Proteins > delta-type opioid receptor
Page last updated: 2024-08-07 15:15:25

delta-type opioid receptor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (46)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
chloroxineHomo sapiens (human)IC5032.000010
clioquinolHomo sapiens (human)IC5032.000010
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)IC5032.000010
3,4-dichloro-n-methyl-n-(2-(1-pyrrolidinyl)cyclohexyl)-benzeneacetamide, (trans)-(+-)-isomerHomo sapiens (human)IC5032.000010
2-[5-[(2-chlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)IC5032.000010
2-[5-[(2,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)IC5032.000020
2-[5-[(4-bromophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)IC5032.000020
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-propyl-2-pyridinecarboxamideHomo sapiens (human)IC5032.000010
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-2-pyridinecarboxamideHomo sapiens (human)IC5032.000010
6-[2-(2-methoxyphenyl)imino-3-(2-oxolanylmethyl)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneHomo sapiens (human)IC5032.000010
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) esterHomo sapiens (human)IC5032.000010
4-[[(4-methylphenyl)sulfonylamino]methyl]-N-[2-[(phenylmethyl)-propan-2-ylamino]ethyl]benzamideHomo sapiens (human)IC5032.000030
N-[1-(cyclopentylamino)-2-methyl-1-oxobutan-2-yl]-N-(thiophen-2-ylmethyl)-2-pyridinecarboxamideHomo sapiens (human)IC5032.000020
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(2-furanylmethyl)-2-pyridinecarboxamideHomo sapiens (human)IC5032.000020
N-[1-(cyclohexylamino)-2-methyl-1-oxobutan-2-yl]-N-(2-furanylmethyl)-2-pyridinecarboxamideHomo sapiens (human)IC5032.000020
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyrazinecarboxamideHomo sapiens (human)IC5032.000010
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyridinecarboxamideHomo sapiens (human)IC5032.000020
N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)IC5032.000010
4-methyl-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)IC5032.000010
4-methoxy-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)IC5032.000010
2-[5-[(3,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)IC5032.000010
4-[[(4-ethylphenyl)sulfonylamino]methyl]-N-[2-[(phenylmethyl)-propan-2-ylamino]ethyl]benzamideHomo sapiens (human)IC5032.000010
LSM-2536Homo sapiens (human)IC5032.000010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ethylisopropylamilorideHomo sapiens (human)EC5036.820520
chloroxineHomo sapiens (human)EC5032.000010
clioquinolHomo sapiens (human)EC5032.000010
benzethonium chlorideHomo sapiens (human)EC5092.461010
cetylpyridinium chlorideHomo sapiens (human)EC5092.485010
alfentanil hydrochlorideHomo sapiens (human)EC5046.306020
9-methoxyellipticineHomo sapiens (human)EC5064.664010
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)EC5032.000010
ici 204448Homo sapiens (human)EC5016.232020
3,4-dichloro-n-methyl-n-(2-(1-pyrrolidinyl)cyclohexyl)-benzeneacetamide, (trans)-(+-)-isomerHomo sapiens (human)EC5032.000010
chondocurine (1beta)-(+-)-isomerHomo sapiens (human)EC5027.191520
calmidazoliumHomo sapiens (human)EC5047.957520
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)EC5064.558010
2-[5-[(2-chlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)EC5048.000020
2-[5-[(2,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)EC5032.000020
2-[5-[(4-bromophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)EC5032.000020
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-propyl-2-pyridinecarboxamideHomo sapiens (human)EC5032.000010
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-2-pyridinecarboxamideHomo sapiens (human)EC5032.000010
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)EC5092.450010
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideHomo sapiens (human)EC5064.572010
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamineHomo sapiens (human)EC5054.443020
N-[(3-benzamidoanilino)-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)EC5092.473010
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideHomo sapiens (human)EC5050.022010
6-[2-(2-methoxyphenyl)imino-3-(2-oxolanylmethyl)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneHomo sapiens (human)EC5032.000010
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) esterHomo sapiens (human)EC5032.000010
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)EC5092.498020
4-[[(4-methylphenyl)sulfonylamino]methyl]-N-[2-[(phenylmethyl)-propan-2-ylamino]ethyl]benzamideHomo sapiens (human)EC5032.000020
N-[1-(cyclopentylamino)-2-methyl-1-oxobutan-2-yl]-N-(thiophen-2-ylmethyl)-2-pyridinecarboxamideHomo sapiens (human)EC5032.000020
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(2-furanylmethyl)-2-pyridinecarboxamideHomo sapiens (human)EC5032.000020
N-[1-(cyclohexylamino)-2-methyl-1-oxobutan-2-yl]-N-(2-furanylmethyl)-2-pyridinecarboxamideHomo sapiens (human)EC5032.000020
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyrazinecarboxamideHomo sapiens (human)EC5032.000010
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)EC5092.471010
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaHomo sapiens (human)EC505.924020
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideHomo sapiens (human)EC5092.498010
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyridinecarboxamideHomo sapiens (human)EC5032.000020
trimebutine maleate saltHomo sapiens (human)EC5044.301520
N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)EC5032.000010
4-methyl-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)EC5032.000010
phencyclidine hydrochlorideHomo sapiens (human)EC5017.299020
dihydroxanthohumolHomo sapiens (human)EC5064.584010
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)EC5092.481010
4-methoxy-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)EC5032.000010
cym51010Homo sapiens (human)EC502.364520
2-[5-[(3,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)EC5032.000010
4-[[(4-ethylphenyl)sulfonylamino]methyl]-N-[2-[(phenylmethyl)-propan-2-ylamino]ethyl]benzamideHomo sapiens (human)EC5032.000010