Proteins > relaxin receptor 1 isoform 1
Page last updated: 2024-08-07 21:02:34

relaxin receptor 1 isoform 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (220)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
9-xylosyladenineHomo sapiens (human)Potency7.931020
erythrosineHomo sapiens (human)Potency158.489010
brl 42810Homo sapiens (human)Potency17.782810
pentoxifyllineHomo sapiens (human)Potency24.169520
suprofenHomo sapiens (human)Potency12.589310
isoproterenol hydrochlorideHomo sapiens (human)Potency3.162310
2-chloroadenosineHomo sapiens (human)Potency9.324130
cladribineHomo sapiens (human)Potency19.118010
1,3,7-trimethyl-8-(phenylmethyl)purine-2,6-dioneHomo sapiens (human)Potency28.183810
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineHomo sapiens (human)Potency22.387210
isoetharine mesylateHomo sapiens (human)Potency3.162310
camptothecinHomo sapiens (human)Potency12.589310
flubendazoleHomo sapiens (human)Potency25.118910
colforsinHomo sapiens (human)Potency0.038810
phenylisopropyladenosineHomo sapiens (human)Potency8.355820
n(6)-phenyladenosineHomo sapiens (human)Potency8.334820
n-methyladenosineHomo sapiens (human)Potency20.935920
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosineHomo sapiens (human)Potency15.848910
adenosine amine congenerHomo sapiens (human)Potency7.359130
12-phenyllauric acidHomo sapiens (human)Potency35.481310
2-methyl-N-[4-(propan-2-ylamino)phenyl]-2-propenamideHomo sapiens (human)Potency11.220210
nsc606985Homo sapiens (human)Potency31.622810
adenosine-5'-(n-ethylcarboxamide)Homo sapiens (human)Potency5.109530
N-(1,3-benzodioxol-5-yl)-1-[4-(4-morpholinylsulfonyl)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency31.622810
7-[(4-fluorophenyl)methyl]-1,3-dimethyl-8-[(2-oxo-2-thiophen-2-ylethyl)thio]purine-2,6-dioneHomo sapiens (human)Potency35.481310
2-[(2-ethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency35.481310
2-[(5,6-dimethyl-4-oxo-3-phenyl-2-thieno[2,3-d]pyrimidinyl)thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency35.481310
n(6)-cyclopentyladenosineHomo sapiens (human)Potency11.945420
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]-N-(2-phenylethyl)acetamideHomo sapiens (human)Potency39.810710
5-bromo-3-ethyl-1H-indole-2-carboxylic acidHomo sapiens (human)Potency39.810710
1-[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-4-piperidinecarboxamideHomo sapiens (human)Potency32.087430
2-(4-benzofuro[3,2-d]pyrimidinylthio)-1-thiophen-2-ylethanoneHomo sapiens (human)Potency22.387210
N-(4-fluorophenyl)-2-[(2-methyl-4-benzofuro[3,2-d]pyrimidinyl)thio]acetamideHomo sapiens (human)Potency35.481310
6-amino-1-(4-fluorophenyl)-3-methyl-4-thiophen-2-yl-5-pyrazolo[3,4-b]pyridinecarbonitrileHomo sapiens (human)Potency39.810710
N-(1,3-dioxo-2-phenyl-5-isoindolyl)-2-thiophenecarboxamideHomo sapiens (human)Potency25.118910
2-amino-4-phenyl-6-(1-pyrrolidinyl)pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency35.481310
6-methoxy-2-(4-methoxyphenyl)-1-benzopyran-4-oneHomo sapiens (human)Potency31.622810
2-[(3-cyano-6-cyclopropyl-4-thiophen-2-yl-2-pyridinyl)thio]acetamideHomo sapiens (human)Potency39.810710
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)Potency6.201230
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-oneHomo sapiens (human)Potency15.848910
N-(7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamideHomo sapiens (human)Potency39.810710
7-methoxy-3,5-dimethyl-2-thiazolo[4,5-d]pyrimidinethioneHomo sapiens (human)Potency39.810710
5-cyano-2-methyl-6-sulfanylidene-1H-pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency31.622810
N-(5-acetyl-4-methyl-2-thiazolyl)-2-methylpropanamideHomo sapiens (human)Potency14.597130
5-phenyl-1,3,4-oxadiazole-2-thiolHomo sapiens (human)Potency25.118910
2-amino-4-(4-chlorophenyl)-6-methyl-3-pyridinecarbonitrileHomo sapiens (human)Potency39.810710
3-[(4,8-dimethyl-2-quinolinyl)thio]propanoic acidHomo sapiens (human)Potency15.848910
6-bromo-3-phenyl-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency39.810710
2-(3-cyano-4,5,6-trimethyl-1H-pyridin-2-ylidene)propanedinitrileHomo sapiens (human)Potency28.183810
3-prop-2-enyl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency15.848910
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneHomo sapiens (human)Potency4.774530
2-amino-1-(4-methylphenyl)-6-oxo-4-phenylpyridine-3,5-dicarbonitrileHomo sapiens (human)Potency39.810710
2-phenyl-1H-quinazoline-4-thioneHomo sapiens (human)Potency28.183810
N-cyclopentyl-2-[(6-methoxy-3-methyl-2-quinolinyl)thio]acetamideHomo sapiens (human)Potency35.481310
N-(4-anilinophenyl)-2-methylpropanamideHomo sapiens (human)Potency43.458420
4-chloro-N-(2-pyridinyl)-1-naphthalenesulfonamideHomo sapiens (human)Potency17.782810
4-[[(2-methyl-1,3-benzothiazol-6-yl)-oxomethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency39.810710
3-[[[5-(phenylmethyl)-1,3,4-oxadiazol-2-yl]thio]methyl]benzoic acidHomo sapiens (human)Potency6.309610
1-(4-methyl-1-piperidinyl)-2-[(3-methyl-2-quinoxalinyl)thio]ethanoneHomo sapiens (human)Potency25.118910
2-thiophenecarboxylic acid (6-methyl-2-oxo-1H-quinolin-3-yl)methyl esterHomo sapiens (human)Potency39.810710
3-tert-butyl-7-[[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]thio]-[1,3,4]thiadiazolo[2,3-c][1,2,4]triazin-4-oneHomo sapiens (human)Potency39.810710
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideHomo sapiens (human)Potency32.653020
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamideHomo sapiens (human)Potency31.622810
2-amino-4-(4-chlorophenyl)-1-(4-methylphenyl)-6-oxopyridine-3,5-dicarbonitrileHomo sapiens (human)Potency31.622810
2-[[3-cyano-6-(4-methylphenyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency11.817020
N-(2-methoxyphenyl)-5-methyl-3-[(2-methylphenyl)methyl]-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideHomo sapiens (human)Potency39.810710
8-[1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decaneHomo sapiens (human)Potency31.622810
N-[2-(3-chlorophenyl)ethyl]-2-[[3-cyano-6-(3-methoxyphenyl)-2-pyridinyl]thio]acetamideHomo sapiens (human)Potency35.481310
N-[5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-4-methoxybenzamideHomo sapiens (human)Potency39.810710
4-(1,3-dioxo-2-isoindolyl)-N-(4-methyl-2-pyrimidinyl)benzenesulfonamideHomo sapiens (human)Potency17.333520
N-(phenylmethyl)-2-[[4-(trifluoromethyl)-5,6-dihydrobenzo[h]quinazolin-2-yl]thio]acetamideHomo sapiens (human)Potency31.622810
2-[(3-cyano-6-methoxy-2-quinolinyl)thio]-N-(2-methyl-1,3-benzothiazol-5-yl)acetamideHomo sapiens (human)Potency35.481310
3-[[2-[[6-fluoro-2-(4-fluorophenyl)-4-quinazolinyl]thio]-1-oxoethyl]amino]benzoic acidHomo sapiens (human)Potency25.118910
3-[[1-oxo-2-[(4,6,9-trimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)thio]ethyl]amino]benzoic acidHomo sapiens (human)Potency39.810710
N-(4-acetylphenyl)-2-[[1-(3,5-dimethoxyphenyl)-5-tetrazolyl]thio]acetamideHomo sapiens (human)Potency14.125410
N-(2-ethylphenyl)-2-[[2-(4-methoxyphenyl)-4-oxo-1-benzopyran-6-yl]oxy]acetamideHomo sapiens (human)Potency14.919530
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency39.810710
5-bromo-N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency35.481310
LSM-28559Homo sapiens (human)Potency35.872130
8-chloro-N-(4-fluorophenyl)-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency15.750330
4-[[2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency35.481310
N-(4-fluorophenyl)-3-([1,2,4]triazolo[4,3-a]quinolin-1-ylthio)propanamideHomo sapiens (human)Potency28.183810
LSM-17286Homo sapiens (human)Potency25.118910
N-[[3-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency39.810710
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneHomo sapiens (human)Potency22.387210
6-[[2-(4-morpholinyl)-2-oxoethyl]thio]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrileHomo sapiens (human)Potency35.481310
N',2-dimethyl-N'-[3-(trifluoromethyl)-2-quinoxalinyl]benzohydrazideHomo sapiens (human)Potency28.183810
N-[2,5-dioxo-6-(4-phenoxyphenyl)-3-pyrano[3,2-c]pyridinyl]benzamideHomo sapiens (human)Potency35.481310
6-(4-methyl-1-piperazinyl)-2-(3,4,5-trimethoxyphenyl)-1H-benzimidazoleHomo sapiens (human)Potency31.622810
4-methoxy-N-(8-methyl-[1,3]dioxolo[4,5-g]quinazolin-6-yl)benzamideHomo sapiens (human)Potency39.810710
2-[(4-cyano-1-methyl-5,6,7,8-tetrahydroisoquinolin-3-yl)thio]-N-(3-ethoxyphenyl)acetamideHomo sapiens (human)Potency28.183810
N-(2,4-dichlorophenyl)-4-phenylbenzamideHomo sapiens (human)Potency39.810710
1-amino-3-[3-(2-sulfanylidene-3H-1,3,4-oxadiazol-5-yl)phenyl]thioureaHomo sapiens (human)Potency10.000010
2-[(2-methyl-4-benzofuro[3,2-d]pyrimidinyl)thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency39.810710
6-(4-bromophenyl)-3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4-(trifluoromethyl)pyrazolo[3,4-b]pyridineHomo sapiens (human)Potency16.258130
2-(1,3-dimethyl-2-benzimidazolylidene)-4-[(6-ethyl-4-thieno[2,3-d]pyrimidinyl)thio]-3-oxobutanenitrileHomo sapiens (human)Potency35.481310
3,5-dimethyl-4-isoxazolecarboxylic acid [2-(4-amino-1-methyl-2,6-dioxo-3-propyl-5-pyrimidinyl)-2-oxoethyl] esterHomo sapiens (human)Potency17.782810
4-[2-[[3-(4-methylphenyl)-5-triazolo[1,5-a]quinazolinyl]amino]ethyl]benzenesulfonamideHomo sapiens (human)Potency14.125410
N-(4-acetylphenyl)-5-[(phenylthio)methyl]-2-furancarboxamideHomo sapiens (human)Potency22.387210
3-phenyl-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneHomo sapiens (human)Potency15.848910
N-(4,7-dimethoxy-3-methyl-1,3-benzothiazol-2-ylidene)butanamideHomo sapiens (human)Potency39.810710
LSM-26967Homo sapiens (human)Potency14.125410
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]acetic acid ethyl esterHomo sapiens (human)Potency39.810710
5-(2-ethoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)Potency17.782810
N-[4-[(4-sulfamoylphenyl)sulfamoyl]phenyl]cyclopropanecarboxamideHomo sapiens (human)Potency39.810710
N-[(phenacylamino)-sulfanylidenemethyl]cyclohexanecarboxamideHomo sapiens (human)Potency39.810710
1-(2-chlorophenyl)-N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency35.481310
N-(3,5-dichloro-2-pyridinyl)-2-methoxy-4-(methylthio)benzamideHomo sapiens (human)Potency39.810710
2-[(4-methylphenyl)sulfonylamino]acetic acid [2-(5-bromo-2-thiophenyl)-2-oxoethyl] esterHomo sapiens (human)Potency17.782810
2-[[2-furanyl(oxo)methyl]amino]-4,5-dimethoxybenzoic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency31.622810
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideHomo sapiens (human)Potency28.183810
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency39.810710
6-(4-chlorophenyl)-4-(methylthio)-2-oxo-1H-pyridine-3-carbonitrileHomo sapiens (human)Potency14.125410
5-cyano-2-(methoxymethyl)-6-sulfanylidene-1H-pyridine-3-carboxylic acid methyl esterHomo sapiens (human)Potency25.118910
2-(4-nitrophenyl)-N-(2-oxolanylmethyl)-4-quinazolinamineHomo sapiens (human)Potency25.118910
2-({[2-acetyl-5-(tert-butyl)-3-thienyl]amino}carbonyl)benzoic acidHomo sapiens (human)Potency15.848910
5-methyl-N-[1-(phenylmethyl)-4-piperidinyl]-4-thieno[2,3-d]pyrimidinamineHomo sapiens (human)Potency22.387210
2-[(7-chloro-4-quinazolinyl)oxy]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethanoneHomo sapiens (human)Potency39.810710
3-(2,4-dimethoxyphenyl)-6-phenyl-2-sulfanylidene-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency15.848910
4-amino-7,8,9,10-tetrahydro-6H-pyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileHomo sapiens (human)Potency33.426830
1-cyclopentyl-2-imino-10-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideHomo sapiens (human)Potency31.372930
6-[[(2-methoxycarbonyl-3-thiophenyl)amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidHomo sapiens (human)Potency15.848910
N-[[(5-bromo-6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-2-(2-chlorophenoxy)acetamideHomo sapiens (human)Potency39.810710
[4-(benzenesulfonyl)-1-piperazinyl]-[6-bromo-2-(2-pyridinyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency31.622810
1,3-dimethyl-8-[2-(1-pyrrolidinyl)ethylthio]-6-sulfanylidene-7H-purin-2-oneHomo sapiens (human)Potency22.387210
4-amino-N5-(4-butoxyphenyl)-N5-[2-(cyclohexylamino)-2-oxoethyl]isothiazole-3,5-dicarboxamideHomo sapiens (human)Potency31.622810
2-[(5,6-dimethyl-2-propyl-4-thieno[2,3-d]pyrimidinyl)thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency31.622810
N-(2,4-dioxo-1H-pyrimidin-5-yl)-2-[(3-ethyl-5,8-dimethyl-2-quinolinyl)thio]acetamideHomo sapiens (human)Potency35.481310
2-(3-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency28.183810
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency39.810710
5-(6,7-diethoxy-4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)-N-(2-furanylmethyl)pentanamideHomo sapiens (human)Potency25.118910
2-(4-methoxyphenyl)-N-[4-[5-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]acetamideHomo sapiens (human)Potency22.387210
2-(4-methyl-1-oxo-[1]benzothiolo[2,3-d]pyridazin-2-yl)propanoic acidHomo sapiens (human)Potency15.848910
2-(2-ethoxyphenyl)-8-oxo-9-phenyl-7H-purine-6-carboxamideHomo sapiens (human)Potency39.810710
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1H-quinoline-4-carboxamideHomo sapiens (human)Potency11.220210
2-(4-benzofuro[3,2-d]pyrimidinylthio)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency39.810710
6-[4-oxo-2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-thieno[3,2-d]pyrimidinyl]hexanoic acidHomo sapiens (human)Potency15.848910
3-[4-oxo-2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-thieno[3,2-d]pyrimidinyl]propanoic acidHomo sapiens (human)Potency14.125410
6-bromo-2-(4-methylphenyl)-N-[(1-methyl-4-pyrazolyl)methyl]-4-quinolinecarboxamideHomo sapiens (human)Potency22.387210
5-chloro-N-(1,3-dioxo-5-isoindolyl)-2-thiophenecarboxamideHomo sapiens (human)Potency39.810710
2-thiophen-2-yl-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)Potency31.622810
6,8-dibromo-2-thiophen-2-ylquinolineHomo sapiens (human)Potency28.183810
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency15.848910
4-(5-bromo-2-thiophenyl)-6-methyl-2-(1-pyrrolyl)pyrimidineHomo sapiens (human)Potency17.782810
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency11.075830
N-(4-fluorophenyl)-5-methyl-1H-indole-2-carboxamideHomo sapiens (human)Potency39.810710
4-[[2-[(1,1-dioxo-3-thiolanyl)amino]-2-oxoethyl]thio]-2,5-dimethyl-6-thieno[2,3-d]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency28.183810
N-(2,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideHomo sapiens (human)Potency39.810710
N-(1,3-benzodioxol-5-ylmethyl)-6-[6-(4-morpholinyl)-4-oxo-2-sulfanylidene-1H-quinazolin-3-yl]hexanamideHomo sapiens (human)Potency28.183810
N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency20.085010
3-methoxy-N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)benzamideHomo sapiens (human)Potency39.810710
1-(3-methyl-1-piperidinyl)-2-(2-quinoxalinylthio)ethanoneHomo sapiens (human)Potency17.782810
2-(5-bromo-2-thiophenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency17.782810
2-[(2,2-dichloro-3,3-dimethylcyclopropyl)methylthio]-1H-benzimidazoleHomo sapiens (human)Potency31.622810
1-cyclohexyl-3-[(1,2-dimethyl-5-indolyl)methyl]ureaHomo sapiens (human)Potency39.810710
N-(4-methylphenyl)-6-(1-pyrazolyl)-3-pyridinecarboxamideHomo sapiens (human)Potency35.481310
3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency17.782810
2-(2-quinoxalinylthio)propanoic acidHomo sapiens (human)Potency15.848910
5-[3-(2-chloro-6-methoxy-3-quinolinyl)-5-(2-furanyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acidHomo sapiens (human)Potency28.183810
4-(2,5-dioxo-1-pyrrolidinyl)-N-[4-(4-methoxyphenyl)-2-thiazolyl]benzamideHomo sapiens (human)Potency35.481310
LSM-16446Homo sapiens (human)Potency17.782810
N-(1,3-dioxo-5-isoindolyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency15.255830
3-(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)-N-(3-fluoro-4-methylphenyl)propanamideHomo sapiens (human)Potency39.810710
6-(6-bromo-4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)-N-[2-(4-sulfamoylphenyl)ethyl]hexanamideHomo sapiens (human)Potency35.481310
2-(1,3-dimethyl-2,6-dioxo-7-purinyl)-N'-[2-(2-ethoxyphenoxy)-1-oxoethyl]acetohydrazideHomo sapiens (human)Potency28.597930
4-[bis(2-methoxyethyl)sulfamoyl]-N-[5-(methoxymethyl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)Potency25.118910
4-methoxy-N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)benzamideHomo sapiens (human)Potency31.622810
N-[5-(1-azepanylsulfonyl)-2-chlorophenyl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)Potency13.111330
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamideHomo sapiens (human)Potency25.118910
4-(4-chlorophenyl)-3-phenyl-1H-imidazole-2-thioneHomo sapiens (human)Potency31.622810
4-(4-chlorophenyl)-3-(phenylmethyl)-1H-imidazole-2-thioneHomo sapiens (human)Potency39.810710
3-[(2,5,6-trimethyl-4-thieno[2,3-d]pyrimidinyl)thio]-2-oxolanoneHomo sapiens (human)Potency28.183810
7-chloro-3-[2-(1-cyclohexenyl)ethyl]-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency35.481310
2-(3-methyl-1-oxo-2-isoquinolinyl)-N-(3,4,5-trimethoxyphenyl)acetamideHomo sapiens (human)Potency37.646010
2-cyano-N'-[2,6-dinitro-4-(trifluoromethyl)phenyl]acetohydrazideHomo sapiens (human)Potency39.810710
2-[2-(7-methoxy-2-oxo-1H-quinolin-3-yl)ethyl]isoindole-1,3-dioneHomo sapiens (human)Potency35.481310
ncgc00099374Homo sapiens (human)Potency15.848910
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1-benzopyran-3-carboxamideHomo sapiens (human)Potency28.183810
N-(5-acetyl-4-methyl-2-thiazolyl)-2-(2,4-dichlorophenoxy)acetamideHomo sapiens (human)Potency14.125410
N-[(1,2-dimethyl-5-indolyl)methyl]-2-(4-nitrophenyl)acetamideHomo sapiens (human)Potency39.810710
sulfuretinHomo sapiens (human)Potency48.943110
7-hydroxy-8-[[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-4-methyl-1-benzopyran-2-oneHomo sapiens (human)Potency28.183810
3-ethyl-2-sulfanylidene-6,7,8,9-tetrahydro-1H-pyrimido[4,5-b]quinolin-4-oneHomo sapiens (human)Potency35.481310
8-(1-piperidinylsulfonyl)-6-pyrido[1,2-a]quinazolinoneHomo sapiens (human)Potency32.740830
1-(2-phenylethyl)-4-([1,2,4]triazolo[4,3-a]quinoxalin-4-yl)piperazine-2,6-dioneHomo sapiens (human)Potency21.810310
N-(2-oxolanylmethyl)-2-(7-oxo-3-phenyl-6-triazolo[4,5-d]pyrimidinyl)acetamideHomo sapiens (human)Potency12.589310
1-(4-morpholinyl)-2-[[3-(3-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]ethanoneHomo sapiens (human)Potency17.782810
4-methyl-2,7-diphenyl-8H-pyrido[2,3-d]pyrimidin-5-oneHomo sapiens (human)Potency39.810710
urolithin bHomo sapiens (human)Potency14.125410
Adenosine 5'-monophosphate monohydrateHomo sapiens (human)Potency22.387210
1-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-N-(phenylmethyl)-3-piperidinecarboxamideHomo sapiens (human)Potency39.810710
epinephrine bitartrateHomo sapiens (human)Potency19.952610
3-(3-methylphenyl)-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneHomo sapiens (human)Potency28.183810
6-(4-bromophenyl)-2-methyl-3-pyridinecarboxylic acidHomo sapiens (human)Potency25.118910
N-[2-methyl-5-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-phenoxyacetamideHomo sapiens (human)Potency39.810710
lissamine rhodamine bHomo sapiens (human)Potency28.183810
(1S)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-6-methoxy-2-methyl-2-oxido-3,4-dihydro-1H-isoquinolin-2-ium-7-olHomo sapiens (human)Potency35.481310
N-(3,5-dichlorophenyl)-4-[(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)methyl]benzamideHomo sapiens (human)Potency39.810710
N'-butan-2-yl-N-[2-(3,5-dimethyl-1-piperidinyl)-4-methyl-6-quinolinyl]butanediamideHomo sapiens (human)Potency39.810710
1-butyl-3-(5-methyl-6-oxo-3-benzo[b][1,4]benzothiazepinyl)ureaHomo sapiens (human)Potency39.810710
2-[[1,3-dimethyl-7-(4-methylphenyl)-2,4-dioxo-5-pyrimido[4,5-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency39.810710
2-[[3-(3,4-dimethoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency28.183810
N,8-dimethyl-N-(3-methylphenyl)-4-oxo-5H-thieno[3,2-c]quinoline-2-carboxamideHomo sapiens (human)Potency39.810710
N-[3-[butyl(ethyl)amino]propyl]-1-(9-fluoro-[1]benzothiolo[3,2-d]pyrimidin-4-yl)-4-piperidinecarboxamideHomo sapiens (human)Potency17.782810
3-methoxy-N-(5-methyl-2-pyridinyl)-2-naphthalenecarboxamideHomo sapiens (human)Potency39.810710
LSM-16753Homo sapiens (human)Potency28.183810
LSM-26549Homo sapiens (human)Potency1.584910
2-(2,5-dichlorophenoxy)-1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-butanoneHomo sapiens (human)Potency31.622810
bucladesineHomo sapiens (human)Potency0.719630
cyclic amp, monosodium saltHomo sapiens (human)Potency0.524830
(2R)-2-[[(3S)-3-acetamido-3-carboxy-1-oxopropyl]amino]pentanedioic acidHomo sapiens (human)Potency6.309610
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency35.481310
2-[[2-(phenoxymethyl)-4-quinazolinyl]thio]acetic acid methyl esterHomo sapiens (human)Potency25.118910
3-[(2-chlorophenyl)methyl]-N-(2-fluorophenyl)-5-methyl-7-triazolo[4,5-d]pyrimidinamineHomo sapiens (human)Potency39.810710
N-(2-fluorophenyl)-2-[[7-(2-fluorophenyl)-1,3-dimethyl-2,4-dioxo-5-pyrimido[4,5-d]pyrimidinyl]thio]acetamideHomo sapiens (human)Potency25.118910
4-hydroxy-1-methyl-3-(phenylthio)-1,2-dihydroquinolin-2-oneHomo sapiens (human)Potency39.810710
LSM-17430Homo sapiens (human)Potency10.000010
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-6-methyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency25.118910
2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]acetamideHomo sapiens (human)Potency17.782810
2-[[2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]-4-methylpentanoic acid methyl esterHomo sapiens (human)Potency31.622810