Proteins > caspase-3 isoform a preproprotein
Page last updated: 2024-08-07 18:24:17

caspase-3 isoform a preproprotein

[no definition available]

Synonyms

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (86)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ipriflavoneHomo sapiens (human)IC5019.700010
methyldimethylaminoazobenzeneHomo sapiens (human)IC505.570010
methylene blueHomo sapiens (human)IC5017.000010
1-amino-2-methylanthraquinoneHomo sapiens (human)IC5011.800010
9,10-phenanthrenequinoneHomo sapiens (human)IC500.903010
pyronineHomo sapiens (human)IC5016.800010
benzethonium chlorideHomo sapiens (human)IC5046.700010
glaucineHomo sapiens (human)IC500.907010
neutral red baseHomo sapiens (human)IC5014.500010
dimidium bromideHomo sapiens (human)IC507.890010
2,2'-((3,3'-dimethoxy(1,1'-biphenyl)-4,4'-diyl)diimino)bis-benzoic acidHomo sapiens (human)IC5018.200010
2-phenylisatogenHomo sapiens (human)IC506.360010
witisolHomo sapiens (human)IC505.390010
papaveraldineHomo sapiens (human)IC506.490020
tanshinone ii aHomo sapiens (human)IC5011.200010
4',6-dihydroxyflavoneHomo sapiens (human)IC5016.800010
(R)-RoemerineHomo sapiens (human)IC502.730010
nsc 95397Homo sapiens (human)IC509.830010
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl esterHomo sapiens (human)IC5031.100010
discretamineHomo sapiens (human)IC504.300010
doxorubicin hydrochlorideHomo sapiens (human)IC5034.600010
6-bromoindirubin-3'-oximeHomo sapiens (human)IC5064.300010
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)IC500.025610
2-[(4-nitrophenyl)methylthio]-1,3-benzoxazoleHomo sapiens (human)IC5025.600010
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineHomo sapiens (human)IC50100.000010
calmidazoliumHomo sapiens (human)IC507.140010
N-(1,3-benzothiazol-2-yl)-N-methylbenzamideHomo sapiens (human)IC5015.600010
N-(2-fluorophenyl)-4-phenylmethoxybenzamideHomo sapiens (human)IC5010.300010
5-amino-3-(4-methoxyphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterHomo sapiens (human)IC5023.000010
vu0038882Homo sapiens (human)IC5059.700010
spiro[1,3-dihydroperimidine-2,1'-cycloheptane]Homo sapiens (human)IC5022.500010
2-[(2-fluorophenyl)methylthio]-5-(4-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)IC5017.700010
[4-[(2-fluorophenyl)methoxy]phenyl]-(1-pyrrolidinyl)methanethioneHomo sapiens (human)IC505.366020
4-methyl-N,5-diphenyl-3-thiophenecarboxamideHomo sapiens (human)IC5019.300010
js 3Homo sapiens (human)IC5022.700010
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideHomo sapiens (human)IC5028.000010
5-amino-3-(2-methylphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterHomo sapiens (human)IC5093.300010
2-[[anilino(oxo)methyl]amino]-N-(phenylmethyl)benzamideHomo sapiens (human)IC5039.400010
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)IC500.145010
5-[(4-methylphenoxy)methyl]-3-phenyl-1,2,4-oxadiazoleHomo sapiens (human)IC5042.100010
3-amino-2-(4-methylphenyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)IC5012.700010
N-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)IC5019.200010
N-(1-naphthalenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineHomo sapiens (human)IC5018.500010
5-(2-chlorophenyl)-N-phenyl-2-furancarboxamideHomo sapiens (human)IC5074.300010
3-[[3-(4-morpholinyl)-1,4-dioxo-2-naphthalenyl]amino]benzoic acidHomo sapiens (human)IC5015.700010
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamineHomo sapiens (human)IC5028.000010
4-(2-quinoxalinylamino)benzoic acid ethyl esterHomo sapiens (human)IC5064.600010
4-(3-chloro-2-thiophenyl)-2-(3-pyridinyl)thiazoleHomo sapiens (human)IC5019.400010
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneHomo sapiens (human)IC503.620010
fm19g11Homo sapiens (human)IC5022.200010
1-[(3,4-dichlorophenyl)methyl]indole-2,3-dioneHomo sapiens (human)IC5022.700010
4-(6-fluoro-3-methyl-4-oxo-1-benzopyran-2-yl)-2-methyl-1-phthalazinoneHomo sapiens (human)IC509.540010
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideHomo sapiens (human)IC5035.100010
5-bromo-N-(4,7-dimethoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)IC5099.000010
3-[[[3-[(3-nitrophenyl)sulfamoyl]phenyl]-oxomethyl]amino]benzoic acidHomo sapiens (human)IC5019.200010
2,4-dithiophen-2-ylthiazoleHomo sapiens (human)IC5025.300010
4-(4-methylphenyl)-2-(3-nitrophenyl)-3-pyrazolamineHomo sapiens (human)IC5023.700010
4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-dioneHomo sapiens (human)IC5019.800010
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)IC50100.000010
2-(2-hydroxyethylamino)-3-(4-methoxyanilino)naphthalene-1,4-dioneHomo sapiens (human)IC5010.600010
N-[(2-chlorophenyl)methyl]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-5-nitro-4-triazolimineHomo sapiens (human)IC50100.000010
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-(1-phenylethylamino)ethyl] esterHomo sapiens (human)IC50100.000010
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneHomo sapiens (human)IC506.790010
N-[3-(4-methyl-1-piperazinyl)-1,4-dioxo-2-naphthalenyl]benzenesulfonamideHomo sapiens (human)IC5027.100010
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-oneHomo sapiens (human)IC5013.500010
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamideHomo sapiens (human)IC5016.200010
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] esterHomo sapiens (human)IC5023.400010
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterHomo sapiens (human)IC5028.200010
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[[oxo-[(phenylmethyl)amino]methyl]amino]ethyl] esterHomo sapiens (human)IC5013.700010
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideHomo sapiens (human)IC5026.000010
2'-hydroxy-4-methoxychalconeHomo sapiens (human)IC5023.100010
reumycinHomo sapiens (human)IC5011.400010
methylbenzethonium chlorideHomo sapiens (human)IC5039.100010
3,3'-diethylthiacarbocyanine iodideHomo sapiens (human)IC5052.800010
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamideHomo sapiens (human)IC5031.200010
dihydroxanthohumolHomo sapiens (human)IC50100.000010
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluoro-4-methylphenyl)propanamideHomo sapiens (human)IC5021.600010
2-chloro-3-[2-(4-methylphenyl)-5-tetrazolyl]pyridineHomo sapiens (human)IC509.030010
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)IC5024.000010
1-(2,3-dihydro-1H-inden-5-yl)-3-(2-ethoxyphenyl)ureaHomo sapiens (human)IC5030.800010
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineHomo sapiens (human)IC5012.500010
2-(4-methoxyphenyl)-1H-quinazolin-4-oneHomo sapiens (human)IC506.830010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
diacereinHomo sapiens (human)EC5014.284521
N-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-2-furancarboxamideHomo sapiens (human)EC50100.000020
2-(3,4-dimethoxyphenyl)-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)EC5085.318010
cefiximeHomo sapiens (human)EC50100.000010