Page last updated: 2024-08-07 13:09:42
Thymidine kinase, cytosolic
[no definition available]
Synonyms
EC 2.7.1.21
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 2 (66.67) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (12)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
stavudine | Rattus norvegicus (Norway rat) | Ki | 1,700.0000 | 1 | 1 |
ibacitabine | Rattus norvegicus (Norway rat) | Ki | 7,450.0000 | 2 | 2 |
methylthymidine | Rattus norvegicus (Norway rat) | Ki | 14,125.0000 | 2 | 2 |
2',3'-dideoxythymidine | Rattus norvegicus (Norway rat) | Ki | 400.0000 | 1 | 1 |
5'-amino-2',5'-dideoxythymidine | Rattus norvegicus (Norway rat) | Ki | 2.4000 | 1 | 1 |
3'-amino-2',3'-dideoxythymidine | Rattus norvegicus (Norway rat) | Ki | 380.0000 | 1 | 1 |
5-amino-2'-deoxyuridine | Rattus norvegicus (Norway rat) | Ki | 370.0000 | 1 | 1 |
5-methyldeoxycytidine | Rattus norvegicus (Norway rat) | Ki | 1,700.0000 | 2 | 2 |
TTP | Rattus norvegicus (Norway rat) | Ki | 5.1000 | 2 | 2 |
5-(1-propenyl)-2'-deoxyuridine | Rattus norvegicus (Norway rat) | Ki | 8,005.0000 | 2 | 2 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
thymidine | Rattus norvegicus (Norway rat) | Km | 4.8000 | 2 | 2 |
thymidine | Rattus norvegicus (Norway rat) | Phosphorylation rate | 100.0000 | 1 | 1 |
zidovudine | Rattus norvegicus (Norway rat) | Phosphorylation rate | 4.0000 | 1 | 1 |