Page last updated: 2024-08-05 14:48:33

antiviral agent

A substance that destroys or inhibits replication of viruses.

ChEBI ID: 22587

Members (73)

MemberDefinitionClass
2,2'-spirobi[3,6,7,8-tetrahydro-1H-cyclopenta[g]naphthalene]-5,5'-dioneA spiro compound that consists of two units of 1,2,3,6,7,8-hexahydro-5H-cyclopenta[b]naphthalen-5-one fused together at position 2. It is an inhibitor of Hepatitis C virus E2 protein that exhibits inhibitory activity against hepatitis C virus infections.2,2'-spirobi[3,6,7,8-tetrahydro-1H-cyclopenta[g]naphthalene]-5,5'-dione
3'-deoxyadenosine 5'-triphosphatecordycepin triphosphate
9-deoxy-9,10-didehydro-12,13-didehydro-13,14-dihydroprostaglandin d2A member of the class of prostaglandins J that is prosta-5,9,12-trien-1-oic acid carrying oxo and hydsroxy substituents at positions 11 and 15 respectively (the 5Z,12E,15S-stereoisomer).13,14-dihydro-Delta(12)-prostaglandin J2
agathisflavoneA biflavonoid that is obtained by oxidative coupling of two molecules of apigenin resulting in a bond between positions C-6 and C-8 of the two chromene rings.agathisflavone
amantadine hydrochlorideA hydrochloride obtained by combining amantadine and hydrochloric acid in equimolar amounts.amantadine hydrochloride
amentoflavoneA biflavonoid that is obtained by oxidative coupling of two molecules of apigenin resulting in a bond between positions C-3 of the hydroxyphenyl ring and C-8 of the chromene ring. A natural product found particularly in Ginkgo biloba and Hypericum perforatum.amentoflavone
antofineAn organic heteropentacyclic compound that is (13aR)-9,11,12,13,13a,14-hexahydrodibenzo[f,h]pyrrolo[1,2-b]isoquinoline substituted at positions 2, 3 and 6 by methoxy groups. It is an alkaloid produced by relatives of the milkweed family and exhibits antiviral, anti-inflammatory, antiadipogenic and antitumorigenic activities.(-)-antofine
ARS-1620A qinazoline derivative carrying chloro and fluoro substituents at positions 6 and 8 respectively, a 2-fluoro-6-hydroxyphenyl group at position 7, and a 4-(prop-2-enoyl)piperazin-1-yl group at position 4. A potent, selective, and orally bioavailable covalent KRAS-G12C inhibitor, it inhibits the protein coding gene KRAS (Kirsten rat sarcoma virus) with high potency in cells and animals.ARS-1620
aspulvinone EA 4-hydroxy-5-(4-hydroxybenzylidene)-3-(4-hydroxyphenyl)furan-2(5H)-one in which the double bond adopts a Z-configuration. It is a marine metabolite isolated from the fungus Aspergillus terreus and exhibits antiviral activity.aspulvinone E
baricitinibA pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted by a 1-[3-(cyanomethyl)-1-(ethanesulfonyl)azetidin-3-yl]-1H-pyrazol-4-yl group at position 5. It is an FDA approved selective Janus Kinase 1 and 2 (JAK1 and JAK2) inhibitor used for the treatment of rheumatoid arthritis.baricitinib
benzethonium chlorideA (synthetic) quaternary ammonium salt that is benzyldimethylamine in which the nitrogen is quaternised by a 2-{2-[p-(2,4,4-trimethylpentan-2-yl)phenoxy]ethoxy}ethyl group, with chloride as the counter-ion. An antiseptic and disinfectant, it is active against a broad spectrum of bacteria, fungi, moulds and viruses.benzethonium chloride
betulinA pentacyclic triterpenoid that is lupane having a double bond at position 20(29) as well as 3beta-hydroxy and 28-hydroxymethyl substituents.betulin
brequinarA quinolinemonocarboxylic acid that is quinoline substituted by 2'-fluoro[1,1'-biphenyl]-4-yl, methyl, carboxy and fluoro groups at positions 2, 3, 4, and 6, respectively. It is an inhibitor of dihydroorotate dehydrogenase, an enzyme that is required for de novo pyrimidine biosynthesis. The compound exhibits antineoplastic and antiviral properties.brequinar
brequinar sodiumAn organic sodium salt of brequinar.brequinar sodium
buforminA member of the class of biguanides that is biguanide substituted by a butyl group at position 1. It is an antidiabetic drug with potential antitumor effect.buformin
caffeic acid phenethyl esterAn alkyl caffeate ester in which 2-phenylethyl is the alkyl component.phenethyl caffeate
camostatA benzoate ester resulting from the formal condensation of the carboxy group of 4-guanidinobenzoic acid with the hydroxy group of 2-(dimethylamino)-2-oxoethyl (4-hydroxyphenyl)acetate. It is a potent inhibitor of the human transmembrane protease serine 2 (TMPRSS2) and its mesylate salt is currently under investigation for its effectiveness in COVID-19 patients.camostat
camostat mesylateA methanesulfonate (mesylate) salt prepared from equimolar amounts of camostat and methanesulfonic acid. It is a serine protease inhibitor approved and marketed in Japan in 1985 for the alleviation of acute symptoms associated with chronic pancreatitis. In 1994, it was approved for the treatment of postoperative reflux esophagitis.camostat mesylate
chrysophanic acidA trihydroxyanthraquinone that is chrysazin with a methyl substituent at C-3. It has been isolated from Aloe vera and exhibits antiviral and anti-inflammatory activity.chrysophanol
chrysosplenetin bA tetramethoxyflavone that is the 3,6,7,3'-tetramethyl ether derivative of quercetagetin.chrysosplenetin
chrysosplenol cA trimethoxyflavone that is the 3,7,3'-trimethyl ether derivative of quercetagetin.chrysosplenol C
cinanserinAn aryl sulfide that is (2E)-3-phenyl-N-(2-sulfanylphenyl)prop-2-enamide in which the hydrogen of the thiol group is substituted by a 3-(dimethylamino)propyl group. It is a 5-hydroxytryptamine receptor antagonist and an inhibitor of SARS-CoV replication.cinanserin
cryptopleurineAn organic heteropentacyclic compound that is (14aR)-11,12,13,14,14a,15-hexahydro-9H-dibenzo[f,h]pyrido[1,2-b]isoquinoline substituted at positions 2, 3 and 6 by methoxy groups.cryptopleurine
cytarabineA pyrimidine nucleoside in which cytosine is attached to D-arabinofuranose via a beta-N(1)-glycosidic bond. Used mainly in the treatment of leukaemia, especially acute non-lymphoblastic leukaemia, cytarabine is an antimetabolite antineoplastic agent that inhibits the synthesis of DNA. It also has antiviral and immunosuppressant properties.cytarabine
d-alpha tocopherolAn alpha-tocopherol that has R,R,R configuration. The naturally occurring stereoisomer of alpha-tocopherol, it is found particularly in sunflower and olive oils.(R,R,R)-alpha-tocopherol
daphnoretinA member of the class of coumarins that is coumarin substituted by a hydroxy group at position 7, a methoxy group at position 6 and a (2-oxo-2H-chromen-7-yl)oxy group at position 3.daphnoretin
deguelinA rotenone that is 13,13a-dihydro-3H-chromeno[3,4-b]pyrano[2,3-h]chromen-7(7aH)-one substituted by methoxy groups at positions 9 and 10, and by two methyl groups at position 3 (the 7aS,13aS-stereoisomer). It exists in abundant quantities in the bark, roots, and leaves of the Leguminosae family of plants and reported to exert anti-tumour effects in various cancers.deguelin
diazooxonorleucineA non-proteinogenic L-alpha-amino acid that is L-norleucine which is substituted at position 5 by an oxo group and at position 6 by a diazo group. It is as inhibitor of various glutamine-utilising enzymes.6-diazo-5-oxo-L-norleucine zwitterion; 6-diazo-5-oxo-L-norleucine
dioscinA spirostanyl glycoside that consists of the trisaccharide alpha-L-Rha-(1->4)-[alpha-L-Rha-(1->2)]-beta-D-Glc attached to position 3 of diosgenin via a glycosidic linkage.dioscin
diosgeninA sapogenin that is spirostan which is substituted by a hydroxy group at the 3beta position, contains a double bond at the 5-6 position, and has R- configuration at position 25. A natural product found in Dioscorea (wild yam) species, it is used as the starting point for the commercial synthesis of a number of steroids, including cortisone, pregnenolone and progesterone.diosgenin
emetineA pyridoisoquinoline comprising emetam having methoxy substituents at the 6'-, 7'-, 10- and 11-positions. It is an antiprotozoal agent and emetic. It inhibits SARS-CoV2, Zika and Ebola virus replication and displays antimalarial, antineoplastic and antiamoebic properties.emetine
emetine dihydrochlorideThe dihydrochloride salt of emetine.emetine dihydrochloride
etravirineAn aminopyrimidine that consists of 2,6-diaminopyrimidine bearing a bromo substituent at position 5, a 4-cyano-2,6-dimethylphenoxy substituent at position 4 and having a 4-cyanophenyl substituent attached to the 2-amino group. NNRTI of HIV-1, binds directly to RT and blocks RNA-dependent and DNA-dependent DNA polymerase activitiesetravirine
flavasperoneA naphtho-gamma-pyrone that is 4H-naphtho[1,2-b]pyran-4-one carrying a methyl substituent at position2, a hydroxy substituent at position 5 and two methoxy substotuents at positions 8 and 10. Originally isolated from Aspergillus niger.flavasperone
fludarabine phosphateA purine arabinonucleoside monophosphate having 2-fluoroadenine as the nucleobase. A prodrug, it is rapidly dephosphorylated to 2-fluoro-ara-A and then phosphorylated intracellularly by deoxycytidine kinase to the active triphosphate, 2-fluoro-ara-ATP. Once incorporated into DNA, 2-fluoro-ara-ATP functions as a DNA chain terminator. It is used for the treatment of adult patients with B-cell chronic lymphocytic leukemia (CLL) who have not responded to, or whose disease has progressed during, treatment with at least one standard alkylating-agent containing regimenas.fludarabine phosphate
ganodermadiolA tetracyclic triterpenoid that is lanosta-7,9(11),24-triene which is substituted by hydroxy groups at positions 3 and 27. It has been isolated from several Ganoderma species.ganoderol B
geldanamycinAn ansamycin consisting of a 19-membered macrocyle incorporating a benzoquinone ring and a lactam functionality. It shows antimicrobial activity against many Gram-positive and some Gram-negative bacteria.geldanamycin
germacroneA germacrane sesquiterpenoid that has formula C15H22O. It is a natural product found in traditional medicinal plants of the family Zingiberaceae. The compound exhibits a range of pharmacological activities including anti-inflammatory, anticancer, antiviral, anti-androgenic, antioxidant, antimicrobial, antifungal, neuroprotective and insecticidal activities.(E,E)-germacrone
ginsenoside rb2A ginsenoside found in Panax ginseng that is dammarane which is substituted by hydroxy groups at the 3beta, 12beta and 20 pro-S positions, in which the hydroxy groups at positions 3 and 20 have been converted to the corresponding beta-D-glucopyranosyl-(1->2)-beta-D-glucopyranoside and alpha-L-arabinopyranosyl-(1->6)-beta-D-glucopyranoside respectively, and in which a double bond has been introduced at the 24-25 position.ginsenoside Rb2
goitrinA 5-ethenyl-1,3-oxazolidine-2-thione that has R-configuration. It is a constituent of a traditional Chinese herbal medicine, Radix isatidis.(R)-goitrin
gramineAn aminoalkylindole that is indole carrying a dimethylaminomethyl substituent at postion 3.gramine
GS-441524A C-nucleoside analog that is (2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-carbonitrile substituted by a 4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl group at position 2. It is the active metabolite of remdesivir and exhibits a broad range of inhibitory activity against various RNA viruses including HCV, parainfluenza and SARS-CoV.GS-441524
hydroxyguanidineA member of the class of guanidines that is guanidine in which one of the hydrogens attached to the nitrogen at position 1 is substituted by a hydroxy group.N-hydroxyguanidine
hypothiocyanite ionA sulfur oxoacid that is sulfenic acid in which the hydrogen attached to the sulfur has been replaced by a cyano group.hypothiocyanous acid
ladaneinA dimethoxyflavone that is scutellarein in which the hydroxy groups at positions 4' and 7 are replaced by methoxy groups. It is an effective anti-HCV agent.ladanein
ldc4297A pyrazolotriazine that is pyrazolo[1,5-a][1,3,5]triazine substituted by a piperidin-3-yloxy group, [2-(1H-pyrazol-1-yl)benzyl]nitrilo group and an isopropyl group at positions 2, 4 and 8 respectively. It is a potent and selective CDK7 inhibitor and exhibits antiviral activity.LDC4297
minquartynoic acidA straight-chain, C18 polyunsaturated fatty acid having four conjugated C#C bonds at positions 9, 11, 13 and 15 as well as an (S)-hydroxy group at position 17.minquartynoic acid
monolinoleinA 1-monoglyceride that has octadecadienoyl (linoleoyl) as the acyl group.1-monolinolein; rac-1-monolinoleoylglycerol
N-[(5-methyl-1,2-oxazol-3-yl)carbonyl]-L-alanyl-L-valyl-N-{(2S,3E)-5-(benzyloxy)-5-oxo-1-[(3S)-2-oxopyrrolidin-3-yl]pent-3-en-2-yl}-L-leucinamideA tripeptide resulting from the formal condensation of the carboxy group of N-[(5-methyl-1,2-oxazol-3-yl)carbonyl]-L-alanyl-L-valine with the amino group of benzyl (2E,4S)-4-(L-leucylamino)-5-[(3S)-2-oxopyrrolidin-3-yl]pent-2-enoate. It is an inhibitor of the main protease of SARS-CoV-2.N-[(5-methyl-1,2-oxazol-3-yl)carbonyl]-L-alanyl-L-valyl-N-{(2S,3E)-5-(benzyloxy)-5-oxo-1-[(3S)-2-oxopyrrolidin-3-yl]pent-3-en-2-yl}-L-leucinamide
n-nonyl-1-deoxynojirimycinA hydroxypiperidine that is deoxynojirimycin (duvoglustat) in which the amino hydrogen is replaced by a nonyl group.N-nonyldeoxynojirimycin
n(4)-hydroxycytidineA nucleoside analogue that is cytidine which carries a hydroxy group at the N(4)-positon. It has broad-spectrum antiviral activity against influenza, SARS-CoV , SARS-CoV-2 and MERS-CoV.N(4)-hydroxycytidine
nsc 23766An aminopyrimidine that is 6-methylpyrimidine-2,4-diamine in which the amino groups at positions 2 and 4 are substituted by 5-(diethylamino)pentan-2-yl and 4-amino-2-methylquinolin-6-yl groups respectively. An inhibitor of the signalling G-protein known as RAC1 (Ras-related C3 botulinum toxin substrate 1).NSC 23766
nsc 23766A hydrochloride resulting from the formal reaction of NSC 23766 with 3 mol eq. of hydrogen chloride. An inhibitor of the signalling G-protein known as RAC1 (Ras-related C3 botulinum toxin substrate 1).NSC 23766 trihydrochloride
pateamine aA marine macrodiolide that is isolated from the sponge Mycale hentscheli and exhibits anticancer and antiviral propertiespateamine
phosphonoacetic acidA member of the class of phosphonic acids that is phosphonic acid in which the hydrogen attached to the phosphorous is replaced by a carboxymethyl group.phosphonoacetic acid
quercetagetinA hexahydroxyflavone that is flavone substituted by hydroxy groups at positions 3, 5, 6, 7, 3' and 4' respectively.quercetagetin
ribavirinA 1-ribosyltriazole that is the 1-ribofuranosyl derivative of 1,2,4-triazole-3-carboxamide. A synthetic guanosine analogue, it is an inhibitor of HCV polymerase and possesses a broad spectrum of activity against DNA and RNA viruses.ribavirin
ribavirin 5'-diphosphateA 1-ribosyltriazole that is ribavirin in which the hydroxy group at the 5'-position is replaced by a phosphonooxy group. It is the active metabolite of the antiviral agent ribavirin.ribavirin 5'-monophosphate
ribavirin 5'-diphosphateA 1-ribosyltriazole that is ribavirin in which the hydroxy group at the 5'-position is replaced by a diphosphate group. It is the metabolite of the antiviral agent ribavirin.ribavirin 5'-diphosphate
ribavirin 5'-triphosphateA 1-ribosyltriazole that is ribavirin in which the hydroxy group at the 5'-position is replaced by a triphosphate group. It is the active metabolite of the antiviral agent ribavirin.ribavirin 5'-triphosphate
rtki cpdA member of the class of quinazolines that is quinazoline substituted by methoxy groups at positions 6 and 7 and a (3-chlorophenyl)nitrilo group at position 4. It acts as an epidermal growth factor receptor antagonist.tyrphostin AG 1478
simalikalactone DA quassinoid isolated from Quassia amara and Quassia africana. It has been shown to exhibit antimalarial, cytotoxic and antiviral activities.simalikalactone D
stavudineA nucleoside analogue obtained by formal dehydration across positions 2 and 3 of thymidine. An inhibitor of HIV-1 reverse transcriptasestavudine
sugiolAn abietane diterpenoid that is ferruginol in which the methylene group para to the phenolic hydroxy group has been substituted by an oxo group.sugiol
surfactin AA cyclodepsipeptide that is N-[(3R)-3-hydroxy-11-methyldodecanoyl]-L-alpha-glutamyl-L-leucyl-D-leucyl-L-valyl-L-alpha-aspartyl-D-leucyl-L-leucine in which the C-terminal carboxy group has been lactonised by condensation with the alcoholic hydroxy group.surfactin A
surfactin cA cyclodepsipeptide that is N-[(3R)-3-hydroxy-13-methyltetradecanoyl]-L-alpha-glutamyl-L-leucyl-D-leucyl-L-valyl-L-alpha-aspartyl-D-leucyl-L-leucine in which the C-terminal carboxy group has been lactonised by condensation with the alcoholic hydroxy group.surfactin C
tiloroneA member of the class of fluoren-9-ones that is 9H-fluoren-9-one which is substituted by a 2-(diethylamino)ethoxy group at positions 2 and 7. It is an interferon inducer and a selective alpha7 nicotinic acetylcholine receptor (alpha7 nAChR) agonist. Its hydrochloride salt is used as an antiviral drug.tilorone
topopyrone cA naphthochromene that is 4H-naphtho[2,3-h]chromene-4,7,12-trione substituted by hydroxy groups at positions 5, 9 and 11 and a methyl group at position 2. It is isolated from fungal strains Phoma and Penicillium and acts as an inhibitor of the enzyme topoisomerase I.topopyrone C
u 18666aA hydrochloride obtained by reaction of 3beta-(2-diethylaminoethoxy)androst-5-en-17-one with one equivalent of hydrochloric acid. It is a cholesterol synthesis and transport inhibitor.3beta-(2-diethylaminoethoxy)androst-5-en-17-one hydrochloride
valinomycinA twelve-membered cyclodepsipeptide composed of three repeating D-alpha-hydroxyisovaleryl-D-valyl-L-lactoyl-L-valyl units joined in sequence. An antibiotic found in several Streptomyces strains.valinomycin
win 53338An isoxazole compound having a methyl substituent at the 3-position and a 5-[2-chloro-4-(4,5-dihydro-1,3-oxazol-2-yl)phenoxy]pentyl substituent at the 5-position.5-{5-[2-chloro-4-(4,5-dihydro-1,3-oxazol-2-yl)phenoxy]pentyl}-3-methylisoxazole
xanthohumolA member of the class of chalcones that is trans-chalcone substituted by hydroxy groups at positions 4, 2' and 4', a methoxy group at position 6' and a prenyl group at position 3'. Isolated from Humulus lupulus, it induces apoptosis in human malignant glioblastoma cells.xanthohumol
zanamivirzanamivir

Research

Studies (72,152)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-199018,108 (25.10)18.7374
1990's12,550 (17.39)18.2507
2000's18,194 (25.22)29.6817
2010's18,551 (25.71)24.3611
2020's4,749 (6.58)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials8,059 (10.40%)5.53%
Reviews6,940 (8.96%)6.00%
Case Studies4,372 (5.64%)4.05%
Observational309 (0.40%)0.25%
Other57,813 (74.60%)84.16%

Protein Targets (832)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1Homo sapiens (human)Potency28.082118
15-lipoxygenase, partialHomo sapiens (human)Potency8.175012
67.9K proteinVaccinia virusPotency15.1859210
acetylcholinesteraseHomo sapiens (human)Potency13.5135412
acid sphingomyelinaseHomo sapiens (human)Potency100.663612
activating transcription factor 6Homo sapiens (human)Potency29.521827
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency27.8074115
alpha-galactosidaseHomo sapiens (human)Potency47.393612
Alpha-synucleinHomo sapiens (human)Potency10.241013
apical membrane antigen 1, AMA1Plasmodium falciparum 3D7Potency35.481311
AR proteinHomo sapiens (human)Potency13.35151158
aryl hydrocarbon receptorHomo sapiens (human)Potency37.261624
arylsulfatase AHomo sapiens (human)Potency25.376012
ATAD5 protein, partialHomo sapiens (human)Potency13.2061919
Ataxin-2Homo sapiens (human)Potency8.514428
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency8.816414
ATPase family AAA domain-containing protein 5Homo sapiens (human)Potency3.671528
Bloom syndrome protein isoform 1Homo sapiens (human)Potency11.9865212
bromodomain adjacent to zinc finger domain 2BHomo sapiens (human)Potency50.354012
caspase 7, apoptosis-related cysteine proteaseHomo sapiens (human)Potency51.145212
caspase-3Cricetulus griseus (Chinese hamster)Potency30.731411
caspase-3Homo sapiens (human)Potency51.145212
Caspase-7Cricetulus griseus (Chinese hamster)Potency30.731411
Cellular tumor antigen p53Homo sapiens (human)Potency22.8253322
cellular tumor antigen p53 isoform aHomo sapiens (human)Potency16.840613
Chain A, 2-oxoglutarate OxygenaseHomo sapiens (human)Potency25.207218
Chain A, ATP-DEPENDENT DNA HELICASE Q1Homo sapiens (human)Potency7.079511
Chain A, Beta-lactamaseEscherichia coli K-12Potency18.527623
Chain A, Breast cancer type 1 susceptibility proteinHomo sapiens (human)Potency39.810711
Chain A, CruzipainTrypanosoma cruziPotency39.810711
Chain A, Ferritin light chainEquus caballus (horse)Potency34.293824
Chain A, GlucosylceramidaseHomo sapiens (human)Potency0.085811
Chain A, HADH2 proteinHomo sapiens (human)Potency26.134025
Chain A, JmjC domain-containing histone demethylation protein 3AHomo sapiens (human)Potency74.306213
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency23.0843212
Chain A, Putative fructose-1,6-bisphosphate aldolaseGiardia intestinalisPotency12.363913
Chain A, TYROSYL-DNA PHOSPHODIESTERASEHomo sapiens (human)Potency31.804615
Chain B, HADH2 proteinHomo sapiens (human)Potency26.134025
chromobox protein homolog 1Homo sapiens (human)Potency69.033026
cytochrome P450 2C19 precursorHomo sapiens (human)Potency18.317412
cytochrome P450 2C9, partialHomo sapiens (human)Potency23.769013
cytochrome P450 2D6Homo sapiens (human)Potency15.951915
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency10.461114
cytochrome P450 3A4 isoform 1Homo sapiens (human)Potency12.9221219
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency15.9169211
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aHomo sapiens (human)Potency7.661619
D(1A) dopamine receptorHomo sapiens (human)Potency22.387211
D(1A) dopamine receptorSus scrofa (pig)Potency0.791412
Disintegrin and metalloproteinase domain-containing protein 17Homo sapiens (human)Potency25.118911
DNA dC->dU-editing enzyme APOBEC-3F isoform aHomo sapiens (human)Potency6.309611
DNA dC->dU-editing enzyme APOBEC-3G isoform 1Homo sapiens (human)Potency17.541622
DNA polymerase betaHomo sapiens (human)Potency58.073313
DNA polymerase eta isoform 1Homo sapiens (human)Potency32.086323
DNA polymerase III, partialBacillus subtilisPotency21.192311
DNA polymerase iota isoform a (long)Homo sapiens (human)Potency49.108214
DNA polymerase kappa isoform 1Homo sapiens (human)Potency28.522915
endonuclease IVEscherichia coliPotency8.354324
enteropeptidase precursorHomo sapiens (human)Potency28.183811
estrogen nuclear receptor alphaHomo sapiens (human)Potency18.00971164
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency33.608239
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency6.53941062
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency18.2467112
EWS/FLI fusion proteinHomo sapiens (human)Potency13.6074420
farnesoid X nuclear receptorHomo sapiens (human)Potency32.3892512
flap endonuclease 1Homo sapiens (human)Potency32.944926
Fumarate hydrataseHomo sapiens (human)Potency16.938414
GVesicular stomatitis virusPotency23.769013
GABA theta subunitRattus norvegicus (Norway rat)Potency12.4341110
GALC proteinHomo sapiens (human)Potency0.707911
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)Potency12.4341110
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)Potency12.4341110
gemininHomo sapiens (human)Potency8.5102423
GLI family zinc finger 3Homo sapiens (human)Potency7.3768314
glp-1 receptor, partialHomo sapiens (human)Potency10.832515
GLS proteinHomo sapiens (human)Potency22.665123
glucocerebrosidaseHomo sapiens (human)Potency9.355923
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency18.6993515
Glutamate receptor 2Rattus norvegicus (Norway rat)Potency17.319019
GTP-binding nuclear protein Ran isoform 1Homo sapiens (human)Potency3.468914
Guanine nucleotide-binding protein GHomo sapiens (human)Potency4.466811
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)Homo sapiens (human)Potency14.028127
heat shock protein beta-1Homo sapiens (human)Potency29.300326
Histamine H2 receptorCavia porcellus (domestic guinea pig)Potency12.812716
histone acetyltransferase KAT2A isoform 1Homo sapiens (human)Potency35.481311
histone deacetylase 9 isoform 3Homo sapiens (human)Potency7.230926
Histone H2A.xCricetulus griseus (Chinese hamster)Potency32.6944216
histone-lysine N-methyltransferase 2A isoform 2 precursorHomo sapiens (human)Potency39.810711
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency23.769013
huntingtin isoform 2Homo sapiens (human)Potency28.183811
hypoxia-inducible factor 1 alpha subunitHomo sapiens (human)Potency27.212426
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)Homo sapiens (human)Potency37.043533
IDH1Homo sapiens (human)Potency9.141813
importin subunit beta-1 isoform 1Homo sapiens (human)Potency30.104327
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency23.769016
Inositol monophosphatase 1Rattus norvegicus (Norway rat)Potency8.822513
Interferon betaHomo sapiens (human)Potency15.7031318
interleukin 8Homo sapiens (human)Potency67.119813
lamin isoform A-delta10Homo sapiens (human)Potency7.1833215
lethal factor (plasmid)Bacillus anthracis str. A2012Potency15.167816
LuciferasePhotinus pyralis (common eastern firefly)Potency38.901811
M-phase phosphoprotein 8Homo sapiens (human)Potency55.540513
Microtubule-associated protein tauHomo sapiens (human)Potency18.5674220
mitogen-activated protein kinase 1Homo sapiens (human)Potency9.379438
muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)Potency8.694224
muscleblind-like protein 1 isoform 1Homo sapiens (human)Potency6.309611
neuropeptide S receptor isoform AHomo sapiens (human)Potency7.550612
NFKB1 protein, partialHomo sapiens (human)Potency15.848922
nonstructural protein 1Influenza A virus (A/WSN/1933(H1N1))Potency5.809214
NPC intracellular cholesterol transporter 1 precursorHomo sapiens (human)Potency58.047911
Nrf2Homo sapiens (human)Potency12.224022
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency31.0801420
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency12.074216
nuclear factor NF-kappa-B p105 subunit isoform 1Homo sapiens (human)Potency42.239512
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency29.751426
Nuclear receptor ROR-gammaHomo sapiens (human)Potency16.922814
nuclear receptor ROR-gamma isoform 1Mus musculus (house mouse)Potency113.5964212
nuclear receptor subfamily 1, group I, member 2Rattus norvegicus (Norway rat)Potency0.100011
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency17.4380326
parathyroid hormone/parathyroid hormone-related peptide receptor precursorHomo sapiens (human)Potency107.508612
ParkinHomo sapiens (human)Potency19.146512
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1Homo sapiens (human)Potency62.202024
peripheral myelin protein 22Rattus norvegicus (Norway rat)Potency10.299223
peripheral myelin protein 22 isoform 1Homo sapiens (human)Potency35.112415
peroxisome proliferator activated receptor gammaHomo sapiens (human)Potency36.5912513
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency37.210859
phosphopantetheinyl transferaseBacillus subtilisPotency64.660717
plasminogen precursorMus musculus (house mouse)Potency7.262315
Platelet-activating factor receptorHomo sapiens (human)Potency39.810711
polyproteinZika virusPotency16.938414
polyunsaturated fatty acid lipoxygenase ALOX12Homo sapiens (human)Potency28.183811
Polyunsaturated fatty acid lipoxygenase ALOX15BHomo sapiens (human)Potency12.812713
potassium voltage-gated channel subfamily H member 2 isoform dHomo sapiens (human)Potency5.650514
PPM1D proteinHomo sapiens (human)Potency14.013018
pregnane X nuclear receptorHomo sapiens (human)Potency14.7306312
progesterone receptorHomo sapiens (human)Potency29.542726
putative alpha-glucosidaseOryza sativa Japonica Group (Japanese rice)Potency0.053111
RAF proto-oncogene serine/threonine-protein kinase isoform bHomo sapiens (human)Potency18.044812
Rap guanine nucleotide exchange factor 3Homo sapiens (human)Potency58.896625
RAR-related orphan receptor gammaMus musculus (house mouse)Potency13.9821220
ras-related protein Rab-9AHomo sapiens (human)Potency18.356411
regulator of G-protein signaling 4Homo sapiens (human)Potency9.819412
retinoic acid nuclear receptor alpha variant 1Homo sapiens (human)Potency24.4082326
retinoid X nuclear receptor alphaHomo sapiens (human)Potency19.5412411
serine/threonine-protein kinase mTOR isoform 1Homo sapiens (human)Potency2.823038
serine/threonine-protein kinase PLK1Homo sapiens (human)Potency21.192311
SMAD family member 2Homo sapiens (human)Potency29.219412
SMAD family member 3Homo sapiens (human)Potency29.219412
Smad3Homo sapiens (human)Potency14.448716
snurportin-1Homo sapiens (human)Potency30.104327
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency21.475923
survival motor neuron protein isoform dHomo sapiens (human)Potency18.8932110
TAR DNA-binding protein 43Homo sapiens (human)Potency21.306513
TDP1 proteinHomo sapiens (human)Potency8.2907244
thioredoxin reductaseRattus norvegicus (Norway rat)Potency1.081226
ThrombopoietinHomo sapiens (human)Potency12.589322
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency11.5427322
thyroid hormone receptor beta isoform aHomo sapiens (human)Potency348.553247
thyroid stimulating hormone receptorHomo sapiens (human)Potency19.2432718
thyrotropin-releasing hormone receptorHomo sapiens (human)Potency33.210423
transcriptional regulator ERG isoform 3Homo sapiens (human)Potency15.848911
ubiquitin carboxyl-terminal hydrolase 2 isoform aHomo sapiens (human)Potency25.527933
urokinase plasminogen activator surface receptor precursorMus musculus (house mouse)Potency7.262315
urokinase-type plasminogen activator precursorMus musculus (house mouse)Potency7.262315
USP1 protein, partialHomo sapiens (human)Potency37.139527
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency20.464125
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency27.370738
vitamin D3 receptor isoform VDRAHomo sapiens (human)Potency43.793815
Voltage-dependent calcium channel gamma-2 subunitMus musculus (house mouse)Potency17.319019
VprHuman immunodeficiency virus 1Potency39.810711
WRNHomo sapiens (human)Potency50.118711

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1Bos taurus (cattle)IC5029.000011
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1Homo sapiens (human)IC5029.000011
10 kDa chaperonin Escherichia coliIC5025.000022
10 kDa heat shock protein, mitochondrialHomo sapiens (human)IC5023.000011
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)IC506.600011
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)Ki3.500011
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)Ki2.250022
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)Ki3.500011
5-hydroxytryptamine receptor 1DSus scrofa (pig)Ki4.094011
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)Ki3.500011
5-hydroxytryptamine receptor 2AHomo sapiens (human)IC500.129011
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)IC500.002011
5-hydroxytryptamine receptor 2AHomo sapiens (human)Ki0.022655
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)Ki0.004033
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)IC500.002011
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)Ki0.004033
5-hydroxytryptamine receptor 2CHomo sapiens (human)IC501.027011
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)IC500.002011
5-hydroxytryptamine receptor 2CHomo sapiens (human)Ki1.097733
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)Ki0.004033
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)IC501.027011
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)Ki0.538011
5'-nucleotidaseHomo sapiens (human)IC5022.660022
5'-nucleotidaseMus musculus (house mouse)IC5050.320011
60 kDa chaperoninEscherichia coli K-12IC50250.000011
60 kDa chaperonin Escherichia coliIC5025.000022
60 kDa heat shock protein, mitochondrialHomo sapiens (human)IC5023.000011
72 kDa type IV collagenaseHomo sapiens (human)IC5030.310011
AcetylcholinesteraseHomo sapiens (human)IC5051.908733
Acyl-CoA desaturase 1Mus musculus (house mouse)IC500.001011
Adenosine receptor A1Homo sapiens (human)Ki7.410022
Adenosine receptor A1Mus musculus (house mouse)Ki4.430011
Adenosine receptor A2aHomo sapiens (human)Ki7.410011
Adenosine receptor A3Homo sapiens (human)Ki7.410011
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1Homo sapiens (human)IC5048.600011
Aldo-keto reductase family 1 member A1Homo sapiens (human)IC5050.000011
Aldo-keto reductase family 1 member B1Homo sapiens (human)IC502.065022
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)IC502.347012
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)Ki2.328012
Aldo-keto reductase family 1 member B10Homo sapiens (human)IC500.183333
Aldo-keto reductase family 1 member B10Homo sapiens (human)Ki0.046011
Aldo-keto reductase family 1 member C1Homo sapiens (human)IC5021.120022
Aldo-keto reductase family 1 member C2 Homo sapiens (human)IC5015.880022
Aldo-keto reductase family 1 member C3Homo sapiens (human)IC502.705022
Aldo-keto reductase family 1 member C4Homo sapiens (human)IC505.275022
Alpha-2A adrenergic receptorHomo sapiens (human)IC501.570012
Alpha-2A adrenergic receptorHomo sapiens (human)Ki0.588512
Alpha-2B adrenergic receptorHomo sapiens (human)IC500.643011
Alpha-2B adrenergic receptorHomo sapiens (human)Ki0.294011
Alpha-2C adrenergic receptorHomo sapiens (human)IC501.071512
Alpha-2C adrenergic receptorHomo sapiens (human)Ki0.155512
Alpha-amylase 1A Homo sapiens (human)IC5010.200022
Alpha-galactosidaseCoffea arabica (coffee)IC5065.000022
Amyloid-beta precursor proteinHomo sapiens (human)IC504.800011
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)IC500.108511
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)Ki0.088911
Angiotensin-converting enzyme 2 Homo sapiens (human)IC508.300011
AP2-associated protein kinase 1Homo sapiens (human)IC500.017011
Apoptotic peptidase activating factor 1Homo sapiens (human)IC5061.750022
ATP-binding cassette sub-family C member 3Homo sapiens (human)IC50117.012528
ATP-dependent molecular chaperone HSP82Saccharomyces cerevisiae S288CIC503.966723
ATP-dependent translocase ABCB1Homo sapiens (human)IC5057.788999
Aurora kinase BHomo sapiens (human)IC502.620011
Beta-galactosidaseBos taurus (cattle)IC5065.000022
Beta-galactosidaseMus musculus (house mouse)IC50200.000011
Beta-secretase 1Homo sapiens (human)IC501.540011
Bile salt export pumpHomo sapiens (human)IC5098.0327311
Breakpoint cluster region proteinHomo sapiens (human)IC503.000022
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)IC506.000011
Canalicular multispecific organic anion transporter 1Homo sapiens (human)IC50117.350028
Cannabinoid receptor 2Mus musculus (house mouse)IC50100.000011
Carbonic anhydrase 1Homo sapiens (human)Ki10.000011
Carbonic anhydrase 2Homo sapiens (human)Ki10.000011
Carbonic anhydrase 5A, mitochondrialHomo sapiens (human)Ki0.130911
caspase-3 isoform a preproproteinHomo sapiens (human)IC5046.700011
caspase-9 isoform alpha precursorHomo sapiens (human)IC5046.700011
Cathepsin GHomo sapiens (human)IC50100.000011
Ceramide glucosyltransferaseMus musculus (house mouse)IC504.000011
Chain A, ALKALINE PHOSPHATASEEscherichia coliKi5,500.000012
Chain A, Inosine-5'-monophosphate DehydrogenaseTritrichomonas suisKi0.065014
Chain A, Mitogen-activated protein kinase 8Homo sapiens (human)IC504.600011
Chain A, NeuraminidaseInfluenza A virusIC500.004011
Chain A, NeuraminidaseInfluenza B virus (STRAIN B/BEIJING/1/87)IC500.004012
Chain A, NeuraminidaseInfluenza A virusKi0.033015
Chain A, Reverse transcriptase/ribonuclease HHIV-1 M:B_HXB2RIC500.002112
Chain B, p51 RTHIV-1 M:B_HXB2RIC500.002112
CholinesteraseHomo sapiens (human)IC50200.000011
Chymotrypsinogen ABos taurus (cattle)IC50100.000011
CruzipainTrypanosoma cruziIC50102.000022
Cyclin-dependent kinase 1Homo sapiens (human)IC500.053011
Cyclin-dependent kinase 2Homo sapiens (human)IC500.006411
Cyclin-dependent kinase 4Homo sapiens (human)IC5010.000011
Cyclin-dependent kinase 6Homo sapiens (human)IC5010.000011
Cyclin-dependent kinase 7Homo sapiens (human)IC500.003433
Cyclin-dependent kinase 9Homo sapiens (human)IC501.711011
Cyclin-G-associated kinaseHomo sapiens (human)IC500.136011
Cystathionine beta-synthaseHomo sapiens (human)IC5017.100011
Cystathionine gamma-lyaseHomo sapiens (human)IC50400.000011
cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)IC5030.250011
Cytidine deaminaseHomo sapiens (human)Ki190.000011
Cytochrome P450 1A2Homo sapiens (human)IC500.019522
Cytochrome P450 2A6Homo sapiens (human)IC5030.000011
Cytochrome P450 2C19Homo sapiens (human)IC500.074011
Cytochrome P450 2C9 Homo sapiens (human)IC5010.030333
Cytochrome P450 2D6Homo sapiens (human)IC500.023022
Cytochrome P450 3A4Homo sapiens (human)IC500.016522
Cytochrome P450 3A4Homo sapiens (human)Ki190.000011
Cytochrome P450 3A43 Homo sapiens (human)IC500.014011
Cytochrome P450 3A5Homo sapiens (human)IC500.014011
Cytochrome P450 3A7Homo sapiens (human)IC500.014011
Cytosolic phospholipase A2Homo sapiens (human)IC50100.000011
D(2) dopamine receptorRattus norvegicus (Norway rat)IC500.007411
D(3) dopamine receptorHomo sapiens (human)Ki1.241011
Delta-type opioid receptorHomo sapiens (human)Ki0.036222
Delta-type opioid receptorSus scrofa (pig)Ki0.036511
Deoxynucleoside kinaseDrosophila melanogaster (fruit fly)IC505,319.000022
Dihydrofolate reductaseHomo sapiens (human)IC500.001811
Dihydroorotate dehydrogenase Leishmania majorIC501,037.000012
Dihydroorotate dehydrogenase Schistosoma mansoniIC5020.000022
Dihydroorotate dehydrogenase (quinone), mitochondrialHomo sapiens (human)IC500.01152626
Dihydroorotate dehydrogenase (quinone), mitochondrialRattus norvegicus (Norway rat)IC500.204245
Dihydroorotate dehydrogenase (quinone), mitochondrialHomo sapiens (human)Ki0.012022
DNA polymerase betaRattus norvegicus (Norway rat)IC50122.300011
DNA primaseMycobacterium tuberculosis CDC1551IC5038.050012
DNA topoisomerase 2-alphaHomo sapiens (human)IC5038.600011
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)IC500.020011
Ectonucleoside triphosphate diphosphohydrolase 1Mus musculus (house mouse)IC5049.760011
EndoplasminCanis lupus familiaris (dog)IC500.010011
Endothelial PAS domain-containing protein 1Homo sapiens (human)IC500.067233
Enoyl-[acyl-carrier-protein] reductase [NADH] Francisella tularensis subsp. tularensis SCHU S4IC5059.000011
Epidermal growth factor receptorHomo sapiens (human)IC500.20421010
Epidermal growth factor receptorMus musculus (house mouse)IC500.100011
Estrogen receptorHomo sapiens (human)IC507.912011
Estrogen receptorHomo sapiens (human)Ki2.260011
exodeoxyribonuclease V subunit RecBEscherichia coli str. K-12 substr. MG1655IC5062.711012
exodeoxyribonuclease V subunit RecCEscherichia coli str. K-12 substr. MG1655IC5062.711012
exodeoxyribonuclease V subunit RecDEscherichia coli str. K-12 substr. MG1655IC5062.711012
Fe(3+)-Zn(2+) purple acid phosphatasePhaseolus vulgarisKi590.000011
Fructose-1,6-bisphosphatase 1Homo sapiens (human)IC501.300011
Fructose-1,6-bisphosphatase 1Sus scrofa (pig)IC5010.000011
Fructose-1,6-bisphosphatase 1 Rattus norvegicus (Norway rat)IC5010.000011
FurinHomo sapiens (human)IC500.018011
FurinHomo sapiens (human)Ki3.439416
GABA theta subunitRattus norvegicus (Norway rat)IC500.014911
Gag-Pol polyproteinHuman immunodeficiency virus type 1 (NEW YORK-5 ISOLATE)IC500.370011
GalactocerebrosidaseHomo sapiens (human)IC5030.000011
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)IC50281,838.000011
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-4Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit beta-1Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)IC50281,838.000011
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit deltaHomo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit epsilonHomo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit gamma-1Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)IC50281,838.000011
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit gamma-3Homo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)IC500.014911
Gamma-aminobutyric acid receptor subunit piHomo sapiens (human)Ki0.006022
Gamma-aminobutyric acid receptor subunit thetaHomo sapiens (human)Ki0.006022
Genome polyprotein IC50215.000012
Glucose transporterLeishmania mexicanaIC500.081011
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)IC50144.470033
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)IC50144.470033
Glutathione S-transferase PHomo sapiens (human)IC500.500011
Glycogen phosphorylase, muscle formOryctolagus cuniculus (rabbit)IC5021.896545
Group 10 secretory phospholipase A2Homo sapiens (human)IC50100.000011
GTPase KRasHomo sapiens (human)IC500.900066
GTPase KRasHomo sapiens (human)Ki47.500022
Heat shock protein 75 kDa, mitochondrialHomo sapiens (human)IC500.661011
Heat shock protein HSP 90Oryctolagus cuniculus (rabbit)IC501.141022
Heat shock protein HSP 90-alphaHomo sapiens (human)IC500.16502121
Heat shock protein HSP 90-betaHomo sapiens (human)IC500.098077
Heme oxygenase 2Homo sapiens (human)IC507.640011
Hepatocyte growth factor activatorHomo sapiens (human)IC5032.000011
Hexose transporter 1 Plasmodium falciparum (malaria parasite P. falciparum)IC500.090011
Histamine H1 receptorCavia porcellus (domestic guinea pig)IC500.007711
Histamine H3 receptorRattus norvegicus (Norway rat)IC501.300012
hypothetical protein SA1422Staphylococcus aureus subsp. aureus N315IC5019.390022
Hypoxia-inducible factor 1-alphaHomo sapiens (human)IC500.067233
Integrase Human immunodeficiency virus 1IC5013.12171113
Kallikrein-1Homo sapiens (human)IC5034.100011
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)IC500.097011
KiSS-1 receptorHomo sapiens (human)Ki3.600011
Lysine-specific demethylase 4BHomo sapiens (human)IC500.700011
Lysine-specific demethylase 4CHomo sapiens (human)IC500.700011
Lysine-specific demethylase 5AHomo sapiens (human)IC500.130011
Lysine-specific demethylase 6BHomo sapiens (human)IC500.400011
Lysosomal acid glucosylceramidaseHomo sapiens (human)IC501.26391515
Lysosomal acid glucosylceramidaseHomo sapiens (human)Ki0.442977
Lysosomal alpha-glucosidaseHomo sapiens (human)IC50400.000011
Lysosomal alpha-glucosidaseMus musculus (house mouse)IC508.000011
M1-family alanyl aminopeptidasePlasmodium falciparum 3D7IC50108.390011
Maltase-glucoamylase, intestinalHomo sapiens (human)IC50400.000011
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)IC500.530011
Matrix metalloproteinase-9Homo sapiens (human)IC502.580011
Mcl-1Homo sapiens (human)IC501.634111
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)IC5037.300044
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Ki16.488545
Mitogen-activated protein kinase 1Homo sapiens (human)IC500.686011
Mitogen-activated protein kinase 14Homo sapiens (human)IC500.560011
Mitogen-activated protein kinase 8Mus musculus (house mouse)IC504.600011
Multidrug and toxin extrusion protein 1Homo sapiens (human)IC502.900011
Multidrug and toxin extrusion protein 2Homo sapiens (human)IC5012.700011
Multidrug resistance-associated protein 1 Homo sapiens (human)IC508.500011
Multidrug resistance-associated protein 4Homo sapiens (human)IC50133.000017
Muscarinic acetylcholine receptor M1Homo sapiens (human)IC500.412011
Muscarinic acetylcholine receptor M1Homo sapiens (human)Ki0.099011
Muscarinic acetylcholine receptor M2Homo sapiens (human)IC500.574011
Muscarinic acetylcholine receptor M2Homo sapiens (human)Ki0.204011
Muscarinic acetylcholine receptor M3Homo sapiens (human)IC500.383011
Muscarinic acetylcholine receptor M3Homo sapiens (human)Ki0.081011
Muscarinic acetylcholine receptor M4Homo sapiens (human)IC500.257011
Muscarinic acetylcholine receptor M4Homo sapiens (human)Ki0.036011
Muscarinic acetylcholine receptor M5Homo sapiens (human)IC500.134011
Muscarinic acetylcholine receptor M5Homo sapiens (human)Ki0.096011
NAD-dependent protein deacetylase HST2Saccharomyces cerevisiae S288CIC50700.000011
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)IC50600.000022
NeuraminidaseInfluenza A virus (A/Aichi/2/1968(H3N2))IC500.002711
NeuraminidaseInfluenza A virus (A/budgerigar/Hokkaido/1/1977(H4N6))IC500.022811
NeuraminidaseInfluenza A virus (A/duck/Ukraine/1/1963(H3N8))IC500.007411
NeuraminidaseInfluenza A virus (A/Memphis/1/1971(H3N2))IC500.014744
NeuraminidaseInfluenza A virus (A/Puerto Rico/8/1934(H1N1))IC500.00431616
NeuraminidaseInfluenza A virus (A/Singapore/1/1957(H2N2))IC500.007024
NeuraminidaseInfluenza A virus (A/udorn/1972(H3N2))IC500.015411
NeuraminidaseInfluenza A virus (A/Wilson-Smith/1933(H1N1))IC500.001755
NeuraminidaseInfluenza B virus (B/Lee/1940)IC500.080999
NeuraminidaseInfluenza B virus (STRAIN B/VICTORIA/3/85)IC500.004512
NeuraminidaseInfluenza B virus (B/Lee/1940)Ki0.000111
Neuraminidase Influenza A virus (A/Brisbane/59/2007(H1N1))IC500.027622
Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1))IC500.000822
Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1))IC500.002733
Neuraminidase Influenza A virus (A/RI/5+/1957(H2N2))IC501.400011
Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1))IC500.002433
Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1))IC500.005444
Neuraminidase Influenza A virus (A/udorn/1972(H3N2))IC500.022911
Neuraminidase Influenza A virus (A/Wilson-Smith/1933(H1N1))IC5041.7026122122
Neuraminidase Influenza B virus (B/Perth/211/2001)IC500.088122
Neuraminidase Influenza A virus (A/chicken/Yogjakarta/BBVet-IX/2004(H5N1))Ki0.000411
Neuraminidase Influenza A virus (A/duck/Laos/25/2006(H5N1))Ki0.000511
Neuraminidase Influenza A virus (A/Thailand/1(KAN-1)/2004(H5N1))Ki0.000511
Neuraminidase Influenza A virus (A/Turkey/651242/2006(H5N1))Ki0.001011
Neuraminidase Influenza A virus (A/Wilson-Smith/1933(H1N1))Ki0.000244
Neutrophil elastaseHomo sapiens (human)IC5039.756733
Non-lysosomal glucosylceramidaseHomo sapiens (human)IC500.005022
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)IC5013.47941315
Nuclear factor NF-kappa-B p100 subunit Homo sapiens (human)IC5030.000011
Nuclear factor NF-kappa-B p105 subunitHomo sapiens (human)IC5030.000011
nuclear receptor coactivator 1 isoform 1 [Homo sapiens]Homo sapiens (human)IC5025.587011
nuclear receptor coactivator 3 isoform aHomo sapiens (human)IC507.533011
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)IC500.108511
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)Ki0.088911
Oligo-1,6-glucosidase IMA1Saccharomyces cerevisiae S288CIC50100.000011
P2Y purinoceptor 12Homo sapiens (human)Ki10.000011
Pancreatic alpha-amylaseSus scrofa (pig)IC50200.000011
Phospholipase A2Rattus norvegicus (Norway rat)IC50100.000011
Phospholipase A2, membrane associatedHomo sapiens (human)IC5023.800011
Plasminogen Rattus norvegicus (Norway rat)IC502.620011
Platelet glycoprotein VIHomo sapiens (human)IC5037.500022
Platelet-derived growth factor receptor alphaHomo sapiens (human)IC5010.000011
Platelet-derived growth factor receptor betaHomo sapiens (human)IC5010.000011
Poly [ADP-ribose] polymerase 1Homo sapiens (human)IC500.102333
Poly [ADP-ribose] polymerase 2Homo sapiens (human)IC5010.300022
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiens (human)IC501.990033
Polyunsaturated fatty acid lipoxygenase ALOX15Homo sapiens (human)IC500.130011
Potassium voltage-gated channel subfamily D member 3Homo sapiens (human)IC503,162.280011
Potassium voltage-gated channel subfamily E member 1Homo sapiens (human)IC501,258.930011
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)IC50145.455944
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)Ki0.088911
Potassium voltage-gated channel subfamily KQT member 1Homo sapiens (human)IC501,258.930011
Probable alpha-glucosidase Os06g0675700Oryza sativa Japonica Group (Japanese rice)IC50100.000011
Probable maltase-glucoamylase 2Homo sapiens (human)IC50400.000011
Procathepsin LHomo sapiens (human)IC504.159022
Procathepsin LHomo sapiens (human)Ki3.439416
Prostaglandin G/H synthase 1Homo sapiens (human)IC5029.416522
Prostaglandin G/H synthase 1Ovis aries (sheep)IC5046.210011
Prostaglandin G/H synthase 2Homo sapiens (human)IC5082.000011
Prostaglandin G/H synthase 2Ovis aries (sheep)IC5036.120011
Protein kinase C alpha typeHomo sapiens (human)IC50100.000022
Protein kinase C beta typeHomo sapiens (human)IC50150.000011
Protein kinase C epsilon typeHomo sapiens (human)IC50150.000011
Protein kinase C theta typeHomo sapiens (human)IC50100.000011
Protein-lysine 6-oxidaseHomo sapiens (human)IC501.500011
Protein-lysine 6-oxidaseHomo sapiens (human)Ki0.300011
ProthrombinHomo sapiens (human)IC5010.799333
ProthrombinHomo sapiens (human)Ki3.439416
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC502.700011
Putative heat shock protein HSP 90-alpha A4Homo sapiens (human)IC500.140011
Quinone oxidoreductaseHomo sapiens (human)IC508.440011
Ras-related C3 botulinum toxin substrate 1Homo sapiens (human)IC5095.000011
Ras-related C3 botulinum toxin substrate 1Mus musculus (house mouse)IC506.300022
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)IC501.706512
Replicase polyprotein 1aSevere acute respiratory syndrome-related coronavirusIC508.300011
Replicase polyprotein 1abBetacoronavirus England 1IC508.650022
Replicase polyprotein 1abHuman coronavirus 229EIC508.300011
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2IC5036.9320913
Replicase polyprotein 1abSevere acute respiratory syndrome-related coronavirusIC507.780045
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2Ki8.425024
Replicase polyprotein 1abSevere acute respiratory syndrome-related coronavirusKi9.625024
Reticulon-4Homo sapiens (human)IC5014.610011
Reverse transcriptase Human immunodeficiency virus 1IC500.018677
Reverse transcriptase/RNaseH Human immunodeficiency virus 1IC502.4806100103
RNA-directed RNA polymerase IC507.200022
Serine hydrolase RBBP9Homo sapiens (human)IC507.800011
Serine protease hepsinHomo sapiens (human)IC500.023522
Serine protease hepsinHomo sapiens (human)Ki3.439416
Serine/threonine-protein kinase pim-1Homo sapiens (human)IC500.340066
Sialidase AStreptococcus pneumoniaeKi720.000011
Sialidase-1Homo sapiens (human)IC50952.166766
Sialidase-1Mus musculus (house mouse)IC50500.000011
Sialidase-2Homo sapiens (human)IC509.792299
Sialidase-2Homo sapiens (human)Ki8.525044
Sialidase-3Homo sapiens (human)IC505.661766
Sialidase-3Homo sapiens (human)Ki0.620033
Sialidase-4Homo sapiens (human)IC50350.000088
Sialidase-4Homo sapiens (human)Ki26.000033
Sigma non-opioid intracellular receptor 1Homo sapiens (human)IC500.182011
Sodium channel protein type 5 subunit alphaHomo sapiens (human)IC502,241.128522
Sodium-dependent dopamine transporter Homo sapiens (human)IC501.365011
Sodium-dependent dopamine transporter Homo sapiens (human)Ki1.085011
Sodium-dependent noradrenaline transporter Homo sapiens (human)IC502.347012
Sodium-dependent noradrenaline transporter Homo sapiens (human)Ki2.328012
Sodium-dependent serotonin transporterHomo sapiens (human)IC502.438011
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)IC500.560011
Sodium-dependent serotonin transporterHomo sapiens (human)Ki1.295011
Sodium/bile acid cotransporterHomo sapiens (human)IC50109.000011
Solute carrier family 2, facilitated glucose transporter member 1Homo sapiens (human)IC500.108011
Solute carrier family 22 member 2Homo sapiens (human)IC5016.500011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)Ki3.825044
Spike glycoproteinBetacoronavirus England 1IC508.300011
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusIC508.300011
Stromelysin-1Homo sapiens (human)IC50100.000011
Substance-K receptorHomo sapiens (human)IC501.925011
Substance-K receptorHomo sapiens (human)Ki0.642011
Sucrase-isomaltase Mus musculus (house mouse)IC500.400011
Sucrase-isomaltase, intestinalHomo sapiens (human)IC50400.000011
Synapsin-1Bos taurus (cattle)IC500.150011
Synaptic vesicle membrane protein VAT-1 homologHomo sapiens (human)IC504.510022
Thioredoxin reductase 1, cytoplasmicHomo sapiens (human)IC5040.000011
Thioredoxin reductase 1, cytoplasmicRattus norvegicus (Norway rat)IC50194.000011
Thioredoxin reductase 2, mitochondrialHomo sapiens (human)IC5040.000011
Thioredoxin reductase 2, mitochondrialRattus norvegicus (Norway rat)IC50181.000011
Thioredoxin reductase 3Homo sapiens (human)IC5040.000011
Thiosulfate sulfurtransferaseHomo sapiens (human)IC50100.000011
Thymidine kinaseHuman alphaherpesvirus 1 (Herpes simplex virus type 1)IC501,000.000011
Thymidine kinaseHuman alphaherpesvirus 1 strain SC16IC501,000.000011
Thymidine kinaseHuman herpesvirus 3 strain DumasIC501,000.000022
Thymidine kinase 2 Rattus norvegicus (Norway rat)Ki3,250.000011
Thymidine kinase 2, mitochondrialHomo sapiens (human)IC501,000.000022
Thymidine kinase, cytosolicHomo sapiens (human)IC501,000.000022
Thymidine kinase, cytosolicHomo sapiens (human)Ki597.500022
Thymidine kinase, cytosolic Rattus norvegicus (Norway rat)Ki1,700.000011
transactivating tegument protein VP16 [Human herpesvirus 1]Human alphaherpesvirus 1 (Herpes simplex virus type 1)IC5016.247011
Transcription factor p65Homo sapiens (human)IC5019.400022
Transmembrane protease serine 2Homo sapiens (human)IC504.159022
Transmembrane protease serine 2Homo sapiens (human)Ki3.439416
Transmembrane protease serine 6Homo sapiens (human)IC500.018011
Transmembrane protease serine 6Homo sapiens (human)Ki3.439416
TransthyretinHomo sapiens (human)IC50100.000011
Trypsin-1Homo sapiens (human)IC500.027022
Trypsin-2Homo sapiens (human)IC500.003511
Trypsin-3Homo sapiens (human)IC500.003511
Tyrosine-protein kinase ABL1Homo sapiens (human)IC502.041733
Tyrosine-protein kinase ABL2Homo sapiens (human)IC500.125011
Tyrosine-protein kinase FynHomo sapiens (human)IC502.491012
Tyrosine-protein kinase JAK1Homo sapiens (human)IC500.07392021
Tyrosine-protein kinase JAK2Homo sapiens (human)IC500.12332123
Tyrosine-protein kinase JAK3Homo sapiens (human)IC501.12561111
Tyrosine-protein kinase LckHomo sapiens (human)IC502.887011
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)IC507.400011
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)Ki7.800011
ubiquitin-conjugating enzyme E2 NHomo sapiens (human)IC5020.000011
Valosin-containing proteinHomo sapiens (human)IC5036.328023
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)IC50622.500011
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)IC50622.500011
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)IC50622.500011
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)IC50622.500011
Xanthine dehydrogenase/oxidaseBos taurus (cattle)IC5035.300011

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase catalytic subunit alpha-2Homo sapiens (human)EC500.016811
5'-AMP-activated protein kinase subunit beta-1Homo sapiens (human)EC500.016811
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)EC500.016811
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.000011
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.000011
Actin-related protein 2Homo sapiens (human)Kd30.000011
Actin-related protein 3Homo sapiens (human)Kd30.000011
Activated CDC42 kinase 1Homo sapiens (human)Kd30.000012
Activin receptor type-1Homo sapiens (human)Kd30.000011
Activin receptor type-1BHomo sapiens (human)Kd30.000011
Activin receptor type-2BHomo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000012
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000011
Adenosine kinaseHomo sapiens (human)Kd30.000011
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000011
ADP/ATP translocase 2Homo sapiens (human)Kd30.000011
ADP/ATP translocase 3Homo sapiens (human)Kd30.000011
AlbuminHomo sapiens (human)Kd44.000011
Alpha-tocopherol transfer proteinHomo sapiens (human)Kd2.420011
Amyloid-beta precursor proteinHomo sapiens (human)EC508.410011
Angiotensin-converting enzyme 2 Homo sapiens (human)EC5025.913015
AP2-associated protein kinase 1Homo sapiens (human)Kd0.014566
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000011
ATP-dependent molecular chaperone HSP82Saccharomyces cerevisiae S288CKd1.200011
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DHX30Homo sapiens (human)Kd30.000011
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd30.000011
Aurora kinase AHomo sapiens (human)Kd30.000011
Aurora kinase BHomo sapiens (human)Kd30.000012
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000011
BMP-2-inducible protein kinaseHomo sapiens (human)Kd0.085333
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd30.000011
Breakpoint cluster region proteinHomo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd0.312011
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd0.243011
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd3.597011
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd30.000012
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000011
Casein kinase I isoform alphaHomo sapiens (human)Kd30.000011
Casein kinase I isoform deltaHomo sapiens (human)Kd30.000011
Casein kinase I isoform epsilonHomo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-1Homo sapiens (human)Kd1.753011
Casein kinase I isoform gamma-2Homo sapiens (human)Kd0.265011
Casein kinase I isoform gamma-3Homo sapiens (human)Kd30.000011
Casein kinase II subunit alpha'Homo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd30.000012
Chain A, Calmodulin-sensitive adenylate cyclaseBacillus anthracisKd130.000011
Chain A, NDP kinaseDictyostelium discoideumKd24.000011
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000011
Citron Rho-interacting kinaseHomo sapiens (human)Kd4.361011
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 13Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 16Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 17Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 2Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 3Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 4Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 6Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 7Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 9Homo sapiens (human)Kd30.000011
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd30.000011
Cyclin-G-associated kinaseHomo sapiens (human)Kd1.068455
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000011
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000011
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000011
delta-type opioid receptorHomo sapiens (human)EC5092.461011
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000011
Deoxycytidine kinaseHomo sapiens (human)Kd30.000011
Dihydroorotate dehydrogenase (quinone), mitochondrialHomo sapiens (human)EC500.055011
Discoidin domain-containing receptor 2Homo sapiens (human)Kd30.000011
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000011
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000011
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000011
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK1Homo sapiens (human)Kd0.778011
Dual specificity protein kinase CLK2Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK3Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK4Homo sapiens (human)Kd30.000011
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd30.000011
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd30.000011
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000011
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd30.000011
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000011
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000011
Ephrin type-A receptor 1Homo sapiens (human)Kd30.000012
Ephrin type-A receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 5Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 7Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 3Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 6Homo sapiens (human)Kd30.000011
Epidermal growth factor receptorHomo sapiens (human)Kd30.000011
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd30.000011
Estrogen receptorRattus norvegicus (Norway rat)EC50150.000012
Estrogen receptor betaRattus norvegicus (Norway rat)EC50150.000012
Eukaryotic peptide chain release factor GTP-binding subunit ERF3BHomo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd0.335011
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000011
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000011
Ferrochelatase, mitochondrialHomo sapiens (human)Kd30.000011
Fibroblast growth factor receptor 1Homo sapiens (human)Kd30.000011
Focal adhesion kinase 1Homo sapiens (human)Kd30.000011
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000011
G-protein coupled bile acid receptor 1Homo sapiens (human)EC5010.000011
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)EC503.600011
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)EC503.600011
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)EC503.600011
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.000011
Genome polyproteinHuman enterovirus 71 (strain BRCR)EC50100.000011
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000011
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.000011
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd30.000012
glycogen synthase kinase-3 beta isoform 1Homo sapiens (human)EC50300.000011
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000011
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000011
Heat shock protein 90, putativePlasmodium falciparum 3D7Kd0.243522
Heat shock protein HSP 90-alphaHomo sapiens (human)EC500.035011
Heat shock protein HSP 90-alphaHomo sapiens (human)Kd1.020855
Heat shock protein HSP 90-betaHomo sapiens (human)EC500.035011
Heat shock protein HSP 90-betaHomo sapiens (human)Kd0.730066
Heme oxygenase 2Homo sapiens (human)Kd30.000011
Hepatocyte growth factor receptorHomo sapiens (human)Kd30.000012
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd30.000011
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000011
Insulin receptorHomo sapiens (human)Kd30.000011
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd30.000011
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd30.000012
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd30.000011
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000011
LIM domain kinase 1Homo sapiens (human)Kd30.000011
LIM domain kinase 2Homo sapiens (human)Kd30.000012
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000011
Lymphocyte antigen 96Homo sapiens (human)Kd460.000011
Macrophage-stimulating protein receptorHomo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd30.000011
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd0.104011
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd30.000011
Matrix metalloproteinase-9Homo sapiens (human)Kd2.180011
melanocortin receptor 4Homo sapiens (human)EC5089.188012
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000011
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd30.000011
MidasinHomo sapiens (human)Kd30.000011
Misshapen-like kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 10Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 11Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 14Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 15Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 7Homo sapiens (human)Kd30.000012
Mitogen-activated protein kinase 8Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 9Homo sapiens (human)Kd30.000012
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd1.891011
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd30.000011
mu-type opioid receptor isoform MOR-1Homo sapiens (human)EC5092.461011
Multifunctional protein ADE2Homo sapiens (human)Kd30.000011
Myosin light chain kinase 3Homo sapiens (human)Kd30.000011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd30.000011
Myosin-10Homo sapiens (human)Kd30.000012
Myosin-14Homo sapiens (human)Kd30.000011
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000011
NeuraminidaseInfluenza A virus (A/udorn/1972(H3N2))Kd0.004711
Neuronal acetylcholine receptor subunit alpha-3Homo sapiens (human)EC5010.000022
Neuronal acetylcholine receptor subunit alpha-4Homo sapiens (human)EC5010.000022
Neuronal acetylcholine receptor subunit alpha-7Homo sapiens (human)EC502.500011
Neuronal acetylcholine receptor subunit alpha-7Rattus norvegicus (Norway rat)EC5010.000011
Neuronal acetylcholine receptor subunit beta-2Homo sapiens (human)EC5010.000022
Neuronal acetylcholine receptor subunit beta-4Homo sapiens (human)EC5010.000022
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd0.622011
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd30.000011
NS5 Zika virusEC506.953933
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd30.000011
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000011
Obg-like ATPase 1Homo sapiens (human)Kd30.000011
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000011
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000011
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd30.000011
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd30.000011
Placenta growth factorHomo sapiens (human)Kd0.008211
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd30.000011
Polymerase acidic proteinInfluenza A virus (A/Puerto Rico/8/1934(H1N1))EC5021.266733
Polymerase basic protein 2Influenza A virus (A/Puerto Rico/8/1934(H1N1))EC5020.000022
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000011
Procathepsin LHomo sapiens (human)EC5025.913015
Protein kinase C alpha typeHomo sapiens (human)Kd2.071011
Protein kinase C beta typeHomo sapiens (human)Kd26.324011
Protein kinase C delta typeHomo sapiens (human)Kd1.075011
Protein kinase C iota typeHomo sapiens (human)Kd30.000011
Protein kinase C theta typeHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 6Homo sapiens (human)Kd30.000011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd0.973011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd30.000011
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000011
Pyridoxal kinaseHomo sapiens (human)Kd30.000011
Rab-like protein 3Homo sapiens (human)Kd30.000011
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Ras-related protein Rab-10Homo sapiens (human)Kd30.000012
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000011
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000011
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd30.000011
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000011
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd30.000011
Replicase polyprotein 1aSevere acute respiratory syndrome-related coronavirusEC5025.913015
Replicase polyprotein 1abBetacoronavirus England 1EC5025.913015
Replicase polyprotein 1abHuman coronavirus 229EEC5025.913015
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2EC5020.906637
Replicase polyprotein 1abSevere acute respiratory syndrome-related coronavirusEC5025.913015
Reverse transcriptase Human immunodeficiency virus 1EC500.01211010
Reverse transcriptase/RNaseH Human immunodeficiency virus 1EC500.05762222
Rho-associated protein kinase 1Homo sapiens (human)Kd0.482011
Rho-associated protein kinase 2Homo sapiens (human)Kd0.756011
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd30.000011
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd30.000011
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000011
RNA-directed RNA polymerase catalytic subunitInfluenza A virus (A/Puerto Rico/8/1934(H1N1))EC5021.266733
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000011
Septin-9Homo sapiens (human)Kd0.084011
Serine/threonine-protein kinase 10Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 16Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 24Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 26Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 4Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ATRHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase D2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase D3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd0.125011
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase N1Homo sapiens (human)Kd0.104011
Serine/threonine-protein kinase N2Homo sapiens (human)Kd0.269011
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd30.000012
Serine/threonine-protein kinase receptor R3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd30.000012
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd0.810011
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.000011
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000011
Spike glycoproteinBetacoronavirus England 1EC5025.913015
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusEC5025.913015
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd30.000011
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd30.000011
streptokinase A precursorStreptococcus pyogenes M1 GASEC5076.149022
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000011
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000011
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000011
TGF-beta receptor type-1Homo sapiens (human)Kd30.000011
TGF-beta receptor type-2Homo sapiens (human)Kd30.000011
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000011
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd30.000011
Transmembrane protease serine 2Homo sapiens (human)EC5021.760826
TransthyretinHomo sapiens (human)EC508.600011
TransthyretinHomo sapiens (human)Kd12.000011
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase BTKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase CSKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FerHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FRKHomo sapiens (human)Kd30.000012
Tyrosine-protein kinase FynHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase HCKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase LckHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase LynHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase SYKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase TecHomo sapiens (human)Kd30.000012
Tyrosine-protein kinase YesHomo sapiens (human)Kd30.000011
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000011
UMP-CMP kinase Homo sapiens (human)Kd30.000011
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000012
Uncharacterized protein FLJ45252Homo sapiens (human)Kd0.078011
Vascular endothelial growth factor AHomo sapiens (human)Kd0.016511
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000011
Wee1-like protein kinaseHomo sapiens (human)Kd15.000722

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
AdenosylhomocysteinaseHomo sapiens (human)Kinact266.000011
AdenosylhomocysteinaseHomo sapiens (human)KR407.000011
ATP-dependent translocase ABCB1Homo sapiens (human)Km3.500012
Cytidine deaminaseHomo sapiens (human)Km118.000033
Delta-type opioid receptorHomo sapiens (human)Ke6.000011
Deoxycytidine kinaseHomo sapiens (human)Km3.040011
DNA repair protein RAD52 homolog isoform aHomo sapiens (human)AC5031.330011
Endothelial PAS domain-containing protein 1Homo sapiens (human)MIC0.300011
Heat shock protein HSP 90-alphaHomo sapiens (human)Concentration5.000011
Heat shock protein HSP 90-betaHomo sapiens (human)Activity0.165522
Hypoxia-inducible factor 1-alphaHomo sapiens (human)MIC0.300011
Kappa-type opioid receptorHomo sapiens (human)Ke0.490011
Liver carboxylesterase 1Homo sapiens (human)Km707.000011
LMP1 [Human herpesvirus 4]human gammaherpesvirus 4 (Epstein-Barr virus)AbsAC35_uM7.240011
LMP1 [Human herpesvirus 4]human gammaherpesvirus 4 (Epstein-Barr virus)AC500.918022
Mu-type opioid receptorHomo sapiens (human)Ke10.000011
NAD(P)H dehydrogenase [quinone] 1Mus musculus (house mouse)CD1.300011
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)INH0.036011
Pancreatic triacylglycerol lipaseSus scrofa (pig)ED5010.000011
Probable deoxycytidylate deaminaseCaenorhabditis elegansKm160.000011
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Activity50.000011
Reverse transcriptase/RNaseH Human immunodeficiency virus 1IC900.100011
Reverse transcriptase/RNaseH Human immunodeficiency virus 1ID500.045522
Serine/threonine-protein kinase pim-1Homo sapiens (human)-Log IC500.470011
Serine/threonine-protein kinase pim-1Homo sapiens (human)ED505.500011
Solute carrier family 22 member 1Rattus norvegicus (Norway rat)Km48.800011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)Km2.080011
Thymidine kinase, cytosolicHomo sapiens (human)Km133.000011
Thymidylate synthaseMus musculus (house mouse)ED500.030011
Tissue factorHomo sapiens (human)Concentration5.000011
Tyrosine-protein kinase JAK1Homo sapiens (human)INH0.011522
Tyrosine-protein kinase JAK2Homo sapiens (human)INH0.158022
Tyrosine-protein kinase JAK3Homo sapiens (human)INH0.180011
UDP-glucuronosyltransferase 1A4Homo sapiens (human)Km13.000011