2091 | 3 | 22 |
| Cyclin-dependent kinase 11B | Homo sapiens (human) | Kd | 9.2818 | 3 | 22 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 20.9677 | 2 | 31 |
| Cyclin-dependent kinase 14 | Homo sapiens (human) | Kd | 8.6409 | 3 | 22 |
| Cyclin-dependent kinase 15 | Homo sapiens (human) | Kd | 8.4933 | 2 | 15 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 16.6111 | 4 | 40 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 16.1465 | 4 | 40 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 12.4000 | 4 | 25 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | Kd | 8.2614 | 3 | 22 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 20.2170 | 5 | 41 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 18.4500 | 4 | 41 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 17.9911 | 3 | 49 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 18.0688 | 4 | 41 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | Kd | 8.3148 | 4 | 23 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 19.2683 | 4 | 41 |
| Cyclin-dependent kinase-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Cyclin-dependent kinase-like 2 | Homo sapiens (human) | Kd | 8.0527 | 2 | 15 |
| Cyclin-dependent kinase-like 3 | Homo sapiens (human) | Kd | 8.7320 | 2 | 15 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 18.0000 | 3 | 25 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 17.9512 | 5 | 41 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 9.7211 | 9 | 52 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Cystic fibrosis transmembrane conductance regulator | Homo sapiens (human) | EC50 | 8.2900 | 5 | 5 |
| Cystic fibrosis transmembrane conductance regulator | Rattus norvegicus (Norway rat) | Kd | 40.0000 | 1 | 1 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Cytochrome P450 2D6 | Homo sapiens (human) | Kd | 0.0037 | 1 | 1 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | Kd | 7.2450 | 4 | 23 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Death-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Death-associated protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Death-associated protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 4 | 29 |
| Delta-type opioid receptor | Mus musculus (house mouse) | EC50 | 0.0030 | 1 | 2 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | EC50 | 8.9063 | 1 | 2 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 6.6541 | 8 | 52 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 28.0324 | 1 | 15 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Dual serine/threonine and tyrosine protein kinase | Homo sapiens (human) | Kd | 9.0557 | 1 | 14 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 15.4901 | 4 | 40 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 15.1545 | 4 | 41 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 18.9707 | 4 | 41 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | Kd | 11.6965 | 4 | 26 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 14.1276 | 2 | 32 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 18.6244 | 4 | 41 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | Kd | 7.8814 | 1 | 14 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 14.7915 | 6 | 42 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 17.1189 | 5 | 37 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 15.4727 | 5 | 33 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 14.8147 | 6 | 36 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 16.5427 | 4 | 38 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 15.6300 | 4 | 37 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 26.6669 | 1 | 9 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 20.3779 | 3 | 33 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 12.8000 | 4 | 26 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | Kd | 9.2333 | 2 | 15 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Echinoderm microtubule-associated protein-like 4 | Homo sapiens (human) | EC50 | 6.2580 | 1 | 1 |
| eIF-2-alpha kinase GCN2 | Homo sapiens (human) | Kd | 7.8905 | 3 | 22 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 15 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| endoribonuclease toxin MazF | Escherichia coli str. K-12 substr. MG1655 | EC50 | 99.0000 | 2 | 2 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 11.9665 | 4 | 35 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 11.1805 | 6 | 50 |
| Ephrin type-A receptor 3 | Homo sapiens (human) | Kd | 4.6149 | 4 | 25 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 14.1565 | 5 | 44 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 12.9444 | 6 | 45 |
| Ephrin type-A receptor 6 | Homo sapiens (human) | Kd | 4.1007 | 5 | 26 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 14.3110 | 6 | 39 |
| Ephrin type-A receptor 8 | Homo sapiens (human) | Kd | 3.3705 | 5 | 27 |
| Ephrin type-B receptor 1 | Homo sapiens (human) | Kd | 5.0423 | 4 | 25 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 14.5065 | 4 | 41 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 16.2778 | 4 | 42 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 12.6970 | 5 | 43 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 17.0904 | 3 | 34 |
| Epidermal growth factor receptor | Homo sapiens (human) | EC50 | 0.1210 | 11 | 11 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 5.2635 | 37 | 277 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 7.1976 | 6 | 44 |
| Estrogen receptor | Homo sapiens (human) | EC50 | 0.9980 | 6 | 6 |
| Estrogen receptor | Mus musculus (house mouse) | EC50 | 55.9410 | 1 | 2 |
| Estrogen receptor beta | Homo sapiens (human) | EC50 | 0.1635 | 9 | 9 |
| Estrogen receptor beta | Mus musculus (house mouse) | EC50 | 55.9410 | 1 | 2 |
| Eukaryotic peptide chain release factor GTP-binding subunit ERF3B | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 20.0405 | 2 | 32 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 11 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 21.3473 | 2 | 24 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 15.4145 | 5 | 42 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | Kd | 5.6157 | 4 | 23 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | Kd | 7.0283 | 7 | 45 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | Kd | 8.5632 | 3 | 22 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 18.8407 | 4 | 41 |
| G protein-coupled receptor kinase 4 | Homo sapiens (human) | Kd | 9.1467 | 2 | 15 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 13 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Glycine receptor subunit alpha-1 | Homo sapiens (human) | EC50 | 1.8000 | 1 | 1 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| glycogen synthase kinase-3 beta isoform 1 | Homo sapiens (human) | EC50 | 300.0000 | 1 | 1 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 14 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | EC50 | 0.0250 | 1 | 1 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Kd | 4.1438 | 7 | 9 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | EC50 | 0.0250 | 1 | 1 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Kd | 0.0106 | 2 | 2 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 11.4515 | 9 | 70 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 15.5734 | 5 | 38 |
| Histamine H1 receptor | Rattus norvegicus (Norway rat) | Kd | 0.0027 | 1 | 1 |
| Histone deacetylase 1 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 11 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 2 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 3 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 4 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 5 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 6 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 7 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 8 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Histone deacetylase 9 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | Kd | 8.3280 | 2 | 15 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | Kd | 8.3533 | 2 | 15 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | Kd | 8.2687 | 2 | 15 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | Kd | 5.6037 | 2 | 15 |
| Hormonally up-regulated neu tumor-associated kinase | Homo sapiens (human) | Kd | 8.4667 | 2 | 15 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 18.0223 | 4 | 40 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Insulin receptor | Homo sapiens (human) | Kd | 19.3571 | 4 | 42 |
| Insulin receptor-related protein | Homo sapiens (human) | Kd | 9.7545 | 3 | 22 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 19.5238 | 4 | 42 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 28.3344 | 1 | 18 |
| Interferon-induced, double-stranded RNA-activated protein kinase | Homo sapiens (human) | Kd | 9.1455 | 3 | 22 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 17.9424 | 3 | 35 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 18.6472 | 4 | 42 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 19.6066 | 2 | 33 |
| Isoleucine--tRNA ligase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 12 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 7.7657 | 2 | 28 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | Kd | 8.4545 | 3 | 22 |
| Leukotriene C4 synthase | Cavia porcellus (domestic guinea pig) | Kd | 10.0000 | 1 | 14 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 14.4086 | 5 | 42 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 16.3648 | 4 | 41 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| Lysine--tRNA ligase | Homo sapiens (human) | Kd | 3.1623 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Kd | 2.1478 | 5 | 25 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 19.6343 | 3 | 33 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 15.4299 | 4 | 40 |
| MAP kinase-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 18.7179 | 4 | 39 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 6.5332 | 3 | 22 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 6.1576 | 4 | 25 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 19.0176 | 4 | 42 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 18.1081 | 4 | 37 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | EC50 | 0.5214 | 2 | 2 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Kd | 2.8299 | 29 | 200 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 18.0094 | 4 | 41 |
| matrix metalloproteinase 1, partial | Homo sapiens (human) | EC50 | 5.6500 | 1 | 1 |
| Megakaryocyte-associated tyrosine-protein kinase | Homo sapiens (human) | Kd | 9.7200 | 2 | 15 |
| melanocortin receptor 4 | Homo sapiens (human) | EC50 | 50.0000 | 1 | 1 |
| Membrane-associated progesterone receptor component 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 15.7899 | 5 | 42 |
| Microtubule-associated serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 9.0567 | 2 | 15 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 11.3015 | 3 | 21 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 4 | 44 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 15.4822 | 5 | 41 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 13.8457 | 6 | 42 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | Kd | 9.6826 | 4 | 23 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | Kd | 9.5467 | 2 | 15 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | EC50 | 2.5350 | 2 | 2 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 10.7330 | 11 | 48 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 17.8150 | 4 | 41 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 19.5238 | 4 | 42 |
| Mitogen-activated protein kinase 4 | Homo sapiens (human) | Kd | 9.3864 | 3 | 22 |
| Mitogen-activated protein kinase 6 | Homo sapiens (human) | Kd | 8.0259 | 3 | 22 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 18.5205 | 4 | 39 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 17.6288 | 5 | 42 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 15.8602 | 5 | 44 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 16.1640 | 3 | 33 |
| Mitogen-activated protein kinase kinase kinase 10 | Homo sapiens (human) | Kd | 8.8227 | 3 | 22 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 16.2044 | 5 | 43 |
| Mitogen-activated protein kinase kinase kinase 12 | Homo sapiens (human) | Kd | 8.0529 | 1 | 14 |
| Mitogen-activated protein kinase kinase kinase 13 | Homo sapiens (human) | Kd | 8.4347 | 2 | 15 |
| Mitogen-activated protein kinase kinase kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Mitogen-activated protein kinase kinase kinase 19 | Homo sapiens (human) | Kd | 3.5626 | 2 | 15 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 17.5179 | 3 | 33 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 9.8695 | 4 | 42 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 18.4032 | 3 | 33 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 15.7104 | 5 | 43 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 19.2683 | 4 | 41 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 20.3226 | 3 | 31 |
| Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens (human) | Kd | 6.4929 | 4 | 17 |
| Mitogen-activated protein kinase kinase kinase 9 | Homo sapiens (human) | Kd | 7.8223 | 3 | 22 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 13.7394 | 4 | 40 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 15.2138 | 3 | 35 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 14.5957 | 5 | 42 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 13.9769 | 4 | 42 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 11.7907 | 5 | 44 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Muscle, skeletal receptor tyrosine-protein kinase | Homo sapiens (human) | Kd | 8.6541 | 3 | 22 |
| Myosin light chain kinase 2, skeletal/cardiac muscle | Homo sapiens (human) | Kd | 7.6387 | 4 | 23 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 19.5272 | 2 | 31 |
| Myosin light chain kinase family member 4 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Myosin light chain kinase, smooth muscle | Gallus gallus (chicken) | Kd | 10.0000 | 1 | 7 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 16.7724 | 5 | 42 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Myosin-IIIa | Homo sapiens (human) | Kd | 9.4591 | 3 | 22 |
| Myosin-IIIb | Homo sapiens (human) | Kd | 9.5182 | 3 | 22 |
| Myotonin-protein kinase | Homo sapiens (human) | Kd | 8.6223 | 3 | 22 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 15.5021 | 4 | 42 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 15.3650 | 6 | 56 |
| NT-3 growth factor receptor | Homo sapiens (human) | Kd | 7.8227 | 3 | 22 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | Kd | 9.4273 | 3 | 22 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 18.2915 | 4 | 40 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | EC50 | 55.9410 | 1 | 1 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 13 |
| Peripheral plasma membrane protein CASK | Homo sapiens (human) | Kd | 9.3450 | 1 | 14 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 28.1259 | 1 | 16 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 29.2685 | 1 | 19 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | Kd | 8.7933 | 2 | 15 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | Homo sapiens (human) | Kd | 9.3780 | 2 | 15 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | Homo sapiens (human) | Kd | 9.8333 | 2 | 15 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha | Homo sapiens (human) | Kd | 9.6955 | 3 | 22 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma | Homo sapiens (human) | Kd | 9.4214 | 1 | 14 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | Kd | 10.0000 | 21 | 163 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 18.9980 | 2 | 33 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 16.8996 | 5 | 41 |
| Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | Homo sapiens (human) | Kd | 8.3017 | 4 | 23 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | EC50 | 0.3851 | 2 | 2 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Kd | 2.3569 | 5 | 24 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 9.9496 | 7 | 46 |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | EC50 | 100.0000 | 1 | 1 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Procathepsin L | Homo sapiens (human) | EC50 | 62.5093 | 1 | 7 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Kd | 8.7000 | 1 | 14 |
| Protein cereblon | Homo sapiens (human) | EC50 | 5.0053 | 1 | 2 |
| Protein delta homolog 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 29.0000 | 2 | 20 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 18.7900 | 4 | 40 |
| Protein kinase C epsilon type | Homo sapiens (human) | Kd | 9.6545 | 3 | 22 |
| Protein kinase C eta type | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 21.5152 | 2 | 33 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 18.0405 | 4 | 40 |
| Protein kinase C zeta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 14 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 17.6323 | 4 | 41 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 14.5762 | 5 | 43 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 6.9698 | 12 | 94 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Kd | 8.8655 | 3 | 22 |
| Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | Kd | 0.0075 | 3 | 11 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 12.3914 | 9 | 48 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Rab-like protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 15 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Kd | 5.4979 | 3 | 22 |
| Ras-related C3 botulinum toxin substrate 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 20 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | EC50 | 0.1305 | 6 | 6 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | Kd | 4.6620 | 4 | 24 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | Kd | 5.3691 | 2 | 15 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | Kd | 4.4765 | 3 | 16 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 8.4782 | 3 | 22 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 9.8271 | 5 | 43 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 18.8620 | 1 | 18 |
| Receptor-interacting serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 8.8013 | 2 | 15 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 6.4360 | 31 | 171 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | EC50 | 62.5093 | 1 | 7 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | EC50 | 62.5093 | 1 | 7 |
| Replicase polyprotein 1ab | Human coronavirus 229E | EC50 | 62.5093 | 1 | 7 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | EC50 | 62.5093 | 1 | 7 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | EC50 | 62.5093 | 1 | 7 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 21.1677 | 3 | 35 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 20.4230 | 3 | 33 |
| Rhodopsin kinase GRK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Rhodopsin kinase GRK7 | Homo sapiens (human) | Kd | 9.4467 | 2 | 15 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 15.3323 | 7 | 62 |
| Ribosomal protein S6 kinase alpha-2 | Homo sapiens (human) | Kd | 9.7114 | 6 | 44 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 18.7800 | 4 | 40 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 15.7592 | 7 | 63 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 16.2500 | 7 | 64 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 15.3775 | 7 | 63 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 20.0706 | 3 | 32 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 25.5997 | 1 | 20 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| RuvB-like 2 | Homo sapiens (human) | Kd | 22.0000 | 1 | 1 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| Septin-9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 9.8685 | 6 | 45 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 18.5632 | 4 | 41 |
| Serine/threonine-protein kinase 17A | Homo sapiens (human) | Kd | 8.3267 | 4 | 24 |
| Serine/threonine-protein kinase 17B | Homo sapiens (human) | Kd | 9.4727 | 3 | 22 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 14.9397 | 4 | 33 |
| Serine/threonine-protein kinase 25 | Homo sapiens (human) | Kd | 8.5005 | 3 | 22 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 17.5334 | 4 | 41 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 18.2438 | 4 | 42 |
| Serine/threonine-protein kinase 32A | Homo sapiens (human) | Kd | 8.5214 | 1 | 14 |
| Serine/threonine-protein kinase 32B | Homo sapiens (human) | Kd | 9.4364 | 3 | 22 |
| Serine/threonine-protein kinase 32C | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase 33 | Homo sapiens (human) | Kd | 7.3171 | 3 | 22 |
| serine/threonine-protein kinase 33 isoform a | Homo sapiens (human) | EC50 | 12.7900 | 1 | 1 |
| Serine/threonine-protein kinase 35 | Homo sapiens (human) | Kd | 6.5725 | 2 | 15 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | Kd | 5.6675 | 4 | 24 |
| Serine/threonine-protein kinase 38 | Homo sapiens (human) | Kd | 11.2500 | 3 | 16 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 12.4000 | 4 | 25 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 17.8990 | 4 | 40 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.1924 | 1 | 19 |
| Serine/threonine-protein kinase ATR | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | EC50 | 0.0030 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 11.4280 | 8 | 64 |
| Serine/threonine-protein kinase BRSK1 | Homo sapiens (human) | Kd | 9.7000 | 3 | 22 |
| Serine/threonine-protein kinase BRSK2 | Homo sapiens (human) | Kd | 9.9500 | 3 | 22 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 19.2548 | 4 | 42 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | Kd | 8.7313 | 2 | 15 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | Kd | 9.5827 | 3 | 22 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 18.7775 | 4 | 40 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 18.9512 | 4 | 41 |
| Serine/threonine-protein kinase DCLK1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase DCLK2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase DCLK3 | Homo sapiens (human) | Kd | 9.7909 | 3 | 22 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 20.3226 | 3 | 31 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 19.2683 | 4 | 41 |
| Serine/threonine-protein kinase LATS2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase MAK | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Serine/threonine-protein kinase MARK1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 18.9975 | 4 | 40 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 18.0125 | 4 | 40 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 17.6503 | 4 | 40 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 17.9262 | 4 | 40 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 18.6490 | 4 | 42 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 18.6475 | 4 | 40 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 12 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 19.4833 | 4 | 42 |
| Serine/threonine-protein kinase Nek11 | Homo sapiens (human) | Kd | 8.1514 | 1 | 14 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 17.7605 | 4 | 40 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 21.5412 | 2 | 34 |
| Serine/threonine-protein kinase Nek4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Serine/threonine-protein kinase Nek5 | Homo sapiens (human) | Kd | 9.4632 | 3 | 22 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 17.4286 | 4 | 35 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 19.0000 | 4 | 40 |
| Serine/threonine-protein kinase NIM1 | Homo sapiens (human) | Kd | 9.1933 | 2 | 15 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 16.6764 | 4 | 41 |
| Serine/threonine-protein kinase OSR1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | Kd | 9.2050 | 3 | 22 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 18.8288 | 4 | 41 |
| Serine/threonine-protein kinase PAK 3 | Homo sapiens (human) | Kd | 9.8045 | 3 | 22 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 18.6963 | 4 | 42 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 15.7258 | 4 | 31 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 19.0561 | 4 | 41 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 18.1081 | 4 | 37 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | Kd | 9.5782 | 3 | 22 |
| Serine/threonine-protein kinase PknB | Mycobacterium tuberculosis H37Rv | Kd | 9.6786 | 1 | 14 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 17.5500 | 4 | 36 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Kd | 9.3973 | 2 | 15 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Kd | 9.6409 | 3 | 22 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 15.1080 | 5 | 43 |
| Serine/threonine-protein kinase PRP4 homolog | Homo sapiens (human) | Kd | 10.0000 | 2 | 15 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 8.7795 | 4 | 23 |
| Serine/threonine-protein kinase RIO1 | Homo sapiens (human) | Kd | 9.1727 | 3 | 22 |
| Serine/threonine-protein kinase RIO2 | Homo sapiens (human) | Kd | 8.8207 | 2 | 15 |
| Serine/threonine-protein kinase RIO3 | Homo sapiens (human) | Kd | 8.5250 | 4 | 24 |
| Serine/threonine-protein kinase SBK1 | Homo sapiens (human) | Kd | 9.0000 | 1 | 14 |
| Serine/threonine-protein kinase Sgk3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Kd | 5.9347 | 3 | 22 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 15.4715 | 4 | 40 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 18.0911 | 3 | 34 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 19.5238 | 4 | 42 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 19.4483 | 4 | 35 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 20.3055 | 2 | 33 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 18.3059 | 3 | 35 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 20.0374 | 3 | 34 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | Kd | 4.6573 | 4 | 23 |
| Serine/threonine-protein kinase tousled-like 1 | Homo sapiens (human) | Kd | 9.5714 | 3 | 22 |
| Serine/threonine-protein kinase tousled-like 2 | Homo sapiens (human) | Kd | 9.6409 | 3 | 22 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 20.3500 | 3 | 32 |
| Serine/threonine-protein kinase ULK2 | Homo sapiens (human) | Kd | 9.3567 | 2 | 15 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 19.6729 | 3 | 35 |
| Serine/threonine-protein kinase VRK2 | Homo sapiens (human) | Kd | 8.8507 | 1 | 14 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 20.3836 | 3 | 34 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Sex hormone-binding globulin | Homo sapiens (human) | Kd | 39.8107 | 1 | 1 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 16 |
| signal transducer and activator of transcription 1-alpha/beta isoform alpha | Homo sapiens (human) | EC50 | 2.0600 | 1 | 1 |
| SNF-related serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Spike glycoprotein | Betacoronavirus England 1 | EC50 | 62.5093 | 1 | 7 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | EC50 | 62.5093 | 1 | 7 |
| SRSF protein kinase 1 | Homo sapiens (human) | Kd | 9.6273 | 3 | 22 |
| SRSF protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 3 | 22 |
| SRSF protein kinase 3 | Homo sapiens (human) | Kd | 9.0800 | 2 | 15 |
| STAT3, partial | Homo sapiens (human) | EC50 | 55.7000 | 1 | 1 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 11.8578 | 5 | 44 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| STE20/SPS1-related proline-alanine-rich protein kinase | Homo sapiens (human) | Kd | 9.5800 | 2 | 15 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 19 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| Testis-specific serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 9.7545 | 3 | 22 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 17.8752 | 4 | 41 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 15.9608 | 4 | 39 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 17 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 13.2220 | 5 | 42 |
| transcription factor p65 isoform 1 | Homo sapiens (human) | EC50 | 55.9410 | 1 | 1 |
| Transient receptor potential cation channel subfamily M member 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 14 |
| Transmembrane protease serine 2 | Homo sapiens (human) | EC50 | 62.5093 | 1 | 7 |
| Transthyretin | Homo sapiens (human) | Kd | 3.1000 | 1 | 1 |
| Tubulin alpha-1A chain | Rattus norvegicus (Norway rat) | Kd | 4.3740 | 1 | 7 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | EC50 | 1.3483 | 4 | 9 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 2.5563 | 46 | 353 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 7.4065 | 9 | 49 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | Kd | 2.7510 | 3 | 22 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 12.8771 | 5 | 42 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 13.5299 | 5 | 43 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 17.4828 | 4 | 43 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 17.3418 | 4 | 40 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 7.9150 | 5 | 33 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 8.8194 | 7 | 49 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 12.4866 | 6 | 43 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 11.8506 | 5 | 43 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | Kd | 8.8227 | 3 | 22 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 16.3696 | 6 | 55 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 12.1606 | 4 | 29 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Kd | 6.5200 | 4 | 23 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 8.3954 | 6 | 45 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 10.0287 | 5 | 43 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 10.5468 | 5 | 28 |
| Tyrosine-protein kinase receptor Tie-1 | Homo sapiens (human) | Kd | 4.2996 | 3 | 22 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | Kd | 7.0778 | 4 | 23 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | Kd | 6.1570 | 4 | 23 |
| Tyrosine-protein kinase Srms | Homo sapiens (human) | Kd | 6.4694 | 3 | 22 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | EC50 | 15.0000 | 2 | 2 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 16.5146 | 4 | 40 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 16.2250 | 4 | 40 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | Kd | 5.2005 | 3 | 22 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 12.8528 | 5 | 43 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | Kd | 9.6182 | 3 | 22 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 12 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 27.3451 | 1 | 11 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 26.8698 | 1 | 18 |
| Uncharacterized serine/threonine-protein kinase SBK3 | Homo sapiens (human) | Kd | 9.4067 | 2 | 15 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Kd | 5.1392 | 4 | 23 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | EC50 | 0.5000 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Kd | 4.8511 | 6 | 26 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Kd | 5.5300 | 6 | 26 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 18 |
| Virulence sensor histidine kinase PhoQ | Salmonella enterica subsp. enterica serovar Typhimurium str. LT2 | Kd | 715.0000 | 2 | 2 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 16.5371 | 5 | 43 |
| Wee1-like protein kinase 2 | Homo sapiens (human) | Kd | 6.6022 | 3 | 17 |