Page last updated: 2024-08-07 20:59:06

Apoptotic peptidase activating factor 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (40)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
methylene blueHomo sapiens (human)IC5057.750020
9,10-phenanthrenequinoneHomo sapiens (human)IC5050.274520
pyronineHomo sapiens (human)IC5042.000020
benzethonium chlorideHomo sapiens (human)IC5061.750020
neutral red baseHomo sapiens (human)IC5067.000020
dimidium bromideHomo sapiens (human)IC5062.250020
2,2'-((3,3'-dimethoxy(1,1'-biphenyl)-4,4'-diyl)diimino)bis-benzoic acidHomo sapiens (human)IC5063.350020
2-phenylisatogenHomo sapiens (human)IC5052.900020
papaveraldineHomo sapiens (human)IC5062.200020
tanshinone ii aHomo sapiens (human)IC5052.410020
(R)-RoemerineHomo sapiens (human)IC5055.100020
nsc 95397Homo sapiens (human)IC5056.350020
2,3-diaminophenazineHomo sapiens (human)IC50100.000020
discretamineHomo sapiens (human)IC5058.150020
doxorubicin hydrochlorideHomo sapiens (human)IC5060.600020
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)IC5050.018820
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineHomo sapiens (human)IC5065.750020
calmidazoliumHomo sapiens (human)IC5056.350020
spiro[1,3-dihydroperimidine-2,1'-cycloheptane]Homo sapiens (human)IC5053.290020
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)IC5050.039520
3-[[3-(4-morpholinyl)-1,4-dioxo-2-naphthalenyl]amino]benzoic acidHomo sapiens (human)IC5071.600020
1-[(3,4-dichlorophenyl)methyl]indole-2,3-dioneHomo sapiens (human)IC5034.000010
4-(6-fluoro-3-methyl-4-oxo-1-benzopyran-2-yl)-2-methyl-1-phthalazinoneHomo sapiens (human)IC5055.800020
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideHomo sapiens (human)IC5061.550020
4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-dioneHomo sapiens (human)IC5056.550020
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)IC5060.825020
2-(2-hydroxyethylamino)-3-(4-methoxyanilino)naphthalene-1,4-dioneHomo sapiens (human)IC5064.700020
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneHomo sapiens (human)IC5052.085020
N-[3-(4-methyl-1-piperazinyl)-1,4-dioxo-2-naphthalenyl]benzenesulfonamideHomo sapiens (human)IC5069.550020
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-oneHomo sapiens (human)IC5059.650020
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideHomo sapiens (human)IC5055.000020
reumycinHomo sapiens (human)IC5057.700020
methylbenzethonium chlorideHomo sapiens (human)IC5060.650020
3,3'-diethylthiacarbocyanine iodideHomo sapiens (human)IC5060.400020
3-bromo-N-[2-[(3R,6S)-6-[(4-methoxyphenyl)methyl]-3-(phenylmethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]imidazol-7-yl]ethyl]-4-methylbenzamideHomo sapiens (human)IC50100.000020
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineHomo sapiens (human)IC5058.000020

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
alpha-methylhydrocinnamic acidHomo sapiens (human)EC50100.000010
N-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-2-furancarboxamideHomo sapiens (human)EC5070.450030
4-fluoro-N-(7-methyl-4-oxo-2-thieno[3,2-d][1,3]thiazinyl)benzamideHomo sapiens (human)EC50100.000010
cefiximeHomo sapiens (human)EC5069.693320