Page last updated: 2024-08-07 18:44:03

Solute carrier family 22 member 7

A solute carrier family 22 member 7 that is encoded in the genome of rat. [OMA:Q5RLM2, PRO:DNx]

Synonyms

Novel liver transporter;
Organic anion transporter 2

Research

Bioassay Publications (3)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (16)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
glyburideRattus norvegicus (Norway rat)Ki12.300010
ketoprofenRattus norvegicus (Norway rat)Ki1.840010
probenecidRattus norvegicus (Norway rat)IC50977.000011
cephaloridineRattus norvegicus (Norway rat)IC505,000.000011
cephalothinRattus norvegicus (Norway rat)IC501,500.000011
cefoperazoneRattus norvegicus (Norway rat)IC501,620.000011
pravastatinRattus norvegicus (Norway rat)IC50449.000011
cefamandoleRattus norvegicus (Norway rat)IC503,180.000011
cefotaximeRattus norvegicus (Norway rat)IC505,000.000011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
alpha-ketoglutaric acidRattus norvegicus (Norway rat)Km17.800011
salicylic acidRattus norvegicus (Norway rat)Km85.000021
indomethacinRattus norvegicus (Norway rat)Km0.366010
zalcitabineRattus norvegicus (Norway rat)Km3,000.000010
zidovudineRattus norvegicus (Norway rat)Km26.000010
dinoprostoneRattus norvegicus (Norway rat)Km38.500010
dinoprostRattus norvegicus (Norway rat)Km0.414011