Page last updated: 2024-08-07 16:34:08
Nociceptin receptor
A nociceptin receptor that is encoded in the genome of rat. [OMA:P35370, PRO:DNx]
Synonyms
Kappa-type 3 opioid receptor;
KOR-3;
Orphanin FQ receptor;
ROR-C;
XOR1
Research
Bioassay Publications (5)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
nociceptin | Rattus norvegicus (Norway rat) | IC50 | 0.0006 | 5 | 9 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
prednisolone | Rattus norvegicus (Norway rat) | EC50 | 0.0034 | 1 | 1 |
nociceptin | Rattus norvegicus (Norway rat) | EC50 | 0.0160 | 6 | 9 |
nociceptin | Rattus norvegicus (Norway rat) | Kd | 0.0004 | 5 | 5 |