An agent that suppresses immune function by one of several mechanisms of action. Classical cytotoxic immunosuppressants act by inhibiting DNA synthesis. Others may act through activation of T-cells or by inhibiting the activation of helper cells. In addition, an immunosuppressive agent is a role played by a compound which is exhibited by a capability to diminish the extent and/or voracity of an immune response.
| Member | Definition | Class |
|---|
| 4'-demethyldesoxypodophyllotoxin | A member of the class of furonaphthodioxoles that is (5R,5aR,8aR)-5,8,8a,9-tetrahydro-2H-furo[3',4':6,7]naphtho[2,3-d][1,3]dioxol-6(5aH)-one substituted at position 5 by a 4-hydroxy-3,5-dimethoxyphenyl group. | 4'-demethyldeoxypodophyllotoxin |
| 5-(4-phenylbutoxy)psoralen | A member of the class of psoralens that is psoralen substituted by a 4-phenylbutoxy group at position 5. It is a potent inhibitor of the voltage-gated potassium channel Kv1.3 (EC50 = 3 nM). | psora 4 |
| azaserine | A carboxylic ester resulting from the formal condensation of the carboxy group of diazoacetic acid with the alcoholic hydroxy group of L-serine. An antibiotic produced by a Streptomyces species. | azaserine |
| azathioprine | A thiopurine that is 6-mercaptopurine in which the mercapto hydrogen is replaced by a 1-methyl-4-nitroimidazol-5-yl group. It is a prodrug for mercaptopurine and is used as an immunosuppressant, prescribed for the treatment of inflammatory conditions and after organ transplantation and also for treatment of Crohn's didease and MS. | azathioprine |
| baricitinib | A pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted by a 1-[3-(cyanomethyl)-1-(ethanesulfonyl)azetidin-3-yl]-1H-pyrazol-4-yl group at position 5. It is an FDA approved selective Janus Kinase 1 and 2 (JAK1 and JAK2) inhibitor used for the treatment of rheumatoid arthritis. | baricitinib |
| betamethasone | | betamethasone |
| brasilicardin a | A diterpenoid antibiotic isolated from the culture broth of Nocardia brasiliensis IFM0406. It exhibits antitumour and strong immunosuppressive activity. | brasilicardin A |
| brequinar | A quinolinemonocarboxylic acid that is quinoline substituted by 2'-fluoro[1,1'-biphenyl]-4-yl, methyl, carboxy and fluoro groups at positions 2, 3, 4, and 6, respectively. It is an inhibitor of dihydroorotate dehydrogenase, an enzyme that is required for de novo pyrimidine biosynthesis. The compound exhibits antineoplastic and antiviral properties. | brequinar |
| brequinar sodium | An organic sodium salt of brequinar. | brequinar sodium |
| chetomin | An organic heteropentacyclic compound of the class of epipolythiodioxopiperazine. Isolated from Chaetomium globosum and Farrowia seminuda, it exhibits immunosuppressive activity. | chetomin |
| chlorambucil | A monocarboxylic acid that is butanoic acid substituted at position 4 by a 4-[bis(2-chloroethyl)amino]phenyl group. A chemotherapy drug that can be used in combination with the antibody obinutuzumab for the treatment of chronic lymphocytic leukemia. | chlorambucil |
| cladribine | 2'-Deoxyadenosine in which the hydrogen at position 2 on the purine ring has been substituted by chlorine. It inhibits the synthesis and repair of DNA, particularly in lymphocytes and monocytes, and is used as an antimetabolite antineoplastic drug for the treatment of lymphoid malignancies including hairy-cell leukaemia and chronic lymphocytic leukaemia. | cladribine |
| cyclophosphamide | The monohydrate of cyclophosphamide. | cyclophosphamide hydrate |
| cyclosporine | A cyclic nonribosomal peptide of eleven amino acids; an immunosuppressant drug widely used in post-allogeneic organ transplant to reduce the activity of the patient's immune system, and therefore the risk of organ rejection. Also causes reversible inhibition of immunocompetent lymphocytes in the G0- and G1-phase of the cell cycle. | cyclosporin A |
| cytarabine | A pyrimidine nucleoside in which cytosine is attached to D-arabinofuranose via a beta-N(1)-glycosidic bond. Used mainly in the treatment of leukaemia, especially acute non-lymphoblastic leukaemia, cytarabine is an antimetabolite antineoplastic agent that inhibits the synthesis of DNA. It also has antiviral and immunosuppressant properties. | cytarabine |
| demethylzeylasteral | A carbopolycyclic compound with formula C29H36O6, originally isolated from Tripterygium wilfordii. | demethylzeylasteral |
| dexrazoxane | | (+)-dexrazoxane |
| dimethyl sulfate | The dimethyl ester of sulfuric acid. | dimethyl sulfate |
| euonine | A sesquiterpene alkaloid that has been isolated from Tripterygium wilfordii and exhibits immunosuppressive and insecticidal properties. It was found to be identical with euonine, previously isolated from Euonymous sieboldiana. | wilformine |
| everolimus | A macrocyclic lactone that is rapamycin in which the hydroxy group attached to the cyclohexyl moiety has been converted into the corresponding 2-hydroxyethyl ether. It is an immunosuppressant and antineoplastic agent. | everolimus |
| fingolimod | An aminodiol that consists of propane-1,3-diol having amino and 2-(4-octylphenyl)ethyl substituents at the 2-position. It is a sphingosine 1-phosphate receptor modulator used for the treatment of relapsing-remitting multiple sclerosis. A prodrug, fingolimod is phosphorylated by sphingosine kinase to active metabolite fingolimod-phosphate, a structural analogue of sphingosine 1-phosphate. | fingolimod |
| fingolimod hydrochloride | The hydrochloride salt of 2-amino-2-[2-(4-octylphenyl) ethyl]-1,3-propanediol (fingolimod). | fingolimod hydrochloride |
| fludarabine phosphate | A purine arabinonucleoside monophosphate having 2-fluoroadenine as the nucleobase. A prodrug, it is rapidly dephosphorylated to 2-fluoro-ara-A and then phosphorylated intracellularly by deoxycytidine kinase to the active triphosphate, 2-fluoro-ara-ATP. Once incorporated into DNA, 2-fluoro-ara-ATP functions as a DNA chain terminator. It is used for the treatment of adult patients with B-cell chronic lymphocytic leukemia (CLL) who have not responded to, or whose disease has progressed during, treatment with at least one standard alkylating-agent containing regimenas. | fludarabine phosphate |
| flunisolide | | flunisolide |
| fluorouracil | A nucleobase analogue that is uracil in which the hydrogen at position 5 is replaced by fluorine. It is an antineoplastic agent which acts as an antimetabolite - following conversion to the active deoxynucleotide, it inhibits DNA synthesis (by blocking the conversion of deoxyuridylic acid to thymidylic acid by the cellular enzyme thymidylate synthetase) and so slows tumour growth. | 5-fluorouracil |
| fty 720p | A primary amino compound that is fingolimod in which one on the hydroxy groups has been converted into its dihydrogen phosphate derivative. It is the active metabolite of fingolimod. | fingolimod phosphate |
| gemcitabine | A 2'-deoxycytidine having geminal fluoro substituents in the 2'-position. An inhibitor of ribonucleotide reductase, gemcitabine is used in the treatment of various carcinomas, particularly non-small cell lung cancer, pancreatic cancer, bladder cancer and breast cancer. | gemcitabine |
| gemcitabine hydrochloride | A 2'-deoxycytidine hydrochloriode having geminal fluoro substituents in the 2'-position. An inhibitor of ribonucleotide reductase, gemcitabine hydrochloride is used in the treatment of various carcinomas, including non-small cell lung cancer, pancreatic cancer, bladder cancer and breast cancer. | gemcitabine hydrochloride |
| ginsenoside rd | A ginsenoside found in Panax ginseng and Panax japonicus var. major that is (20S)-ginsenoside Rg3 in which the hydroxy group at position 20 has been converted to its beta-D-glucopyranoside. | ginsenoside Rd |
| gliotoxin | A pyrazinoindole with a disulfide bridge spanning a dioxo-substituted pyrazine ring; mycotoxin produced by several species of fungi. | gliotoxin |
| hydrocortamate | | hydrocortamate |
| ifosfamide | The simplest member of the class of ifosfamides that is 1,3,2-oxazaphosphinan-2-amine 2-oxide substituted by 2-chloroethyl groups on both the nitrogen atoms respectively. It is a nitrogen mustard alkylating agent used in the treatment of advanced breast cancer. | ifosfamide |
| l 683590 | A macrolide that is produced by the fermentation of Streptomyces hygroscopicus and exhibits strong immunosuppressant properties. | ascomycin |
| leflunomide | A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 5-methyl-1,2-oxazole-4-carboxylic acid with the anilino group of 4-(trifluoromethyl)aniline. The prodrug of teriflunomide. | leflunomide |
| melphalan | A phenylalanine derivative comprising L-phenylalanine having [bis(2-chloroethyl)amino group at the 4-position on the phenyl ring. | melphalan |
| methotrexate | | methotrexate |
| mycophenolate mofetil | A carboxylic ester resulting from the formal condensation between the carboxylic acid group of mycophenolic acid and the hydroxy group of 2-(morpholin-4-yl)ethanol. In the liver, it is metabolised to mycophenolic acid, an immunosuppressant for which it is a prodrug. It is widely used to prevent tissue rejection following organ transplants as well as for the treatment of certain autoimmune diseases. | mycophenolate mofetil |
| mycophenolic acid | A member of the class of 2-benzofurans that is 2-benzofuran-1(3H)-one which is substituted at positions 4, 5, 6, and 7 by methyl, methoxy, (2E)-5-carboxy-3-methylpent-2-en-1-yl, and hydroxy groups, respectively. It is an antibiotic produced by Penicillium brevi-compactum, P. stoloniferum, P. echinulatum and related species. An immunosuppressant, it is widely used (partiularly as its sodium salt and as the 2-(morpholin-4-yl)ethyl ester prodrug, mycophenolate mofetil) to prevent tissue rejection following organ transplants and for the treatment of certain autoimmune diseases. | mycophenolic acid |
| perfosfamide | A phosphorodiamide that is the active metabolite of the nitrogen mustard cyclophosphamide. It has potent antineoplastic and immunosuppressive properties. | 4-hydroperoxycyclophosphamide |
| phenanthridone | A member of the class of phenanthridines that is phenanthridine with an oxo substituent at position 6. A poly(ADP-ribose) polymerase (PARP) inhibitor, it has been shown to exhibit immunosuppressive activity. | phenanthridone |
| physalin f | A physalin with antimalarial and antitumour activities isolated from Physalis angulata. | physalin F |
| prednisolone | A glucocorticoid that is prednisone in which the oxo group at position 11 has been reduced to the corresponding beta-hydroxy group. It is a drug metabolite of prednisone. | prednisolone |
| prednisone | A synthetic glucocorticoid drug that is particularly effective as an immunosuppressant, and affects virtually all of the immune system. Prednisone is a prodrug that is converted by the liver into prednisolone (a beta-hydroxy group instead of the oxo group at position 11), which is the active drug and also a steroid. | prednisone |
| scoparone | A member of the class of coumarins that is esculetin in which the two hydroxy groups at positions 6 and 7 are replaced by methoxy groups. It is a major constituent of the Chinese herbal medicine Yin Chen Hao, and exhibits a variety of pharmacological activities such as anti-inflammatory, anti-allergic, and anti-tumor activities. | scoparone |
| sirolimus | A macrolide lactam isolated from Streptomyces hygroscopicus consisting of a 29-membered ring containing 4 trans double bonds, three of which are conjugated. It is an antibiotic, immunosupressive and antineoplastic agent. | sirolimus |
| sotrastaurin | A member of the class of maleimides that is maleimide which is substituted at position 3 by an indol-3-yl group and at position 4 by a quinazolin-4-yl group, which in turn is substituted at position 2 by a 4-methylpiperazin-1-yl group. It is a potent and selective inhibitor of protein kinase C and has been investigated as an immunosuppresant in renal transplant patients. | sotrastaurin |
| spermine | A polyazaalkane that is tetradecane in which the carbons at positions 1, 5, 10 and 14 are replaced by nitrogens. Spermine has broad actions on cellular metabolism. | spermine |
| tacrolimus | A macrolide lactam containing a 23-membered lactone ring, originally isolated from the fermentation broth of a Japanese soil sample that contained the bacteria Streptomyces tsukubaensis. | tacrolimus (anhydrous) |
| thermozymocidin | An amino acid-based antibiotic derived from certain thermophilic fungi; acts as a potent inhibitor of serine palmitoyltransferase, the first step in sphingosine biosynthesis. Myriocin also possesses immunosuppressant activity. | myriocin |
| thiamphenicol | | thiamphenicol |
| triphenyltin chloride | An organotin compound that is triphenylstannane in which the hydrogen attached to tin is replaced by a chloro group. A fungicide used to control blights on potatoes, leaf spot diseases on sugar beet and anthracnose on beans. | fentin chloride |
| triptonide | A diterpene triepoxide that is triptobenzene K in which the acylhydroquinone moiety has undergone oxidation to the corresponding triepoxyketone derivative. It has been isolated from the roots of Tripterygium wilfordii. | triptonide |
| undecylprodigiosin | A member of the class of tripyrroles that is 1H-pyrrole substituted by (4'-methoxy-1H,5'H-[2,2'-bipyrrol]-5'-ylidene)methyl and undecyl groups at positions 2 and 5, respectively. It is a pigment produced by Stveptomyces coelicolor. | undecylprodigiosin |
| vincaleukoblastine | | vincaleukoblastine |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 29.7002 | 1 | 6 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 19.4640 | 1 | 5 |
| 67.9K protein | Vaccinia virus | Potency | 5.1180 | 2 | 21 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 39.9340 | 2 | 8 |
| acid sphingomyelinase | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 28.0959 | 2 | 9 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 26.3148 | 1 | 11 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 19.6222 | 1 | 2 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 8.9698 | 1 | 3 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Potency | 18.3564 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 23.8770 | 1 | 2 |
| AR protein | Homo sapiens (human) | Potency | 11.7700 | 12 | 174 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 19.8524 | 2 | 15 |
| arylsulfatase A | Homo sapiens (human) | Potency | 21.6211 | 1 | 3 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 7.5732 | 4 | 11 |
| Ataxin-2 | Homo sapiens (human) | Potency | 16.7237 | 2 | 18 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 16.8916 | 1 | 6 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 18.3415 | 2 | 26 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 16.9399 | 2 | 12 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 24.1907 | 1 | 6 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| caspase-3 | Cricetulus griseus (Chinese hamster) | Potency | 16.9089 | 1 | 2 |
| caspase-3 | Homo sapiens (human) | Potency | 24.1907 | 1 | 6 |
| Caspase-7 | Cricetulus griseus (Chinese hamster) | Potency | 16.9089 | 1 | 2 |
| Caspase-7 | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 15.3637 | 3 | 57 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 7.9850 | 2 | 9 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 29.9525 | 1 | 10 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 7.0193 | 2 | 2 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 12.5893 | 1 | 1 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 31.4571 | 2 | 8 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 23.5901 | 2 | 9 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 12.8577 | 2 | 8 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 19.0728 | 1 | 2 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 63.2438 | 1 | 5 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 23.5901 | 2 | 9 |
| chaperonin GroEL | Methanococcus maripaludis S2 | Potency | 79.4328 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 56.9918 | 2 | 7 |
| ClpP | Bacillus subtilis | Potency | 23.7358 | 1 | 2 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 7.9518 | 1 | 3 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 15.8614 | 1 | 2 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 24.3866 | 1 | 8 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 18.8509 | 1 | 6 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 0.0501 | 1 | 1 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 6.1624 | 2 | 14 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 13.0257 | 2 | 12 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 6.7808 | 1 | 21 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 0.9268 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 68.5229 | 1 | 7 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 36.1871 | 1 | 3 |
| dopamine D1 receptor | Homo sapiens (human) | Potency | 4.6109 | 1 | 2 |
| endonuclease IV | Escherichia coli | Potency | 9.3587 | 2 | 3 |
| Endothelin receptor type B | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 1 |
| Endothelin-1 receptor | Rattus norvegicus (Norway rat) | Potency | 17.7828 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 14.4896 | 11 | 149 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 15.1137 | 2 | 12 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 14.3178 | 10 | 123 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 12.2933 | 1 | 22 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 10.1670 | 4 | 49 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 14.8332 | 4 | 22 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 18.5307 | 1 | 3 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 16.5137 | 1 | 8 |
| G | Vesicular stomatitis virus | Potency | 24.3866 | 1 | 8 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| GALC protein | Homo sapiens (human) | Potency | 0.5773 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 6.1624 | 1 | 7 |
| geminin | Homo sapiens (human) | Potency | 10.5013 | 3 | 35 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 14.0777 | 3 | 38 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 6.8886 | 1 | 7 |
| GLS protein | Homo sapiens (human) | Potency | 25.2855 | 1 | 2 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 4.6930 | 5 | 36 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 10.9655 | 1 | 14 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 35.5473 | 2 | 3 |
| hemoglobin subunit beta | Homo sapiens (human) | Potency | 7.7121 | 5 | 11 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 15.8025 | 2 | 10 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 28.6855 | 1 | 5 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 1.7561 | 2 | 4 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 38.0803 | 2 | 29 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 24.3866 | 1 | 8 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 3.1004 | 3 | 4 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 31.6228 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 14.2187 | 2 | 7 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 19.7559 | 3 | 10 |
| IDH1 | Homo sapiens (human) | Potency | 4.1726 | 1 | 6 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 119.0470 | 1 | 2 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 24.3866 | 1 | 16 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 11.7396 | 1 | 3 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 11.7396 | 1 | 3 |
| Interferon beta | Homo sapiens (human) | Potency | 14.7135 | 3 | 30 |
| interleukin 8 | Homo sapiens (human) | Potency | 69.5421 | 1 | 3 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 4.9172 | 3 | 26 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 1.8854 | 2 | 2 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 19.3766 | 3 | 8 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 39.5209 | 1 | 4 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 22.2893 | 2 | 11 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 5.3778 | 2 | 3 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 16.7490 | 2 | 8 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 57.1368 | 1 | 5 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 6.3344 | 1 | 2 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 4.6796 | 2 | 4 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 10.0630 | 1 | 4 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 2.2882 | 1 | 3 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 25.4912 | 4 | 46 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 3.2780 | 2 | 17 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 24.7028 | 1 | 3 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 34.6258 | 1 | 4 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 17.3057 | 2 | 11 |
| nuclear receptor subfamily 1, group I, member 2 | Rattus norvegicus (Norway rat) | Potency | 10.7170 | 1 | 4 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 9.1212 | 3 | 51 |
| P53 | Homo sapiens (human) | Potency | 56.2341 | 1 | 2 |
| Parkin | Homo sapiens (human) | Potency | 1.6360 | 1 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 27.0327 | 1 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 7.6164 | 2 | 18 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 32.4566 | 1 | 6 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 12.9829 | 5 | 29 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 22.7816 | 4 | 19 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 53.9282 | 1 | 7 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 3.0946 | 1 | 7 |
| polyprotein | Zika virus | Potency | 16.5137 | 1 | 8 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 15.7142 | 1 | 2 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 22.3916 | 1 | 4 |
| PPM1D protein | Homo sapiens (human) | Potency | 10.6358 | 1 | 12 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 24.6326 | 3 | 25 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 31.0967 | 1 | 4 |
| progesterone receptor | Homo sapiens (human) | Potency | 18.3448 | 3 | 25 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 17.7828 | 2 | 2 |
| Rap guanine nucleotide exchange factor 3 | Homo sapiens (human) | Potency | 2.5119 | 1 | 1 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 11.3142 | 2 | 35 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 1.0716 | 1 | 2 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 0.4744 | 1 | 1 |
| relaxin receptor 1 isoform 1 | Homo sapiens (human) | Potency | 19.1180 | 1 | 2 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 18.9393 | 3 | 40 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 14.6591 | 4 | 34 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 6.3976 | 3 | 4 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 15.2163 | 2 | 5 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 15.2163 | 2 | 5 |
| Smad3 | Homo sapiens (human) | Potency | 15.2741 | 1 | 5 |
| snurportin-1 | Homo sapiens (human) | Potency | 119.0470 | 1 | 2 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 16.8493 | 2 | 9 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 6.8889 | 2 | 25 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 23.2867 | 1 | 5 |
| TDP1 protein | Homo sapiens (human) | Potency | 6.6477 | 2 | 87 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 20.2196 | 1 | 5 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 22.0491 | 4 | 20 |
| Thrombopoietin | Homo sapiens (human) | Potency | 6.4748 | 2 | 8 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 11.1414 | 3 | 48 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 389.7796 | 3 | 6 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 13.4688 | 6 | 13 |
| thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 6.4895 | 2 | 2 |
| transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 79.2586 | 1 | 1 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 3.0946 | 1 | 7 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 3.0946 | 1 | 7 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 78.1571 | 2 | 9 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 36.9533 | 2 | 14 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 15.0545 | 5 | 15 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 55.8143 | 1 | 7 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 10.9655 | 1 | 14 |
| Vpr | Human immunodeficiency virus 1 | Potency | 10.0000 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial | Homo sapiens (human) | IC50 | 6.7000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | IC50 | 0.0011 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus (Norway rat) | IC50 | 0.0146 | 2 | 2 |
| 6-phosphogluconate dehydrogenase, decarboxylating | Homo sapiens (human) | Ki | 136.7000 | 1 | 1 |
| Acetolactate synthase catalytic subunit, mitochondrial | Saccharomyces cerevisiae S288C | IC50 | 0.2000 | 1 | 1 |
| Adenosine receptor A3 | Rattus norvegicus (Norway rat) | Ki | 207.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 4.6300 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 4.5910 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 9.3400 | 1 | 1 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 9.3400 | 1 | 1 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 9.3400 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 20.6960 | 1 | 1 |
| Androgen receptor | Homo sapiens (human) | IC50 | 18.0000 | 2 | 2 |
| Androgen receptor | Rattus norvegicus (Norway rat) | IC50 | 42.6579 | 1 | 1 |
| Androgen receptor | Homo sapiens (human) | Ki | 2.6807 | 3 | 3 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | IC50 | 0.0170 | 1 | 1 |
| Aromatase | Homo sapiens (human) | IC50 | 0.6300 | 1 | 1 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 119.1253 | 2 | 21 |
| ATP-binding cassette sub-family C member 3 | Rattus norvegicus (Norway rat) | Ki | 90.0000 | 1 | 1 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 3.0046 | 42 | 43 |
| ATP-dependent translocase ABCB1 | Mus musculus (house mouse) | IC50 | 6.2167 | 5 | 6 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | Ki | 1.7183 | 6 | 6 |
| ATP-dependent translocase ABCB1 | Mus musculus (house mouse) | Ki | 3.5750 | 2 | 2 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Bifunctional dihydrofolate reductase-thymidylate synthase | Plasmodium falciparum K1 | IC50 | 0.0840 | 1 | 1 |
| Bifunctional dihydrofolate reductase-thymidylate synthase | Toxoplasma gondii | IC50 | 5.7614 | 29 | 39 |
| Bifunctional dihydrofolate reductase-thymidylate synthase | Trypanosoma cruzi | IC50 | 0.1100 | 1 | 1 |
| Bifunctional dihydrofolate reductase-thymidylate synthase | Leishmania major | Ki | 0.0001 | 1 | 1 |
| Bifunctional purine biosynthesis protein ATIC | Homo sapiens (human) | IC50 | 10.0050 | 2 | 2 |
| Bifunctional purine biosynthesis protein ATIC | Homo sapiens (human) | Ki | 0.8800 | 1 | 1 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 197.0182 | 8 | 44 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | IC50 | 528.0500 | 1 | 4 |
| Bile salt export pump | Homo sapiens (human) | Ki | 9.5000 | 1 | 1 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | Ki | 0.3000 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 15.8327 | 3 | 5 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Calcineurin subunit B type 1 | Homo sapiens (human) | IC50 | 34.0000 | 1 | 1 |
| Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A | Bos taurus (cattle) | IC50 | 500.0000 | 1 | 1 |
| Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B | Bos taurus (cattle) | IC50 | 500.0000 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 100.1071 | 5 | 24 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | Ki | 11.2700 | 3 | 3 |
| Canalicular multispecific organic anion transporter 1 | Rattus norvegicus (Norway rat) | Ki | 207.1920 | 5 | 5 |
| Cannabinoid receptor 1 | Rattus norvegicus (Norway rat) | Ki | 22.6000 | 1 | 1 |
| Carbonic anhydrase 1 | Homo sapiens (human) | Ki | 130.5000 | 4 | 4 |
| Carbonic anhydrase 12 | Homo sapiens (human) | Ki | 35.0667 | 3 | 3 |
| Carbonic anhydrase 13 | Mus musculus (house mouse) | Ki | 22.6000 | 1 | 1 |
| Carbonic anhydrase 14 | Homo sapiens (human) | Ki | 0.8600 | 1 | 1 |
| Carbonic anhydrase 15 | Mus musculus (house mouse) | Ki | 74.0000 | 1 | 1 |
| Carbonic anhydrase 2 | Homo sapiens (human) | Ki | 57.0000 | 4 | 4 |
| Carbonic anhydrase 3 | Homo sapiens (human) | Ki | 167.0000 | 1 | 1 |
| Carbonic anhydrase 4 | Homo sapiens (human) | Ki | 0.0100 | 1 | 1 |
| Carbonic anhydrase 5A, mitochondrial | Homo sapiens (human) | Ki | 0.4854 | 2 | 2 |
| Carbonic anhydrase 5B, mitochondrial | Homo sapiens (human) | Ki | 0.8300 | 1 | 1 |
| Carbonic anhydrase 6 | Homo sapiens (human) | Ki | 0.9900 | 1 | 1 |
| Carbonic anhydrase 7 | Homo sapiens (human) | Ki | 0.7100 | 1 | 1 |
| Carbonic anhydrase 9 | Homo sapiens (human) | Ki | 25.5333 | 3 | 3 |
| cGMP-dependent 3',5'-cyclic phosphodiesterase | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Chain A, DEOXYNUCLEOSIDE KINASE | Drosophila melanogaster (fruit fly) | IC50 | 0.7600 | 1 | 1 |
| Chain A, Inosine-5'-Monophosphate Dehydrogenase 2 | Cricetulus griseus (Chinese hamster) | Ki | 0.0060 | 1 | 1 |
| Chain A, Uracil Phosphoribosyltransferase | Toxoplasma gondii | Ki | 25.0000 | 1 | 1 |
| Collagenase ColH | Hathewaya histolytica | IC50 | 0.0240 | 1 | 1 |
| Corticosteroid-binding globulin | Homo sapiens (human) | Ki | 0.0309 | 1 | 1 |
| Cyclin-A1 | Homo sapiens (human) | IC50 | 2.3000 | 1 | 1 |
| Cyclin-A2 | Homo sapiens (human) | IC50 | 2.3000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 2.3000 | 1 | 1 |
| Cyclin-G-associated kinase | Homo sapiens (human) | IC50 | 0.1360 | 1 | 1 |
| Cysteine protease | Trypanosoma brucei rhodesiense | IC50 | 50.0000 | 1 | 1 |
| Cytidine deaminase | Homo sapiens (human) | Ki | 190.0000 | 1 | 1 |
| Cytochrome P450 11B1, mitochondrial | Bos taurus (cattle) | IC50 | 0.0012 | 2 | 5 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 33.5053 | 2 | 3 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 5.5000 | 2 | 2 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 30.2667 | 3 | 3 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 82.5500 | 2 | 2 |
| Cytochrome P450 2J2 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 2.0375 | 9 | 11 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Ki | 42.8440 | 3 | 5 |
| Cytochrome P450 3A43 | Homo sapiens (human) | IC50 | 2.0600 | 1 | 1 |
| Cytochrome P450 3A43 | Homo sapiens (human) | Ki | 7.6000 | 1 | 2 |
| Cytochrome P450 3A5 | Homo sapiens (human) | IC50 | 0.9433 | 3 | 3 |
| Cytochrome P450 3A5 | Homo sapiens (human) | Ki | 7.6000 | 1 | 2 |
| Cytochrome P450 3A7 | Homo sapiens (human) | IC50 | 2.0600 | 1 | 1 |
| Cytochrome P450 3A7 | Homo sapiens (human) | Ki | 7.6000 | 1 | 2 |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0030 | 1 | 1 |
| Deoxynucleoside kinase | Drosophila melanogaster (fruit fly) | IC50 | 5,319.0000 | 2 | 2 |
| Dihydrofolate reductase | Enterococcus faecium | IC50 | 0.0014 | 1 | 1 |
| Dihydrofolate reductase | Escherichia coli K-12 | IC50 | 4.1688 | 24 | 34 |
| Dihydrofolate reductase | Gallus gallus (chicken) | IC50 | 0.0545 | 2 | 2 |
| Dihydrofolate reductase | Homo sapiens (human) | IC50 | 1.4921 | 81 | 95 |
| Dihydrofolate reductase | Lacticaseibacillus casei | IC50 | 0.0138 | 29 | 30 |
| Dihydrofolate reductase | Mus musculus (house mouse) | IC50 | 0.0331 | 11 | 11 |
| Dihydrofolate reductase | Mycobacterium tuberculosis H37Rv | IC50 | 0.0174 | 3 | 3 |
| Dihydrofolate reductase | Pneumocystis carinii | IC50 | 0.0717 | 12 | 13 |
| Dihydrofolate reductase | Rattus norvegicus (Norway rat) | IC50 | 0.0047 | 10 | 11 |
| Dihydrofolate reductase | Escherichia coli K-12 | Ki | 34.5460 | 5 | 5 |
| Dihydrofolate reductase | Homo sapiens (human) | Ki | 0.4019 | 11 | 11 |
| Dihydrofolate reductase | Lacticaseibacillus casei | Ki | 0.0000 | 1 | 1 |
| Dihydrofolate reductase | Mus musculus (house mouse) | Ki | 0.2167 | 17 | 18 |
| Dihydrofolate reductase | Pneumocystis carinii | Ki | 0.0000 | 1 | 1 |
| Dihydrofolate reductase | Staphylococcus aureus | Ki | 0.0005 | 2 | 2 |
| Dihydrofolate reductase | Bacillus anthracis | IC50 | 0.0136 | 1 | 2 |
| Dihydrofolate reductase | Bos taurus (cattle) | IC50 | 722.1480 | 11 | 11 |
| Dihydroorotate dehydrogenase | Schistosoma mansoni | IC50 | 20.0000 | 2 | 2 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | IC50 | 2.4700 | 29 | 30 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Mus musculus (house mouse) | IC50 | 0.0300 | 1 | 1 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Rattus norvegicus (Norway rat) | IC50 | 0.1717 | 5 | 6 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | Ki | 0.0120 | 2 | 2 |
| DNA topoisomerase 1 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | IC50 | 430.0000 | 3 | 3 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| E3 ubiquitin-protein ligase Mdm2 | Homo sapiens (human) | IC50 | 0.0200 | 1 | 1 |
| E3 ubiquitin-protein ligase RNF31 | Homo sapiens (human) | IC50 | 0.5100 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] | Francisella tularensis subsp. tularensis SCHU S4 | IC50 | 59.0000 | 1 | 1 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 5.1600 | 2 | 2 |
| Equilibrative nucleoside transporter 1 | Homo sapiens (human) | IC50 | 0.1900 | 1 | 1 |
| Estrogen receptor | Homo sapiens (human) | IC50 | 55.0000 | 2 | 2 |
| Estrogen receptor | Homo sapiens (human) | Ki | 3.6667 | 3 | 3 |
| Estrogen receptor beta | Homo sapiens (human) | IC50 | 55.0000 | 2 | 2 |
| Estrogen receptor beta | Homo sapiens (human) | Ki | 1.0000 | 1 | 1 |
| Fatty acid-binding protein, liver | Rattus norvegicus (Norway rat) | Ki | 51.8300 | 2 | 2 |
| Fatty-acid amide hydrolase 1 | Mus musculus (house mouse) | IC50 | 0.0800 | 1 | 1 |
| fMet-Leu-Phe receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Focal adhesion kinase 1 | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| Folate receptor alpha | Homo sapiens (human) | IC50 | 0.2262 | 4 | 4 |
| Folate receptor beta | Homo sapiens (human) | IC50 | 0.1585 | 4 | 4 |
| Folylpolyglutamate synthase, mitochondrial | Homo sapiens (human) | IC50 | 3.2000 | 1 | 1 |
| Folylpolyglutamate synthase, mitochondrial | Mus musculus (house mouse) | Ki | 166.0000 | 1 | 1 |
| galanin receptor type 3 | Homo sapiens (human) | IC50 | 29.9000 | 1 | 1 |
| Geranylgeranyl transferase type-1 subunit beta | Homo sapiens (human) | IC50 | 17.0000 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | IC50 | 0.0737 | 41 | 44 |
| Glucocorticoid receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0565 | 3 | 3 |
| Glucocorticoid receptor | Homo sapiens (human) | Ki | 0.0323 | 15 | 18 |
| Glucose-6-phosphate 1-dehydrogenase | Homo sapiens (human) | Ki | 91.0000 | 1 | 1 |
| Glutamate receptor 1 | Rattus norvegicus (Norway rat) | IC50 | 0.0140 | 1 | 1 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | IC50 | 0.0140 | 1 | 1 |
| Glutamate receptor 3 | Rattus norvegicus (Norway rat) | IC50 | 0.0140 | 1 | 1 |
| Glutamate receptor 4 | Rattus norvegicus (Norway rat) | IC50 | 0.0140 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2D | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3A | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3B | Rattus norvegicus (Norway rat) | IC50 | 232.0000 | 1 | 1 |
| Glycine receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 0.2938 | 1 | 4 |
| Glycine receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Ki | 0.1336 | 1 | 4 |
| Glycine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 0.2938 | 1 | 4 |
| Glycine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Ki | 0.1336 | 1 | 4 |
| Glycine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 0.2938 | 1 | 4 |
| Glycine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Ki | 0.1336 | 1 | 4 |
| Glycine receptor subunit beta | Rattus norvegicus (Norway rat) | IC50 | 0.2938 | 1 | 4 |
| Glycine receptor subunit beta | Rattus norvegicus (Norway rat) | Ki | 0.1336 | 1 | 4 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 0.8700 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Histidine decarboxylase | Rattus norvegicus (Norway rat) | IC50 | 0.0014 | 1 | 1 |
| Histone-lysine N-methyltransferase EHMT2 | Homo sapiens (human) | IC50 | 3.4650 | 2 | 2 |
| Histone-lysine N-methyltransferase SUV39H1 | Homo sapiens (human) | IC50 | 0.2600 | 1 | 1 |
| Ileal sodium/bile acid cotransporter | Homo sapiens (human) | Ki | 24.0000 | 1 | 1 |
| Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens (human) | IC50 | 25.1400 | 1 | 1 |
| Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens (human) | Ki | 9.5400 | 1 | 1 |
| Inosine-5'-monophosphate dehydrogenase | Cryptococcus neoformans var. neoformans JEC21 | IC50 | 0.1200 | 1 | 1 |
| Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens (human) | IC50 | 3.3977 | 6 | 6 |
| Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens (human) | Ki | 0.0365 | 8 | 8 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | IC50 | 1.1421 | 20 | 20 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Ki | 0.0084 | 8 | 8 |
| Insulin receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Interleukin-2 | Mus musculus (house mouse) | IC50 | 0.0050 | 1 | 1 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 250.0000 | 1 | 1 |
| Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0030 | 1 | 1 |
| Large neutral amino acids transporter small subunit 1 | Rattus norvegicus (Norway rat) | Ki | 55.0000 | 1 | 1 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mineralocorticoid receptor | Homo sapiens (human) | IC50 | 0.0322 | 5 | 5 |
| Mineralocorticoid receptor | Homo sapiens (human) | Ki | 0.0186 | 2 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0030 | 1 | 1 |
| Multidrug resistance associated protein | Homo sapiens (human) | Ki | 1,200.0000 | 1 | 1 |
| Multidrug resistance-associated protein 1 | Homo sapiens (human) | IC50 | 3.5082 | 10 | 10 |
| Multidrug resistance-associated protein 1 | Homo sapiens (human) | Ki | 5.0000 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 123.7050 | 1 | 20 |
| Mycothiol S-conjugate amidase | Mycobacterium tuberculosis H37Rv | IC50 | 50.0000 | 1 | 1 |
| NF-kappa-B inhibitor alpha | Homo sapiens (human) | IC50 | 27.1000 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | IC50 | 13.4794 | 13 | 15 |
| nuclear receptor coactivator 1 isoform 1 [Homo sapiens] | Homo sapiens (human) | IC50 | 32.4483 | 2 | 3 |
| nuclear receptor coactivator 3 isoform a | Homo sapiens (human) | IC50 | 14.5410 | 2 | 3 |
| Peptidyl-prolyl cis-trans isomerase A | Homo sapiens (human) | IC50 | 0.0252 | 12 | 12 |
| Peptidyl-prolyl cis-trans isomerase A | Homo sapiens (human) | Ki | 0.0645 | 8 | 8 |
| Peptidyl-prolyl cis-trans isomerase B | Homo sapiens (human) | IC50 | 0.0088 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase D | Homo sapiens (human) | IC50 | 0.0036 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase D | Homo sapiens (human) | Ki | 0.0129 | 4 | 4 |
| Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens (human) | IC50 | 3.0260 | 10 | 13 |
| Peptidyl-prolyl cis-trans isomerase FKBP1A | Mus musculus (house mouse) | IC50 | 0.0010 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens (human) | Ki | 0.9037 | 4 | 6 |
| Peptidyl-prolyl cis-trans isomerase FKBP1B | Homo sapiens (human) | Ki | 0.0060 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase FKBP4 | Homo sapiens (human) | IC50 | 4.0080 | 1 | 2 |
| Peptidyl-prolyl cis-trans isomerase FKBP5 | Homo sapiens (human) | Ki | 0.0540 | 2 | 3 |
| Peptidylglycine alpha-amidating monooxygenase | Rattus norvegicus (Norway rat) | Ki | 0.0060 | 1 | 1 |
| Peroxisome proliferator-activated receptor alpha | Homo sapiens (human) | IC50 | 0.0031 | 1 | 6 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Mus musculus (house mouse) | IC50 | 0.5700 | 1 | 1 |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens (human) | IC50 | 0.3445 | 7 | 8 |
| Poly [ADP-ribose] polymerase 1 | Bos taurus (cattle) | IC50 | 0.3000 | 1 | 1 |
| Poly [ADP-ribose] polymerase 2 | Mus musculus (house mouse) | IC50 | 0.2080 | 1 | 2 |
| Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens (human) | IC50 | 0.1111 | 1 | 2 |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens (human) | IC50 | 0.0139 | 1 | 2 |
| Potassium voltage-gated channel subfamily A member 3 | Homo sapiens (human) | IC50 | 0.7240 | 1 | 1 |
| Potassium voltage-gated channel subfamily D member 3 | Homo sapiens (human) | IC50 | 10,000.0000 | 1 | 1 |
| Potassium voltage-gated channel subfamily E member 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 5,714.8050 | 3 | 3 |
| Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Progesterone receptor | Homo sapiens (human) | IC50 | 6.0133 | 6 | 6 |
| Progesterone receptor | Homo sapiens (human) | Ki | 5.4286 | 7 | 7 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Ki | 5.0000 | 1 | 2 |
| Proteasome subunit beta type-1 | Homo sapiens (human) | IC50 | 22.1400 | 2 | 2 |
| Proteasome subunit beta type-2 | Homo sapiens (human) | IC50 | 9.7000 | 2 | 2 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 22.2900 | 2 | 2 |
| Protein farnesyltransferase subunit beta | Homo sapiens (human) | IC50 | 40.5500 | 2 | 2 |
| Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha | Homo sapiens (human) | IC50 | 32.7000 | 3 | 3 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 0.0026 | 5 | 10 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 0.0025 | 5 | 10 |
| Protein kinase C beta type | Mus musculus (house mouse) | IC50 | 0.2340 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 0.0025 | 4 | 9 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 0.0040 | 5 | 10 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 0.0041 | 4 | 9 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 0.0094 | 6 | 11 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 5.4000 | 1 | 1 |
| Protein mono-ADP-ribosyltransferase PARP15 | Homo sapiens (human) | IC50 | 2.4559 | 1 | 2 |
| Protein-arginine deiminase type-4 | Homo sapiens (human) | IC50 | 6,833.3333 | 1 | 3 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Proton-coupled folate transporter | Homo sapiens (human) | IC50 | 0.1208 | 2 | 2 |
| Pteridine reductase 1 | Leishmania major | Ki | 0.1095 | 2 | 2 |
| Pyruvate kinase PKM | Homo sapiens (human) | IC50 | 22.6400 | 1 | 1 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| RanBP-type and C3HC4-type zinc finger-containing protein 1 | Homo sapiens (human) | IC50 | 0.5100 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Reduced folate transporter | Homo sapiens (human) | IC50 | 0.0120 | 2 | 2 |
| Reduced folate transporter | Homo sapiens (human) | Ki | 3.5000 | 1 | 1 |
| Regulatory-associated protein of mTOR | Homo sapiens (human) | IC50 | 0.1500 | 2 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 5.8200 | 1 | 1 |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | IC50 | 0.4550 | 1 | 1 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 69.5000 | 1 | 2 |
| Serine palmitoyltransferase 2 | Homo sapiens (human) | IC50 | 0.0001 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 0.0021 | 1 | 1 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | IC50 | 0.6817 | 13 | 16 |
| Serine/threonine-protein kinase mTOR | Mus musculus (house mouse) | IC50 | 0.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 0.0501 | 1 | 1 |
| Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 0.0989 | 2 | 2 |
| Serum paraoxonase/arylesterase 1 | Homo sapiens (human) | Ki | 8,973.0000 | 1 | 1 |
| Sharpin | Homo sapiens (human) | IC50 | 0.5100 | 1 | 1 |
| Sodium channel protein type 5 subunit alpha | Homo sapiens (human) | IC50 | 415.2415 | 2 | 2 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | IC50 | 2.8840 | 1 | 1 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | Ki | 2.2910 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 4.6300 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 4.5910 | 1 | 1 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | IC50 | 0.0150 | 1 | 1 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | IC50 | 0.0110 | 1 | 1 |
| Sodium/bile acid cotransporter | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Solute carrier family 22 member 20 | Mus musculus (house mouse) | Ki | 599.7800 | 1 | 2 |
| Solute carrier family 22 member 6 | Mus musculus (house mouse) | Ki | 896.1255 | 1 | 2 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | IC50 | 1.3643 | 6 | 7 |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | Ki | 0.4845 | 4 | 4 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | IC50 | 41.0000 | 2 | 2 |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | Ki | 19.3000 | 2 | 2 |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens (human) | IC50 | 37.0000 | 1 | 1 |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens (human) | Ki | 36.0000 | 1 | 1 |
| Sphingosine 1-phosphate receptor 1 | Homo sapiens (human) | IC50 | 0.2407 | 5 | 6 |
| Sphingosine 1-phosphate receptor 1 | Homo sapiens (human) | Ki | 0.2117 | 1 | 5 |
| Sphingosine 1-phosphate receptor 2 | Homo sapiens (human) | IC50 | 3.7003 | 2 | 3 |
| Sphingosine 1-phosphate receptor 2 | Homo sapiens (human) | Ki | 0.2117 | 1 | 5 |
| Sphingosine 1-phosphate receptor 3 | Homo sapiens (human) | IC50 | 3.3375 | 2 | 3 |
| Sphingosine 1-phosphate receptor 3 | Homo sapiens (human) | Ki | 0.2117 | 1 | 5 |
| Sphingosine 1-phosphate receptor 4 | Homo sapiens (human) | IC50 | 3.3433 | 2 | 3 |
| Sphingosine 1-phosphate receptor 4 | Homo sapiens (human) | Ki | 0.2117 | 1 | 5 |
| Sphingosine 1-phosphate receptor 5 | Homo sapiens (human) | IC50 | 1.0504 | 1 | 2 |
| Sphingosine 1-phosphate receptor 5 | Homo sapiens (human) | Ki | 0.2117 | 1 | 5 |
| Sphingosine-1-phosphate lyase 1 | Homo sapiens (human) | IC50 | 34.5000 | 2 | 2 |
| Sphingosine-1-phosphate lyase 1 | Mus musculus (house mouse) | IC50 | 52.4000 | 1 | 1 |
| Splicing factor 3B subunit 3 | Homo sapiens (human) | IC50 | 0.0124 | 2 | 2 |
| Substance-K receptor | Homo sapiens (human) | IC50 | 4.1390 | 1 | 1 |
| Substance-K receptor | Homo sapiens (human) | Ki | 1.3800 | 1 | 1 |
| Target of rapamycin complex subunit LST8 | Homo sapiens (human) | IC50 | 0.1500 | 2 | 3 |
| Thymidine kinase | Human alphaherpesvirus 1 (Herpes simplex virus type 1) | IC50 | 1,000.0000 | 1 | 1 |
| Thymidine kinase | Human alphaherpesvirus 1 strain SC16 | IC50 | 1,000.0000 | 1 | 1 |
| Thymidine kinase | Human herpesvirus 3 strain Dumas | IC50 | 1,000.0000 | 2 | 2 |
| Thymidine kinase 2, mitochondrial | Homo sapiens (human) | IC50 | 1,000.0000 | 2 | 2 |
| Thymidine kinase, cytosolic | Homo sapiens (human) | IC50 | 1,000.0000 | 2 | 2 |
| Thymidylate synthase | Escherichia coli K-12 | IC50 | 11.4303 | 3 | 12 |
| Thymidylate synthase | Homo sapiens (human) | IC50 | 33.6082 | 12 | 21 |
| Thymidylate synthase | Lacticaseibacillus casei | IC50 | 158.1000 | 10 | 10 |
| Thymidylate synthase | Mus musculus (house mouse) | IC50 | 7.2375 | 8 | 8 |
| Thymidylate synthase | Homo sapiens (human) | Ki | 0.6000 | 1 | 1 |
| Thymidylate synthase | Mus musculus (house mouse) | Ki | 45.0000 | 1 | 1 |
| Thymidylate synthase | Escherichia coli | IC50 | 60.6000 | 3 | 3 |
| Thymidylate synthase | Escherichia coli LF82 | IC50 | 18.0000 | 1 | 1 |
| Toll-like receptor 4 | Homo sapiens (human) | IC50 | 1.0400 | 1 | 1 |
| transactivating tegument protein VP16 [Human herpesvirus 1] | Human alphaherpesvirus 1 (Herpes simplex virus type 1) | IC50 | 29.3350 | 2 | 3 |
| Transthyretin | Homo sapiens (human) | Ki | 0.0026 | 1 | 1 |
| Trifunctional purine biosynthetic protein adenosine-3 | Homo sapiens (human) | IC50 | 10.0050 | 2 | 2 |
| Trifunctional purine biosynthetic protein adenosine-3 | Mus musculus (house mouse) | IC50 | 20.0000 | 2 | 2 |
| Tubulin alpha-1A chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin alpha-1B chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin alpha-1C chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin alpha-3C chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin alpha-3E chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin alpha-4A chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-1 chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-2A chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-2B chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-3 chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-4A chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-4B chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-6 chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tubulin beta-8 chain | Homo sapiens (human) | IC50 | 1.3700 | 2 | 2 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 3.3000 | 1 | 1 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 5.5000 | 1 | 1 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | IC50 | 0.4023 | 21 | 22 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | IC50 | 0.5348 | 22 | 24 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | IC50 | 1.1568 | 12 | 12 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | IC50 | 9.1000 | 1 | 1 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| UDP-glucuronosyltransferase 1-6 | Homo sapiens (human) | IC50 | 211.8333 | 1 | 6 |
| UDP-glucuronosyltransferase 1A1 | Homo sapiens (human) | IC50 | 211.8333 | 1 | 6 |
| UDP-glucuronosyltransferase 1A4 | Homo sapiens (human) | IC50 | 211.8333 | 1 | 6 |
| UDP-glucuronosyltransferase 2B10 | Homo sapiens (human) | IC50 | 211.8333 | 1 | 6 |
| UDP-glucuronosyltransferase 2B7 | Homo sapiens (human) | IC50 | 211.8333 | 1 | 6 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 3.9000 | 1 | 1 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | IC50 | 4.6000 | 1 | 1 |
| Zinc finger protein GLI1 | Homo sapiens (human) | IC50 | 0.6600 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit beta-1 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | EC50 | 0.0168 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Adenosine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | EC50 | 5.2867 | 1 | 3 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0097 | 6 | 9 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | EC50 | 25.7799 | 8 | 8 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Aurora kinase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Aurora kinase B | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| bcl-2-like protein 11 isoform 1 | Homo sapiens (human) | EC50 | 350.0000 | 1 | 1 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 15.0427 | 3 | 6 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | EC50 | 1.7500 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 22.5780 | 1 | 4 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 22.5608 | 1 | 4 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 23.3992 | 1 | 4 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Carbonic anhydrase 2 | Homo sapiens (human) | EC50 | 0.0010 | 1 | 1 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 22.9382 | 1 | 4 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 20.0883 | 1 | 3 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Caspase-2 | Homo sapiens (human) | EC50 | 8.5000 | 1 | 1 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Chain A, BCL-2-RELATED PROTEIN A1 | Homo sapiens (human) | EC50 | 350.0000 | 1 | 1 |
| Chain B, DIHYDROFOLATE REDUCTASE | Escherichia coli | Kd | 0.1344 | 1 | 5 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 23.5902 | 1 | 4 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | EC50 | 0.0010 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 11.9178 | 5 | 8 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cytochrome P450 3A4 | Homo sapiens (human) | EC50 | 0.0001 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Kd | 0.0130 | 1 | 1 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dihydrofolate reductase | Escherichia coli K-12 | EC50 | 0.0010 | 1 | 1 |
| Dihydrofolate reductase | Escherichia coli K-12 | Kd | 0.3062 | 10 | 10 |
| Dihydroorotate dehydrogenase (quinone), mitochondrial | Homo sapiens (human) | EC50 | 0.0550 | 1 | 1 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 22.6945 | 1 | 4 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 22.5302 | 1 | 4 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Estrogen receptor | Rattus norvegicus (Norway rat) | EC50 | 4.0180 | 1 | 2 |
| Estrogen receptor beta | Rattus norvegicus (Norway rat) | EC50 | 4.0180 | 1 | 2 |
| Eukaryotic peptide chain release factor GTP-binding subunit ERF3B | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 24.0670 | 1 | 5 |
| Eukaryotic translation initiation factor 4E | Homo sapiens (human) | Kd | 0.0005 | 1 | 1 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Glucocorticoid receptor | Homo sapiens (human) | EC50 | 0.0291 | 41 | 41 |
| Glucocorticoid receptor | Mus musculus (house mouse) | EC50 | 0.0046 | 2 | 2 |
| Glucocorticoid receptor | Rattus norvegicus (Norway rat) | EC50 | 0.0196 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | Kd | 0.0290 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | EC50 | 100.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Homo sapiens (human) | EC50 | 126.0000 | 2 | 2 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | EC50 | 90.5000 | 2 | 2 |
| Glutamine synthetase | Homo sapiens (human) | EC50 | 0.0320 | 1 | 1 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 24.2402 | 1 | 5 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 24.1418 | 1 | 5 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| High mobility group protein B1 | Homo sapiens (human) | Kd | 0.2620 | 2 | 2 |
| Histamine H1 receptor | Cavia porcellus (domestic guinea pig) | EC50 | 0.0026 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Insulin receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Isoleucine--tRNA ligase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| MAP kinase-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 22.5260 | 1 | 4 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| matrix metalloproteinase 1, partial | Homo sapiens (human) | EC50 | 5.6500 | 1 | 1 |
| Membrane-associated progesterone receptor component 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mineralocorticoid receptor | Homo sapiens (human) | EC50 | 0.0010 | 2 | 2 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 20.0137 | 1 | 3 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 22.9727 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 22.8950 | 1 | 4 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Multidrug resistance-associated protein 1 | Homo sapiens (human) | EC50 | 1.7000 | 1 | 1 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Nociceptin receptor | Rattus norvegicus (Norway rat) | EC50 | 0.0034 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 22.6555 | 1 | 4 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Nuclear receptor subfamily 1 group I member 2 | Homo sapiens (human) | EC50 | 5.2967 | 2 | 3 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 24.5495 | 1 | 4 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| ORF73 | Human gammaherpesvirus 8 | EC50 | 75.0000 | 1 | 1 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Peptidyl-prolyl cis-trans isomerase A | Homo sapiens (human) | Kd | 0.6225 | 11 | 11 |
| Peptidyl-prolyl cis-trans isomerase B | Homo sapiens (human) | Kd | 0.0098 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase D | Homo sapiens (human) | Kd | 0.0215 | 2 | 2 |
| Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens (human) | EC50 | 0.0101 | 4 | 4 |
| Peptidyl-prolyl cis-trans isomerase FKBP1B | Homo sapiens (human) | Kd | 0.0003 | 1 | 2 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Peroxisome proliferator-activated receptor gamma | Homo sapiens (human) | Kd | 110.0000 | 1 | 1 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Procathepsin L | Homo sapiens (human) | EC50 | 5.2867 | 1 | 3 |
| Programmed cell death protein 4 | Homo sapiens (human) | EC50 | 0.0500 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 15.5210 | 1 | 4 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 21.5870 | 1 | 4 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 15.2700 | 1 | 4 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 22.5032 | 1 | 4 |
| Protein kinase C zeta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 22.7432 | 1 | 4 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Rab-like protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ras-related C3 botulinum toxin substrate 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | EC50 | 5.2867 | 1 | 3 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | EC50 | 5.2867 | 1 | 3 |
| Replicase polyprotein 1ab | Human coronavirus 229E | EC50 | 5.2867 | 1 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | EC50 | 5.2867 | 1 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | EC50 | 5.2867 | 1 | 3 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 22.6205 | 1 | 4 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 24.1512 | 1 | 5 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 22.8930 | 1 | 4 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Septin-9 | Homo sapiens (human) | Kd | 22.5210 | 1 | 4 |
| Serine palmitoyltransferase 1 | Homo sapiens (human) | EC50 | 0.0495 | 1 | 1 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase ATR | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 24.1722 | 1 | 4 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 22.5312 | 1 | 4 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 0.0013 | 1 | 2 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 15.7645 | 1 | 4 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 22.5672 | 1 | 4 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 24.7105 | 1 | 4 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 22.7025 | 1 | 4 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Sphingosine 1-phosphate receptor 1 | Homo sapiens (human) | EC50 | 1.0469 | 21 | 22 |
| Sphingosine 1-phosphate receptor 2 | Homo sapiens (human) | EC50 | 10.0000 | 1 | 2 |
| Sphingosine 1-phosphate receptor 3 | Homo sapiens (human) | EC50 | 1.7449 | 12 | 13 |
| Sphingosine 1-phosphate receptor 4 | Homo sapiens (human) | EC50 | 1.4356 | 6 | 7 |
| Sphingosine 1-phosphate receptor 5 | Homo sapiens (human) | EC50 | 1.3227 | 9 | 10 |
| Spike glycoprotein | Betacoronavirus England 1 | EC50 | 5.2867 | 1 | 3 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | EC50 | 5.2867 | 1 | 3 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| streptokinase A precursor | Streptococcus pyogenes M1 GAS | EC50 | 2.3790 | 2 | 2 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 22.5095 | 1 | 4 |
| Transmembrane protease serine 2 | Homo sapiens (human) | EC50 | 5.2867 | 1 | 3 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | EC50 | 0.0010 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 22.5195 | 1 | 4 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |