Page last updated: 2024-08-07 15:19:16

signal transducer and activator of transcription 1-alpha/beta isoform alpha

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (40)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ouabainHomo sapiens (human)IC5055.700010
digitoxinHomo sapiens (human)IC5055.700010
2-(1-benzimidazolylmethyl)-5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazoleHomo sapiens (human)IC5055.700010
4-[(2-bromophenoxy)methyl]-N-[4-[(3,5-dimethyl-1-pyrazolyl)methyl]phenyl]benzamideHomo sapiens (human)IC5055.700010
6-chloro-4-phenyl-3-(1-phenyl-5-tetrazolyl)quinolineHomo sapiens (human)IC5055.700010
(4-chlorophenyl)-[4-(7-chloro-4-quinolinyl)-1-piperazinyl]methanoneHomo sapiens (human)IC5055.700010
4-(dimethylsulfamoyl)-N-(4-thiophen-2-yl-2-thiazolyl)benzamideHomo sapiens (human)IC5055.700010
N-[2-methoxy-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]-2-(4-methylphenoxy)acetamideHomo sapiens (human)IC5018.930010
4-[4-(phenylmethyl)-1-piperidinyl]thieno[2,3-d]pyrimidineHomo sapiens (human)IC5055.700010
digoxinHomo sapiens (human)IC5055.700010
N-[1-(4-methyl-6-oxo-1-pyrimidinyl)-2-oxo-2-phenylethyl]benzamideHomo sapiens (human)IC509.254010
N-[(2-methyl-4-thiazolyl)methyl]-4-phenoxybenzenesulfonamideHomo sapiens (human)IC5055.700010
6-chloro-N-[3-[(2-chlorophenyl)sulfamoyl]phenyl]-3-pyridinecarboxamideHomo sapiens (human)IC5055.700010
2-(dimethylaminostyryl)-1-ethylpyridiniumHomo sapiens (human)IC5055.700010
beta-zearalenolHomo sapiens (human)IC5055.700010
LSM-34734Homo sapiens (human)IC5055.700010
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[3-(4-fluorophenyl)-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetamideHomo sapiens (human)IC5014.050010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ipriflavoneHomo sapiens (human)EC500.418010
7-(methoxymethyl)-3-(2-methoxyphenyl)-1H-[1,2,4]triazolo[4,3-a]pyrimidin-5-oneHomo sapiens (human)EC5055.700010
1H-indazole-3-carboxylic acid methyl esterHomo sapiens (human)EC5055.700010
arachinHomo sapiens (human)EC5055.700010
N-[2-(1-cyclohexenyl)ethyl]-4-fluorobenzamideHomo sapiens (human)EC500.687010
2-amino-4-(4-chlorophenyl)-6-methyl-3-pyridinecarbonitrileHomo sapiens (human)EC5055.700010
6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-amineHomo sapiens (human)EC500.516010
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)EC501.002010
5-(4-methylphenyl)-2-phenyl-3-pyrazolamineHomo sapiens (human)EC502.998010
1-(4-methoxyphenyl)-3-(6-quinoxalinyl)thioureaHomo sapiens (human)EC5013.320010
N-[4-[2-[(6-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideHomo sapiens (human)EC501.647010
4-(5-formyl-2-furanyl)benzoic acid propyl esterHomo sapiens (human)EC500.436010
5-(2-ethoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)EC5055.700010
N2-(5-phenyl-1H-pyrazol-3-yl)benzene-1,2-diamineHomo sapiens (human)EC502.716010
2-(1,3-benzoxazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneHomo sapiens (human)EC500.229010
6-[[4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)anilino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidHomo sapiens (human)EC5055.700010
5-methyl-N-(3-methylphenyl)-4-nitro-1H-pyrazol-3-amineHomo sapiens (human)EC501.237010
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamideHomo sapiens (human)EC5055.700010
LSM-16446Homo sapiens (human)EC5055.700010
biochanin aHomo sapiens (human)EC502.060010
3-(4-chlorophenyl)-1-methyl-N-[3-(1-pyrrolidinyl)propyl]-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)EC5021.560010
N-(4-chloro-2,5-dimethoxyphenyl)-5-cyclopropyl-3-isoxazolecarboxamideHomo sapiens (human)EC5055.700010
N-(6-fluoro-1,3-benzothiazol-2-yl)-6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-amineHomo sapiens (human)EC501.286010