Page last updated: 2024-09-27

Myxoid Liposarcoma

Synonyms(2)

Synonym
Round Cell Liposarcoma
Myxoid Liposarcoma

Research Excerpts

Overview

ExcerptReference
"Myxoid liposarcoma is the most common type of liposarcoma (approximately 40 to 50% of all liposarcomas)."( Boyer, B; Cordoliani, YS; Le Friant, G; Lescop, J; Pujol, A; Soulié, D, 1995)
"Metastatic myxoid liposarcoma is an important condition because it may indicate distant micrometastatic disease."( Hirose, Y; Matsuo, M; Nishimoto, Y; Ohno, T; Tomita, H; Yamaguchi, K, 2006)
"Myxoid liposarcomas are soft tissue sarcomas, with a high prevalence of extrapulmonary metastases."( Bredella, MA; Kattapuram, S; Nielsen, GP; Ouellette, HA; Sheah, K; Torriani, M, 2008)
"Myxoid liposarcoma is a common subtype of liposarcoma."( Bello, E; Casali, P; D'Incalci, M; Frapolli, R; Gronchi, A; Grosso, F; Marchini, S; Peloso, G; Pilotti, S; Sanfilippo, R; Tamborini, E; Tarantino, E; Tercero, JC; Virdis, E, 2010)
"Myxoid liposarcoma is a relatively common malignant soft tissue tumor, characterized by a (12;16) translocation resulting in a FUS-DDIT3 fusion gene playing a pivotal role in its tumorigenesis."( Bovée, JV; Bruijn, IH; Hogendoorn, PC; Schrage, YM; Szuhai, K; Willems, SM, 2010)
"Myxoid liposarcoma is a soft tissue tumor in adults with rare cardiac involvement."( Alizadeh, L; Amini, S; Asadi, M; Mottahedi, B, 2013)
"Myxoid liposarcoma is a histological subtype of liposarcoma particularly sensitive to trabectedin."( Ballabio, S; Bello, E; Brich, S; Carrassa, L; Casali, PG; Craparotta, I; D'Incalci, M; Frapolli, R; Gatta, R; Gronchi, A; Mannarino, L; Marchini, S; Matteo, C; Pilotti, S; Sanfilippo, R, 2019)

Context

ExcerptReference
"Myxoid liposarcoma has a relatively good prognosis but tends to recur locally."( Clarke, PM; Sandison, A; Tysome, JR, 2006)

Treatment

ExcerptReference
"We describe a patient with a myxoid liposarcoma of the thigh and a secondary lesion in the interventricular septum, which was treated with radiotherapy."( Judson, I; Ng, C; Stebbing, J, 2001)
"51 patients with advanced pretreated myxoid liposarcoma who started treatment with trabectedin between April 4, 2001, and Sept 18, 2006 at five institutions in a compassionate-use programme were analysed retrospectively."( Blay, JY; Casali, PG; Casieri, P; Collini, P; D'Incalci, M; Demetri, GD; Dileo, P; Fletcher, JA; Gronchi, A; Grosso, F; Jimeno, J; Jones, RL; Judson, IR; Le Cesne, A; Pilotti, S; Sanfilippo, R; Spreafico, C; Stacchiotti, S; Tamborini, E; Tercero, JC, 2007)
"Treatment of the myxoid liposarcoma cell lines MLS 402 and MLS 1765 with the FGFR inhibitors PD173074, TKI258 (dovitinib) and BGJ398 as well as specific siRNAs reduced cell proliferation, induced apoptosis and delayed cell migration."( Brors, B; Büttner, R; Fassunke, J; Heydt, C; Ihle, MA; Künstlinger, H; Mechtersheimer, G; Merkelbach-Bruse, S; Schildhaus, HU; Wardelmann, E, 2015)
"As the understanding of the biology of myxoid liposarcomas progresses, more targeted therapies are being developed that will lead to better tolerated treatments and improved survival for patients."( Abaricia, S; Hirbe, AC, 2018)

Research

Studies (82)

TimeframeStudies, This Condition (%)All Conditions %
pre-19900 (0.00)23.3326
1990's8 (9.76)12.5806
2000's26 (31.71)18.1394
2010's41 (50.00)28.8240
2020's7 (8.54)9.53
DrugIndicatedRelationship StrengthStudiesTrials
salicylic acid0low20
formaldehyde0low10
pd 1730740low10
4,5,6,7-tetrabromo-2-azabenzimidazole0low10
ifosfamide0low30
pioglitazone0low10
temozolomide0low10
bromodeoxyuridine0low10
cycloheximide0low10
isoxazoles0low10
thiazoles0low10
reticulin0low10
gadolinium0low20
camptothecin0low10
barium sulfate0low10
propiconazole0low10
3-iodobenzylguanidine0low10
triazoles0low10
fluorodeoxyglucose f180low50
ecteinascidin 7430medium292
iodofiltic acid0low10
imatinib mesylate0low10
methotrexate0low10
bromochloroacetic acid0low10
amrubicin0medium11
dasatinib0low10
17-(dimethylaminoethylamino)-17-demethoxygeldanamycin0low10
casein kinase ii0low10
gadolinium dtpa0low10
panobinostat0medium11
rivaroxaban0low10
er-0865260low10
oligonucleotides0low10
mesna0low10
incb-0184240low10
interleukin-80low20
transforming growth factor beta0low10
pm 011830low10
hyaluronoglucosaminidase0low10
dacarbazine0low30

Protein Targets (930)

ProteinPotency MeasurementsInhibition MeasurementsActivation MeasurementsDrugs
Gamma-aminobutyric acid receptor subunit pi4015
Lysine-specific demethylase 6B0101
Lysine-specific demethylase 4B0101
Heat shock protein HSP 90-alpha0224
Heat shock protein HSP 90-beta0123
Cholesteryl ester transfer protein0011
Gamma-aminobutyric acid receptor subunit beta-14015
Gamma-aminobutyric acid receptor subunit delta4015
Gamma-aminobutyric acid receptor subunit gamma-24015
5-hydroxytryptamine receptor 1A0101
Gamma-aminobutyric acid receptor subunit alpha-54015
Gamma-aminobutyric acid receptor subunit alpha-34015
Gamma-aminobutyric acid receptor subunit gamma-14015
Gamma-aminobutyric acid receptor subunit alpha-24015
Gamma-aminobutyric acid receptor subunit alpha-44015
Gamma-aminobutyric acid receptor subunit gamma-34015
Lysine-specific demethylase 5A0101
Gamma-aminobutyric acid receptor subunit alpha-64015
Endoplasmin0011
Gamma-aminobutyric acid receptor subunit alpha-14015
Gamma-aminobutyric acid receptor subunit beta-34015
Gamma-aminobutyric acid receptor subunit beta-24015
Hypoxia-inducible factor 1-alpha0202
GABA theta subunit4015
Endothelial PAS domain-containing protein 10202
Gamma-aminobutyric acid receptor subunit epsilon4015
Lysine-specific demethylase 4C0101
dopamine D1 receptor3003
thioredoxin reductase7007
GLS protein2002
Thrombopoietin4004
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)2002
cytochrome P450 2D6 isoform 11001
cytochrome P450 2C19 precursor2002
ras-related protein Rab-9A5005
histone acetyltransferase KAT2A isoform 15005
lethal factor (plasmid)3003
POU domain, class 2, transcription factor 10001
Spike glycoprotein7029
ATP-dependent phosphofructokinase4004
Chain A, Cell division protein kinase 20101
Chain A, HADH2 protein3003
Chain B, HADH2 protein3003
Chain A, 2-oxoglutarate Oxygenase6006
Chain A, ATP-DEPENDENT DNA HELICASE Q11001
Chain A, Ferritin light chain5005
Genome polyprotein 0202
15-lipoxygenase, partial4004
ATAD5 protein, partial7007
USP1 protein, partial3003
NFKB1 protein, partial3003
Microtubule-associated protein tau4004
aldehyde dehydrogenase 1 family, member A19009
regulator of G-protein signaling 42002
nonstructural protein 12002
estrogen-related nuclear receptor alpha100010
euchromatic histone-lysine N-methyltransferase 25005
Bloom syndrome protein isoform 14004
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 14004
vitamin D3 receptor isoform VDRA3003
chromobox protein homolog 17007
flap endonuclease 12002
DNA polymerase iota isoform a (long)6006
geminin110011
DNA polymerase kappa isoform 14004
cytochrome P450 3A4 isoform 14004
M-phase phosphoprotein 83003
lamin isoform A-delta106006
Replicase polyprotein 1ab0134
Ribosyldihydronicotinamide dehydrogenase [quinone]0246
Casein kinase II subunit alpha'0426
Alpha-synuclein2002
Casein kinase II subunit beta0415
Casein kinase II subunit alpha0437
Dual specificity tyrosine-phosphorylation-regulated kinase 1A0224
Casein kinase II subunit alpha 30404
Ataxin-28008
RAR-related orphan receptor gamma7007
AR protein100010
nuclear receptor subfamily 1, group I, member 37007
retinoic acid nuclear receptor alpha variant 17007
thyroid stimulating hormone receptor4004
nuclear factor erythroid 2-related factor 2 isoform 16006
Cellular tumor antigen p536006
Nuclear receptor ROR-gamma3003
interleukin 83003
pregnane X receptor3003
TDP1 protein110011
progesterone receptor7007
glucocorticoid receptor [Homo sapiens]7007
retinoid X nuclear receptor alpha8008
pregnane X nuclear receptor5005
estrogen nuclear receptor alpha100010
bromodomain adjacent to zinc finger domain 2B1001
arylsulfatase A2002
IDH15005
nuclear receptor subfamily 1, group I, member 23003
cellular tumor antigen p53 isoform a4004
Nuclear hormone receptor family member daf-120011
nuclear factor erythroid 2-related factor 2 isoform 25005
thyroid hormone receptor beta isoform 28008
serine/threonine-protein kinase mTOR isoform 15005
oxysterols receptor LXR-beta isoform 10011
urokinase-type plasminogen activator precursor3003
plasminogen precursor3003
urokinase plasminogen activator surface receptor precursor3003
peripheral myelin protein 223003
survival motor neuron protein isoform d6006
muscarinic acetylcholine receptor M11001
Voltage-dependent calcium channel gamma-2 subunit6006
Thymidine kinase, cytosolic0101
Glutamate receptor 26006
Thymidine phosphorylase0001
Thymidylate kinase0101
Thymidine kinase0001
Thymidylate kinase0101
ATPase family AAA domain-containing protein 57007
Chain A, Cruzipain1001
DNA topoisomerase 0101
Fumarate hydratase5005
PPM1D protein8008
thyroid stimulating hormone receptor2002
EWS/FLI fusion protein100010
polyprotein5005
67.9K protein5005
glucocerebrosidase2002
putative alpha-glucosidase1001
alpha-galactosidase3003
lysosomal alpha-glucosidase preproprotein1001
peripheral myelin protein 22 isoform 12002
hemoglobin subunit beta1001
huntingtin isoform 22002
eukaryotic translation initiation factor 2-alpha kinase 3 isoform 1 precursor0011
nuclear receptor ROR-gamma isoform 14004
muscleblind-like protein 1 isoform 13003
relaxin receptor 1 isoform 11001
Telomerase reverse transcriptase0101
Serine/threonine-protein kinase Chk10033
Histone deacetylase 30314
ATP-binding cassette sub-family C member 30909
Multidrug resistance-associated protein 409010
Type-2 restriction enzyme ScaI0101
Deoxyribonuclease-2-alpha0101
Bile salt export pump010010
Tyrosyl-DNA phosphodiesterase 20101
Deoxyribonuclease-10101
Type-2 restriction enzyme PstI0101
Type-2 restriction enzyme EcoRI0101
Prothrombin0102
DNA ligase0101
Interferon beta8008
Integrin beta-32002
Integrin alpha-IIb2002
Heterogeneous nuclear ribonucleoprotein A10011
DNA topoisomerase 10116
DNA topoisomerase 2-alpha0101
Type-2 restriction enzyme BamHI0101
Somatostatin receptor type 10101
Somatostatin receptor type 20101
Somatostatin receptor type 40101
Somatostatin receptor type 30101
Somatostatin receptor type 50101
5-hydroxytryptamine receptor 2B0202
Type-2 restriction enzyme HindIII0101
D(1A) dopamine receptor2002
Histone deacetylase 40303
Ribonuclease pancreatic0101
Inositol monophosphatase 12002
DNA topoisomerase 2-beta0023
DNA topoisomerase 10102
Histone deacetylase 10314
DNA topoisomerase 10101
Integrase 0101
Histone deacetylase 70303
Histone deacetylase 20314
Canalicular multispecific organic anion transporter 10808
DNA topoisomerase type IB small subunit 0011
Polyamine deacetylase HDAC100303
Histone deacetylase 11 0303
Histone deacetylase 80303
Tyrosyl-DNA phosphodiesterase 10101
Histone deacetylase 60415
Histone deacetylase 90303
Histone deacetylase 50303
Chain A, Protein kinase CK2, alpha Subunit0101
Chain A, PROTEIN KINASE CK2, alpha SUBUNIT0101
Chain A, Protein Kinase Ck2, Alpha Subunit0101
endonuclease IV1001
Parkin1001
NPC intracellular cholesterol transporter 1 precursor2002
mitogen-activated protein kinase 11001
Serine/threonine-protein kinase Sgk10101
Casein kinase II subunit alpha 0101
Cyclin-A20101
Cyclin-dependent kinase 20235
Casein kinase II subunit beta0101
Cyclin-A10101
Dual specificity mitogen-activated protein kinase kinase 10325
Ribosomal protein S6 kinase alpha-10224
Single-stranded DNA cytosine deaminase1001
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE5005
glp-1 receptor, partial4004
GLI family zinc finger 36006
Smad33003
estrogen receptor 2 (ER beta)5005
farnesoid X nuclear receptor5005
P531001
peroxisome proliferator-activated receptor delta6006
peroxisome proliferator activated receptor gamma6006
vitamin D (1,25- dihydroxyvitamin D3) receptor3003
RPL19A0011
aryl hydrocarbon receptor5005
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a5005
activating transcription factor 62002
v-jun sarcoma virus 17 oncogene homolog (avian)1001
Histone H2A.x3003
Spike glycoprotein0022
Replicase polyprotein 1ab0022
thyroid hormone receptor beta isoform a2002
nuclear factor NF-kappa-B p105 subunit isoform 11001
heat shock protein HSP 90-alpha isoform 20002
transactivating tegument protein VP16 [Human herpesvirus 1]0202
COUP transcription factor 2 isoform a0101
Transmembrane protease serine 20022
Glucose transporter0101
Hexose transporter 1 0101
Procathepsin L0022
Polyunsaturated fatty acid 5-lipoxygenase0101
Replicase polyprotein 1a0022
Replicase polyprotein 1ab0022
Replicase polyprotein 1ab0022
Solute carrier family 2, facilitated glucose transporter member 10101
Eukaryotic initiation factor 4A-I0101
Peptidyl-prolyl cis-trans isomerase FKBP1A0202
Peptidyl-prolyl cis-trans isomerase FKBP30101
Peptidyl-prolyl cis-trans isomerase FKBP40101
TAR DNA-binding protein 433003
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 10101
Angiotensin-converting enzyme 2 0022
Peptidyl-prolyl cis-trans isomerase FKBP140101
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 40101
heat shock protein 90, putative0002
hypoxia-inducible factor 1 alpha subunit1001
cytochrome P450 2D61001
Matrix metalloproteinase-90101
Isocitrate lyase0101
Leukotriene C4 synthase0022
acetylcholinesterase2002
GALC protein2002
caspase 7, apoptosis-related cysteine protease1001
cytochrome P450 family 3 subfamily A polypeptide 43003
caspase-31001
tyrosine-protein kinase Yes4004
Bone morphogenetic protein receptor type-1B0022
Membrane-associated progesterone receptor component 10011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform0224
Serine/threonine-protein kinase PLK40022
Serine/threonine-protein kinase 250022
ATP-dependent RNA helicase DDX3X0022
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta0022
Pyridoxal kinase0022
Citron Rho-interacting kinase0022
Serine/threonine-protein kinase RIO30022
Dual specificity mitogen-activated protein kinase kinase 70022
Inhibitor of nuclear factor kappa-B kinase subunit beta0124
Peripheral plasma membrane protein CASK0022
Aurora kinase A0123
Cyclin-G-associated kinase0123
Serine/threonine-protein kinase DCLK10022
Inhibitor of nuclear factor kappa-B kinase subunit alpha0123
Muscle, skeletal receptor tyrosine-protein kinase0022
Ephrin type-B receptor 60022
Peroxisomal acyl-coenzyme A oxidase 30022
Mitogen-activated protein kinase 130123
3-phosphoinositide-dependent protein kinase 10022
Mitogen-activated protein kinase kinase kinase 130022
Death-associated protein kinase 30022
Mitogen-activated protein kinase kinase kinase 70022
Receptor-interacting serine/threonine-protein kinase 20224
Mitotic checkpoint serine/threonine-protein kinase BUB10022
NUAK family SNF1-like kinase 10022
Dynamin-like 120 kDa protein, mitochondrial0022
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma0022
Tyrosine-protein kinase JAK20235
Voltage-dependent L-type calcium channel subunit alpha-1F0101
Eukaryotic translation initiation factor 5B0022
Rho-associated protein kinase 20022
Serine/threonine-protein kinase ULK10022
Serine/threonine-protein kinase/endoribonuclease IRE10022
Ribosomal protein S6 kinase alpha-50022
U5 small nuclear ribonucleoprotein 200 kDa helicase0022
Ribosomal protein S6 kinase alpha-40022
Serine/threonine-protein kinase 160022
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma0022
Serine/threonine-protein kinase PAK 30022
Cyclin-dependent kinase-like 50022
Serine/threonine-protein kinase 17B0022
Serine/threonine-protein kinase 100022
Serine/threonine-protein kinase D30022
Cyclin-dependent kinase 140022
Structural maintenance of chromosomes protein 20022
Mitogen-activated protein kinase kinase kinase 60022
Serine/threonine-protein kinase OSR10022
Mitogen-activated protein kinase kinase kinase kinase 40022
Serine/threonine-protein kinase LATS10022
Serine/threonine-protein kinase PAK 40022
Serine/threonine-protein kinase Chk20022
Tyrosine-protein kinase ABL105511
Tyrosine-protein kinase ABL10101
Proto-oncogene tyrosine-protein kinase Src0213
Epidermal growth factor receptor0224
Transthyretin0011
RAF proto-oncogene serine/threonine-protein kinase0123
Receptor tyrosine-protein kinase erbB-20123
High affinity nerve growth factor receptor0022
Guanine nucleotide-binding protein G(i) subunit alpha-20022
ADP/ATP translocase 20022
Cytochrome P450 1A20202
Neuronal proto-oncogene tyrosine-protein kinase Src 0001
Protein kinase C beta type0022
Insulin receptor0224
Tyrosine-protein kinase Lck0325
Proto-oncogene tyrosine-protein kinase LCK 0202
Tyrosine-protein kinase Fyn0325
Cyclin-dependent kinase 10022
Glycogen phosphorylase, liver form0022
Tyrosine-protein kinase Fes/Fps0022
Macrophage colony-stimulating factor 1 receptor0224
Adenine phosphoribosyltransferase0011
Tyrosine-protein kinase Yes0123
Tyrosine-protein kinase Lyn0123
Proto-oncogene tyrosine-protein kinase receptor Ret0123
Insulin-like growth factor 1 receptor0123
Signal recognition particle receptor subunit alpha0011
Cytochrome c1, heme protein, mitochondrial0022
Hepatocyte growth factor receptor0022
Tyrosine-protein kinase HCK0224
Proto-oncogene tyrosine-protein kinase ROS0022
Platelet-derived growth factor receptor beta0224
Tyrosine-protein kinase Fgr0022
Quinolone resistance protein NorA0101
Wee1-like protein kinase 20022
Uncharacterized serine/threonine-protein kinase SBK30022
Serine/threonine-protein kinase A-Raf0022
Cytochrome P450 2D60101
Mast/stem cell growth factor receptor Kit0235
Glycogen phosphorylase, brain form0022
Breakpoint cluster region protein0247
Serine/threonine-protein kinase pim-10022
Fibroblast growth factor receptor 10235
Cytochrome P450 2A60101
Cytochrome P450 2C9 0101
Myosin light chain kinase, smooth muscle0011
Cyclin-dependent kinase 40022
ADP/ATP translocase 30022
Inosine-5'-monophosphate dehydrogenase 20022
Angiotensin-converting enzyme 0101
Proto-oncogene tyrosine-protein kinase Src0426
cAMP-dependent protein kinase type II-alpha regulatory subunit0022
Insulin receptor-related protein0022
Serine/threonine-protein kinase B-raf0022
Potassium voltage-gated channel subfamily E member 10101
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform0022
Platelet-derived growth factor receptor alpha0336
Tyrosine-protein kinase Blk0101
Tyrosine-protein kinase Fer0022
Protein kinase C alpha type0123
cAMP-dependent protein kinase catalytic subunit alpha0022
Vascular endothelial growth factor receptor 1 0123
General transcription and DNA repair factor IIH helicase subunit XPD0022
Interferon-induced, double-stranded RNA-activated protein kinase0022
Ras-related protein Rab-6A0011
Serine/threonine-protein kinase MAK0022
Cytochrome P450 2B60101
Cyclin-dependent kinase 11B0022
Ephrin type-A receptor 10022
Fibroblast growth factor receptor 20123
Receptor tyrosine-protein kinase erbB-30022
Multifunctional protein ADE20022
Fibroblast growth factor receptor 40123
Fibroblast growth factor receptor 30134
cAMP-dependent protein kinase catalytic subunit gamma0022
cAMP-dependent protein kinase catalytic subunit beta0022
Ferrochelatase, mitochondrial0022
Ribosomal protein S6 kinase beta-10022
Tyrosine-protein kinase JAK10235
Protein kinase C eta type0022
Beta-adrenergic receptor kinase 10022
Probable ATP-dependent RNA helicase DDX60022
Activin receptor type-2A0022
Mitogen-activated protein kinase 3 0022
MAP/microtubule affinity-regulating kinase 30022
Deoxycytidine kinase0022
Mitogen-activated protein kinase 10022
Ephrin type-A receptor 20123
Ephrin type-A receptor 30022
Ephrin type-A receptor 80022
Ephrin type-B receptor 20123
Leukocyte tyrosine kinase receptor0022
Non-receptor tyrosine-protein kinase TYK20235
UMP-CMP kinase 0011
Phosphatidylethanolamine-binding protein 10022
Wee1-like protein kinase0022
Heme oxygenase 20022
Tyrosine-protein kinase receptor UFO0022
Mitogen-activated protein kinase 40022
S-adenosylmethionine synthase isoform type-20022
DnaJ homolog subfamily A member 10022
RAC-alpha serine/threonine-protein kinase0123
RAC-beta serine/threonine-protein kinase0123
G protein-coupled receptor kinase 40022
Cytochrome P450 2C190101
Dual specificity protein kinase TTK0022
DNA replication licensing factor MCM40022
Prostaglandin G/H synthase 20123
Tyrosine-protein kinase receptor Tie-10022
Vascular endothelial growth factor receptor 30123
Vascular endothelial growth factor receptor 20235
Dual specificity mitogen-activated protein kinase kinase 20123
Receptor-type tyrosine-protein kinase FLT30123
Bone morphogenetic protein receptor type-1A0022
Activin receptor type-1B0022
TGF-beta receptor type-10022
Serine/threonine-protein kinase receptor R30022
TGF-beta receptor type-20022
Electron transfer flavoprotein subunit beta0022
Tyrosine-protein kinase CSK0224
Glycine--tRNA ligase0022
Protein kinase C iota type0022
Exosome RNA helicase MTR40022
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform0123
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform0224
Serine/threonine-protein kinase mTOR0123
Megakaryocyte-associated tyrosine-protein kinase0022
Tyrosine-protein kinase Tec0123
Tyrosine-protein kinase TXK0123
Tyrosine-protein kinase ABL20123
Tyrosine-protein kinase FRK0022
G protein-coupled receptor kinase 60011
Tyrosine-protein kinase ZAP-700022
Tyrosine-protein kinase SYK0123
26S proteasome regulatory subunit 6B0022
Mitogen-activated protein kinase 80022
Mitogen-activated protein kinase 90022
Dual specificity mitogen-activated protein kinase kinase 40022
Dual specificity mitogen-activated protein kinase kinase 30022
Casein kinase I isoform alpha0123
Casein kinase I isoform delta0022
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 0224
MAP kinase-activated protein kinase 20123
Cyclin-dependent kinase 80022
Elongation factor Tu, mitochondrial0022
Choline-phosphate cytidylyltransferase A0011
Cysteine--tRNA ligase, cytoplasmic0022
Casein kinase I isoform epsilon0022
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial0022
Dual specificity protein kinase CLK10022
Dual specificity protein kinase CLK20022
Dual specificity protein kinase CLK30022
Glycogen synthase kinase-3 alpha0022
Glycogen synthase kinase-3 beta0022
Cyclin-dependent kinase 70022
Cyclin-dependent kinase 90022
Ras-related protein Rab-27A0022
Tyrosine-protein kinase Blk0123
Interleukin-1 receptor-associated kinase 10022
Potassium voltage-gated channel subfamily KQT member 10101
Ribosomal protein S6 kinase alpha-30123
Cytoplasmic tyrosine-protein kinase BMX0022
cAMP-dependent protein kinase catalytic subunit PRKX0022
Serine/threonine-protein kinase Nek20022
Serine/threonine-protein kinase Nek30022
Serine/threonine-protein kinase Nek40022
Tyrosine-protein kinase JAK30224
Dual specificity mitogen-activated protein kinase kinase 60022
Serine/threonine-protein kinase PLK10022
Death-associated protein kinase 10022
LIM domain kinase 10123
LIM domain kinase 20123
Mitogen-activated protein kinase 120123
Mitogen-activated protein kinase 100022
Tyrosine--tRNA ligase, cytoplasmic0022
5'-AMP-activated protein kinase subunit gamma-10023
5'-AMP-activated protein kinase catalytic subunit alpha-20023
Ephrin type-B receptor 30022
Ephrin type-A receptor 50022
Ephrin type-B receptor 40123
Ephrin type-B receptor 10022
Ephrin type-A receptor 40022
Adenylate kinase 2, mitochondrial0022
Adenosine kinase0022
Hormonally up-regulated neu tumor-associated kinase0022
Serine/threonine-protein kinase SIK10224
Receptor-interacting serine/threonine-protein kinase 40022
Ras-related protein Rab-100022
Cell division control protein 2 homolog0022
Actin-related protein 30022
Actin-related protein 20022
Calcium-dependent protein kinase 10022
GTP-binding nuclear protein Ran0022
Tubulin alpha-1A chain0011
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta0022
SRSF protein kinase 20022
Casein kinase I isoform gamma-20022
DNA-dependent protein kinase catalytic subunit0101
Mitogen-activated protein kinase kinase kinase 90022
Serine/threonine-protein kinase PknB0022
Cyclin-dependent kinase 30022
Cyclin-dependent kinase-like 10022
Cyclin-dependent kinase 60022
Cyclin-dependent-like kinase 5 0022
Cyclin-dependent kinase 160022
Cyclin-dependent kinase 170022
Myelin transcription factor 10101
Voltage-dependent L-type calcium channel subunit alpha-1D 0101
ATP-dependent 6-phosphofructokinase, platelet type0022
Protein kinase C epsilon type0022
Angiopoietin-1 receptor0022
Mitogen-activated protein kinase kinase kinase 100022
Protein kinase C theta type0022
Activin receptor type-10022
Macrophage-stimulating protein receptor0022
Focal adhesion kinase 10123
Protein kinase C zeta type0112
Protein kinase C delta type0123
Tyrosine-protein kinase BTK0224
Tyrosine-protein kinase receptor TYRO30022
Cyclin-dependent kinase 180022
Activated CDC42 kinase 10123
Epithelial discoidin domain-containing receptor 10325
Tyrosine-protein kinase ITK/TSK0123
Myotonin-protein kinase0022
Potassium voltage-gated channel subfamily H member 20101
Mitogen-activated protein kinase kinase kinase kinase 20022
Mitogen-activated protein kinase kinase kinase 120022
Tyrosine-protein kinase Mer0022
Serine/threonine-protein kinase 40022
5'-AMP-activated protein kinase catalytic subunit alpha-10023
Serine/threonine-protein kinase PAK 10022
Dual specificity mitogen-activated protein kinase kinase 50022
Mitogen-activated protein kinase 70022
Serine/threonine-protein kinase PAK 20022
Serine/threonine-protein kinase 30022
Mitogen-activated protein kinase kinase kinase 10022
cGMP-dependent protein kinase 20022
Integrin-linked protein kinase0022
Rho-associated protein kinase 10022
Non-receptor tyrosine-protein kinase TNK10022
Serine/threonine-protein kinase PRP4 homolog0022
Receptor-interacting serine/threonine-protein kinase 10022
Calcium/calmodulin-dependent protein kinase type II subunit beta0022
Calcium/calmodulin-dependent protein kinase type II subunit gamma0022
Calcium/calmodulin-dependent protein kinase type II subunit delta0022
Voltage-dependent L-type calcium channel subunit alpha-1S0101
Activin receptor type-2B0022
Bone morphogenetic protein receptor type-20022
Protein-tyrosine kinase 60123
Voltage-dependent L-type calcium channel subunit alpha-1C0101
cGMP-dependent protein kinase 1 0022
Cyclin-dependent kinase 130022
Calcium/calmodulin-dependent protein kinase type 10022
Inhibitor of nuclear factor kappa-B kinase subunit epsilon0022
Protein-tyrosine kinase 2-beta0022
Sodium channel protein type 5 subunit alpha0101
Maternal embryonic leucine zipper kinase0022
Structural maintenance of chromosomes protein 1A0022
Chromodomain-helicase-DNA-binding protein 40022
Peroxisomal acyl-coenzyme A oxidase 10022
Serine/threonine-protein kinase D10022
Serine/threonine-protein kinase 380022
Receptor tyrosine-protein kinase erbB-40022
Ribosomal protein S6 kinase alpha-20022
Ephrin type-A receptor 70022
Delta(24)-sterol reductase0022
Dual specificity testis-specific protein kinase 10022
Myosin light chain kinase, smooth muscle0022
Mitogen-activated protein kinase 110123
Serine/threonine-protein kinase STK110022
Rhodopsin kinase GRK10022
NT-3 growth factor receptor0022
Serine/threonine-protein kinase N10022
Serine/threonine-protein kinase N20022
Mitogen-activated protein kinase 140134
Calcium/calmodulin-dependent protein kinase type IV0022
Mitogen-activated protein kinase kinase kinase 110022
BDNF/NT-3 growth factors receptor0022
Mitogen-activated protein kinase 60022
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform0022
Discoidin domain-containing receptor 20224
AP2-associated protein kinase 10123
Myosin light chain kinase 30022
Uncharacterized aarF domain-containing protein kinase 50011
Serine/threonine-protein kinase SBK10022
Mitogen-activated protein kinase kinase kinase 190022
Putative heat shock protein HSP 90-beta 20022
Serine/threonine-protein kinase TNNI3K0022
Leucine-rich repeat serine/threonine-protein kinase 20022
Serine/threonine-protein kinase MRCK alpha0022
Serine/threonine-protein kinase MRCK gamma0022
Acyl-CoA dehydrogenase family member 100022
Serine/threonine-protein kinase Nek50022
Serine/threonine-protein kinase N30022
Breakpoint cluster region protein0101
Serine/threonine-protein kinase ULK30022
Dual serine/threonine and tyrosine protein kinase0022
Mitogen-activated protein kinase kinase kinase 150022
Uncharacterized protein FLJ452520022
Acyl-CoA dehydrogenase family member 110022
Serine/threonine-protein kinase/endoribonuclease IRE20022
Serine/threonine-protein kinase MARK20022
Serine/threonine-protein kinase TAO10022
STE20-related kinase adapter protein alpha0022
Myosin-140022
AarF domain-containing protein kinase 10022
Serine/threonine-protein kinase tousled-like 20022
Serine/threonine-protein kinase 32C0022
Serine/threonine-protein kinase pim-30022
ATP-dependent RNA helicase DDX420011
Serine/threonine-protein kinase VRK20022
Myosin light chain kinase family member 40022
Homeodomain-interacting protein kinase 10022
Calcium/calmodulin-dependent protein kinase type 1D0022
Mitogen-activated protein kinase kinase kinase kinase 30022
Cyclin-dependent kinase-like 30022
MAP kinase-activated protein kinase 50022
Serine/threonine-protein kinase BRSK20022
Serine/threonine-protein kinase NIM10022
Eukaryotic peptide chain release factor GTP-binding subunit ERF3B0022
Serine/threonine-protein kinase ULK20022
Misshapen-like kinase 10022
Serine/threonine-protein kinase DCLK20022
Calcium/calmodulin-dependent protein kinase kinase 10022
Casein kinase I isoform alpha-like0022
Homeodomain-interacting protein kinase 40022
Myosin-IIIa0022
Ankyrin repeat and protein kinase domain-containing protein 10022
Serine/threonine-protein kinase Nek110022
Atypical kinase COQ8A, mitochondrial0022
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma0022
Mitogen-activated protein kinase 150022
Serine/threonine-protein kinase Nek90022
Serine/threonine-protein kinase BRSK10022
Serine/threonine-protein kinase 350022
Serine/threonine-protein kinase Nek70022
Rhodopsin kinase GRK70022
Serine/threonine-protein kinase 32A0022
Myosin-IIIb0022
ATP-dependent RNA helicase DDX10022
Dual specificity tyrosine-phosphorylation-regulated kinase 20022
Cyclin-dependent kinase-like 20022
Mitogen-activated protein kinase kinase kinase kinase 10022
Serine/threonine-protein kinase Sgk30022
Atypical kinase COQ8B, mitochondrial0022
Aurora kinase B0123
MAP/microtubule affinity-regulating kinase 40022
Calcium/calmodulin-dependent protein kinase type 1G0022
Serine/threonine-protein kinase Nek10022
Cyclin-dependent kinase 150022
PAS domain-containing serine/threonine-protein kinase0022
Calcium/calmodulin-dependent protein kinase kinase 20022
EKC/KEOPS complex subunit TP53RK0022
Dual specificity testis-specific protein kinase 20011
SRSF protein kinase 10022
Protein cereblon0012
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase0224
Mitogen-activated protein kinase kinase kinase 50022
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha0022
Mitogen-activated protein kinase kinase kinase 30022
Eukaryotic translation initiation factor 2-alpha kinase 10022
Serine/threonine-protein kinase RIO10022
MAP kinase-interacting serine/threonine-protein kinase 10022
Serine/threonine-protein kinase RIO20022
Cyclin-dependent kinase 190022
Transient receptor potential cation channel subfamily M member 60022
Testis-specific serine/threonine-protein kinase 10022
Serine/threonine-protein kinase 330022
Nucleolar GTP-binding protein 10022
Serine/threonine-protein kinase D20022
Serine/threonine-protein kinase DCLK30022
NUAK family SNF1-like kinase 20022
RNA cytidine acetyltransferase0022
Serine/threonine-protein kinase SIK20123
Myosin light chain kinase 2, skeletal/cardiac muscle0022
STE20-like serine/threonine-protein kinase 0022
Serine/threonine-protein kinase TAO30022
Homeodomain-interacting protein kinase 20022
Tyrosine-protein kinase Srms0022
Homeodomain-interacting protein kinase 30022
Serine/threonine-protein kinase PLK30022
dCTP pyrophosphatase 10022
Dual specificity protein kinase CLK40022
MAP kinase-interacting serine/threonine-protein kinase 20022
Serine/threonine-protein kinase Nek60022
Casein kinase I isoform gamma-10022
Serine/threonine-protein kinase PAK 60022
SNF-related serine/threonine-protein kinase0022
Serine/threonine-protein kinase LATS20022
Serine/threonine-protein kinase 360022
Phenylalanine--tRNA ligase beta subunit0022
Isoleucine--tRNA ligase, mitochondrial0022
BMP-2-inducible protein kinase0022
Obg-like ATPase 10011
Midasin0022
Interleukin-1 receptor-associated kinase 40022
Serine/threonine-protein kinase 32B0022
Mitogen-activated protein kinase kinase kinase 200022
Cyclin-dependent kinase 120022
Serine/threonine-protein kinase PLK20022
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 130022
Serine/threonine-protein kinase MARK10022
Serine/threonine-protein kinase pim-20022
Serine/threonine-protein kinase PAK 50022
Serine/threonine-protein kinase 260022
eIF-2-alpha kinase GCN20022
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial0022
Serine/threonine-protein kinase NLK0022
Phosphatidylinositol 4-kinase beta0022
Serine/threonine-protein kinase 17A0022
STE20/SPS1-related proline-alanine-rich protein kinase0022
Ephrin type-A receptor 60022
5'-AMP-activated protein kinase subunit gamma-20023
Serine/threonine-protein kinase TBK10022
Septin-90022
Death-associated protein kinase 20022
Potassium voltage-gated channel subfamily D member 30101
Ribosomal protein S6 kinase alpha-60022
TRAF2 and NCK-interacting protein kinase0022
Serine/threonine-protein kinase tousled-like 10022
Serine/threonine-protein kinase TAO20022
Long-chain-fatty-acid--CoA ligase 50011
ALK tyrosine kinase receptor0022
Broad substrate specificity ATP-binding cassette transporter ABCG20102
SRSF protein kinase 30022
Serine/threonine-protein kinase ICK0022
Cyclin-dependent kinase 11A0022
Aurora kinase C0022
Calcium/calmodulin-dependent protein kinase type II subunit alpha0022
RAC-gamma serine/threonine-protein kinase0123
Serine/threonine-protein kinase 38-like0022
Microtubule-associated serine/threonine-protein kinase 10022
Serine/threonine-protein kinase SIK30123
Mitogen-activated protein kinase kinase kinase 20022
Thyroid hormone receptor-associated protein 30022
Dual specificity tyrosine-phosphorylation-regulated kinase 1B0022
Mitogen-activated protein kinase kinase kinase kinase 50022
Receptor-interacting serine/threonine-protein kinase 30022
Serine/threonine-protein kinase MRCK beta0022
Interleukin-1 receptor-associated kinase 30022
Serine/threonine-protein kinase 240022
NF-kappa-B essential modulator0101
Casein kinase I isoform gamma-30022
Mitogen-activated protein kinase kinase kinase 40022
UDP-glucuronosyltransferase 2B70001
Chain A, Beta-lactamase3003
Serum paraoxonase/arylesterase 10101
Luciferase2002
SMAD family member 22002
SMAD family member 32002
parathyroid hormone/parathyroid hormone-related peptide receptor precursor1001
DNA repair protein RAD52 homolog isoform a0001
Cytochrome P450 3A40102
Cytochrome P450 2C80001
Cytochrome P450 3A50102
Cell division cycle 7-related protein kinase0011
Myosin-100011
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha0011
Oxysterols receptor LXR-beta0101
Tyrosine-protein kinase JAK2 0011
Chain B, DIHYDROFOLATE REDUCTASE0011
Chain B, DIHYDROFOLATE REDUCTASE0011
Chain A, TYROSYL-DNA PHOSPHODIESTERASE1001
Chain B, DIHYDROFOLATE REDUCTASE0011
acid sphingomyelinase1001
ClpP1001
phosphopantetheinyl transferase2002
Thymidylate synthase 0101
Thymidylate synthase 0101
polyunsaturated fatty acid lipoxygenase ALOX121001
transcriptional regulator ERG isoform 31001
importin subunit beta-1 isoform 11001
DNA polymerase beta1001
nuclear receptor coactivator 1 isoform 1 [Homo sapiens]0101
snurportin-11001
peptidyl-prolyl cis-trans isomerase NIMA-interacting 11001
DNA polymerase eta isoform 11001
caspase-1 isoform alpha precursor1001
nuclear receptor coactivator 3 isoform a0101
Toll-like receptor 40101
Fatty-acid amide hydrolase 10101
Bile salt export pump0303
ATP-binding cassette sub-family C member 30102
Dihydrofolate reductase0203
Dihydrofolate reductase0203
Dihydrofolate reductase 0101
Dihydrofolate reductase0101
Dihydrofolate reductase0101
Dihydrofolate reductase0203
Thymidylate synthase0101
Carbonic anhydrase 20415
Thymidylate synthase0202
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Thymidylate synthase0202
5-hydroxytryptamine receptor 2C0102
High mobility group protein B10022
Dihydrofolate reductase0101
Thymidylate synthase0101
Dihydrofolate reductase0224
Glucose-6-phosphate 1-dehydrogenase0101
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Folate receptor beta0101
5-hydroxytryptamine receptor 2A0101
Cytochrome P450 11B1, mitochondrial 0101
Folate receptor alpha0101
Dihydrofolate reductase0202
Histidine decarboxylase0101
Trifunctional purine biosynthetic protein adenosine-30101
Bifunctional purine biosynthesis protein ATIC0202
Multidrug resistance-associated protein 1 0001
Delta-type opioid receptor0101
Mu-type opioid receptor0101
Kappa-type opioid receptor0101
Reduced folate transporter0202
Folylpolyglutamate synthase, mitochondrial0103
6-phosphogluconate dehydrogenase, decarboxylating0101
Caspase-71001
Solute carrier organic anion transporter family member 1A30001
Dihydrofolate reductase0101
Pteridine reductase 10101
Folylpolyglutamate synthase, mitochondrial0103
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Bifunctional dihydrofolate reductase-thymidylate synthase0101
Solute carrier family 22 member 60102
Canalicular multispecific organic anion transporter 10102
Trifunctional purine biosynthetic protein adenosine-30101
Solute carrier family 22 member 200202
Dihydrofolate reductase 0101
Solute carrier family 22 member 80102
Solute carrier family 22 member 60202
Dihydrofolate reductase0101
ATP-binding cassette sub-family C member 110001
Proton-coupled folate transporter0101
Multidrug resistance associated protein0102
Solute carrier organic anion transporter family member 1B30001
Solute carrier family 22 member 110001
Protein-arginine deiminase type-40101
Histone deacetylase 80101
Bromodomain-containing protein 40101
Protein Tat0011
Leukotriene A-4 hydrolase0101
Phosphatidylinositol 3-kinase regulatory subunit alpha0101
NAD-dependent protein deacetylase sirtuin-20202
NAD-dependent protein deacetylase sirtuin-10202
NAD-dependent protein deacetylase sirtuin-70101
NAD-dependent protein deacetylase sirtuin-3, mitochondrial0202
Histone deacetylase 0101
Nuclear receptor corepressor 20101
Chain A, Protein (fibroblast Growth Factor (fgf) Receptor 1)0101
serine-protein kinase ATM isoform a1001
histone-lysine N-methyltransferase 2A isoform 2 precursor1001
Platelet-derived growth factor receptor beta0101
Platelet-derived growth factor receptor alpha0101
Platelet-derived growth factor receptor beta0101
Serine-protein kinase ATM0101
CDGSH iron-sulfur domain-containing protein 10101
Free fatty acid receptor 10011
Peroxisome proliferator-activated receptor gamma0101
Muscarinic acetylcholine receptor M10011
Muscarinic acetylcholine receptor M30011
Muscarinic acetylcholine receptor M40011
Steryl-sulfatase0101
Muscarinic acetylcholine receptor M50011
Muscarinic acetylcholine receptor M20011
Tyrosine-protein phosphatase non-receptor type 10204
Carnitine O-palmitoyltransferase 2, mitochondrial0101
Amine oxidase [flavin-containing] B0101
Amine oxidase [flavin-containing] A 0101
Amine oxidase [flavin-containing] A0101
Peroxisome proliferator-activated receptor alpha0101
Carnitine O-palmitoyltransferase 2, mitochondrial0101
Amine oxidase [flavin-containing] B0202
Peroxisome proliferator-activated receptor gamma0225
Peroxisome proliferator-activated receptor gamma0112
Carnitine O-palmitoyltransferase 1, liver isoform0101
Peroxisome proliferator-activated receptor alpha0112
Enoyl-[acyl-carrier-protein] reductase [NADH] 0101
CDGSH iron-sulfur domain-containing protein 20101
CDGSH iron-sulfur domain-containing protein 10202
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)1001
Polyunsaturated fatty acid lipoxygenase ALOX15B1001
Histamine H2 receptor1001
Guanine nucleotide-binding protein G1001
Chain A, Activated Factor Xa Heavy Chain0101
Coagulation factor X0202
Coagulation factor XII0101
Suppressor of tumorigenicity 14 protein0101
chaperonin-containing TCP-1 beta subunit homolog1001
Estrogen receptor beta0001
Solute carrier family 22 member 60101
Polyphenol oxidase 20102
Carbonic anhydrase 120202
5'-AMP-activated protein kinase subunit beta-20001
Carbonic anhydrase 10303
Albumin0101
Polymerase acidic protein0011
Carbonic anhydrase 30101
Stromelysin-10011
Tyrosine-protein phosphatase YopH0101
Aldo-keto reductase family 1 member B10101
Prolyl 4-hydroxylase subunit alpha-10101
Estrogen receptor0001
Acetylcholinesterase0101
Carbonic anhydrase 40101
Prostaglandin G/H synthase 10101
Carbonic anhydrase 60101
Cystathionine gamma-lyase0101
Carbonic anhydrase 5A, mitochondrial0101
Carbonic anhydrase 70101
Xanthine dehydrogenase/oxidase0101
Carbonic anhydrase 90202
Carbonic anhydrase0101
Solute carrier family 22 member 70001
Nicotinate phosphoribosyltransferase0101
Ubiquitin-like domain-containing CTD phosphatase 10101
Carbonic anhydrase 150101
Carbonic anhydrase 130101
5'-AMP-activated protein kinase subunit gamma-30001
Carbonic anhydrase 140101
Carbonic anhydrase 5B, mitochondrial0101
5'-AMP-activated protein kinase subunit beta-10001
polyadenylate-binding protein 10101
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023]