Page last updated: 2024-08-07 21:16:27
Tyrosine-protein kinase JAK2
A tyrosine-protein kinase JAK2 that is encoded in the genome of mouse. [OMA:Q62120, PRO:DNx]
Synonyms
EC 2.7.10.2;
Janus kinase 2;
JAK-2
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 3 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
sb 1518 | Mus musculus (house mouse) | IC50 | 1.0613 | 1 | 1 |
bms-911543 | Mus musculus (house mouse) | IC50 | 0.0650 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
incb-018424 | Mus musculus (house mouse) | EC50 | 0.1860 | 1 | 1 |