Page last updated: 2024-08-08 00:10:52

Multidrug resistance associated protein

[no definition available]

Synonyms

Research

Bioassay Publications (6)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (7)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
taurocholic acidHomo sapiens (human)IC5040.000011
methotrexateHomo sapiens (human)Ki1,200.000011
E3040 glucuronideHomo sapiens (human)Ki5.600011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
taurocholic acidHomo sapiens (human)Km30.000011
glycocholic acidHomo sapiens (human)Km248.000011
methotrexateHomo sapiens (human)Km768.666733
estradiol-17 beta-glucuronideHomo sapiens (human)Km28.800044
folic acidHomo sapiens (human)Km1,960.000011
leucovorinHomo sapiens (human)Km1,740.000011