Page last updated: 2024-08-07 14:46:41
Heat shock protein HSP 90
[no definition available]
Synonyms
Eukaryotic peptide initiation factor 2 kinase, alpha-chain-associated phosphopeptide
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 2 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| geldanamycin | Oryctolagus cuniculus (rabbit) | IC50 | 1.1410 | 2 | 2 |
| novobiocin | Oryctolagus cuniculus (rabbit) | IC50 | 382.0000 | 2 | 2 |
Potential C-terminal-domain inhibitors of heat shock protein 90 derived from a C-terminal peptide helix.Bioorganic & medicinal chemistry, , Aug-01, Volume: 22, Issue:15, 2014
Identification and initial SAR of silybin: an Hsp90 inhibitor.Bioorganic & medicinal chemistry letters, , May-01, Volume: 21, Issue:9, 2011
Potential C-terminal-domain inhibitors of heat shock protein 90 derived from a C-terminal peptide helix.Bioorganic & medicinal chemistry, , Aug-01, Volume: 22, Issue:15, 2014
Identification and initial SAR of silybin: an Hsp90 inhibitor.Bioorganic & medicinal chemistry letters, , May-01, Volume: 21, Issue:9, 2011