Page last updated: 2024-08-07 23:42:51
Solute carrier organic anion transporter family member 1A3
A protein that is a translation product of the Slc21a4 gene in rat. [PRO:DNx, UniProtKB:P70502]
Synonyms
OAT-K2;
Sodium-independent organic anion transporter K1;
OAT-K1;
Solute carrier family 21 member 4;
rOAT-K
Research
Bioassay Publications (6)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (66.67) | 18.2507 |
2000's | 2 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (15)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
indomethacin | Rattus norvegicus (Norway rat) | Ki | 1,000.0000 | 1 | 1 |
ketoprofen | Rattus norvegicus (Norway rat) | Ki | 1,900.0000 | 1 | 1 |
sulfobromophthalein sodium | Rattus norvegicus (Norway rat) | Ki | 21.0000 | 1 | 1 |
taurocholic acid | Rattus norvegicus (Norway rat) | Ki | 183.0000 | 1 | 1 |
aminopterin | Rattus norvegicus (Norway rat) | Ki | 0.5000 | 1 | 1 |
5-methyltetrahydrofolate | Rattus norvegicus (Norway rat) | Ki | 1.2000 | 1 | 1 |
folic acid | Rattus norvegicus (Norway rat) | Ki | 14.1000 | 1 | 1 |
leucovorin | Rattus norvegicus (Norway rat) | Ki | 8.2000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
thyroxine | Rattus norvegicus (Norway rat) | Km | 16.1000 | 2 | 2 |
triiodothyronine | Rattus norvegicus (Norway rat) | Km | 34.3000 | 2 | 2 |
taurocholic acid | Rattus norvegicus (Norway rat) | Km | 20.7000 | 2 | 2 |
dehydroepiandrosterone sulfate | Rattus norvegicus (Norway rat) | Km | 8.0500 | 2 | 2 |
zidovudine | Rattus norvegicus (Norway rat) | Km | 70.3000 | 2 | 2 |
methotrexate | Rattus norvegicus (Norway rat) | Km | 1.6333 | 3 | 3 |
ochratoxin a | Rattus norvegicus (Norway rat) | Km | 11.1000 | 2 | 2 |
estradiol-17 beta-glucuronide | Rattus norvegicus (Norway rat) | Km | 40.1000 | 2 | 2 |