Page last updated: 2024-08-07 23:42:51

Solute carrier organic anion transporter family member 1A3

A protein that is a translation product of the Slc21a4 gene in rat. [PRO:DNx, UniProtKB:P70502]

Synonyms

OAT-K2;
Sodium-independent organic anion transporter K1;
OAT-K1;
Solute carrier family 21 member 4;
rOAT-K

Research

Bioassay Publications (6)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's4 (66.67)18.2507
2000's2 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (15)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
indomethacinRattus norvegicus (Norway rat)Ki1,000.000011
ketoprofenRattus norvegicus (Norway rat)Ki1,900.000011
sulfobromophthalein sodiumRattus norvegicus (Norway rat)Ki21.000011
taurocholic acidRattus norvegicus (Norway rat)Ki183.000011
aminopterinRattus norvegicus (Norway rat)Ki0.500011
5-methyltetrahydrofolateRattus norvegicus (Norway rat)Ki1.200011
folic acidRattus norvegicus (Norway rat)Ki14.100011
leucovorinRattus norvegicus (Norway rat)Ki8.200011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
thyroxineRattus norvegicus (Norway rat)Km16.100022
triiodothyronineRattus norvegicus (Norway rat)Km34.300022
taurocholic acidRattus norvegicus (Norway rat)Km20.700022
dehydroepiandrosterone sulfateRattus norvegicus (Norway rat)Km8.050022
zidovudineRattus norvegicus (Norway rat)Km70.300022
methotrexateRattus norvegicus (Norway rat)Km1.633333
ochratoxin aRattus norvegicus (Norway rat)Km11.100022
estradiol-17 beta-glucuronideRattus norvegicus (Norway rat)Km40.100022